Outros inibidores
Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.
Foram encontrados 37827 produtos de "Outros inibidores"
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DS69910557
<p>DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism & osteoporosis research.</p>Fórmula:C32H33Cl2FN4O3Cor e Forma:SolidPeso molecular:611.53PEN-866
CAS:<p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>Fórmula:C49H49N7O9Cor e Forma:SolidPeso molecular:879.95Dinordrin I diacetate
CAS:<p>Dinordrin I diacetate is an implantation inhibitor and hormone.</p>Fórmula:C25H32O4Pureza:98%Cor e Forma:SolidPeso molecular:396.52BRD-9526
CAS:BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Fórmula:C26H31Cl2N3O6SPureza:98%Cor e Forma:SolidPeso molecular:584.51Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Fórmula:C21H36O7Cor e Forma:SolidPeso molecular:400.506Naltalimide
CAS:<p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>Fórmula:C28H28N2O5Pureza:98%Cor e Forma:SolidPeso molecular:472.53DGY-08-097
CAS:<p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>Fórmula:C60H76N10O14Cor e Forma:SolidPeso molecular:1161.3CY208-243 Mandelate
CAS:<p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>Fórmula:C27H26N2O3Cor e Forma:SolidPeso molecular:426.52Nnc 09-0026
CAS:<p>Nnc 09-0026 is a neuronal calcium channel blocker</p>Fórmula:C25H35Cl2F3N2OCor e Forma:SolidPeso molecular:507.46S24-14
CAS:S24-14 serves as an effective anti-osteoporosis agent by inhibiting osteoclastogenesis, promoting osteoblast differentiation, and reducing bone resorption.Fórmula:C19H12N2O3SCor e Forma:SolidPeso molecular:348.38T-3861174
CAS:<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Fórmula:C26H25FN6O2Cor e Forma:SolidPeso molecular:472.51Chrymutasin C
CAS:<p>Chrymutasin C is a glycoside antitumor antibiotic with cytotoxic properties.</p>Fórmula:C39H43NO17Cor e Forma:SolidPeso molecular:797.755Epelmycin D
CAS:<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Fórmula:C30H35NO11Cor e Forma:SolidPeso molecular:585.599L 767679
CAS:<p>L 767679 is an antagonist of the fibrinogen receptors.</p>Fórmula:C20H24N4O4Pureza:98%Cor e Forma:SolidPeso molecular:384.43Menoxymycin A
CAS:<p>Menoxymycin A is an antibiotic with cytotoxic properties. It inhibits the growth of KB and N18-RE-105 cells, with IC50 values of 0.86 μM and 0.14 μM, respectively.</p>Fórmula:C24H27NO9Cor e Forma:SolidPeso molecular:473.473DDCPPB-Glu
CAS:<p>DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.</p>Fórmula:C22H27N5O5Pureza:98%Cor e Forma:SolidPeso molecular:441.48S-1033
CAS:<p>S-1033 is an FP receptor agonist.</p>Fórmula:C20H33NaO4Cor e Forma:SolidPeso molecular:360.4698Atiratecan
CAS:<p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>Fórmula:C31H34N6O6Pureza:98%Cor e Forma:SolidPeso molecular:586.64CH5447240
CAS:<p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>Fórmula:C26H39N5O4SPureza:98%Cor e Forma:SolidPeso molecular:517.68Pluracidomycin C2
CAS:<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C11H15NO9S2Cor e Forma:SolidPeso molecular:369.37hCA IX-IN-1
<p>hCA IX-IN-1 inhibits human carbonic anhydrases I, II, IX, and XII with Ki values of 331.4, 28.4, 9.4, 17.8 nM and exhibits anticancer properties.</p>Fórmula:C19H18N2O3SCor e Forma:SolidPeso molecular:354.42L 739749
CAS:<p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>Fórmula:C24H41N3O6S2Pureza:98%Cor e Forma:SolidPeso molecular:531.73Hetrombopag olamine
CAS:<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Fórmula:C29H36N6O7Pureza:98%Cor e Forma:SolidPeso molecular:580.63Arterolane
CAS:<p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>Fórmula:C22H36N2O4Cor e Forma:SolidPeso molecular:392.53Hydranthomycin
CAS:<p>Hydranthomycin is an antibiotic with moderate antifungal activity, exhibiting a minimum inhibitory concentration (MIC) of 25 μg/mL against the rice blast fungus. Additionally, it inhibits the growth of Chlorella (tiny naked algae) and possesses herbicidal properties.</p>Fórmula:C20H20O5Cor e Forma:SolidPeso molecular:340.37Dinordrin
CAS:Dinordrin is an implantation inhibitor and hormone.Fórmula:C27H36O4Pureza:98%Cor e Forma:SolidPeso molecular:424.57MRS2179 tetrasodium hydrate
<p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>Fórmula:C11H15N5Na4O10P2Cor e Forma:SolidPeso molecular:576.2118:0-LPS
CAS:<p>18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.</p>Fórmula:C24H48NO9PCor e Forma:SolidPeso molecular:525.6132-PPA
CAS:2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.Fórmula:C11H10N2Cor e Forma:SolidPeso molecular:170.21Retelliptine
CAS:Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Fórmula:C25H32N4OPureza:98%Cor e Forma:SolidPeso molecular:404.55KY-02327 acetate
<p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>Fórmula:C22H31N3O6Cor e Forma:SolidPeso molecular:433.5SLC4101431
<p>SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.</p>Fórmula:C29H28ClN7OSCor e Forma:SolidPeso molecular:558.1Methyl Streptonigrin
CAS:<p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>Fórmula:C26H24N4O8Pureza:98%Cor e Forma:SolidPeso molecular:520.49BGC-638
CAS:<p>BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.</p>Fórmula:C32H33N5O9Cor e Forma:SolidPeso molecular:631.63JBJ-08-178-01
CAS:JBJ-08-178-01, a mutant-selective tyrosine kinase inhibitor, targets (HER2) human epidermal growth factor receptor 2 and exhibits antitumoral activity. This compound not only diminishes HER2's kinase activity and protein levels through the induction of proteasomal degradation of the receptor but also shows promise in non-small-cell lung cancer research.Fórmula:C31H30N8O3Cor e Forma:SolidPeso molecular:562.62Anti-TSWV agent 1
<p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>Fórmula:C22H27ClN4OS3Cor e Forma:SolidPeso molecular:495.12Sekdel sequence
CAS:Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.Fórmula:C29H49N7O14Cor e Forma:SolidPeso molecular:719.74J-104132
CAS:<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Fórmula:C31H33NO7Pureza:98%Cor e Forma:SolidPeso molecular:531.60Nevirapine dimer
CAS:<p>Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).</p>Fórmula:C30H26N8O2Cor e Forma:SolidPeso molecular:530.58PTP1B-IN-21
<p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>Fórmula:C22H22O11Cor e Forma:SolidPeso molecular:462.4TCMDC-125431
<p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>Fórmula:C25H27N3O2SCor e Forma:SolidPeso molecular:433.57A 74273
CAS:<p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>Fórmula:C44H74N4O8Pureza:98%Cor e Forma:SolidPeso molecular:787.08PD-1-IN-17 TFA
<p>PD-1-IN-17 TFA is a potent PD-1 inhibitor, blocking 92% of splenocyte growth at 100 nM.</p>Fórmula:C15H23F3N6O9Cor e Forma:SolidPeso molecular:488.37Dermostatin A
CAS:<p>Dermostatin A is a polyene antibiotic with antifungal properties suitable for studying fungal infections.</p>Fórmula:C40H64O11Cor e Forma:SolidPeso molecular:720.93S39625
CAS:<p>S39625 is a stable, potent topoisomerase I inhibitor with anticancer properties, resistant to efflux transporters, inducing gamma-H2AX at nanomolar levels.</p>Fórmula:C25H22N2O5Pureza:98%Cor e Forma:SolidPeso molecular:430.45Narbomycin
CAS:<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Fórmula:C28H47NO7Cor e Forma:SolidPeso molecular:509.675GZN39838
CAS:<p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>Fórmula:C22H30O6Cor e Forma:SolidPeso molecular:390.47Haliangicin A
CAS:<p>Haliangicin A exhibits antifungal activity against filamentous fungi and also affects oomycetes, though it does not possess antibacterial properties.</p>Fórmula:C22H32O5Cor e Forma:SolidPeso molecular:376.49Resolvin E4
CAS:<p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.45Purine phosphoribosyltransferase-IN-2
<p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>Fórmula:C11H15N5Na4O10P2Cor e Forma:SolidPeso molecular:531.172-n-Heptyl-4-quinolinol
CAS:<p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>Fórmula:C16H21NOCor e Forma:SolidPeso molecular:243.345(S),6(S)-DiHETE
CAS:<p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.474"-Demethylgentamicin C2
CAS:<p>4"-Demethylgentamicin C2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C19H39N5O7Cor e Forma:SolidPeso molecular:449.54YM-355179
CAS:<p>YM-355179 is a novel, selective antagonist of CC chemokine receptor 3 with oral activity.</p>Fórmula:C33H34FN4O7Pureza:98%Cor e Forma:SolidPeso molecular:617.64Epithienamycin D
CAS:<p>Epithienamycin D is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C13H16N2O5SCor e Forma:SolidPeso molecular:312.342PGDM
CAS:<p>PGD2 is involved in allergy, asthma, sleep, temperature regulation, inhibits clotting, and relaxes blood vessels; PGDM, its metabolite, is a biomarker.</p>Fórmula:C16H24O7Cor e Forma:SolidPeso molecular:328.36NRX-2663
CAS:<p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>Fórmula:C20H13F3N2O5Cor e Forma:SolidPeso molecular:418.32FW 34569
CAS:<p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>Fórmula:C30H43N5O7SPureza:98%Cor e Forma:SolidPeso molecular:617.76FTI-2628
CAS:<p>FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.</p>Fórmula:C31H34N4O3SCor e Forma:SolidPeso molecular:542.69PD-1/PD-L1-IN-23
CAS:<p>PD-1/PD-L1-IN-23: potent, oral PD-1/PD-L1 inhibitor; L7's ester prodrug; exhibits strong antitumor effects.</p>Fórmula:C32H30BrCl2N3O6Cor e Forma:SolidPeso molecular:703.412-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H41N5O8Cor e Forma:SolidPeso molecular:479.568Cytosaminomycin C
CAS:<p>Cytosaminomycin C exhibits anti-Eimeria Tenella coccidial activity.</p>Fórmula:C23H36N4O8Cor e Forma:SolidPeso molecular:496.554KOS-1584
CAS:<p>KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.</p>Fórmula:C27H39NO5SCor e Forma:SolidPeso molecular:489.67Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Fórmula:C26H36N2O4Cor e Forma:SolidPeso molecular:440.58ITK inhibitor 6
CAS:<p>ITK inhibitor 6 selectively targets ITK, BTK, JAK3, EGFR, LCK, blocks PLCγ1 and ERK1/2 phosphorylation, and inhibits cell proliferation.</p>Fórmula:C28H24F2N4O2Cor e Forma:SolidPeso molecular:486.51Pralatrexate, (R)-
CAS:<p>Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.</p>Fórmula:C23H23N7O5Pureza:98%Cor e Forma:SolidPeso molecular:477.47PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Fórmula:C21H23N5O2Cor e Forma:SolidPeso molecular:377.44Anti-inflammatory agent 13
<p>Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.</p>Fórmula:C30H48O4Cor e Forma:SolidPeso molecular:472.7Kahweol linoleate
CAS:<p>Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.</p>Fórmula:C38H56O4Cor e Forma:SolidPeso molecular:576.85PLP_Snyder530
<p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>Fórmula:C24H24N2O2Cor e Forma:SolidPeso molecular:372.46KNI 10033
CAS:<p>KNI 10033 is a potent inhibitor of HIV protease</p>Fórmula:C40H45N5O7S2Cor e Forma:SolidPeso molecular:771.95ONO-8809
CAS:<p>ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.</p>Fórmula:C30H46BrNO4SPureza:98%Cor e Forma:SolidPeso molecular:596.66Carazostatin
CAS:<p>Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.</p>Fórmula:C20H25NOPureza:98%Cor e Forma:Pale Yellow SolidPeso molecular:295.42TRPC5-IN-4
CAS:<p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>Fórmula:C18H11ClF4N4O3Cor e Forma:SolidPeso molecular:442.75GR-71251
CAS:<p>GR-71251 is a Tachykinin receptor antagonist.</p>Fórmula:C74H105N19O13Cor e Forma:SolidPeso molecular:1468.74Pochonin D
CAS:<p>Pochonin D is an inhibitor of heat shock protein 90 (Hsp90) with antiviral and anti-inflammatory properties. It disrupts Hsp90, affecting the stability, folding, and assembly of viral proteins, thereby diminishing viral replication. Additionally, Pochonin D reduces the infiltration of inflammatory cells and decreases the secretion of inflammatory cytokines such as TNF-α and IL-1β, alleviating inflammatory responses. This compound shows potential for research in human rhinovirus (HRV) infections and cancer.</p>Fórmula:C18H19ClO5Cor e Forma:SolidPeso molecular:350.793Halomicin D
CAS:<p>Halomicin D is an ansamycin-class antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C43H56N2O12Cor e Forma:SolidPeso molecular:792.911Isoleucyl tRNA synthetase-IN-2
CAS:<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Fórmula:C22H33N5O8SCor e Forma:SolidPeso molecular:527.594α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Fórmula:C40H64O8Cor e Forma:SolidPeso molecular:672.93P-gp modulator 1
CAS:<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Fórmula:C41H72N2O6Pureza:98%Cor e Forma:SolidPeso molecular:689.02Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Fórmula:C27H25FN6O2Cor e Forma:SolidPeso molecular:484.52Ceclazepide
CAS:<p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>Fórmula:C30H32N6O5Pureza:98%Cor e Forma:SolidPeso molecular:556.61FCE-27262
CAS:<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Fórmula:C23H31N3O3Cor e Forma:SolidPeso molecular:397.51L 731735
CAS:<p>L 731735 is a farnesyltransferase inhibitor.</p>Fórmula:C19H40N4O4SPureza:98%Cor e Forma:SolidPeso molecular:420.61Mopivabil
<p>Mopivabil is the angiotensin II receptor antagonist[1].</p>Fórmula:C14H20O3Cor e Forma:SolidPeso molecular:236.31Alentemol hydrobromide
CAS:<p>Alentemol hydrobromide is a Dopamine agonist.</p>Fórmula:C19H26BrNOPureza:98%Cor e Forma:SolidPeso molecular:364.32L 668750
CAS:<p>L 668750 is an inhibitor of platelet-activating factor.</p>Fórmula:C25H34O9SPureza:98%Cor e Forma:SolidPeso molecular:510.6Vulolisib
CAS:<p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>Fórmula:C18H19F2N5O3SCor e Forma:SolidPeso molecular:423.44ADH-353
CAS:<p>ADH-353 inhibits Aβ fibrillization and mitigates Aβ-induced cytotoxicity in SH-SY5Y and N2a cells, making it useful for studies related to Alzheimer's disease.</p>Fórmula:C27H38N8O6Cor e Forma:SolidPeso molecular:570.64Hesperidin dihydrochalcone
CAS:Hesperidin dihydrochalcone, a non-toxic sweetener with high sweetness and low calories, exhibits multiple biological activities including anti-oxidation, liver and kidney protection, bacteriostasis, and enhancement of gastrointestinal health.Fórmula:C28H36O15Cor e Forma:SolidPeso molecular:612.58Hit 1
<p>Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.</p>Fórmula:C22H24N4O3S2Cor e Forma:SolidPeso molecular:456.58PDE4-IN-6
<p>PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.</p>Fórmula:C25H20FNO5SCor e Forma:SolidPeso molecular:465.49MRS2500
CAS:<p>MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.</p>Fórmula:C13H18IN5O8P2Pureza:98%Cor e Forma:SolidPeso molecular:561.16PI3K-IN-27
CAS:<p>PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.</p>Fórmula:C30H26F2N6O2SCor e Forma:SolidPeso molecular:572.63AKR1C3-IN-8
<p>AKR1C3-IN-8 (Compound 5) is an effective and selective AKR1C3 inhibitor (IC50=0.069 μM). AKR1C3-IN-8 has antitumor activity.</p>Fórmula:C23H20N4O3Cor e Forma:SolidPeso molecular:400.43Gunacin
CAS:<p>Gunacin is a quinone antibiotic that exhibits significant activity against Gram-positive bacteria, Gram-negative bacteria, and mycoplasmas.</p>Fórmula:C17H16O8Cor e Forma:SolidPeso molecular:348.30416(R)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Fórmula:C22H32O4Cor e Forma:SolidPeso molecular:360.49RK-582
CAS:<p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>Fórmula:C27H35FN6O3Cor e Forma:SolidPeso molecular:510.6Peridinin
CAS:<p>Peridinin is an exceptionally potent and membrane-embedded inhibitor of bilayer lipid peroxidation.</p>Fórmula:C39H50O7Cor e Forma:SolidPeso molecular:630.81Tacrolimus anhydrous 8-epimer
CAS:<p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>Fórmula:C44H69NO12Cor e Forma:SolidPeso molecular:804.02DAD dichloride
<p>DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.</p>Fórmula:C26H42Cl2N6OCor e Forma:SolidPeso molecular:525.56Nonsteroidal aromatase inhibitor 1
<p>Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.</p>Fórmula:C22H16N4O2Cor e Forma:SolidPeso molecular:368.39AB 5046A
CAS:<p>AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.</p>Fórmula:C10H14O4Cor e Forma:SolidPeso molecular:198.22DMP 728
CAS:<p>DMP 728 is an antagonist of Glycoprotein IIb-IIIa.</p>Fórmula:C26H40N8O10SPureza:98%Cor e Forma:SolidPeso molecular:656.71Cilobamine (free base)
CAS:<p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>Fórmula:C17H23Cl2NOCor e Forma:SolidPeso molecular:328.28PPARα agonist 1
<p>PPARα agonist 1 is a complete and potent PPARα agonist.</p>Fórmula:C27H34O4Cor e Forma:SolidPeso molecular:422.56Plumbemycin A
CAS:<p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Fórmula:C12H20N3O9PCor e Forma:SolidPeso molecular:381.28TRK-IN-19
<p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.</p>Fórmula:C22H26FN5O2Cor e Forma:SolidPeso molecular:411.47Tzc 5665
CAS:<p>Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.</p>Fórmula:C31H38ClN5O7Cor e Forma:SolidPeso molecular:628.12Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Fórmula:C32H33N5O4Pureza:98%Cor e Forma:SolidPeso molecular:551.647(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Fórmula:C29H56Cor e Forma:SolidPeso molecular:404.75NRMA-8
CAS:<p>NRMA-8 is a small-molecule nuclear receptor modulator capable of penetrating the brain. It holds potential for research into central nervous system (CNS) diseases, including Alzheimer's disease, Parkinson's disease, demyelinating diseases, and glioblastoma.</p>Fórmula:C20H23ClN2O3Cor e Forma:SolidPeso molecular:374.86LY3325656
CAS:<p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>Fórmula:C21H23F3N6O2Cor e Forma:SolidPeso molecular:448.44[R-(Z)]-4-Amino-3-chloro-2-pen-tenedioicacid
CAS:<p>[R-(Z)]-4-Amino-3-chloro-2-pentenedioic acid inhibits Micrococcus luteus.</p>Fórmula:C5H6ClNO4Cor e Forma:SolidPeso molecular:179.56Cystothiazole A
CAS:<p>Cystothiazole A exhibits antifungal properties, effectively inhibiting Candida albicans, Saccharomyces cerevisiae, and Aspergillus fumigatus with minimum inhibitory concentrations (MIC) of 0.4 μg/mL, 0.1 μg/mL, and 1.6 μg/mL, respectively. It also demonstrates inhibitory activity against human tumor cells such as HPT-116 and K562, with MIC values of 130 ng/mL and 110 ng/mL. However, it shows no antibacterial activity.</p>Fórmula:C20H26N2O4S2Cor e Forma:SolidPeso molecular:422.561hTrkA-IN-2
<p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>Fórmula:C24H22F3N5O3Cor e Forma:SolidPeso molecular:485.46DWN-12088 HCl
CAS:<p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>Fórmula:C15H21Cl4N3OCor e Forma:SolidPeso molecular:401.15O-Demethylpaulomycin A
CAS:<p>O-Demethylpaulomycin A is an antibiotic known for its antibacterial properties. It is particularly effective against Gram-positive bacteria, including Staphylococcus aureus.</p>Fórmula:C33H44N2O17SCor e Forma:SolidPeso molecular:772.771Urease-IN-16
CAS:<p>Urease-IN-16, with an IC50 of 132 µmol/L, is a urease inhibitor that coordinates with nickel atoms through the oxygen atoms of either carbonyl or boronic acid groups. This compound holds significant potential as an additive in the development of efficient fertilizers and medical applications.</p>Fórmula:C14H17BN2O4SCor e Forma:SolidPeso molecular:320.17Imolamine hydrochloride
CAS:<p>Imolamine hydrochloride is a blood platelet aggregation antagonist.</p>Fórmula:C14H21ClN4OCor e Forma:SolidPeso molecular:296.80Fusarochromanone
CAS:Fusarochromanone (FC-101) is a mycotoxin produced by Fusarium oxysporum with potent antiangiogenic, anticancer and antimalarial activities.Fórmula:C15H20N2O4Pureza:95.31% - 96%Cor e Forma:SolidPeso molecular:292.33TCMDC-136230
<p>TCMDC-136230 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystallisation.</p>Fórmula:C24H34N4O2SCor e Forma:SolidPeso molecular:442.62BXL0124
CAS:<p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>Fórmula:C32H44F6O4Cor e Forma:SolidPeso molecular:606.68Dermostatin B
CAS:<p>Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.</p>Fórmula:C41H66O11Cor e Forma:SolidPeso molecular:734.956Kaitocephalin
CAS:<p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>Fórmula:C18H21Cl2N3O9Cor e Forma:SolidPeso molecular:494.28Monorden diacetate
CAS:<p>Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.</p>Fórmula:C22H21ClO8Cor e Forma:SolidPeso molecular:448.85Sannamycin J
CAS:<p>Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C14H30N4O4Cor e Forma:SolidPeso molecular:318.41PTP1B-IN-16
<p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>Fórmula:C26H18ClN3O4SCor e Forma:SolidPeso molecular:503.96GSK3527497
CAS:<p>GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).</p>Fórmula:C17H16ClFN4O4SCor e Forma:SolidPeso molecular:426.85Topoisomerase I inhibitor 8
CAS:<p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>Fórmula:C24H21FN2O4Cor e Forma:SolidPeso molecular:420.43Freselestat
CAS:<p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>Fórmula:C23H28N6O4Cor e Forma:SolidPeso molecular:452.51CEP-7055
CAS:<p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>Fórmula:C32H35N3O4Cor e Forma:SolidPeso molecular:525.64MtDTBS-IN-1
<p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>Fórmula:C16H16N4O5Cor e Forma:SolidPeso molecular:344.32Cryptopleurine
CAS:<p>Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.</p>Fórmula:C24H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:377.48ASB14780
<p>ASB14780 is a 4-phenoxy derivative and an inhibitor of cytoplasmic phospholipase cPLA2α (IC50: 20 nM).</p>Cor e Forma:SolidDeoxyfuconojirimycin hydrochloride
CAS:<p>Deoxyfuconojirimycin hydrochloride acts as a specific competitive inhibitor targeting human liver α-L-fucosidase.</p>Fórmula:C6H14ClNO3Cor e Forma:SolidPeso molecular:183.63Salvinorin A Propionate
CAS:<p>Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.</p>Fórmula:C24H30O8Cor e Forma:SolidPeso molecular:446.49MK-1220
CAS:<p>MK-1220 is a novel Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure.</p>Fórmula:C40H53N5O9SCor e Forma:SolidPeso molecular:779.94Squalestatin 2
CAS:<p>Squalestatin 2 is an inhibitor of squalene synthase.</p>Fórmula:C33H44O13Pureza:98%Cor e Forma:SolidPeso molecular:648.69LAF-153
CAS:<p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>Fórmula:C18H32N2O7Cor e Forma:SolidPeso molecular:388.46STA 2
CAS:<p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>Fórmula:C21H34O3SCor e Forma:SolidPeso molecular:366.56Unoprostone
CAS:<p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>Fórmula:C22H38O5Pureza:98%Cor e Forma:SolidPeso molecular:382.53Oral antiplatelet agent 1
CAS:<p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>Fórmula:C23H24N4O5SPureza:98%Cor e Forma:SolidPeso molecular:468.53Calphostin A
CAS:<p>Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.</p>Fórmula:C44H38O12Cor e Forma:SolidPeso molecular:758.77Sdz 210-096
CAS:<p>Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.</p>Fórmula:C27H31NO2Cor e Forma:SolidPeso molecular:401.54Bacithrocin C
CAS:<p>Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.</p>Fórmula:C18H27N5O3Cor e Forma:SolidPeso molecular:361.439H-Glu(4MβNA)-OH
CAS:H-Glu(4MβNA)-OH serves as a substrate for aminopeptidases (APs).Fórmula:C16H18N2O4Cor e Forma:SolidPeso molecular:302.33TLN-232
CAS:<p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>Fórmula:C36H49N9O7S2Cor e Forma:SolidPeso molecular:783.96VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Fórmula:C20H21N3O2Cor e Forma:SolidPeso molecular:335.4Acetoxycycloheximide
CAS:<p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>Fórmula:C17H25NO6Cor e Forma:SolidPeso molecular:339.38ONO-DI-004
CAS:<p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>Fórmula:C24H38O6Cor e Forma:SolidPeso molecular:422.55Juglomycin B
CAS:<p>Juglomycin B exhibits broad-spectrum antibacterial and antimycobacterial properties and is capable of inhibiting Ehrlich ascites carcinoma in mice.</p>Fórmula:C14H10O6Cor e Forma:SolidPeso molecular:274.226MK-7445
CAS:<p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>Fórmula:C21H13Cl2N7OCor e Forma:SolidPeso molecular:450.28CGP 22979
CAS:<p>CGP 22979 is a renal selective vasodilator prodrug.</p>Fórmula:C16H24N4O4Cor e Forma:SolidPeso molecular:336.39Tyk2-IN-10
CAS:<p>Tyk2-IN-10 acts as an inhibitor of the Tyrosine Kinase 2 (Tyk2)-mediated signaling pathway, which plays a role in inflammation regulation.</p>Fórmula:C25H27N5O3Cor e Forma:SolidPeso molecular:445.51Oxeclosporin
CAS:<p>Oxeclosporin is a hydroxyethyl derivative of serine(8)-cyclosporine; inhibits proliferation and functions of lymphocytes.</p>Fórmula:C64H115N11O14Cor e Forma:SolidPeso molecular:1262.66MDK-3298
CAS:MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).Fórmula:C35H32BN3O7Pureza:98%Cor e Forma:SolidPeso molecular:617.46Orvepitant
CAS:<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Fórmula:C31H35F7N4O2Cor e Forma:SolidPeso molecular:628.62Tazide
<p>Tazide is an antitumor agent [1].</p>Fórmula:C12H16N4OCor e Forma:SolidPeso molecular:232.284-Chloropyridine
CAS:<p>4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.</p>Fórmula:C5H4ClNCor e Forma:SolidPeso molecular:113.55Unoprostone isopropyl
CAS:<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Fórmula:C25H44O5Pureza:98%Cor e Forma:SolidPeso molecular:424.61Cycloepoxydon
CAS:<p>Cycloepoxydon inhibits the NF-KB and AP-1 mediated secretion of alkaline phosphatase (SEAP) induced by Phorbol 12-myristate 13-acetate (PMA), with IC50 values of 1-2 μg/mL (4.2-8.4 μM) and 3-5 μg/mL (12.6-21 μM), respectively.</p>Fórmula:C12H16O5Cor e Forma:SolidPeso molecular:240.252GSK579289A
CAS:<p>GSK579289A is an inhibitor of benzimidazole thiophene.</p>Fórmula:C26H27ClN4O3SPureza:98%Cor e Forma:SolidPeso molecular:511.04VU0463271 quarterhydrate
<p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>Fórmula:C19H20N4O2S2Cor e Forma:SolidPeso molecular:387PTP1B-IN-3 diammonium
<p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>Fórmula:C12H13BrF2N3O3PCor e Forma:SolidPeso molecular:396.12PD 113271
CAS:PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.Fórmula:C19H27O10PPureza:98%Cor e Forma:SolidPeso molecular:446.39PZ-3022
CAS:<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Fórmula:C20H21N5OCor e Forma:SolidPeso molecular:347.41Cytosaminomycin B
CAS:<p>Cytosaminomycin B exhibits activity against Eimeria Tenella coccidia.</p>Fórmula:C26H37N5O8Cor e Forma:SolidPeso molecular:547.601BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Fórmula:C26H30F3N7O2Cor e Forma:SolidPeso molecular:529.56AT-IAP
CAS:AT-IAP is an effective dual antagonist of XIAP and cIAP1.Fórmula:C29H40FN5O2Pureza:98%Cor e Forma:SolidPeso molecular:509.66Formadicin A
CAS:<p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>Fórmula:C30H34N4O16Cor e Forma:SolidPeso molecular:706.608Org-31710
CAS:<p>Org-31710 is a progesterone receptor antagonist potentially for contraception.</p>Fórmula:C30H39NO2Pureza:98%Cor e Forma:SolidPeso molecular:445.64A 70450
CAS:<p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>Fórmula:C42H71ClN6O5Pureza:98%Cor e Forma:SolidPeso molecular:775.50Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Fórmula:C11H15N5Na4O10P2Cor e Forma:SolidPeso molecular:531.17Retezorogant
CAS:<p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>Fórmula:C23H33ClN2O3Cor e Forma:SolidPeso molecular:420.97SORT1-IN-1
CAS:<p>SORT1-IN-1 (compound 2) is a SORT1 inhibitor.</p>Fórmula:C17H13F3N2O4Cor e Forma:SolidPeso molecular:366.29HMGB1-IN-3
CAS:<p>HMGB1-IN-3 (compound E), a derivative of glycyrrhizic acid, exhibits potent inhibitory effects on HMGB1 (high mobility group protein 1). It is utilized in research related to intracerebral hemorrhage.</p>Fórmula:C31H46O4Cor e Forma:SolidPeso molecular:482.69IMR687
CAS:<p>IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.</p>Fórmula:C21H26N6O2Pureza:98%Cor e Forma:SolidPeso molecular:394.47CS-003 HCl
CAS:<p>CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.</p>Fórmula:C34H39Cl3N2O6SCor e Forma:SolidPeso molecular:710.1DI-404
CAS:<p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>Fórmula:C35H45ClN6O6SPureza:98%Cor e Forma:SolidPeso molecular:713.29BM635 mesylate (1493762-74-5 free base)
BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Fórmula:C26H33FN2O4SPureza:98%Cor e Forma:SolidPeso molecular:488.61KMN-80
CAS:<p>KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.</p>Fórmula:C21H33NO4Cor e Forma:SolidPeso molecular:363.495(S),6(R)-DiHETE
CAS:<p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.47G-9791
CAS:<p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>Fórmula:C26H26ClFN6O2Pureza:98%Cor e Forma:SolidPeso molecular:508.98GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Fórmula:C30H29Cl2F3N8O3Cor e Forma:SolidPeso molecular:677.50ROPA
CAS:<p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>Fórmula:C28H32O6Pureza:98%Cor e Forma:SolidPeso molecular:464.55B-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Fórmula:C55H74F3N15O11Cor e Forma:SolidPeso molecular:1178.27SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Fórmula:C21H21N5O5SCor e Forma:SolidPeso molecular:455.49Quorum Sensing-IN-1
<p>Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.</p>Fórmula:C13H10N2O2S2Cor e Forma:SolidPeso molecular:290.36PCSK9-IN-17
CAS:<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Fórmula:C16H19N5OSCor e Forma:SolidPeso molecular:329.42C-di-IMP
CAS:<p>Cyclic-di-IMP (C-di-IMP), a STING agonist, serves as a research tool in tumor studies.</p>Fórmula:C20H22N8O14P2Cor e Forma:SolidPeso molecular:660.38Ambelline
CAS:<p>Ambelline has antitumor activity.</p>Fórmula:C18H21NO5Pureza:98%Cor e Forma:SolidPeso molecular:331.36J-104118
CAS:<p>J-104118 potentially inhibits squalene synthase.</p>Fórmula:C28H26Cl2FNO5Pureza:98%Cor e Forma:SolidPeso molecular:546.41Haliangicin B
CAS:<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Fórmula:C22H32O5Cor e Forma:SolidPeso molecular:376.49Lorajmine
CAS:Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.Fórmula:C22H27ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:402.91Lactoquinomycin B
CAS:<p>Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.</p>Fórmula:C24H27NO9Cor e Forma:SolidPeso molecular:473.473Detoxin D1
CAS:<p>Detoxin D1 is a selective blasticidin S antagonist.</p>Fórmula:C28H41N3O8Pureza:98%Cor e Forma:SolidPeso molecular:547.64Hydrolyzed Fumonisin B2
CAS:Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.Fórmula:C22H47NO4Pureza:98%Cor e Forma:SolidPeso molecular:389.61Haloquinone
CAS:<p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>Fórmula:C17H12O5Cor e Forma:SolidPeso molecular:296.274UTPγS trisodium salt
CAS:<p>P2Y2 and P2Y4 receptor agonist</p>Fórmula:C9H12N2Na3O14P3SPureza:98%Cor e Forma:SolidPeso molecular:566.15
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