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Outros inibidores

Outros inibidores

Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.

Foram encontrados 36770 produtos de "Outros inibidores"

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  • Copper(II) ionophore I

    CAS:
    Copper(II) ionophore I is an active compound.
    Fórmula:C26H44N2S4
    Cor e Forma:Solid
    Peso molecular:512.90
  • AZD-3199 dihydrobromide

    CAS:
    <p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>
    Fórmula:C32H44Br2N4O4S
    Cor e Forma:Solid
    Peso molecular:740.59
  • SENP2-IN-1

    CAS:
    SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.
    Fórmula:C32H29N3O5S2
    Cor e Forma:Solid
    Peso molecular:599.72
  • M-COPA

    CAS:
    M-COPA disrupts Golgi, blocks MET & Arf1 activation, and inhibits angiogenesis via VEGFR & NF-kB pathways.
    Fórmula:C25H34N2O2
    Cor e Forma:Solid
    Peso molecular:394.55
  • Oudenone

    CAS:
    <p>Oudenone is an oxygen-containing heterocyclic antibiotic with mild antibacterial and antifungal properties. It also exhibits antihypertensive effects in rats with spontaneous hypertension.</p>
    Fórmula:C12H16O3
    Cor e Forma:Solid
    Peso molecular:208.254
  • L-739750

    CAS:
    <p>L-739,750 is an inhibitor (FTI) of peptidomimetic farnesyltransferase.</p>
    Fórmula:C23H39N3O6S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:517.7
  • PARP10/15-IN-1


    PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].
    Fórmula:C13H10N2O3S
    Cor e Forma:Solid
    Peso molecular:274.3
  • Ataprost

    CAS:
    Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.
    Fórmula:C21H32O4
    Cor e Forma:Solid
    Peso molecular:348.48
  • PDE4-IN-12


    PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).
    Fórmula:C34H35NO6
    Cor e Forma:Solid
    Peso molecular:553.64
  • BRD-K25923209

    CAS:
    BRD-K25923209 is a novel inhibitor of BAF transcriptional repression.
    Fórmula:C29H36N4O3
    Cor e Forma:Solid
    Peso molecular:488.62
  • MSK-195

    CAS:
    MSK-195 is an effective TRPV1 agonist.
    Fórmula:C28H40N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:484.63
  • Miyakamide B2

    CAS:
    Miyakamide B2 is an antibiotic with insecticidal properties. It suppresses the growth of brine shrimp and shows weak activity against Xanthomonas species. The IC50 for inhibition of P388 cells by Miyakamide B2 is 7.6 μg/mL.
    Fórmula:C31H32N4O4
    Cor e Forma:Solid
    Peso molecular:524.61
  • 2-PPA

    CAS:
    2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.
    Fórmula:C11H10N2
    Cor e Forma:Solid
    Peso molecular:170.21
  • Fumarranol

    CAS:
    Fumarranol inhibits angiogenesis and malaria growth by targeting PfMAP2.
    Fórmula:C16H24O4
    Cor e Forma:Solid
    Peso molecular:280.36
  • Longicoricin

    CAS:
    <p>Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.</p>
    Fórmula:C37H68O6
    Cor e Forma:Solid
    Peso molecular:608.93
  • MRS-2339

    CAS:
    MRS-2339 is a P2X receptor activator.
    Fórmula:C12H15ClN5O6P
    Cor e Forma:Solid
    Peso molecular:391.70
  • Vimirogant hydrochloride


    Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), >1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.
    Fórmula:C27H36ClF3N4O3S
    Cor e Forma:Solid
    Peso molecular:588.21487
  • UTPγS trisodium salt

    CAS:
    P2Y2 and P2Y4 receptor agonist
    Fórmula:C9H12N2Na3O14P3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:566.15
  • CN-716 HCl

    CAS:
    cn-716 is a novel Zika virus (ZIKV) NS2B-NS3pro protease inhibitor.
    Fórmula:C22H33BCl2N6O4
    Cor e Forma:Solid
    Peso molecular:527.25
  • Croconic acid disodium

    CAS:
    <p>Croconic acid (disodium) (Nacr) enhances gene expression related to lysine crotonylation (Kcr) modification, which promotes cell growth and proliferation. This compound also shows promise in boosting somatic cell nuclear transfer (SCNT) efficiency and optimizing research in cell culture conditions.</p>
    Fórmula:C5Na2O5
    Cor e Forma:Solid
    Peso molecular:186.03
  • SGLT1/2-IN-1

    CAS:
    SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.
    Fórmula:C25H28O8
    Cor e Forma:Solid
    Peso molecular:456.48
  • NRMA-8

    CAS:
    <p>NRMA-8 is a small-molecule nuclear receptor modulator capable of penetrating the brain. It holds potential for research into central nervous system (CNS) diseases, including Alzheimer's disease, Parkinson's disease, demyelinating diseases, and glioblastoma.</p>
    Fórmula:C20H23ClN2O3
    Cor e Forma:Solid
    Peso molecular:374.86
  • AP-6

    CAS:
    AP-6, a selective TMEM175 inhibitor, enhances lysosomal macromolecular catabolism by acutely inhibiting TMEM175, thus speeding up macrophage and other digestive activities. This compound holds potential for use in Parkinson's disease research due to its role in modulating lysosomal function.
    Fórmula:C16H14N4
    Cor e Forma:Solid
    Peso molecular:262.31
  • GSK340


    <p>GSK340 is a BET inhibitor.</p>
    Fórmula:C26H31N3O2
    Cor e Forma:Solid
    Peso molecular:417.55
  • OP-2507

    CAS:
    OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.
    Fórmula:C25H41NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:419.6
  • CH-38083

    CAS:
    CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.
    Fórmula:C18H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:337.84
  • GS-9160

    CAS:
    GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.
    Fórmula:C20H18FN3O4S
    Cor e Forma:Solid
    Peso molecular:415.44
  • AM-3189

    CAS:
    <p>AM-3189: potent, selective GPR40 agonist with low CNS penetration, good pharmacokinetics, and efficacy mirroring AMG 837.</p>
    Fórmula:C27H25ClN2O3
    Cor e Forma:Solid
    Peso molecular:460.95
  • NS2B/NS3-IN-4

    CAS:
    <p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>
    Fórmula:C15H11NO4
    Cor e Forma:Solid
    Peso molecular:269.25
  • Butaprost

    CAS:
    <p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>
    Fórmula:C24H40O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:408.57
  • AMG-222 tosylate

    CAS:
    <p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>
    Fórmula:C39H47N9O6S
    Cor e Forma:Solid
    Peso molecular:769.91
  • DC1SMe

    CAS:
    <p>DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.</p>
    Fórmula:C35H30ClN5O4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:684.23
  • Fosfazinomycin B

    CAS:
    <p>Fosfazinomycin B exhibits activity against plant pathogenic fungi such as the rice blast pathogen (Xanthomonas oryzae).</p>
    Fórmula:C10H23N6O6P
    Cor e Forma:Solid
    Peso molecular:354.3
  • GW-597901 cinnamate

    CAS:
    <p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>
    Fórmula:C34H46N2O8S
    Cor e Forma:Solid
    Peso molecular:642.80
  • RORγt inhibitor 2

    CAS:
    <p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>
    Fórmula:C31H33F5N2O7S
    Cor e Forma:Solid
    Peso molecular:672.66
  • P-gp modulator 3


    <p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>
    Fórmula:C31H37N3O5
    Cor e Forma:Solid
    Peso molecular:531.64
  • 3HKT-IN-1

    CAS:
    3HKT-IN-1 (Compound 17122279) is an inhibitor of Anopheles gambiae 3-hydroxykynurenine transaminase (3HKT) and is utilized in malaria research.
    Fórmula:C12H11BrN2O3
    Cor e Forma:Solid
    Peso molecular:311.131
  • Antitumor agent-75


    <p>Antitumor agent-75 is a novel and potent antitumor agent.</p>
    Fórmula:C26H23FN6
    Cor e Forma:Solid
    Peso molecular:438.5
  • Haliangicin D

    CAS:
    <p>Haliangicin D exhibits antifungal activity against filamentous fungi and is also effective against oomycetes, though it lacks antibacterial properties.</p>
    Fórmula:C22H32O5
    Cor e Forma:Solid
    Peso molecular:376.49
  • MK-1220

    CAS:
    MK-1220 is a novel Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure.
    Fórmula:C40H53N5O9S
    Cor e Forma:Solid
    Peso molecular:779.94
  • SL agonist 1

    CAS:
    <p>SL agonist 1, a Strigolactone (SL) agonist, is effective in promoting Arabidopsis seed germination through its recognition by the SL receptors OmKAI2d3 and OmKAI2d4.</p>
    Fórmula:C11H8FNO5
    Cor e Forma:Solid
    Peso molecular:253.18
  • SARS-CoV-2 nsp14-IN-2


    <p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>
    Fórmula:C21H21N5O5S
    Cor e Forma:Solid
    Peso molecular:455.49
  • KT2-962

    CAS:
    <p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>
    Fórmula:C23H27ClNNaO5S2
    Cor e Forma:Solid
    Peso molecular:520.04
  • Memnobotrin B

    CAS:
    Memnobotrin B is an antibiotic that exhibits inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.
    Fórmula:C27H37NO6
    Cor e Forma:Solid
    Peso molecular:471.59
  • Topoisomerase I/II inhibitor 2


    <p>Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.</p>
    Fórmula:C19H16N2O4
    Cor e Forma:Solid
    Peso molecular:336.34
  • Coriolin B

    CAS:
    <p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Fórmula:C23H36O6
    Cor e Forma:Solid
    Peso molecular:408.528
  • Diarylalkane derivative 1

    CAS:
    Diarylalkane derivative 1 is used for the research of pancreatitis.
    Fórmula:C34H51NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:537.77
  • Epicochlioquinone A

    CAS:
    <p>Epicochlioquinone A inhibits rat liver microsomal ACAT with an IC50 of 1.7 μM and inhibits plasma lecithin-cholesterol acyltransferase (LCAT) with an IC50 of 15.8 μM. At a dosage of 75 mg/kg, it can reduce cholesterol absorption in rats by 50%.</p>
    Fórmula:C30H44O8
    Cor e Forma:Solid
    Peso molecular:532.666
  • ASB14780


    ASB14780 is a 4-phenoxy derivative and an inhibitor of cytoplasmic phospholipase cPLA2α (IC50: 20 nM).
    Cor e Forma:Solid
  • Carmegliptin dihydrochloride

    CAS:
    <p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>
    Fórmula:C20H30Cl2FN3O3
    Cor e Forma:Solid
    Peso molecular:450.38
  • Heme Oxygenase-1-IN-2


    <p>Heme Oxygenase-1-IN-2 is a novel inhibitor of heme oxygenase-1 (HO-1), displaying potent antiproliferative activity in vitro, with an IC50 value of 0.95 μM.</p>
    Fórmula:C19H18ClN3O
    Cor e Forma:Solid
    Peso molecular:339.82
  • SK&amp;F 108361

    CAS:
    <p>SK&amp;F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.</p>
    Fórmula:C24H48N6O6
    Cor e Forma:Solid
    Peso molecular:516.67
  • EP-7041 HCl

    CAS:
    EP-7041 is a novel, potent, and selective Factor XIa inhibitor.
    Fórmula:C19H27ClN4O4
    Cor e Forma:Solid
    Peso molecular:410.89
  • STA-1474

    CAS:
    STA-1474, a soluble prodrug of ganetespib (STA-9090), becomes a strong HSP90 inhibitor effective against canine tumors.
    Fórmula:C20H21N4O6P
    Cor e Forma:Solid
    Peso molecular:444.38
  • PTP1B-IN-18


    PTP1B-IN-18 is an orally active, fully mixed protein tyrosine phosphatase 1B (PTP1B) inhibitor (Ki: 35.2 μM).PTP1B-IN-18 can be used to study type 2 diabetes.
    Fórmula:C26H19N3O4S
    Cor e Forma:Solid
    Peso molecular:469.51
  • CU-2010

    CAS:
    <p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>
    Fórmula:C37H42N6O6S
    Cor e Forma:Solid
    Peso molecular:698.83
  • L-2,5-Dihydrophenylalanine

    CAS:
    <p>L-2,5-Dihydrophenylalanine can induce apoptosis in human medulloblastoma leukemia cells [HL-60].</p>
    Fórmula:C9H13NO2
    Cor e Forma:Solid
    Peso molecular:167.21
  • 13-Hydroxyglucopiericidin A

    CAS:
    13-Hydroxyglucopiericidin A is an antibiotic with potent antitumor cell activity.
    Fórmula:C31H47NO10
    Cor e Forma:Solid
    Peso molecular:593.706
  • Pradimicin Q

    CAS:
    Pradimicin Q is an antibiotic exhibiting cytotoxicity against human colon HCT-116 cells and mouse melanoma B16-F10 cells, with IC50 values of 75 μg/mL and 100 μg/mL, respectively.
    Fórmula:C24H16O10
    Cor e Forma:Solid
    Peso molecular:464.378
  • PD-L1-IN-1


    <p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>
    Fórmula:C21H23N5O2
    Cor e Forma:Solid
    Peso molecular:377.44
  • Pulvilloric acid

    CAS:
    Pulvilloric acid is an antifungal antibiotic produced by the organism Pen. pulvillorum 504.
    Fórmula:C15H18O5
    Cor e Forma:Solid
    Peso molecular:278.30
  • LAF-153

    CAS:
    LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.
    Fórmula:C18H32N2O7
    Cor e Forma:Solid
    Peso molecular:388.46
  • KUS121

    CAS:
    <p>KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.</p>
    Fórmula:C22H17FN4NaO3S
    Cor e Forma:Solid
    Peso molecular:459.45
  • PKG1α activator 3


    PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).
    Fórmula:C27H26Cl2N2O6
    Cor e Forma:Solid
    Peso molecular:545.41
  • LY2934747

    CAS:
    <p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>
    Fórmula:C10H13NO4
    Cor e Forma:Solid
    Peso molecular:211.21
  • IACS-8779 disodium

    CAS:
    IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.
    Fórmula:C21H23N9Na2O10P2S2
    Cor e Forma:Solid
    Peso molecular:733.52
  • Defucogilvocarcin V

    CAS:
    <p>Defucogilvocarcin V is an antibiotic with activity against Gram-positive bacteria.</p>
    Fórmula:C21H16O5
    Cor e Forma:Solid
    Peso molecular:348.349
  • Phenazostatin A

    CAS:
    <p>Phenazostatin A is a phenazine compound known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. Phenazostatin A inhibits glutamate toxicity in N18-RE-105 cells with an EC50 of 0.34 μg/mL.</p>
    Fórmula:C28H20N4O3
    Cor e Forma:Solid
    Peso molecular:460.48
  • Curromycin A

    CAS:
    <p>Curromycin A exhibits antibacterial activity against Gram-positive bacteria such as Bacillus subtilis. Additionally, it can inhibit the replication of the human immunodeficiency virus (HIV) and suppresses the growth of mouse melanoma B16 and leukemia P388 cells.</p>
    Fórmula:C38H55N3O10
    Cor e Forma:Solid
    Peso molecular:713.857
  • Bacithrocin C

    CAS:
    Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.
    Fórmula:C18H27N5O3
    Cor e Forma:Solid
    Peso molecular:361.439
  • Dienomycin B

    CAS:
    <p>Dienomycin B exhibits mild antibacterial activity.</p>
    Fórmula:C18H23NO2
    Cor e Forma:Solid
    Peso molecular:285.38
  • Barixibat

    CAS:
    Barixibat is a bile acid transport inhibitor.
    Fórmula:C42H55N5O8
    Cor e Forma:Solid
    Peso molecular:757.91
  • Fusarin C

    CAS:
    Fusarin C is a mutagenic compound found in strains of the Fusarium genus.
    Fórmula:C23H29NO7
    Cor e Forma:Solid
    Peso molecular:431.479
  • Exfoliamycin

    CAS:
    <p>Exfoliamycin is a naphthoquinone antibiotic found in the Streptomyces strain Exfoliamycin Tu 1424, and it exhibits activity against Gram-positive bacteria.</p>
    Fórmula:C22H26O9
    Cor e Forma:Solid
    Peso molecular:434.436
  • Vulolisib

    CAS:
    <p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>
    Fórmula:C18H19F2N5O3S
    Cor e Forma:Solid
    Peso molecular:423.44
  • Antibiotic MA 144M2

    CAS:
    <p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>
    Fórmula:C42H55NO16
    Cor e Forma:Solid
    Peso molecular:829.88
  • Fudecalone

    CAS:
    <p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>
    Fórmula:C15H22O3
    Cor e Forma:Solid
    Peso molecular:250.33
  • Oximidine Ⅲ

    CAS:
    <p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>
    Fórmula:C23H24N2O6
    Cor e Forma:Solid
    Peso molecular:424.45
  • Cremeomycin

    CAS:
    <p>Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.</p>
    Fórmula:C8H6N2O4
    Cor e Forma:Solid
    Peso molecular:194.144
  • RORγt modulator 5

    CAS:
    <p>RORγt modulator 5, a potent RORγt modulator, exhibits a dissociation constant (K_i) of &lt;100 nM.</p>
    Fórmula:C27H22F5N3O6S
    Cor e Forma:Solid
    Peso molecular:611.54
  • 9-cis-13,14-Dihydroretinoic acid

    CAS:
    <p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>
    Fórmula:C20H30O2
    Cor e Forma:Solid
    Peso molecular:302.451
  • AZD-4121

    CAS:
    <p>AZD-4121 is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>
    Fórmula:C36H39F2N3O7S
    Cor e Forma:Solid
    Peso molecular:695.77
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Fórmula:C20H12F3NO5
    Cor e Forma:Solid
    Peso molecular:403.31
  • Terfluranol

    CAS:
    Terfluranol, a benzyl derivative, is utilized as an antitumor medication.
    Fórmula:C17H17F3O2
    Cor e Forma:Solid
    Peso molecular:310.31
  • Rivenprost

    CAS:
    Rivenprost, selective EP4 agonist (Ki: 0.7 nM), promotes bone growth, osteoblast differentiation, and aids wound healing.
    Fórmula:C24H34O6S
    Cor e Forma:Solid
    Peso molecular:450.59
  • Glidobactin G

    CAS:
    <p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>
    Fórmula:C27H44N4O7
    Cor e Forma:Solid
    Peso molecular:536.661
  • 3-O-Demethylmonensin A

    CAS:
    3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).
    Fórmula:C35H60O11
    Cor e Forma:Solid
    Peso molecular:656.84
  • Seldomycin factor 1

    CAS:
    Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.
    Fórmula:C17H34N4O10
    Cor e Forma:Solid
    Peso molecular:454.473
  • Gentamicin C2

    CAS:
    <p>Gentamicin C2 is an aminoglycoside antibiotic.</p>
    Fórmula:C20H41N5O7
    Cor e Forma:Solid
    Peso molecular:463.569
  • Lunacalcipol

    CAS:
    Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.
    Fórmula:C28H42O4S
    Cor e Forma:Solid
    Peso molecular:474.7
  • 9(S),10(S),13(S)-TriHOME

    CAS:
    9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.
    Fórmula:C18H34O5
    Cor e Forma:Solid
    Peso molecular:330.46
  • Deoxyradicinin

    CAS:
    <p>Deoxyradicinin is a biosynthetic precursor of Radicinin. It can inhibit Xylella fastidiosa and Liberibacter crescens, with a minimum inhibitory concentration (MIC) of 3.5 μg/mL against Liberibacter crescens. Deoxyradicinin is applicable for research on controlling plant diseases caused by these pathogens.</p>
    Fórmula:C12H12O4
    Cor e Forma:Solid
    Peso molecular:220.221
  • 1-Hydroxyoxaunomycin

    CAS:
    <p>1-Hydroxyoxaunomycin is an antibiotic that inhibits the growth of U210 cells as well as the synthesis of DNA and RNA, with IC50 values of 0.0005 μg/mL, 1.00 μg/mL, and 0.76 μg/mL, respectively.</p>
    Fórmula:C26H29NO11
    Cor e Forma:Solid
    Peso molecular:531.509
  • 16-Hydroxyroridin L-2

    CAS:
    <p>16-Hydroxyroridin L-2 is a member of the verrucarin subclass of antibiotics with antitumor properties.</p>
    Fórmula:C29H38O10
    Cor e Forma:Solid
    Peso molecular:546.606
  • Antiviral agent 6


    <p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>
    Fórmula:C23H27BrN2O3S2
    Cor e Forma:Solid
    Peso molecular:523.51
  • Avorelin acetate

    CAS:
    <p>Avorelin acetate is a luteinizing hormone releasing hormone (LH-RH) agonist.</p>
    Fórmula:C67H89N17O14
    Cor e Forma:Solid
    Peso molecular:1356.55
  • A 74273

    CAS:
    <p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>
    Fórmula:C44H74N4O8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:787.08
  • LA-810

    CAS:
    LA-810 is a nitrous oxide donor.
    Fórmula:C15H25N5O7S
    Cor e Forma:Solid
    Peso molecular:419.45
  • Chrymutasin C

    CAS:
    Chrymutasin C is a glycoside antitumor antibiotic with cytotoxic properties.
    Fórmula:C39H43NO17
    Cor e Forma:Solid
    Peso molecular:797.755
  • 4"-Demethylgentamicin C1

    CAS:
    <p>4"-Demethylgentamicin C1 exhibits antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C20H41N5O7
    Cor e Forma:Solid
    Peso molecular:463.57
  • Nevirapine dimer

    CAS:
    Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).
    Fórmula:C30H26N8O2
    Cor e Forma:Solid
    Peso molecular:530.58
  • NPEC-caged-(S)-3,4-DCPG

    CAS:
    mGlu8a agonist
    Fórmula:C19H16N2O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:432.34
  • AS1940477

    CAS:
    <p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>
    Fórmula:C24H22FN5O2
    Cor e Forma:Solid
    Peso molecular:431.46
  • RS 2135

    CAS:
    RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.
    Fórmula:C18H21ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:332.83
  • NTPDase-IN-2

    CAS:
    <p>NTPDase-IN-2 inhibits h-NTPDase-2/-8 (IC50: 0.04, 2.27 µM), non-competitive for h-NTPDase-1/-2 (Km: 74 µM); useful in cancer, immune, bacterial research.</p>
    Fórmula:C24H20FN3OS2
    Cor e Forma:Solid
    Peso molecular:449.56
  • G12Si-1


    G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.
    Fórmula:C29H32ClN5O3
    Cor e Forma:Solid
    Peso molecular:534.05
  • AVE-1330A free acid

    CAS:
    AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.
    Fórmula:C7H11N3O6S
    Cor e Forma:Solid
    Peso molecular:265.24
  • 22-HDHA

    CAS:
    22-HDHA is an oxidation product of docosahexaenoic acid .
    Fórmula:C22H32O3
    Cor e Forma:Solid
    Peso molecular:344.49
  • BAY-693

    CAS:
    <p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>
    Fórmula:C26H30F3N7O2
    Cor e Forma:Solid
    Peso molecular:529.56
  • SSM3 TFA

    CAS:
    SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..
    Fórmula:C22H32N12O2
    Cor e Forma:Solid
    Peso molecular:496.57
  • B-3852

    CAS:
    B-3852 is a Bradykinin inhibitor.
    Fórmula:C55H74F3N15O11
    Cor e Forma:Solid
    Peso molecular:1178.27
  • BAY-091

    CAS:
    BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.
    Fórmula:C26H21FN4O2
    Pureza:97.66% - 99.23%
    Cor e Forma:Soild
    Peso molecular:440.47
  • SGK1-IN-3


    SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.
    Fórmula:C23H20Cl2N6O3S
    Cor e Forma:Solid
    Peso molecular:531.41
  • UAWJ9-36-1

    CAS:
    UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.
    Fórmula:C23H29N3O5
    Cor e Forma:Solid
    Peso molecular:427.49
  • STA 2

    CAS:
    STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.
    Fórmula:C21H34O3S
    Cor e Forma:Solid
    Peso molecular:366.56
  • Sannamycin J

    CAS:
    Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.
    Fórmula:C14H30N4O4
    Cor e Forma:Solid
    Peso molecular:318.41
  • J-104132

    CAS:
    J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.
    Fórmula:C31H33NO7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:531.60
  • BMS-748730

    CAS:
    <p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>
    Fórmula:C22H26ClN7O3S
    Cor e Forma:Solid
    Peso molecular:504.01
  • Homopteroic Acid

    CAS:
    Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.
    Fórmula:C15H14N6O3
    Cor e Forma:Solid
    Peso molecular:326.31
  • SIK1 activator 1

    CAS:
    SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.
    Fórmula:C23H32O6
    Cor e Forma:Solid
    Peso molecular:404.50
  • (R)-ONO-2952


    (R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.
    Fórmula:C22H20ClFN2O2
    Cor e Forma:Solid
    Peso molecular:398.86
  • BILA 1906 BS

    CAS:
    BILA 1906 BS is an inhibitor of substrate analog protease.
    Fórmula:C41H52N6O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:724.95
  • Antimalarial agent 9


    <p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>
    Fórmula:C28H32BrN3O2
    Cor e Forma:Solid
    Peso molecular:522.48
  • Mutatochrome

    CAS:
    <p>Mutatochrome (Citroxanthin) is a compound found in plants.</p>
    Fórmula:C40H56O
    Cor e Forma:Solid
    Peso molecular:552.872
  • Plasma kallikrein-IN-2


    Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.
    Fórmula:C28H24ClF3N8O3
    Cor e Forma:Solid
    Peso molecular:612.99
  • FTO-IN-6

    CAS:
    FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).
    Fórmula:C14H12N4O6
    Cor e Forma:Solid
    Peso molecular:332.27
  • GG-43


    GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].
    Fórmula:C21H21NO3
    Cor e Forma:Solid
    Peso molecular:335.4
  • Olanzapine/Samidorphan

    CAS:
    Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.
    Fórmula:C38H46N6O4S
    Cor e Forma:Solid
    Peso molecular:682.88
  • Parimycin

    CAS:
    <p>Parimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as tumors, but shows no efficacy against fungi. It inhibits tumor cells such as GXF 251L, H640, LXFA 629L, MCF-7, and MEXF 514L, with an IC70 range of 0.9-6.7 μg/mL.</p>
    Fórmula:C22H20O7
    Cor e Forma:Solid
    Peso molecular:396.39
  • ATX inhibitor 12


    <p>Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.</p>
    Fórmula:C30H34FN5O2
    Cor e Forma:Solid
    Peso molecular:515.62
  • Pacidamycin 5T

    CAS:
    <p>Pacidamycin 5T is found in the bacterium Streptomyces coeruleorubidus [NRRL 18370].</p>
    Fórmula:C36H44N8O12
    Cor e Forma:Solid
    Peso molecular:780.78
  • Nonsteroidal aromatase inhibitor 1


    Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.
    Fórmula:C22H16N4O2
    Cor e Forma:Solid
    Peso molecular:368.39
  • Pilatin

    CAS:
    <p>Pilatin exhibits inhibitory effects on both bacteria and fungi, and it strongly suppresses the incorporation of thymidine and uridine into DNA and RNA in Ehrlich ascites tumor cells.</p>
    Fórmula:C21H26O7
    Cor e Forma:Solid
    Peso molecular:390.427
  • AGN-204396

    CAS:
    AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).
    Fórmula:C32H44FN3O4
    Cor e Forma:Solid
    Peso molecular:553.71
  • PF-06815345 hydrochloride

    CAS:
    <p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>
    Fórmula:C27H30Cl2FN9O4
    Cor e Forma:Solid
    Peso molecular:634.49
  • Pyrisulfoxin A

    CAS:
    <p>Pyrisulfoxin A is an antibiotic that can be found in Streptomyces callfornicus [BS-75].</p>
    Fórmula:C13H13N3O3S
    Cor e Forma:Solid
    Peso molecular:291.326
  • Nnc 09-0026

    CAS:
    Nnc 09-0026 is a neuronal calcium channel blocker
    Fórmula:C25H35Cl2F3N2O
    Cor e Forma:Solid
    Peso molecular:507.46
  • GSK 932121

    CAS:
    GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.
    Fórmula:C20H15ClF3NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:425.79
  • Dihydrocompactin

    CAS:
    <p>Dihydrocompactin is an antifungal metabolite derived from Penicillium citrinum and acts as an inhibitor of 3-hydroxy-3-methylglutaryl coenzyme-A reductase (HMG-CoA reductase).</p>
    Fórmula:C23H36O5
    Cor e Forma:Solid
    Peso molecular:392.529
  • CY208-243 Mandelate

    CAS:
    CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.
    Fórmula:C27H26N2O3
    Cor e Forma:Solid
    Peso molecular:426.52
  • TAM&Met-IN-1

    CAS:
    TAM&Met-IN-1 inhibits AXL, MER, TYRO3 with IC50s 6.1, 13.2, 21.6 nM, respectively, for cancer research.
    Fórmula:C29H27F2N7O5
    Cor e Forma:Solid
    Peso molecular:591.57
  • AMG-315

    CAS:
    AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.
    Fórmula:C24H41NO2
    Cor e Forma:Solid
    Peso molecular:375.59
  • Roselipin 1A

    CAS:
    <p>Roselipin 1A inhibits diacylglycerol acyltransferase (DGAT) in rats.</p>
    Fórmula:C40H72O14
    Cor e Forma:Solid
    Peso molecular:776.991
  • EBI-907

    CAS:
    EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.
    Fórmula:C23H21ClF2N4O3S
    Cor e Forma:Solid
    Peso molecular:506.95
  • Antidepressant agent 2


    <p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>
    Fórmula:C21H22ClFN2O3S
    Cor e Forma:Solid
    Peso molecular:436.93
  • Artemisiane E

    CAS:
    Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .
    Fórmula:C20H22O5
    Cor e Forma:Solid
    Peso molecular:342.39
  • LY3325656

    CAS:
    LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.
    Fórmula:C21H23F3N6O2
    Cor e Forma:Solid
    Peso molecular:448.44
  • 2-Hydroxybutirosin

    CAS:
    2-Hydroxybutirosin is an antibiotic that can be found in Bacillus circulans.
    Fórmula:C21H41N5O13
    Cor e Forma:Solid
    Peso molecular:571.576
  • Pradimicin B

    CAS:
    Pradimicin B is an antibiotic with potent antifungal and anti-yeast activities.
    Fórmula:C35H36N2O14
    Cor e Forma:Solid
    Peso molecular:708.665
  • Dephostatin

    CAS:
    <p>Dephostatin is a competitive protein tyrosine phosphatase (PTP) inhibitor isolated from Streptomyces spp., exhibiting activity within the micromolar range.</p>
    Fórmula:C7H8N2O3
    Cor e Forma:Solid
    Peso molecular:168.15
  • Cryptosporiopsin

    CAS:
    <p>Cryptosporiopsin can be isolated from strains of Cryptosporiopsis sp. and Sporormia affinis. It exhibits antimicrobial activity against various basidiomycetes, alga fungi, ascomycetes, and glaucomycetes responsible for wood decay. Additionally, it inhibits the germination of Phytophthora potatoes spores. Cryptosporiopsin also shows some activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C10H10Cl2O4
    Cor e Forma:Solid
    Peso molecular:265.09
  • 9-Hydroxyoudemansin A

    CAS:
    <p>9-Hydroxyoudemansin A exhibits antifungal activity with a minimum inhibitory concentration (MIC) of 12.5 μg/mL against Saccharomyces cerevisiae. It shows resistance to fungi such as Candida albicans, Rhodotorula, Penicillium, and Streptomyces, with MIC values all exceeding 50 μg/mL. It does not possess antibacterial properties.</p>
    Fórmula:C16H20O4
    Cor e Forma:Solid
    Peso molecular:276.328
  • 23-De(mycinosyloxy)tylosin

    CAS:
    <p>23-De(mycinosyloxy)tylosin is a macrolide antibiotic exhibiting activity against Gram-positive bacteria, with limited efficacy against Gram-negative bacteria and mycoplasma.</p>
    Fórmula:C38H63NO12
    Cor e Forma:Solid
    Peso molecular:725.91
  • UNC9426

    CAS:
    <p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>
    Fórmula:C32H34F6N6O
    Pureza:98.051%
    Cor e Forma:Solid
    Peso molecular:632.642
  • Cuevaene A

    CAS:
    <p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>
    Fórmula:C21H22O5
    Cor e Forma:Solid
    Peso molecular:354.396
  • Anti-Trypanosoma cruzi agent-2


    Compd 3b: anti-trypanosomal, IC50 0.51 μM (NINOA), 3.06 μM (INC-5), also combats T. gondii.
    Fórmula:C17H10ClNO5
    Cor e Forma:Solid
    Peso molecular:343.72
  • Guanine-7-oxide

    CAS:
    Guanine-7-oxide (Guanine 7-N-oxide) is an antitumor antibiotic with antitumor and anti-Candida albicans activities. It inhibits the replication of viruses such as herpes virus, infectious hematopoietic necrosis virus (IHNV), and infectious pancreatic necrosis virus (IPNV). The compound also demonstrates significant activity against mouse L1210 leukemia cells.
    Fórmula:C5H5N5O2
    Cor e Forma:Solid
    Peso molecular:167.126
  • SSTR5 antagonist 2 hydrochloride


    SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.
    Fórmula:C32H36ClFN2O5
    Cor e Forma:Solid
    Peso molecular:583.09
  • FK-906 HCl

    CAS:
    FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.
    Fórmula:C40H64ClN7O7
    Cor e Forma:Solid
    Peso molecular:790.44
  • NUCC-555

    CAS:
    NUCC-555 is a first-in-class antagonist of activin. It opens a completely new approach to inhibiting the activity of TGF-beta receptor superfamily members.
    Fórmula:C25H25N5O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:443.5
  • BSc5367

    CAS:
    <p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>
    Fórmula:C20H15N3O2
    Cor e Forma:Soild
    Peso molecular:329.35
  • Purine phosphoribosyltransferase-IN-1


    Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.
    Fórmula:C11H15N5Na4O10P2
    Cor e Forma:Solid
    Peso molecular:531.17
  • Clecarmycin C

    CAS:
    <p>Clecarmycin C is an antitumor antibiotic that demonstrates cytotoxic and antitumor properties. Additionally, Clecarmycin C exhibits antibacterial activity.</p>
    Fórmula:C29H26O11
    Cor e Forma:Solid
    Peso molecular:550.51
  • 4-Diazo-3-methoxy-2,5-cyclohexadien-1-one

    CAS:
    <p>4-Diazo-3-methoxy-2,5-cyclohexadien-1-one demonstrates notable activity against anaerobic bacteria. Minimum inhibitory concentrations (MIC) are 0.4 μg/mL for Clostridium and Bacteroidetes, and 0.2 μg/mL for Haemophilus.</p>
    Fórmula:C7H6N2O2
    Cor e Forma:Solid
    Peso molecular:150.14
  • PAD-IN-2

    CAS:
    <p>PAD-IN-2, potent PAD4 inhibitor, IC50 &lt;1 μM; targets autoimmune/cancer disorders.</p>
    Fórmula:C27H28ClN5O2
    Cor e Forma:Solid
    Peso molecular:490
  • 2-Hydroxymethylclavam

    CAS:
    <p>2-Hydroxymethylclavam is a β-lactam antibiotic with antifungal properties, particularly effective against plant pathogenic fungi.</p>
    Fórmula:C6H9NO3
    Cor e Forma:Solid
    Peso molecular:143.141
  • Antitrypanosomal agent 5


    Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).
    Fórmula:C30H30N6O4S
    Cor e Forma:Solid
    Peso molecular:570.66
  • Antimalarial agent 2


    Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.
    Fórmula:C27H25N3O5
    Cor e Forma:Solid
    Peso molecular:471.5
  • Juvenimicin A2

    CAS:
    <p>Juvenimicin A2 is effective against Gram-positive bacteria and certain Gram-negative bacteria.</p>
    Fórmula:C30H51NO8
    Cor e Forma:Solid
    Peso molecular:553.728
  • 1-Deamino-1-hydroxygentamicin C1a

    CAS:
    <p>1-Deamino-1-hydroxygentamicin C1a (AntibioticSU-2) is an aminoglycoside antibiotic effective against both gram-positive and gram-negative bacteria.</p>
    Fórmula:C19H38N4O8
    Cor e Forma:Solid
    Peso molecular:450.527
  • VEGFR-2-IN-12


    VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.
    Fórmula:C22H24N6O3S
    Cor e Forma:Solid
    Peso molecular:452.53
  • Elaiomycin

    CAS:
    Elaiomycin exhibits activity against Gram-positive bacteria, certain anaerobic bacteria, Eimeria tenella, and Eimeria stiedai.
    Fórmula:C13H26N2O3
    Cor e Forma:Solid
    Peso molecular:258.357
  • Acetoxycycloheximide

    CAS:
    <p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>
    Fórmula:C17H25NO6
    Cor e Forma:Solid
    Peso molecular:339.38
  • Deacetylravidomycin N-oxide

    CAS:
    <p>Deacetylravidomycin N-oxide is an antibiotic produced by [Streptomyces ravidus S50905] that exhibits activity against Gram-positive bacteria but is inactive against Gram-negative bacteria. Additionally, Deacetylravidomycin N-oxide demonstrates antitumor properties against P388 leukemia and methylcholanthrene A fibrosarcoma.</p>
    Fórmula:C31H33NO10
    Cor e Forma:Solid
    Peso molecular:579.594
  • FTO-IN-1 TFA


    FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.
    Fórmula:C20H17Cl2F3N4O4
    Cor e Forma:Solid
    Peso molecular:505.27
  • ML-SI1

    CAS:
    ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).
    Fórmula:C23H26Cl2N2O3
    Cor e Forma:Solid
    Peso molecular:449.37
  • Lp-PLA2-IN-5

    CAS:
    <p>Lp-PLA2-IN-5 inhibits Lp-PLA2 and PAF-AH, potentially useful in Alzheimer's and atherosclerosis studies.</p>
    Fórmula:C23H18F5N3O4
    Cor e Forma:Solid
    Peso molecular:495.4
  • Reumycin

    CAS:
    <p>Reumycin is a 7-azaindole antibiotic that exhibits cytotoxicity against tumor cells such as Ellrich carcinoma, Sarcoma-180, Sarcoma-37, and lymphosarcoma.</p>
    Fórmula:C6H5N5O2
    Cor e Forma:Solid
    Peso molecular:179.136
  • Fumaryl-DL-alanine

    CAS:
    Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.
    Fórmula:C7H9NO5
    Cor e Forma:Solid
    Peso molecular:187.15
  • 18:0-LPS

    CAS:
    18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.
    Fórmula:C24H48NO9P
    Cor e Forma:Solid
    Peso molecular:525.613
  • (25S)-δ7-Dafachronic acid

    CAS:
    (25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.
    Fórmula:C27H42O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:414.62
  • Haliangicin B

    CAS:
    Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.
    Fórmula:C22H32O5
    Cor e Forma:Solid
    Peso molecular:376.49
  • Dihydroabikoviromycin

    CAS:
    Dihydroabikoviromycin is a secondary metabolite of Streptomyces anulatus and acts as a polyketide synthase inhibitor.
    Fórmula:C10H13NO
    Cor e Forma:Solid
    Peso molecular:163.216
  • nNOS-IN-25

    CAS:
    nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.
    Fórmula:C21H22N4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:330.43
  • AT-IAP

    CAS:
    AT-IAP is an effective dual antagonist of XIAP and cIAP1.
    Fórmula:C29H40FN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:509.66
  • Haliangicin A

    CAS:
    <p>Haliangicin A exhibits antifungal activity against filamentous fungi and also affects oomycetes, though it does not possess antibacterial properties.</p>
    Fórmula:C22H32O5
    Cor e Forma:Solid
    Peso molecular:376.49
  • 2-n-Heptyl-4-quinolinol

    CAS:
    <p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>
    Fórmula:C16H21NO
    Cor e Forma:Solid
    Peso molecular:243.34
  • Pegcantratinib

    CAS:
    Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.
    Fórmula:C32H28N4O7
    Cor e Forma:Solid
    Peso molecular:580.59
  • Ici D1542

    CAS:
    Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.
    Fórmula:C25H30N2O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:470.51
  • RIPK1-IN-24

    CAS:
    <p>RIPK1-IN-24 is an inhibitor of receptor-interacting protein kinase 1 (RIPK1) with an IC50 of 1.3 μM. It is utilized in research on inflammatory diseases.</p>
    Fórmula:C26H21FN6O2
    Cor e Forma:Solid
    Peso molecular:468.48
  • Coleon-U-quinone

    CAS:
    Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.
    Fórmula:C20H24O5
    Cor e Forma:Solid
    Peso molecular:344.4
  • Schidigera-genin B

    CAS:
    <p>Schidigera-genin B is a steroidal saponin that can be isolated from Yucca glauca. It exhibits mild antifungal activity.</p>
    Fórmula:C27H40O4
    Cor e Forma:Solid
    Peso molecular:428.604
  • 4"-Demethylgentamicin C2

    CAS:
    4"-Demethylgentamicin C2 exhibits activity against both Gram-positive and Gram-negative bacteria.
    Fórmula:C19H39N5O7
    Cor e Forma:Solid
    Peso molecular:449.54
  • Chitinovorin C

    CAS:
    Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.
    Fórmula:C15H20N4O8S
    Cor e Forma:Solid
    Peso molecular:416.406
  • Haloquinone

    CAS:
    <p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>
    Fórmula:C17H12O5
    Cor e Forma:Solid
    Peso molecular:296.274
  • Epithienamycin C

    CAS:
    <p>Epithienamycin C is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C13H18N2O5S
    Cor e Forma:Solid
    Peso molecular:314.357
  • NCATS-SM4487

    CAS:
    NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).
    Fórmula:C25H24ClFN8O2
    Cor e Forma:Solid
    Peso molecular:522.96
  • Ophiobolin D

    CAS:
    Ophiobolin D is a terpene antibiotic with mild inhibitory effects on Staphylococcus aureus.
    Fórmula:C25H36O4
    Cor e Forma:Solid
    Peso molecular:400.55
  • Pradimicin T2

    CAS:
    <p>Pradimicin T2 is an antibiotic with activity against filamentous fungi and yeast-like fungi.</p>
    Fórmula:C37H37NO19
    Cor e Forma:Solid
    Peso molecular:799.685
  • FW 34569

    CAS:
    FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.
    Fórmula:C30H43N5O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:617.76