Outros inibidores
Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.
Foram encontrados 37902 produtos de "Outros inibidores"
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VEGFR-2-IN-12
<p>VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.</p>Fórmula:C22H24N6O3SCor e Forma:SolidPeso molecular:452.53Netobimin
CAS:<p>Netobimin is an anthelmintic effective against naturally acquired gastrointestinal nematodes in cows.</p>Fórmula:C14H20N4O7S2Cor e Forma:SolidPeso molecular:420.46H-Glu(4MβNA)-OH
CAS:<p>H-Glu(4MβNA)-OH serves as a substrate for aminopeptidases (APs).</p>Fórmula:C16H18N2O4Cor e Forma:SolidPeso molecular:302.33Hesperidin dihydrochalcone
CAS:Hesperidin dihydrochalcone, a non-toxic sweetener with high sweetness and low calories, exhibits multiple biological activities including anti-oxidation, liver and kidney protection, bacteriostasis, and enhancement of gastrointestinal health.Fórmula:C28H36O15Cor e Forma:SolidPeso molecular:612.58Tubulosine
CAS:<p>Tubulosine is an anticancer agent that inhibits cancer cell growth.</p>Fórmula:C29H37N3O3Cor e Forma:SolidPeso molecular:475.62Gunacin
CAS:<p>Gunacin is a quinone antibiotic that exhibits significant activity against Gram-positive bacteria, Gram-negative bacteria, and mycoplasmas.</p>Fórmula:C17H16O8Cor e Forma:SolidPeso molecular:348.304Hymenidin
CAS:<p>Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.</p>Fórmula:C11H12BrN5OPureza:96.85% - 99.52%Cor e Forma:SolidPeso molecular:310.15Antitrypanosomal agent 5
<p>Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).</p>Fórmula:C30H30N6O4SCor e Forma:SolidPeso molecular:570.66Antibiotic MA 144M2
CAS:<p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>Fórmula:C42H55NO16Cor e Forma:SolidPeso molecular:829.88Amrubicin HCl
CAS:<p>Amrubicin (SM-5887), an anthracycline, treats lung cancer by inhibiting DNA replication and topoisomerase II, with less cardiac toxicity.</p>Fórmula:C25H25NO9Cor e Forma:SolidPeso molecular:483.47Seldomycin factor 1
CAS:<p>Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.</p>Fórmula:C17H34N4O10Cor e Forma:SolidPeso molecular:454.473METTL3-IN-2
CAS:<p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>Fórmula:C25H26N8OCor e Forma:SolidPeso molecular:454.53Anticancer agent 12
<p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>Fórmula:C16H17BrN4O2SCor e Forma:SolidPeso molecular:409.3Pyrisulfoxin A
CAS:<p>Pyrisulfoxin A is an antibiotic that can be found in Streptomyces callfornicus [BS-75].</p>Fórmula:C13H13N3O3SCor e Forma:SolidPeso molecular:291.326PF1070A
CAS:<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Fórmula:C31H44N4O6Cor e Forma:SolidPeso molecular:568.7Tauro-ω-muricholic acid sodium
<p>Tauro-ω-muricholic acid sodium (TωMCA sodium) is an analogue of tauro-α-muricholic acid, a bile acid of hepatic origin.</p>Fórmula:C26H44NNaO7SCor e Forma:SolidPeso molecular:537.68ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Fórmula:C29H33ClF2N6O9Pureza:98%Cor e Forma:SolidPeso molecular:683.06CYP121A1-IN-1
<p>CYP121A1-IN-1: Strong inhibitor for CYP121A1, hinders Mycobacterium tuberculosis growth (MIC 90 ~6.25 μM), reduces mycocyclosin synthesis.</p>Fórmula:C22H20N4OCor e Forma:SolidPeso molecular:356.42Topoisomerase II inhibitor 6
<p>Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.</p>Fórmula:C19H18N4O2Cor e Forma:SolidPeso molecular:334.37NAZ2329
CAS:<p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>Fórmula:C21H18F3NO4S3Cor e Forma:SoildPeso molecular:501.56Plumbemycin B
CAS:<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Fórmula:C12H21N4O8PCor e Forma:SolidPeso molecular:380.29S-2,3-Dicarboxyaziridine
CAS:<p>S-2,3-Dicarboxyaziridine is a metabolite that can be isolated from Streptomyces species and exhibits antibacterial activity.</p>Fórmula:C4H5NO4Cor e Forma:SolidPeso molecular:131.087Brostallicin HCl
CAS:<p>Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.</p>Fórmula:C30H36BrClN12O5Cor e Forma:SolidPeso molecular:760.04PCSK9-IN-17
CAS:<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Fórmula:C16H19N5OSCor e Forma:SolidPeso molecular:329.42MRS2279 diammonium
CAS:<p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>Fórmula:C13H24ClN7O8P2Cor e Forma:SolidPeso molecular:503.77GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Fórmula:C30H29Cl2F3N8O3Cor e Forma:SolidPeso molecular:677.50MB725
CAS:<p>MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.</p>Fórmula:C18H21IN4O2SCor e Forma:SolidPeso molecular:484.35Tzc 5665
CAS:<p>Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.</p>Fórmula:C31H38ClN5O7Cor e Forma:SolidPeso molecular:628.12SSTR5 antagonist 2 hydrochloride
<p>SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.</p>Fórmula:C32H36ClFN2O5Cor e Forma:SolidPeso molecular:583.09Copper(II) ionophore I
CAS:Copper(II) ionophore I is an active compound.Fórmula:C26H44N2S4Cor e Forma:SolidPeso molecular:512.90Terfluranol
CAS:<p>Terfluranol, a benzyl derivative, is utilized as an antitumor medication.</p>Fórmula:C17H17F3O2Cor e Forma:SolidPeso molecular:310.31LAS195319
CAS:<p>LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.</p>Fórmula:C29H26N10O3SCor e Forma:SolidPeso molecular:594.652,4-Diaminoanisole
CAS:<p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>Fórmula:C7H10N2OCor e Forma:SolidPeso molecular:138.17Octahydrocyclopenta[c]pyrrole
CAS:<p>Octahydrocyclopenta[c]pyrrole has demonstrated promising applications in the fields of anti-inflammatory, anti-tumor, and neuroprotection. The unique structure-activity relationship of Octahydrocyclopenta[c]pyrrole offers fresh insights for the design of new drugs.</p>Fórmula:C7H13NCor e Forma:SolidPeso molecular:111.18Antitumor agent-51
<p>Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.</p>Fórmula:C23H25N5O2SCor e Forma:SolidPeso molecular:435.54Taprostene
CAS:<p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>Fórmula:C24H30O5Cor e Forma:SolidPeso molecular:398.49BMS-824
CAS:<p>BMS-824: potent HCV NS5A inhibitor, IC50 ~5 nM, therapeutic index >10,000, specific to HCV.</p>Fórmula:C27H25F3N4O5Cor e Forma:SolidPeso molecular:542.51SARS-CoV-2 nsp3-IN-1
<p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>Fórmula:C17H15N5O2Cor e Forma:SolidPeso molecular:321.33ZL-Pin13
CAS:<p>ZL-Pin13: potent Pin1 inhibitor (IC50: 67 nM), halts MDA-MB-231 cell growth, reduces Pin1 substrates.</p>Fórmula:C24H23ClN2O3SCor e Forma:SoildPeso molecular:454.97FTI-2148
CAS:<p>FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.</p>Fórmula:C24H28N4O3SPureza:98%Cor e Forma:SolidPeso molecular:452.57SHP2 IN-1
CAS:<p>SHP2 IN-1 is an allergic SHP2 (PTPN11) inhibitor(IC50 : 3 nM).</p>Fórmula:C18H22Cl2N6OSPureza:98%Cor e Forma:SolidPeso molecular:441.38TrxR-IN-5
<p>TrxR-IN-5 (compound 4f) is an effective inhibitor of thioredoxin reductase (TrxR) with an IC₅₀ of 0.16 μM. anti-proliferative and anti-metastatic.</p>Fórmula:C26H22O3Cor e Forma:SolidPeso molecular:382.46Hsp90-IN-16
<p>Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.</p>Fórmula:C30H26FN3O6Cor e Forma:SolidPeso molecular:543.54Feudomycin B
CAS:<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Fórmula:C28H31NO10Cor e Forma:SolidPeso molecular:541.546KOS-1584
CAS:<p>KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.</p>Fórmula:C27H39NO5SCor e Forma:SolidPeso molecular:489.67Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Fórmula:C26H36N2O4Cor e Forma:SolidPeso molecular:440.5818:0-LPS
CAS:<p>18:0-LPS (Lysophosphatidylserine C18:0) is an endogenous lipid identified during the oxidation of phospholipids. It holds potential for use in cardiovascular disease research.</p>Fórmula:C24H48NO9PCor e Forma:SolidPeso molecular:525.613DC41SMe
CAS:<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Fórmula:C38H36ClN5O4S2Pureza:98%Cor e Forma:SolidPeso molecular:726.314α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Fórmula:C40H64O8Cor e Forma:SolidPeso molecular:672.93SARS 3CLpro-IN-1
CAS:<p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>Fórmula:C22H38N4O2Cor e Forma:SolidPeso molecular:390.56MIF2-IN-1
<p>MIF2-IN-1, potent inhibitor of MIF2 (IC50: 1μM), halts non-small cell lung cancer growth via MAPK pathway.</p>Fórmula:C26H19F3N2O2SCor e Forma:SolidPeso molecular:480.5Anti-Trypanosoma cruzi agent-2
<p>Compd 3b: anti-trypanosomal, IC50 0.51 μM (NINOA), 3.06 μM (INC-5), also combats T. gondii.</p>Fórmula:C17H10ClNO5Cor e Forma:SolidPeso molecular:343.72MEIS-IN-1
CAS:<p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>Fórmula:C24H21F3N2O4Cor e Forma:SolidPeso molecular:458.43EBI-907
CAS:<p>EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.</p>Fórmula:C23H21ClF2N4O3SCor e Forma:SolidPeso molecular:506.95Gepotidacin hydrochloride
CAS:<p>Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.</p>Fórmula:C24H29ClN6O3Cor e Forma:SolidPeso molecular:484.989(S),10(S),13(S)-TriHOME
CAS:<p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>Fórmula:C18H34O5Cor e Forma:SolidPeso molecular:330.46PPARγ agonist 1
<p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>Fórmula:C34H39NO3Cor e Forma:SolidPeso molecular:509.68BDZ-h
CAS:<p>BDZ-h inhibits both closed/open states of all 4 homomeric & 2 GluA2R-complex AMPA receptors.</p>Fórmula:C21H21N5O3SCor e Forma:SolidPeso molecular:423.49PF-06815345 hydrochloride
CAS:<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Fórmula:C27H30Cl2FN9O4Cor e Forma:SolidPeso molecular:634.49Napyradiomycin C2
CAS:<p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>Fórmula:C25H27Cl3O5Cor e Forma:SolidPeso molecular:513.838ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Fórmula:C23H26Cl2N2O3Cor e Forma:SolidPeso molecular:449.37MK-1220
CAS:<p>MK-1220 is a novel Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure.</p>Fórmula:C40H53N5O9SCor e Forma:SolidPeso molecular:779.94Steroid sulfatase/17β-HSD1-IN-3
<p>Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).</p>Fórmula:C19H17ClN2O5SCor e Forma:SolidPeso molecular:420.87LAF-153
CAS:<p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>Fórmula:C18H32N2O7Cor e Forma:SolidPeso molecular:388.46STA 2
CAS:<p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>Fórmula:C21H34O3SCor e Forma:SolidPeso molecular:366.56Haliangicin B
CAS:<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Fórmula:C22H32O5Cor e Forma:SolidPeso molecular:376.49AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Fórmula:C32H38N6O3Cor e Forma:SolidPeso molecular:554.7STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Fórmula:C17H12N4O4Cor e Forma:SolidPeso molecular:336.3LLS30
CAS:<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Fórmula:C34H33Cl4N5O3Cor e Forma:SolidPeso molecular:701.47PF-06305591 dihydrate
<p>PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADME</p>Fórmula:C15H26N4O3Cor e Forma:SolidPeso molecular:310.39AZD-3199 dihydrobromide
CAS:<p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>Fórmula:C32H44Br2N4O4SCor e Forma:SolidPeso molecular:740.59NS2B/NS3-IN-5
<p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>Fórmula:C14H9IN2O3SCor e Forma:SolidPeso molecular:412.2PX-316
CAS:<p>PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.</p>Fórmula:C28H57O10PCor e Forma:SolidPeso molecular:584.72GSK2945 hydrochloride
<p>GSK2945 HCl is a specific Rev-erbα antagonist, EC50: 21.5 μM (mouse), 20.8 μM (human), increases cholesterol 7α-hydroxylase.</p>Fórmula:C20H19Cl3N2O2SCor e Forma:SolidPeso molecular:457.8SHR0687
CAS:<p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>Fórmula:C39H60N8O5Cor e Forma:SolidPeso molecular:720.94SK&F 108361
CAS:<p>SK&F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.</p>Fórmula:C24H48N6O6Cor e Forma:SolidPeso molecular:516.67Cilazapril HCl
CAS:<p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>Fórmula:C22H32ClN3O5Cor e Forma:SolidPeso molecular:453.96PDE4-IN-14
CAS:<p>PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, including</p>Fórmula:C19H20F2N4O3SCor e Forma:SolidPeso molecular:422.45Chitinase-IN-4
<p>Chitinase-IN-4 (compound 8f) is a potent and selective inhibitor of OfChi-h with an IC50 value of 0.1 μM and good insecticidal activity.</p>Fórmula:C21H24ClN7Cor e Forma:SolidPeso molecular:409.92P-gp modulator 1
CAS:<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Fórmula:C41H72N2O6Pureza:98%Cor e Forma:SolidPeso molecular:689.02UH 301
CAS:<p>UH 301 is a 5-HT1A receptor antagonist.</p>Fórmula:C16H24FNOCor e Forma:SolidPeso molecular:265.375(S),6(R)-DiHETE
CAS:<p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.47Kalafungin
CAS:<p>Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.</p>Fórmula:C16H12O6Cor e Forma:SolidPeso molecular:300.26CCW 28-3
CAS:<p>CCW 28-3 is a novel potent covalent BRD4 degrader, degrading BRD4 in a proteasome- and RNF4-dependent manner without inhibiting RNF4 autoubiquitination activity</p>Fórmula:C44H42Cl2N6O4SCor e Forma:SolidPeso molecular:821.81L-744832
CAS:<p>L-744832, also known as L-744,832, is a potent Farnesyltransferase inhibitor with potential anticancer activity.</p>Fórmula:C26H45N3O6S2Cor e Forma:SolidPeso molecular:559.78Resolvin E4
CAS:<p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.45Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Fórmula:C24H26O8Cor e Forma:SolidPeso molecular:442.4616(S)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds to human IP & EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>Fórmula:C22H32O4Cor e Forma:SolidPeso molecular:360.49BM635 mesylate (1493762-74-5 free base)
<p>BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).</p>Fórmula:C26H33FN2O4SPureza:98%Cor e Forma:SolidPeso molecular:488.61XR8-69
<p>XR8-69 is a SARS-CoV-2 PLpro inhibitor. XR8-69 has a low micromolar antiviral effect in SARS-CoV-2 infected human cells.</p>Fórmula:C26H30N4O2SCor e Forma:SolidPeso molecular:462.61SORT1-IN-1
CAS:<p>SORT1-IN-1 (compound 2) is a SORT1 inhibitor.</p>Fórmula:C17H13F3N2O4Cor e Forma:SolidPeso molecular:366.29(6S)-CP-470711
CAS:<p>(6S)-CP-470711 (Compound 8) acts as an inhibitor of sorbitol dehydrogenase (SDH) in both humans and rats, exhibiting inhibitory concentrations (IC50) of 19 nM and 27 nM, respectively. Additionally, (6S)-CP-470711 has been shown to ameliorate diabetes in rats induced by Streptozotocin.</p>Fórmula:C18H26N6O2Cor e Forma:SolidPeso molecular:358.44hDDAH-1-IN-2 sulfate
<p>hDDAH-1-IN-2: selective oral hDDAH-1 inhibitor with low cell toxicity.</p>Fórmula:C8H24N4O10S2Cor e Forma:SolidPeso molecular:400.43Idraparinux Na
CAS:<p>Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa Inhibitor</p>Fórmula:C38H55Na9O49S7Cor e Forma:SolidPeso molecular:1727.14Belatacept
CAS:<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Cor e Forma:LiquidPZ-3022
CAS:<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Fórmula:C20H21N5OCor e Forma:SolidPeso molecular:347.41CXN37378
CAS:<p>CXN37378, aka NAP, is a potent MOR-selective antagonist with no official name yet, termed per MedKoo Nomenclature.</p>Fórmula:C27H31N3O4Cor e Forma:SolidPeso molecular:461.55L-Tyrosyl-L-glutamic acid
CAS:<p>L-Tyrosyl-L-glutamic acid acts as an inhibitor of the amino acid permease GAP1.</p>Fórmula:C14H18N2O6Cor e Forma:SolidPeso molecular:310.3VEGFR-2-IN-16
<p>VEGFR-2-IN-16 (Compound 15b) is a potent inhibitor of VEGFR-2 (IC50: 86.36 nM) that exhibits antitumour effects.</p>Fórmula:C21H13Cl2N3O2Cor e Forma:SolidPeso molecular:410.25MDL-27788
CAS:<p>MDL-27788 is a tricyclic inhibitor.</p>Fórmula:C24H26N2O5SCor e Forma:SolidPeso molecular:454.5420-HEDE
CAS:<p>20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.</p>Fórmula:C20H36O3Pureza:98%Cor e Forma:SolidPeso molecular:324.50AZ14145845
<p>AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.</p>Fórmula:C32H35N9OCor e Forma:SolidPeso molecular:561.68Furaquinocin A
CAS:<p>Furaquinocin A has the ability to kill HeLa S3 and B16 melanoma cells, yet it lacks antibacterial activity.</p>Fórmula:C22H26O7Cor e Forma:SolidPeso molecular:402.438CI-1029
CAS:<p>CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.</p>Fórmula:C28H37NO4SCor e Forma:SolidPeso molecular:483.66AVE 0991
CAS:<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Fórmula:C29H32N4O5S2Pureza:98.69%Cor e Forma:SolidPeso molecular:580.72PPARα agonist 1
<p>PPARα agonist 1 is a complete and potent PPARα agonist.</p>Fórmula:C27H34O4Cor e Forma:SolidPeso molecular:422.56AB 5046A
CAS:<p>AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.</p>Fórmula:C10H14O4Cor e Forma:SolidPeso molecular:198.22PDE4-IN-6
<p>PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.</p>Fórmula:C25H20FNO5SCor e Forma:SolidPeso molecular:465.49Canosimibe
CAS:<p>Canosimibe is a cholesterol absorption inhibitor</p>Fórmula:C44H60FN3O10Cor e Forma:SolidPeso molecular:809.96Unoprostone
CAS:<p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>Fórmula:C22H38O5Pureza:98%Cor e Forma:SolidPeso molecular:382.53Rosiptor acetate
CAS:<p>Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.</p>Fórmula:C22H39NO4Pureza:98%Cor e Forma:Solid PowderPeso molecular:381.55Atiratecan
CAS:<p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>Fórmula:C31H34N6O6Pureza:98%Cor e Forma:SolidPeso molecular:586.64Thielavin B
CAS:<p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>Fórmula:C31H34O10Cor e Forma:SolidPeso molecular:566.6Chitinovorin C
CAS:<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Fórmula:C15H20N4O8SCor e Forma:SolidPeso molecular:416.406FTI 276 TFA
CAS:<p>FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).</p>Fórmula:C23H28F3N3O5S2Cor e Forma:SolidPeso molecular:547.61Anti-Trypanosoma cruzi agent-1
<p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>Fórmula:C23H29N3O5Cor e Forma:SolidPeso molecular:427.49BRD-K25923209
CAS:<p>BRD-K25923209 is a novel inhibitor of BAF transcriptional repression.</p>Fórmula:C29H36N4O3Cor e Forma:SolidPeso molecular:488.62TSWV-IN-1
<p>TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.</p>Fórmula:C26H31FO4S2Cor e Forma:SolidPeso molecular:490.65GW311616
CAS:<p>GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>Fórmula:C19H31N3O4SCor e Forma:SolidPeso molecular:397.53Epelmycin D
CAS:<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Fórmula:C30H35NO11Cor e Forma:SolidPeso molecular:585.599NA 0346
CAS:<p>NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.</p>Fórmula:C26H22N4O3Cor e Forma:SolidPeso molecular:438.48Schidigera-genin B
CAS:<p>Schidigera-genin B is a steroidal saponin that can be isolated from Yucca glauca. It exhibits mild antifungal activity.</p>Fórmula:C27H40O4Cor e Forma:SolidPeso molecular:428.604P-gp modulator 2
<p>P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.</p>Fórmula:C22H20BrN3O4Cor e Forma:SolidPeso molecular:470.32RXR antagonist 1
<p>RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.</p>Fórmula:C28H33F3N2O3Cor e Forma:SolidPeso molecular:502.57mPGES-1-IN-1
<p>MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.</p>Fórmula:C21H14N4O2SCor e Forma:SolidPeso molecular:386.43TIY-7
<p>TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.</p>Cor e Forma:SolidTuvatidine
CAS:<p>Tuvatidine is a histamine 2 receptor antagonist.</p>Fórmula:C10H17N9O2S3Cor e Forma:SolidPeso molecular:391.5Streptonigrin (racemate)
CAS:<p>Streptonigrin: aminoquinone antibiotic; antitumor, antibacterial; blocks β-Catenin/Tcf, cytotoxic; alters hamster chromosomes; (-)-isomer, CAS#3930-19-6.</p>Fórmula:C25H22N4O8Cor e Forma:SolidPeso molecular:506.4616(R)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Fórmula:C22H32O4Cor e Forma:SolidPeso molecular:360.49LMD-A
CAS:<p>LMD-A, also known as CCR8 antagonist LMD-A, is a CCR8 antagonist.</p>Fórmula:C27H32N4O4SCor e Forma:SolidPeso molecular:508.63FTO-IN-1 TFA
<p>FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.</p>Fórmula:C20H17Cl2F3N4O4Cor e Forma:SolidPeso molecular:505.27PTP1B-IN-21
<p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>Fórmula:C22H22O11Cor e Forma:SolidPeso molecular:462.4CPX-351
CAS:<p>CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.</p>Fórmula:C36H42N4O15Pureza:98.95% - 99.763%Cor e Forma:SolidPeso molecular:770.74Olanzapine/Samidorphan
CAS:<p>Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.</p>Fórmula:C38H46N6O4SCor e Forma:SolidPeso molecular:682.88SSM3 TFA
CAS:<p>SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..</p>Fórmula:C22H32N12O2Cor e Forma:SolidPeso molecular:496.57LA-810
CAS:<p>LA-810 is a nitrous oxide donor.</p>Fórmula:C15H25N5O7SCor e Forma:SolidPeso molecular:419.45(S)-Butaprost free acid
CAS:<p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>Fórmula:C23H38O5Cor e Forma:SolidPeso molecular:394.54NS2B/NS3-IN-4
CAS:<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Fórmula:C15H11NO4Cor e Forma:SolidPeso molecular:269.25CU-2010
CAS:<p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>Fórmula:C37H42N6O6SCor e Forma:SolidPeso molecular:698.83Glycotriosyl glutamine
CAS:<p>Glycotriosyl glutamine is a nephritogenoside analog.</p>Fórmula:C23H40N2O18Cor e Forma:SolidPeso molecular:632.57LPA5 antagonist 2
<p>LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.</p>Fórmula:C26H25FN2O4SCor e Forma:SolidPeso molecular:480.55Griseolutein A
CAS:<p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C17H14N2O6Cor e Forma:SolidPeso molecular:342.303MetRS-IN-1
CAS:<p>MetRS-IN-1 (Compound 27) is an inhibitor of E. coli methionyl-tRNA synthetase (MetRS) with an IC50 value of 237 nM [1].</p>Fórmula:C15H13N3O4SCor e Forma:SolidPeso molecular:331.35Utrophin modulator 1
<p>UM1 upregulates utrophin, has EC50 of 0.11 μM, useful in DMD research.</p>Fórmula:C22H18N6OCor e Forma:SolidPeso molecular:382.42Harziphilone
CAS:<p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>Fórmula:C15H18O4Cor e Forma:SolidPeso molecular:262.301Bcl-2-IN-8
<p>Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.</p>Fórmula:C36H44O6Cor e Forma:SolidPeso molecular:572.73Everafenib
<p>Everafenib: potent BRAF inhibitor, crosses blood-brain barrier, hinders MAPK, effective on V600EBRAF cells, outperforms other drugs in trials.</p>Fórmula:C20H23ClFN5O2S2Cor e Forma:SolidPeso molecular:484.01EICAR
CAS:<p>EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.</p>Fórmula:C11H13N3O5Cor e Forma:SolidPeso molecular:267.24A1-Phytoprostane-I
CAS:<p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.</p>Fórmula:C18H28O4Cor e Forma:SolidPeso molecular:308.41Latrunculin M
CAS:<p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>Fórmula:C21H33NO5SCor e Forma:SolidPeso molecular:411.55ZINC000104379474
<p>ZINC000104379474 is a compound that targets SARS-CoV-2 endoribonuclease.</p>Fórmula:C27H33N3O10Cor e Forma:SolidPeso molecular:559.57Mycinamicin Ⅵ
CAS:<p>Mycinamicin VI is a macrolide antibiotic with antibacterial activity against Gram-positive bacteria.</p>Fórmula:C35H57NO11Cor e Forma:SolidPeso molecular:667.83G12Si-1
<p>G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.</p>Fórmula:C29H32ClN5O3Cor e Forma:SolidPeso molecular:534.05RMG8-8
<p>RMG8-8 shows the excellent efficacy against C. neoformans (1.56 μg/mL).</p>Fórmula:C41H78N8O5Cor e Forma:SolidPeso molecular:763.11Cilobamine (free base)
CAS:<p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>Fórmula:C17H23Cl2NOCor e Forma:SolidPeso molecular:328.28MRS4738
<p>MRS4738 is a potent antagonist with high affinity for the P2Y14R receptor. It demonstrates in vivo anti-hyperallodynic and antiasthmatic activity [1].</p>Fórmula:C30H24F3NO2Cor e Forma:SolidPeso molecular:487.5111-Demethyltomaymycin
CAS:<p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>Fórmula:C15H18N2O4Cor e Forma:SolidPeso molecular:290.314Glucoallosamidin A
CAS:<p>Glucoallosamidin A is a glycoside antibiotic that inhibits chitinase activity. It effectively suppresses the chitinase enzyme in Candida albicans [ATCC 10231], exhibiting an IC50 of 3.4 μg/mL.</p>Fórmula:C26H44N4O14Cor e Forma:SolidPeso molecular:636.646GRPR antagonist-1
<p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>Fórmula:C29H33F3N4O4Cor e Forma:SolidPeso molecular:558.59SCP1-IN-2
<p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>Fórmula:C19H17F3N2O6S2Cor e Forma:SolidPeso molecular:490.47TY 11223
CAS:<p>TY 11223: stable homoisocarbacyclin analog, potently inhibits platelet aggregation with lasting effect and selective activity.</p>Fórmula:C24H34O5Cor e Forma:SolidPeso molecular:402.52VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Fórmula:C21H14ClN3O2Cor e Forma:SolidPeso molecular:375.81VEGFR-2-IN-5 hydrochloride
<p>VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.</p>Fórmula:C19H25ClN8Cor e Forma:SolidPeso molecular:400.91U 80215
CAS:<p>U 80215 is an enzyme-competitive inhibitor.</p>Fórmula:C42H60N8O6SCor e Forma:SolidPeso molecular:805.04Antitumor agent-65
CAS:<p>Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.</p>Fórmula:C18H17NO10Cor e Forma:SolidPeso molecular:407.33Glucosylceramide synthase-IN-3
<p>Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.</p>Fórmula:C21H20FN3O3Cor e Forma:SolidPeso molecular:381.4Aristoforin
CAS:<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Fórmula:C37H54O6Cor e Forma:SolidPeso molecular:594.82Gallinamide A
CAS:Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.Fórmula:C31H52N4O7Cor e Forma:SolidPeso molecular:592.778(S),15(S)-DiHETE
CAS:<p>8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.47IT-066 HCl
CAS:<p>IT-066 HCl is a histamine H2 receptor antagonist.</p>Fórmula:C19H25ClN4O3Cor e Forma:SolidPeso molecular:392.88PCTR1
CAS:<p>PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.</p>Fórmula:C32H47N3O9SCor e Forma:SolidPeso molecular:649.8Pluracidomycin C2
CAS:<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C11H15NO9S2Cor e Forma:SolidPeso molecular:369.37Mepixetil
<p>Mepixetil is a potent angiotensin II receptor antagonist[1].</p>Fórmula:C12H18N2O3Cor e Forma:SolidPeso molecular:238.288-iso Prostaglandin F3α
CAS:<p>8-iso PGF3α is an isoprostane produced from the free-radical peroxidation of EPA.</p>Fórmula:C20H32O5Cor e Forma:SolidPeso molecular:352.47Lipohexin
CAS:<p>Lipohexin is a peptide antibiotic that exhibits activity against Gram-positive bacteria. It competitively inhibits human placental proline endopeptidase (proline endopeptidase) with an IC50 of 3.5 μM. Additionally, Lipohexin inhibits proline endopeptidase from Flavobacterium meningosepticum, with an IC50 of 25 μM.</p>Fórmula:C39H68N6O9Cor e Forma:SolidPeso molecular:764.992Pefcalcitol
CAS:<p>Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.</p>Fórmula:C26H34F5NO4Cor e Forma:SolidPeso molecular:519.54Coriolin B
CAS:<p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>Fórmula:C23H36O6Cor e Forma:SolidPeso molecular:408.528Unoprostone isopropyl
CAS:<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Fórmula:C25H44O5Pureza:98%Cor e Forma:SolidPeso molecular:424.61di-Val-L-dC
CAS:<p>Di-Val-L-dC, a reverse transcriptase inhibitor, is used potentially for treatment of HBV infection.</p>Fórmula:C19H31N5O6Pureza:98%Cor e Forma:SolidPeso molecular:425.48Salfredin C1
CAS:<p>Salfredin C1 is an inhibitor of aldose reductase.</p>Fórmula:C13H11NO6Cor e Forma:SolidPeso molecular:277.229Orvepitant
CAS:<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Fórmula:C31H35F7N4O2Cor e Forma:SolidPeso molecular:628.62Treloxinate
CAS:<p>Treloxinate is an effective lipid-lowering agent. It specifically influences the triglyceride levels in Sprague-Dawley rats, while impacting both triglyceride and cholesterol levels in Wistar rats.</p>Fórmula:C16H12Cl2O4Cor e Forma:SolidPeso molecular:339.17Diatretyne Ⅰ
CAS:Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.Fórmula:C8H5NO3Cor e Forma:SolidPeso molecular:163.13Azirinomycin
CAS:<p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C4H5NO2Cor e Forma:SolidPeso molecular:99.088Eurocidin E
CAS:<p>Eurocidin E is an antibiotic that inhibits degranulation and histamine release from rat mast cells.</p>Fórmula:C40H61NO14Cor e Forma:SolidPeso molecular:779.911ONO-DI-004
CAS:<p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>Fórmula:C24H38O6Cor e Forma:SolidPeso molecular:422.55COTC
CAS:<p>COTC is an anticancer bacterial metabolite; inhibits glyoxalase with GSH, halts HeLa cell growth, and fights tumor in Ehrlich murine model.</p>Fórmula:C11H14O6Cor e Forma:SolidPeso molecular:242.23Vindeburnol
CAS:<p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>Fórmula:C17H20N2OCor e Forma:SolidPeso molecular:268.35Tetrahydrouridine dihydrate
<p>THU dihydrate, a potent CDA inhibitor, outperforms cytidine by blocking the enzyme's active site.</p>Fórmula:C9H20N2O8Cor e Forma:SolidPeso molecular:284.26O4
CAS:<p>O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.</p>Fórmula:C24H15NO7Pureza:98%Cor e Forma:SolidPeso molecular:429.38Dehatrine
CAS:<p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>Fórmula:C37H38N2O6Cor e Forma:SolidPeso molecular:606.71Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Fórmula:C27H29NO10Cor e Forma:SolidPeso molecular:527.52FTO-IN-6
CAS:<p>FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).</p>Fórmula:C14H12N4O6Cor e Forma:SolidPeso molecular:332.27STING agonist-20
CAS:<p>STING agonist-20: potent, aids in XMT-2056 synthesis, used as a cancer vaccine adjuvant.</p>Fórmula:C36H39N11O8Cor e Forma:SolidPeso molecular:753.76TRPC4/5-IN-1
<p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>Fórmula:C21H21N3OCor e Forma:SolidPeso molecular:331.41Calphostin I
CAS:<p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>Fórmula:C44H38O15Cor e Forma:SolidPeso molecular:806.76Lunacalcipol
CAS:<p>Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.</p>Fórmula:C28H42O4SCor e Forma:SolidPeso molecular:474.7Hetrombopag olamine
CAS:<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Fórmula:C29H36N6O7Pureza:98%Cor e Forma:SolidPeso molecular:580.63SARS-CoV-2-IN-24
<p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>Fórmula:C27H30N4O5Cor e Forma:SolidPeso molecular:490.55SphK2-IN-1
CAS:<p>SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.</p>Fórmula:C23H22ClF3N8OCor e Forma:SolidPeso molecular:518.92
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