Outros inibidores
Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.
Foram encontrados 37827 produtos de "Outros inibidores"
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Haloquinone
CAS:<p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>Fórmula:C17H12O5Cor e Forma:SolidPeso molecular:296.274Hymenidin
CAS:Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.Fórmula:C11H12BrN5OPureza:96.85% - 99.52%Cor e Forma:SolidPeso molecular:310.15Tribenuron
CAS:<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Fórmula:C14H15N5O6SCor e Forma:SolidPeso molecular:381.36Cycloepoxydon
CAS:<p>Cycloepoxydon inhibits the NF-KB and AP-1 mediated secretion of alkaline phosphatase (SEAP) induced by Phorbol 12-myristate 13-acetate (PMA), with IC50 values of 1-2 μg/mL (4.2-8.4 μM) and 3-5 μg/mL (12.6-21 μM), respectively.</p>Fórmula:C12H16O5Cor e Forma:SolidPeso molecular:240.252NVP-CFC218
CAS:<p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>Fórmula:C37H45ClN4O4Cor e Forma:SolidPeso molecular:645.23(S)-Dexfadrostat
CAS:(S)-Dexfadrostat ((S)-Fadrozole), an aromatase inhibitor, exhibits an IC 50 of 4.6 nM in in vitro assays using human placental microsomes. It is applicable for research on estrogen-dependent breast cancer, gynecomastia, and systemic lupus erythematosus.Fórmula:C14H13N3Cor e Forma:SolidPeso molecular:223.27TT15
CAS:<p>TT15 is an agonist of the GLP-1R.</p>Fórmula:C51H44Cl2N4O6Cor e Forma:SolidPeso molecular:879.82Inactone
CAS:<p>Inactone is a biologically active molecule with a 3-pentanoylimino group that inhibits the large ribosomal subunit.</p>Fórmula:C15H21NO4Cor e Forma:SolidPeso molecular:279.332Dermostatin B
CAS:<p>Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.</p>Fórmula:C41H66O11Cor e Forma:SolidPeso molecular:734.956Chitinovorin C
CAS:<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Fórmula:C15H20N4O8SCor e Forma:SolidPeso molecular:416.406Pochonin D
CAS:<p>Pochonin D is an inhibitor of heat shock protein 90 (Hsp90) with antiviral and anti-inflammatory properties. It disrupts Hsp90, affecting the stability, folding, and assembly of viral proteins, thereby diminishing viral replication. Additionally, Pochonin D reduces the infiltration of inflammatory cells and decreases the secretion of inflammatory cytokines such as TNF-α and IL-1β, alleviating inflammatory responses. This compound shows potential for research in human rhinovirus (HRV) infections and cancer.</p>Fórmula:C18H19ClO5Cor e Forma:SolidPeso molecular:350.7934"-Demethylgentamicin C2
CAS:<p>4"-Demethylgentamicin C2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C19H39N5O7Cor e Forma:SolidPeso molecular:449.54BI-1388
CAS:<p>BI-1388 is a potent HCV NS3 protease inhibitor; halts replication across genotypes, including D168V/R155K mutants.</p>Fórmula:C41H53N7O9SCor e Forma:SolidPeso molecular:819.97CGC 11150
CAS:<p>CGC 11150 is a polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Fórmula:C40H100Cl10N10Cor e Forma:SolidPeso molecular:1075.82FTO-IN-5
CAS:<p>FTO-IN-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (FTO).</p>Fórmula:C23H18Cl2N6O6Cor e Forma:SolidPeso molecular:545.33Aquayamycin
CAS:<p>Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..</p>Fórmula:C25H26O10Cor e Forma:SolidPeso molecular:486.47Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Fórmula:C26H27N5O4Cor e Forma:SolidPeso molecular:473.52Leu-AMS R enantiomer
CAS:<p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>Fórmula:C16H25N7O7SPureza:98%Cor e Forma:SolidPeso molecular:459.48Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Fórmula:C18H18O6Cor e Forma:SolidPeso molecular:330.332Ericamycin
CAS:<p>Ericamycin is an antibiotic with antibacterial activity against Gram-positive bacteria. It effectively inhibits Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.004 to 0.016 µg/mL.</p>Fórmula:C28H21NO8Cor e Forma:SolidPeso molecular:499.468TRPC4/5-IN-1
<p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>Fórmula:C21H21N3OCor e Forma:SolidPeso molecular:331.41PTP1B-IN-17
<p>PTP1B-IN-17, a benzimidazole derivative, inhibits PTP1B (Ki: 30.2 μM) and may help study type 2 diabetes.</p>Fórmula:C26H19N3O4SCor e Forma:SolidPeso molecular:469.51Fujianmycin A
CAS:<p>Fujianmycin A exhibits activity against Bacillus subtilis (hay bacillus).</p>Fórmula:C19H14O5Cor e Forma:SolidPeso molecular:322.311Diazaquinomycin A
CAS:<p>Diazaquinomycin A (DAQA) is a diazaquinomycin antibiotic that acts as an inhibitor of thymidylate synthase. DAQA induces DNA damage, cell cycle arrest, and apoptosis through cleavage of PARP.</p>Fórmula:C20H22N2O4Cor e Forma:SolidPeso molecular:354.4Cuevaene B
CAS:<p>Cuevaene B can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. This compound exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and shows moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>Fórmula:C21H24O7Cor e Forma:SolidPeso molecular:388.411Glidobactin F
CAS:<p>Glidobactin F is an antitumor antibiotic effective against pathogenic fungi and yeasts. It has been shown to increase the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C25H40N4O6Cor e Forma:SolidPeso molecular:492.608Cirramycin B1
CAS:<p>Cirramycin B1 exhibits activity against both Gram-positive bacteria, Gram-negative bacteria, and mycoplasmas.</p>Fórmula:C37H59NO12Cor e Forma:SolidPeso molecular:709.864Piperazinomycin
CAS:<p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>Fórmula:C18H20N2O2Cor e Forma:SolidPeso molecular:296.36Collinone
CAS:<p>Collinone is a recombinant polyketide antibiotic with antimicrobial activity against Gram-positive bacteria and exhibits cytotoxicity.</p>Fórmula:C27H18O12Cor e Forma:SolidPeso molecular:534.425ICA-105665
CAS:ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.Fórmula:C19H15F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:355.34DC4SMe
CAS:<p>DC4SMe, a prodrug for targeted tumor therapy and ADC synthesis, has IC50s: 1.9 nM (Ramos), 2.9 nM (Namalwa), 1.8 nM (HL60/s).</p>Fórmula:C35H31ClN5O7PS2Pureza:98%Cor e Forma:SolidPeso molecular:764.21Glucosylquestiomycin
CAS:<p>Glucosylquestiomycin exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and yeast.</p>Fórmula:C18H18N2O7Cor e Forma:SolidPeso molecular:374.345Korormicin
CAS:<p>Korormicin is effective against marine Gram-negative bacteria but does not work against marine Gram-positive bacteria or common bacteria.</p>Fórmula:C25H39NO5Cor e Forma:SolidPeso molecular:433.581Serratamolide
CAS:<p>Serratamolide is a cyclic peptide antibiotic with activity against Gram-positive bacteria, mycobacteria, and fungi, although its potency is relatively weak.</p>Fórmula:C26H46N2O8Cor e Forma:SolidPeso molecular:514.6523-Hydroxyrifamycin S
CAS:<p>3-Hydroxyrifamycin S is an ansamycin antibiotic that exhibits strong activity against Gram-positive bacteria, while its effectiveness against Gram-negative bacteria is relatively limited.</p>Fórmula:C37H45NO13Cor e Forma:SolidPeso molecular:711.752Neoenactin B2
CAS:<p>Neoenactin B2 demonstrates potent antifungal activity against yeast and filamentous fungi.</p>Fórmula:C20H38N2O5Cor e Forma:SolidPeso molecular:386.526Edeine A1
CAS:<p>Edeine A1 inhibits DNA replication and protein biosynthesis, exhibiting activity against Gram-positive and Gram-negative bacteria, fungi, and yeasts.</p>Fórmula:C33H58N10O10Cor e Forma:SolidPeso molecular:754.875Ezomycin B2
CAS:<p>Ezomycin B2 is an antibiotic with antifungal activity.</p>Fórmula:C19H25N5O13Cor e Forma:SolidPeso molecular:531.427Enactin Ⅴa
CAS:<p>EnactinVa is a compound produced by the bacterium Streptomyces roseoviridis and exhibits relatively weak antifungal activity.</p>Fórmula:C19H38N2O5Cor e Forma:SolidPeso molecular:374.515Pluracidomycin A1
CAS:<p>Pluracidomycin A1 is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria, and it also inhibits β-lactamase enzymes.</p>Fórmula:C9H11NO10S2Cor e Forma:SolidPeso molecular:357.314Galactostatin
CAS:<p>Galactostatin is an inhibitor of β-galactosidase.</p>Fórmula:C6H13NO5Cor e Forma:SolidPeso molecular:179.171Flavomycoin
CAS:<p>Flavomycoin is an antibiotic known for its antifungal properties.</p>Fórmula:C40H66O12Cor e Forma:SolidPeso molecular:738.945Porothramycin A
CAS:<p>Porothramycin A is an antibiotic effective against Gram-positive bacteria and anaerobic bacteria.</p>Fórmula:C18H21N3O4Cor e Forma:SolidPeso molecular:343.377Curvularol
CAS:<p>Curvularol exhibits mild antifungal activity but lacks antibacterial effects. At a concentration of 150 ng/mL, it can inhibit the cell cycle progression of normal rat renal cells (G1 phase NRK). Additionally, 100 ng/mL of Curvularol can restore the morphology of deformed NRK cells induced by SRCTS. Curvularol also inhibits protein synthesis.</p>Fórmula:C15H22O4Cor e Forma:SolidPeso molecular:266.333Cytochalasin G
CAS:<p>Cytochalasin G exhibits reversible inhibition of cytokinesis and also inhibits macrophage phagocytosis and exocytosis, among other biological activities.</p>Fórmula:C29H34N2O4Cor e Forma:SolidPeso molecular:474.591Pyralomicin 2c
CAS:<p>Pyralomicin 2c is an antibiotic with antibacterial properties.</p>Fórmula:C19H19Cl2NO8Cor e Forma:SolidPeso molecular:460.262Epicorazine B
CAS:<p>Epicorazine B exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, with an MIC of 25 μg/mL.</p>Fórmula:C18H16N2O6S2Cor e Forma:SolidPeso molecular:420.45931-Homorifamycin W
CAS:<p>31-Homorifamycin W is an antibiotic discovered in Amycolatopsis mediterranei.</p>Fórmula:C36H47NO11Cor e Forma:SolidPeso molecular:669.758Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Fórmula:C21H36O7Cor e Forma:SolidPeso molecular:400.506Ro 0437626
CAS:<p>P2X1 purinergic receptor antagonist</p>Fórmula:C27H35N5O4SPureza:98%Cor e Forma:SolidPeso molecular:525.66Bacithrocin D
CAS:<p>Bacithrocin D (Thiolstatin D) inhibits various proteases and has the capability to prolong clotting time. It exhibits IC50 values of 124, 9, 0.85, and 0.01 μM against thrombin, factor Xa, trypsin, and papain, respectively.</p>Fórmula:C17H25N5O3Cor e Forma:SolidPeso molecular:347.412Schidigera-genin B
CAS:<p>Schidigera-genin B is a steroidal saponin that can be isolated from Yucca glauca. It exhibits mild antifungal activity.</p>Fórmula:C27H40O4Cor e Forma:SolidPeso molecular:428.604Mutatochrome
CAS:<p>Mutatochrome (Citroxanthin) is a compound found in plants.</p>Fórmula:C40H56OCor e Forma:SolidPeso molecular:552.872PPO-IN-15
CAS:PPO-IN-15 (compound (R)-I-5) serves as an inhibitor of protoporphyrinogen IX oxidase (PPO), offering efficacy against resistant weeds while maintaining safety for wheat and rice.Fórmula:C17H18ClFN4O5SCor e Forma:SolidPeso molecular:444.87Juglomycin B
CAS:<p>Juglomycin B exhibits broad-spectrum antibacterial and antimycobacterial properties and is capable of inhibiting Ehrlich ascites carcinoma in mice.</p>Fórmula:C14H10O6Cor e Forma:SolidPeso molecular:274.226MPO-IN-8
CAS:<p>MPO-IN-8, an orally active myeloperoxidase (MPO) inhibitor, effectively inhibits the production of hypochlorous acid in neutrophils and the release of extracellular traps (NETosis). In mice exhibiting gouty arthritis, it reduces swelling, decreases peroxidase activity, and lowers IL-1β levels.</p>Fórmula:C12H9N3O2Cor e Forma:SolidPeso molecular:227.22Dimesna free acid
CAS:<p>Dimesna (BNP-778), when used in conjunction with active cancer chemotherapy agents, can reduce the toxicity associated with uremia.</p>Fórmula:C4H10O6S4Cor e Forma:SolidPeso molecular:282.38Herbimycin B
CAS:<p>Herbimycin B, an ansamycin antibiotic, functions as an inhibitor of Src family kinases. It exhibits herbicidal effects on most monocotyledonous and dicotyledonous plants and can inhibit the activity of tobacco mosaic virus (TMV), HeLa cells, and Ehrlich cells.</p>Fórmula:C29H40N2O7Cor e Forma:SolidPeso molecular:528.637Lactoquinomycin B
CAS:<p>Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.</p>Fórmula:C24H27NO9Cor e Forma:SolidPeso molecular:473.473Netobimin
CAS:<p>Netobimin is an anthelmintic effective against naturally acquired gastrointestinal nematodes in cows.</p>Fórmula:C14H20N4O7S2Cor e Forma:SolidPeso molecular:420.46Halomicin D
CAS:<p>Halomicin D is an ansamycin-class antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C43H56N2O12Cor e Forma:SolidPeso molecular:792.911Resolvin E4
CAS:<p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.45CXCR4 probe 1
CAS:<p>CXCR4 probe 1, a specific PET tracer, targets CXCR4 with antagonist TN14003 (IC50: 6.9 nM), aiding in imaging CXCR4-related diseases and tumors.</p>Fórmula:C24H30FN5O4SCor e Forma:SolidPeso molecular:502.5911-Demethyltomaymycin
CAS:<p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>Fórmula:C15H18N2O4Cor e Forma:SolidPeso molecular:290.314Formadicin A
CAS:<p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>Fórmula:C30H34N4O16Cor e Forma:SolidPeso molecular:706.608Exophilin A
CAS:<p>Exophilin A is an antibiotic that exhibits activity against Gram-positive bacteria.</p>Fórmula:C30H56O10Cor e Forma:SolidPeso molecular:576.76Croconic acid disodium
CAS:<p>Croconic acid (disodium) (Nacr) enhances gene expression related to lysine crotonylation (Kcr) modification, which promotes cell growth and proliferation. This compound also shows promise in boosting somatic cell nuclear transfer (SCNT) efficiency and optimizing research in cell culture conditions.</p>Fórmula:C5Na2O5Cor e Forma:SolidPeso molecular:186.032-n-Heptyl-4-quinolinol
CAS:<p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>Fórmula:C16H21NOCor e Forma:SolidPeso molecular:243.34Haliangicin A
CAS:<p>Haliangicin A exhibits antifungal activity against filamentous fungi and also affects oomycetes, though it does not possess antibacterial properties.</p>Fórmula:C22H32O5Cor e Forma:SolidPeso molecular:376.49Narbomycin
CAS:<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Fórmula:C28H47NO7Cor e Forma:SolidPeso molecular:509.675Dykellic acid
CAS:<p>Dykellic acid is a RhoA inhibitor. It can suppress the migration and motility of B16 cells and inhibit the tubular formation of HUVECs. Dykellic acid shows potential for use in cancer research.</p>Fórmula:C14H16O4Cor e Forma:SolidPeso molecular:248.274Pluracidomycin C2
CAS:<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C11H15NO9S2Cor e Forma:SolidPeso molecular:369.37Epelmycin D
CAS:<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Fórmula:C30H35NO11Cor e Forma:SolidPeso molecular:585.599KY-02327 acetate
<p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>Fórmula:C22H31N3O6Cor e Forma:SolidPeso molecular:433.5Dihydroabikoviromycin
CAS:<p>Dihydroabikoviromycin is a secondary metabolite of Streptomyces anulatus and acts as a polyketide synthase inhibitor.</p>Fórmula:C10H13NOCor e Forma:SolidPeso molecular:163.216Haliangicin B
CAS:<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Fórmula:C22H32O5Cor e Forma:SolidPeso molecular:376.491-Deamino-1-hydroxygentamicin C2
CAS:<p>1-Deamino-1-hydroxygentamicin C2 (AntibioticSU-1) is an aminoglycoside antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H40N4O8Cor e Forma:SolidPeso molecular:464.554Diolmycin A1
CAS:<p>Diolmycin A1 is an antibiotic known for its anticoccidial activity.</p>Fórmula:C18H19NO3Cor e Forma:SolidPeso molecular:297.348Cytosaminomycin C
CAS:<p>Cytosaminomycin C exhibits anti-Eimeria Tenella coccidial activity.</p>Fórmula:C23H36N4O8Cor e Forma:SolidPeso molecular:496.554β-Prumycin hydrochloride
CAS:<p>β-Prumycin hydrochloride is a carbohydrate antibiotic that exhibits antifungal properties and possesses mild antibacterial activity.</p>Fórmula:C8H19Cl2N3O4Cor e Forma:SolidPeso molecular:292.16Cephemimycin
CAS:<p>Cephemimycin exhibits mild antibacterial and antifungal activity.</p>Fórmula:C16H22N4O9SCor e Forma:SolidPeso molecular:446.432Queenslandon
CAS:<p>Queenslandon exhibits moderate antifungal activity against fungi such as Streptomyces, Penicillium, Aspergillus fumigatus, and Aspergillus flavus, and has no effect on bacteria.</p>Fórmula:C20H26O8Cor e Forma:SolidPeso molecular:394.4218:0-LPS
CAS:<p>18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.</p>Fórmula:C24H48NO9PCor e Forma:SolidPeso molecular:525.613Granaticin B
CAS:<p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>Fórmula:C28H30O12Cor e Forma:SolidPeso molecular:558.531Feigrisolide D
CAS:<p>Feigrisolide D is a lactone produced by Streptomyces griseus. It exhibits moderate inhibitory activity against 3α-hydroxysteroid dehydrogenase.</p>Fórmula:C22H38O7Cor e Forma:SolidPeso molecular:414.533Feudomycin B
CAS:<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Fórmula:C28H31NO10Cor e Forma:SolidPeso molecular:541.546Asperenone
CAS:<p>Asperenone is a 15-lipoxygenase (15-LOX) inhibitor with an IC50 of 0.3 mM. Additionally, it acts as a platelet aggregation inhibitor with an IC50 of 0.23 mM. Asperenone also exhibits antifungal properties, inhibiting the growth of pathogenic fungi Ophiostoma crassivaginatum and O. piliferum, and may be utilized in research related to cardiovascular diseases and anti-infective treatments.</p>Fórmula:C20H22OCor e Forma:SolidPeso molecular:278.388Fumaryl-DL-alanine
CAS:<p>Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.</p>Fórmula:C7H9NO5Cor e Forma:SolidPeso molecular:187.15Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Fórmula:C24H26O8Cor e Forma:SolidPeso molecular:442.46Pterulinic acid
CAS:<p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>Fórmula:C15H11ClO4Cor e Forma:SolidPeso molecular:290.70Polyoxin H
CAS:<p>Polyoxin H is a nucleoside antifungal antibiotic that exhibits significant efficacy against rice sheath blight.</p>Fórmula:C23H32N6O13Cor e Forma:SolidPeso molecular:600.53Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Fórmula:C20H24O5Cor e Forma:SolidPeso molecular:344.43-O-Demethylmonensin A
CAS:<p>3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).</p>Fórmula:C35H60O11Cor e Forma:SolidPeso molecular:656.84Monamycin H1
CAS:<p>Monamycin H1 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.</p>Fórmula:C34H56ClN7O8Cor e Forma:SolidPeso molecular:726.30Antileishmanial agent-4
<p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>Fórmula:C17H18N4O4Cor e Forma:SolidPeso molecular:342.35(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Fórmula:C24H24N4O6Cor e Forma:SolidPeso molecular:464.47Bacithrocin B
CAS:<p>Bacithrocin B is a thrombin inhibitor that suppresses the activity of thrombin, Factor Xa, trypsin, and papain, with IC50 values of 84 μM, 17 μM, 1.7 μM, and 0.02 μM, respectively.</p>Fórmula:C19H29N5O3Cor e Forma:SolidPeso molecular:375.465Nebramycin Ⅳ
CAS:<p>Nebramycin IV is an aminoglycoside antibiotic with a broad antimicrobial spectrum, demonstrating significant efficacy against Gram-positive bacteria, Gram-negative bacteria, and mycobacteria.</p>Fórmula:C19H38N6O11Cor e Forma:SolidPeso molecular:526.539Resorcinomycin B
CAS:<p>Resorcinomycin B is an antibiotic found in [Streptoverticillum roseoverticillatum].</p>Fórmula:C13H18N4O5Cor e Forma:SolidPeso molecular:310.3062-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H41N5O8Cor e Forma:SolidPeso molecular:479.568HMGB1-IN-3
CAS:<p>HMGB1-IN-3 (compound E), a derivative of glycyrrhizic acid, exhibits potent inhibitory effects on HMGB1 (high mobility group protein 1). It is utilized in research related to intracerebral hemorrhage.</p>Fórmula:C31H46O4Cor e Forma:SolidPeso molecular:482.69Glidobactin C
CAS:<p>Glidobactin C (GlbC) is an antitumor antibiotic with activity against pathogenic fungi and yeasts. It exhibits antifungal properties against Candida albicans and Aspergillus fumigatus, with a minimum inhibitory concentration (MIC) of 0.8 μg/mL. Additionally, Glidobactin C prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C29H48N4O6Cor e Forma:SolidPeso molecular:548.715ZIKV-IN-5
<p>ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.</p>Fórmula:C36H45NO4SiCor e Forma:SolidPeso molecular:583.83TP-030-2
CAS:<p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>Fórmula:C23H21BrN4O3Cor e Forma:SolidPeso molecular:481.34Menoxymycin A
CAS:<p>Menoxymycin A is an antibiotic with cytotoxic properties. It inhibits the growth of KB and N18-RE-105 cells, with IC50 values of 0.86 μM and 0.14 μM, respectively.</p>Fórmula:C24H27NO9Cor e Forma:SolidPeso molecular:473.47311-Deacetoxywortmannin
CAS:<p>11-Deacetoxywortmannin is an antibiotic with potent antibacterial and anti-inflammatory properties, and it also exhibits anti-edema effects.</p>Fórmula:C21H22O6Cor e Forma:SolidPeso molecular:370.396NRMA-8
CAS:<p>NRMA-8 is a small-molecule nuclear receptor modulator capable of penetrating the brain. It holds potential for research into central nervous system (CNS) diseases, including Alzheimer's disease, Parkinson's disease, demyelinating diseases, and glioblastoma.</p>Fórmula:C20H23ClN2O3Cor e Forma:SolidPeso molecular:374.867β,16α-Dihydroxybufalin
CAS:<p>7β,16α-Dihydroxybufalin, a dihydroxylated derivative of bufalin, demonstrates cytotoxic properties against various cancer cell lines.</p>Fórmula:C24H34O6Cor e Forma:SolidPeso molecular:418.52S24-14
CAS:S24-14 serves as an effective anti-osteoporosis agent by inhibiting osteoclastogenesis, promoting osteoblast differentiation, and reducing bone resorption.Fórmula:C19H12N2O3SCor e Forma:SolidPeso molecular:348.38MB-07344 sodium
<p>"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."</p>Fórmula:C19H25NaO5PPureza:98%Cor e Forma:SolidPeso molecular:387.36Chrymutasin C
CAS:<p>Chrymutasin C is a glycoside antitumor antibiotic with cytotoxic properties.</p>Fórmula:C39H43NO17Cor e Forma:SolidPeso molecular:797.75516(S)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds to human IP & EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>Fórmula:C22H32O4Cor e Forma:SolidPeso molecular:360.492-Hydroxygentamicin B1
CAS:<p>2-Hydroxygentamicin B1 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H40N4O11Cor e Forma:SolidPeso molecular:512.552ONL-1204
CAS:<p>ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.</p>Fórmula:C71H100N18O16Cor e Forma:SolidPeso molecular:1461.66IACS-8779 disodium
CAS:<p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>Fórmula:C21H23N9Na2O10P2S2Cor e Forma:SolidPeso molecular:733.52Memnobotrin A
CAS:<p>Memnobotrin A is an antibiotic with inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.</p>Fórmula:C25H33NO5Cor e Forma:SolidPeso molecular:427.53ADH-353
CAS:<p>ADH-353 inhibits Aβ fibrillization and mitigates Aβ-induced cytotoxicity in SH-SY5Y and N2a cells, making it useful for studies related to Alzheimer's disease.</p>Fórmula:C27H38N8O6Cor e Forma:SolidPeso molecular:570.64Melithiazole K
CAS:<p>Melithiazol K is an antibiotic and functions as a β-methoxyacrylate (MOA) inhibitor, exhibiting strong resistance.</p>Fórmula:C20H26N2O5S2Cor e Forma:SolidPeso molecular:438.561RSV-IN-5
CAS:<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Fórmula:C28H37N7O2Cor e Forma:SolidPeso molecular:503.64SSTR5 antagonist 2 TFA
CAS:<p>Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.</p>Fórmula:C34H36F4N2O7Pureza:98%Cor e Forma:SolidPeso molecular:660.65ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Cor e Forma:SolidGilvusmycin
CAS:<p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>Fórmula:C38H34N6O8Cor e Forma:SolidPeso molecular:702.712Leucomycin U
CAS:<p>Leucomycin U is a macrolide antibiotic. It demonstrates significant activity against Gram-positive bacteria and also exhibits effects on spirochetes, rickettsiae, and chlamydiae.</p>Fórmula:C37H61NO14Cor e Forma:SolidPeso molecular:743.878Celesticetin B
CAS:<p>Celesticetin B is an antibiotic primarily exhibiting antibacterial activity against Gram-positive microorganisms.</p>Fórmula:C21H38N2O8SCor e Forma:SolidPeso molecular:478.6GYKI-53784
CAS:<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Fórmula:C19H20N4O3Cor e Forma:SolidPeso molecular:352.39ATX inhibitor 22
<p>ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.</p>Fórmula:C19H17Cl3F2N2O4SCor e Forma:SolidPeso molecular:513.77Resorcinomycin A
CAS:<p>Resorcinomycin A is an antibiotic with potent antimycobacterial activity and relatively weaker activity against mycoplasma.</p>Fórmula:C14H20N4O5Cor e Forma:SolidPeso molecular:324.332Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Fórmula:C23H31NO7SPureza:98%Cor e Forma:White To Off-White SolidPeso molecular:465.56Rosiptor acetate
CAS:<p>Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.</p>Fórmula:C22H39NO4Pureza:98%Cor e Forma:Solid PowderPeso molecular:381.553'-O-Decarbamoylirumamycin
CAS:<p>3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.</p>Fórmula:C40H64O11Cor e Forma:SolidPeso molecular:720.93Hydrolyzed Fumonisin B2
CAS:Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.Fórmula:C22H47NO4Pureza:98%Cor e Forma:SolidPeso molecular:389.61MEIS-IN-3
<p>MEIS-IN-3 is a potent inhibitor of MEIS.</p>Fórmula:C25H26N2O4Cor e Forma:SolidPeso molecular:418.489-Hydroxyoudemansin A
CAS:<p>9-Hydroxyoudemansin A exhibits antifungal activity with a minimum inhibitory concentration (MIC) of 12.5 μg/mL against Saccharomyces cerevisiae. It shows resistance to fungi such as Candida albicans, Rhodotorula, Penicillium, and Streptomyces, with MIC values all exceeding 50 μg/mL. It does not possess antibacterial properties.</p>Fórmula:C16H20O4Cor e Forma:SolidPeso molecular:276.3282-Hydroxygentamicin B
CAS:<p>2-Hydroxygentamicin B is an aminoglycoside antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C19H38N4O11Cor e Forma:SolidPeso molecular:498.525AP-6
CAS:AP-6, a selective TMEM175 inhibitor, enhances lysosomal macromolecular catabolism by acutely inhibiting TMEM175, thus speeding up macrophage and other digestive activities. This compound holds potential for use in Parkinson's disease research due to its role in modulating lysosomal function.Fórmula:C16H14N4Cor e Forma:SolidPeso molecular:262.3110-Decarbomethoxyaclacinomycin A
CAS:<p>10-Decarbomethoxyaclacinomycin A is an anthracycline antibiotic produced by the mutant strain Streptomyces galilaeus MA144-Mlt KE303. This compound exhibits antibacterial activity.</p>Fórmula:C40H51NO13Cor e Forma:SolidPeso molecular:753.832ODN 2088
CAS:<p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>Cor e Forma:SolidDiphenicillin
CAS:<p>Diphenicillin (Ancillin (free acid); 2-Biphenylyl penicillin (free acid); SKF-12141 (free acid)) is a penicillin that resists Penicillinase and exhibits antibacterial activity. It shows effective activity against Gram-positive cocci. Diphenicillin is promising for research on infectious diseases caused by Gram-positive bacteria such as staphylococci, pneumococci, and group A streptococci.</p>Fórmula:C21H20N2O4SCor e Forma:SolidPeso molecular:396.459Antimalarial agent 2
<p>Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.</p>Fórmula:C27H25N3O5Cor e Forma:SolidPeso molecular:471.5SL agonist 1
CAS:<p>SL agonist 1, a Strigolactone (SL) agonist, is effective in promoting Arabidopsis seed germination through its recognition by the SL receptors OmKAI2d3 and OmKAI2d4.</p>Fórmula:C11H8FNO5Cor e Forma:SolidPeso molecular:253.18JBJ-08-178-01
CAS:JBJ-08-178-01, a mutant-selective tyrosine kinase inhibitor, targets (HER2) human epidermal growth factor receptor 2 and exhibits antitumoral activity. This compound not only diminishes HER2's kinase activity and protein levels through the induction of proteasomal degradation of the receptor but also shows promise in non-small-cell lung cancer research.Fórmula:C31H30N8O3Cor e Forma:SolidPeso molecular:562.62BRD4-IN-9
CAS:<p>BRD4-IN-9, an orally active BRD4 inhibitor, demonstrates a potent IC50 of 9.4 nM. In a murine melanoma xenograft model, it effectively inhibits tumor growth.</p>Fórmula:C24H23N3O3Cor e Forma:SolidPeso molecular:401.46Tezampanel hydrate
CAS:<p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>Fórmula:C13H23N5O3Cor e Forma:SolidPeso molecular:297.35Glidobactin G
CAS:<p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Fórmula:C27H44N4O7Cor e Forma:SolidPeso molecular:536.6619-cis-13,14-Dihydroretinoic acid
CAS:<p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>Fórmula:C20H30O2Cor e Forma:SolidPeso molecular:302.451Demethylblasticidin S
CAS:<p>Demethylblasticidin S is an antifungal antibiotic produced by Streptomyces griseochromogenes.</p>Fórmula:C16H24N8O5Cor e Forma:SolidPeso molecular:408.412Furaprevir
CAS:<p>Furaprevir is an HCV NS3/4A Inhibitor</p>Fórmula:C47H56N6O10SCor e Forma:SolidPeso molecular:897.05BMS-748730
CAS:<p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>Fórmula:C22H26ClN7O3SCor e Forma:SolidPeso molecular:504.01Allosucrose
CAS:<p>Allosucrose is a biochemical.</p>Fórmula:C12H22O11Cor e Forma:SolidPeso molecular:342.30Tyk2-IN-10
CAS:<p>Tyk2-IN-10 acts as an inhibitor of the Tyrosine Kinase 2 (Tyk2)-mediated signaling pathway, which plays a role in inflammation regulation.</p>Fórmula:C25H27N5O3Cor e Forma:SolidPeso molecular:445.51H-Glu(4MβNA)-OH
CAS:H-Glu(4MβNA)-OH serves as a substrate for aminopeptidases (APs).Fórmula:C16H18N2O4Cor e Forma:SolidPeso molecular:302.33Hesperidin dihydrochalcone
CAS:Hesperidin dihydrochalcone, a non-toxic sweetener with high sweetness and low calories, exhibits multiple biological activities including anti-oxidation, liver and kidney protection, bacteriostasis, and enhancement of gastrointestinal health.Fórmula:C28H36O15Cor e Forma:SolidPeso molecular:612.58SGK1-IN-3
<p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>Fórmula:C23H20Cl2N6O3SCor e Forma:SolidPeso molecular:531.41Vanin-1-IN-3
<p>Vanin-1-IN-3 (OMP-7) is a vanin-1 inhibitor with an IC 50 of 0.038 μM [1].</p>Fórmula:C17H22F3NO5Cor e Forma:SolidPeso molecular:377.36AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Fórmula:C32H38N6O3Cor e Forma:SolidPeso molecular:554.7Bis(N-methylthioformohydroxamate)nickel (II)
CAS:<p>Bis(N-methylthioformohydroxamate)nickel (II) is a nickel-containing antibiotic that exhibits significant activity against both Gram-positive and Gram-negative bacteria, as well as antitumor properties.</p>Fórmula:C4H8N2NiO2S2Cor e Forma:SolidPeso molecular:238.942STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Fórmula:C17H12N4O4Cor e Forma:SolidPeso molecular:336.3Phyllosinol
CAS:<p>Phyllosinol is an antifungal antibiotic.</p>Fórmula:C7H8O4Cor e Forma:SolidPeso molecular:156.136ZBH-1205
CAS:<p>ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.</p>Fórmula:C29H31N3O8Cor e Forma:SolidPeso molecular:549.57Enamidonin
CAS:<p>Enamidonin is a lipopeptide antibiotic. It inhibits EGF-dependent [3H] thymidine incorporation in Balb/MK cells with an IC50 of 10 μg/mL and can restore the transformed SRCTS-NRK cells to their normal flat shape with an ED50 of 10 μg/mL. It exhibits no antibacterial activity.</p>Fórmula:C37H51N7O7Cor e Forma:SolidPeso molecular:705.844LLS30
CAS:<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Fórmula:C34H33Cl4N5O3Cor e Forma:SolidPeso molecular:701.47Idraparinux Na
CAS:<p>Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa Inhibitor</p>Fórmula:C38H55Na9O49S7Cor e Forma:SolidPeso molecular:1727.14CXN37378
CAS:<p>CXN37378, aka NAP, is a potent MOR-selective antagonist with no official name yet, termed per MedKoo Nomenclature.</p>Fórmula:C27H31N3O4Cor e Forma:SolidPeso molecular:461.55Deflectin 1a
CAS:<p>Deflectin 1a is an antibiotic with activities such as lysing bacteria, lysing red blood cells, and inhibiting Ehrlich ascites cancer cells. However, its effectiveness can be neutralized by the addition of serum or serum albumin.</p>Fórmula:C21H24O5Cor e Forma:SolidPeso molecular:356.412VEGFR-2-IN-16
<p>VEGFR-2-IN-16 (Compound 15b) is a potent inhibitor of VEGFR-2 (IC50: 86.36 nM) that exhibits antitumour effects.</p>Fórmula:C21H13Cl2N3O2Cor e Forma:SolidPeso molecular:410.25Diarylalkane derivative 1
CAS:<p>Diarylalkane derivative 1 is used for the research of pancreatitis.</p>Fórmula:C34H51NO4Pureza:98%Cor e Forma:SolidPeso molecular:537.77PF-06305591 dihydrate
<p>PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADME</p>Fórmula:C15H26N4O3Cor e Forma:SolidPeso molecular:310.39Pyloricidin A
CAS:<p>Pyloricidin A is an antibiotic effective against Helicobacter pylori, produced by Bacillus sp. HC-70. It exhibits strong anti-Helicobacter pylori activity and shows no efficacy against other bacteria or yeasts.</p>Fórmula:C31H51N5O10Cor e Forma:SolidPeso molecular:653.76ZK159222
CAS:<p>ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.</p>Fórmula:C32H48O5Pureza:98%Cor e Forma:SolidPeso molecular:512.72Piloquinone
CAS:<p>Piloquinone is a type of phenanthrene compound that exhibits mild inhibitory effects on mycobacteria and protozoa.</p>Fórmula:C21H20O5Cor e Forma:SolidPeso molecular:352.38Faldaprevir sodium
CAS:<p>Faldaprevir sodium: HCV treatment, inhibits NS3/NS4A protease, P-glycoprotein, CYP3A4, UGT1A1.</p>Fórmula:C40H48BrN6NaO9SCor e Forma:SolidPeso molecular:891.81Enteromycin
CAS:<p>Enteromycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C6H8N2O5Cor e Forma:SolidPeso molecular:188.138Cervicarcin
CAS:<p>Cervicarcin is an antitumor antibiotic (antibiotic) exhibiting strong inhibitory effects on sarcoma 180 and sarcoma NF, while showing weaker activity against sarcoma 37, Ehrlich ascites carcinoma, and Freund leukemia.</p>Fórmula:C19H20O9Cor e Forma:SolidPeso molecular:392.357Kurasoin A
CAS:<p>Kurasoin A is an inhibitor of the enzyme farnesyltransferase.</p>Fórmula:C16H16O3Cor e Forma:SolidPeso molecular:256.296Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Fórmula:C11H15N5Na4O10P2Cor e Forma:SolidPeso molecular:531.17Enactin Ia
CAS:<p>Enactin Ia is found in Streptomyces roseoviridis and exhibits mild antibacterial activity.</p>Fórmula:C20H38N2O6Cor e Forma:SolidPeso molecular:402.526Dersimelagon phosphate
CAS:<p>Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.</p>Fórmula:C36H48F4N3O9PCor e Forma:SolidPeso molecular:773.75AZD2353
CAS:<p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>Fórmula:C22H19ClFN3O3Cor e Forma:SolidPeso molecular:427.86Crotocin
CAS:<p>Crotocin exhibits bactericidal activity against Cryptococcus neoformans, Candida albicans, and Saccharomyces cerevisiae (brewer’s yeast), but it can be inactivated by blood.</p>Fórmula:C19H24O5Cor e Forma:SolidPeso molecular:332.391Acrylamidine
CAS:<p>Acrylamidine exhibits weak antifungal and yeast activity.</p>Fórmula:C3H6N2Cor e Forma:SolidPeso molecular:70.09Epicochlioquinone A
CAS:<p>Epicochlioquinone A inhibits rat liver microsomal ACAT with an IC50 of 1.7 μM and inhibits plasma lecithin-cholesterol acyltransferase (LCAT) with an IC50 of 15.8 μM. At a dosage of 75 mg/kg, it can reduce cholesterol absorption in rats by 50%.</p>Fórmula:C30H44O8Cor e Forma:SolidPeso molecular:532.666Epoxyquinomicin B
CAS:<p>Epoxyquinomicin B is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus, with a minimum inhibitory concentration (MIC) of 6.25-12.5 µg/mL. It also shows cytotoxicity in cancer cells L1210, with an IC50 of 16.3 µg/mL. Additionally, Epoxyquinomicin B demonstrates anti-inflammatory effects on collagen-induced arthritis.</p>Fórmula:C14H11NO6Cor e Forma:SolidPeso molecular:289.24P2X7 receptor antagonist-1
<p>P2X7 receptor antagonist-1 is a purinergic P2X7 receptor antagonist with anti-neuroinflammatory effects.</p>Fórmula:C22H20F4N2O3Cor e Forma:SolidPeso molecular:436.4Diatretyne Ⅰ
CAS:Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.Fórmula:C8H5NO3Cor e Forma:SolidPeso molecular:163.13LY2934747
CAS:<p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>Fórmula:C10H13NO4Cor e Forma:SolidPeso molecular:211.21Phencomycin
CAS:<p>Phencomycin exhibits mild activity against Gram-positive bacteria and inhibits physiologically important enzymes such as renin, with an IC50 of 440 μg/mL.</p>Fórmula:C15H10N2O4Cor e Forma:SolidPeso molecular:282.251Hynapene C
CAS:<p>Hynapene C exhibits an inhibitory minimum inhibitory concentration (MIC) of 34.7 μM against Eimeria acervulina.</p>Fórmula:C18H24O3Cor e Forma:SolidPeso molecular:288.381Polyozellin
CAS:<p>Polyozellin is a prolyl endopeptidase inhibitor with properties effective against inflammation, cancer, and diseases related to oxidative stress.</p>Fórmula:C22H14O10Cor e Forma:SolidPeso molecular:438.341Leptofuranin C
CAS:<p>Leptofuranin C, found in the Str. tanashiensis strain, is known to arrest normal cell progression and induce cell death.</p>Fórmula:C32H46O5Cor e Forma:SolidPeso molecular:510.705Cremeomycin
CAS:<p>Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.</p>Fórmula:C8H6N2O4Cor e Forma:SolidPeso molecular:194.144SENP2-IN-1
CAS:<p>SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.</p>Fórmula:C32H29N3O5S2Cor e Forma:SolidPeso molecular:599.72GS-9160
CAS:<p>GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.</p>Fórmula:C20H18FN3O4SCor e Forma:SolidPeso molecular:415.44FK-906 HCl
CAS:<p>FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.</p>Fórmula:C40H64ClN7O7Cor e Forma:SolidPeso molecular:790.44BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Fórmula:C26H30F3N7O2Cor e Forma:SolidPeso molecular:529.56Deoxyradicinin
CAS:<p>Deoxyradicinin is a biosynthetic precursor of Radicinin. It can inhibit Xylella fastidiosa and Liberibacter crescens, with a minimum inhibitory concentration (MIC) of 3.5 μg/mL against Liberibacter crescens. Deoxyradicinin is applicable for research on controlling plant diseases caused by these pathogens.</p>Fórmula:C12H12O4Cor e Forma:SolidPeso molecular:220.221Kynapcin-28
CAS:<p>Kynapcin-28 is a non-competitive inhibitor of prolyl endopeptidase (PEP) with an IC50 of 76.80 μM and exhibits weak inhibitory effects on other serine proteases.</p>Fórmula:C19H12O10Cor e Forma:SolidPeso molecular:400.293Antitumor agent-75
<p>Antitumor agent-75 is a novel and potent antitumor agent.</p>Fórmula:C26H23FN6Cor e Forma:SolidPeso molecular:438.5PTP1B-IN-3 diammonium
<p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>Fórmula:C12H13BrF2N3O3PCor e Forma:SolidPeso molecular:396.12Belatacept
CAS:<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Cor e Forma:LiquidDiaporthin
CAS:<p>Diaporthin is a phytotoxin that can be isolated from Cryphonectria parasitica. It exhibits antibacterial activity.</p>Fórmula:C13H14O5Cor e Forma:SolidPeso molecular:250.247
