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Outros inibidores

Outros inibidores

Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.

Foram encontrados 37902 produtos de "Outros inibidores"

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  • Diaporthin

    CAS:
    <p>Diaporthin is a phytotoxin that can be isolated from Cryphonectria parasitica. It exhibits antibacterial activity.</p>
    Fórmula:C13H14O5
    Cor e Forma:Solid
    Peso molecular:250.247
  • 1-Deamino-1-hydroxygentamicin C1a

    CAS:
    <p>1-Deamino-1-hydroxygentamicin C1a (AntibioticSU-2) is an aminoglycoside antibiotic effective against both gram-positive and gram-negative bacteria.</p>
    Fórmula:C19H38N4O8
    Cor e Forma:Solid
    Peso molecular:450.527
  • GNE-616

    CAS:
    <p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>
    Fórmula:C24H23F4N5O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:537.53
  • Prohibitin ligand 1


    <p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>
    Fórmula:C20H22N2O
    Cor e Forma:Solid
    Peso molecular:306.4
  • Epoxyquinomicin C

    CAS:
    <p>Epoxyquinomicin C is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis and is also utilized in the synthesis of the NF-κB inhibitor DHMEQ.</p>
    Fórmula:C14H13NO6
    Cor e Forma:Solid
    Peso molecular:291.256
  • PRN694

    CAS:
    <p>PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.</p>
    Fórmula:C28H35F2N5O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:543.67
  • 6"'-Deamino-6"'-hydroxyneomycin B

    CAS:
    <p>6"'-Deamino-6"'-hydroxyneomycin B is an aminoglycoside antibiotic produced by [Streptomyces fradiaeUC 75]. It is effective against both Gram-positive and Gram-negative bacteria and serves as an intermediate in the biosynthesis of neomycin.</p>
    Fórmula:C23H45N5O14
    Cor e Forma:Solid
    Peso molecular:615.628
  • AMPK Activator SC4

    CAS:
    <p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>
    Fórmula:C26H18ClN3O4
    Cor e Forma:Solid
    Peso molecular:471.89
  • Fostriecin (free base)

    CAS:
    <p>Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.</p>
    Fórmula:C19H27O9P
    Cor e Forma:Solid
    Peso molecular:430.39
  • Ganciclovir monophosphonate

    CAS:
    <p>Ganciclovir monophosphate treats CMV, inhibiting replication in human/animal strains (IC50: 0.01μM).</p>
    Fórmula:C10H16N5O6P
    Cor e Forma:Solid
    Peso molecular:333.24
  • FMK-MEA

    CAS:
    <p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>
    Fórmula:C21H26FN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.46
  • Leptofuranin C

    CAS:
    <p>Leptofuranin C, found in the Str. tanashiensis strain, is known to arrest normal cell progression and induce cell death.</p>
    Fórmula:C32H46O5
    Cor e Forma:Solid
    Peso molecular:510.705
  • Arterolane

    CAS:
    <p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>
    Fórmula:C22H36N2O4
    Cor e Forma:Solid
    Peso molecular:392.53
  • Pillaromycin A

    CAS:
    <p>Pillaromycin A exhibits activity against mycobacteria, Gram-positive bacteria, and Gram-negative bacteria, although it is less effective against Gram-negative bacteria. Additionally, it possesses antitumor properties.</p>
    Fórmula:C28H30O11
    Cor e Forma:Solid
    Peso molecular:542.531
  • Fomecin A

    CAS:
    <p>Fomecin A exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, and weak activity against fungi. It also possesses antiviral activity against the influenza virus PR-8.</p>
    Fórmula:C8H8O5
    Cor e Forma:Solid
    Peso molecular:184.146
  • Cytochalasin L

    CAS:
    <p>Cytochalasin L possesses reversible biological activities, including the inhibition of cytoplasmic division, as well as the suppression of both endocytosis and exocytosis in phagocytic macrophages.</p>
    Fórmula:C32H37NO7
    Cor e Forma:Solid
    Peso molecular:547.639
  • Namitecan

    CAS:
    <p>Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.</p>
    Fórmula:C23H22N4O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.44
  • Gentamicin A

    CAS:
    <p>Gentamicin A is an antibiotic exhibiting effective antibacterial activity against both Gram-positive and Gram-negative bacteria, and it also demonstrates activity against most methicillin-sensitive staphylococci.</p>
    Fórmula:C18H36N4O10
    Cor e Forma:Solid
    Peso molecular:468.499
  • METTL3-IN-3

    CAS:
    METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor .
    Fórmula:C26H28BrFN6O2
    Cor e Forma:Solid
    Peso molecular:555.44
  • PAD2-IN-1 hydrochloride


    <p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>
    Fórmula:C25H30ClFN6O3
    Cor e Forma:Solid
    Peso molecular:517
  • HOE-288

    CAS:
    <p>HOE-288 is a converting enzyme (CE) inhibitor.</p>
    Fórmula:C27H38N2O5
    Cor e Forma:Solid
    Peso molecular:470.60
  • NRX-2663

    CAS:
    <p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>
    Fórmula:C20H13F3N2O5
    Cor e Forma:Solid
    Peso molecular:418.32
  • KF 20274

    CAS:
    <p>KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.</p>
    Fórmula:C21H29N5O
    Cor e Forma:Solid
    Peso molecular:367.49
  • PARP10/15-IN-1


    <p>PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].</p>
    Fórmula:C13H10N2O3S
    Cor e Forma:Solid
    Peso molecular:274.3
  • CGC 11144

    CAS:
    <p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>
    Fórmula:C40H100Cl10N10
    Cor e Forma:Solid
    Peso molecular:1075.82
  • RXR antagonist 1


    <p>RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.</p>
    Fórmula:C28H33F3N2O3
    Cor e Forma:Solid
    Peso molecular:502.57
  • TIY-7


    <p>TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.</p>
    Cor e Forma:Solid
  • Antioxidant agent-3


    <p>Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.</p>
    Fórmula:C18H14O8
    Cor e Forma:Solid
    Peso molecular:358.3
  • 16(R)-Iloprost

    CAS:
    <p>Iloprost, a potent prostacyclin analog, binds IP &amp; EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>
    Fórmula:C22H32O4
    Cor e Forma:Solid
    Peso molecular:360.49
  • β-N-Acetyl-D-hexosaminidase-IN-1


    <p>β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.</p>
    Fórmula:C18H13F2NO2S
    Cor e Forma:Solid
    Peso molecular:345.36
  • Afeletecan HCl

    CAS:
    <p>Afeletecan (BAY 56-3722) is a water-soluble, anti-cancer camptothecin conjugated to a carbohydrate, inhibiting DNA replication and inducing apoptosis.</p>
    Fórmula:C45H50ClN7O11S
    Cor e Forma:Solid
    Peso molecular:932.44
  • Canosimibe

    CAS:
    <p>Canosimibe is a cholesterol absorption inhibitor</p>
    Fórmula:C44H60FN3O10
    Cor e Forma:Solid
    Peso molecular:809.96
  • 10-Decarbomethoxyaclacinomycin A

    CAS:
    <p>10-Decarbomethoxyaclacinomycin A is an anthracycline antibiotic produced by the mutant strain Streptomyces galilaeus MA144-Mlt KE303. This compound exhibits antibacterial activity.</p>
    Fórmula:C40H51NO13
    Cor e Forma:Solid
    Peso molecular:753.832
  • MEIS-IN-2


    <p>MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.</p>
    Fórmula:C23H21ClN2O4
    Cor e Forma:Solid
    Peso molecular:424.88
  • PLP_Snyder530


    <p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>
    Fórmula:C24H24N2O2
    Cor e Forma:Solid
    Peso molecular:372.46
  • TRPC5-IN-4

    CAS:
    <p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>
    Fórmula:C18H11ClF4N4O3
    Cor e Forma:Solid
    Peso molecular:442.75
  • VEGFR-2-IN-25

    CAS:
    <p>VEGFR-2-IN-25 (compound 5d) is a potent inhibitor of VEGFR-2 (IC50: 12.1 nM).</p>
    Fórmula:C24H22N6O2
    Cor e Forma:Solid
    Peso molecular:426.47
  • MMG-11 quarterhydrate


    <p>MMG-11 quarterhydrate, a potent hTLR2 antagonist, inhibits TLR2/1 and TLR2/6 with IC50s of 1.7μM and 5.7μM; low toxicity.</p>
    Fórmula:C15H16O8
    Cor e Forma:Solid
    Peso molecular:310.78
  • Phyllosinol

    CAS:
    <p>Phyllosinol is an antifungal antibiotic.</p>
    Fórmula:C7H8O4
    Cor e Forma:Solid
    Peso molecular:156.136
  • Kri 1314

    CAS:
    Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.
    Fórmula:C38H51N5O7
    Cor e Forma:Solid
    Peso molecular:689.84
  • Polvitolimod

    CAS:
    <p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>
    Fórmula:C13H14FN5O4
    Cor e Forma:Solid
    Peso molecular:323.28
  • Combretastatin A1 phosphate

    CAS:
    <p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>
    Fórmula:C18H22O12P2
    Cor e Forma:Solid
    Peso molecular:492.31
  • Methyl 5-thia-6,8,11,14-eicosatetraenoate

    CAS:
    <p>Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.</p>
    Fórmula:C20H32O2S
    Cor e Forma:Solid
    Peso molecular:336.53
  • EICAR

    CAS:
    <p>EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.</p>
    Fórmula:C11H13N3O5
    Cor e Forma:Solid
    Peso molecular:267.24
  • A1-Phytoprostane-I

    CAS:
    <p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression &amp; increases phytoalexin synthesis.</p>
    Fórmula:C18H28O4
    Cor e Forma:Solid
    Peso molecular:308.41
  • Latrunculin M

    CAS:
    <p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>
    Fórmula:C21H33NO5S
    Cor e Forma:Solid
    Peso molecular:411.55
  • Hydroxymycotrienin A

    CAS:
    <p>Hydroxymycotrienin A is an ansamycin antibiotic with the ability to inhibit human neck tumor cell lines. Its inhibitory effect is more pronounced on HPV-positive neck tumor cells (such as HeLa, CaSKi, and SiHa) compared to HPV-negative cells.</p>
    Fórmula:C36H48N2O9
    Cor e Forma:Solid
    Peso molecular:652.774
  • Juvenimicin A2

    CAS:
    <p>Juvenimicin A2 is effective against Gram-positive bacteria and certain Gram-negative bacteria.</p>
    Fórmula:C30H51NO8
    Cor e Forma:Solid
    Peso molecular:553.728
  • ZINC000104379474


    <p>ZINC000104379474 is a compound that targets SARS-CoV-2 endoribonuclease.</p>
    Fórmula:C27H33N3O10
    Cor e Forma:Solid
    Peso molecular:559.57
  • VRT-18858

    CAS:
    <p>VRT-18858 is a metabolite of VX-740.</p>
    Fórmula:C24H25N5O7
    Cor e Forma:Solid
    Peso molecular:495.48
  • 9(S)-HEPE

    CAS:
    <p>9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.</p>
    Fórmula:C20H30O3
    Cor e Forma:Solid
    Peso molecular:318.45
  • FWM-1


    <p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>
    Fórmula:C15H11ClN4O4S2
    Cor e Forma:Solid
    Peso molecular:410.86
  • M-COPA

    CAS:
    <p>M-COPA disrupts Golgi, blocks MET &amp; Arf1 activation, and inhibits angiogenesis via VEGFR &amp; NF-kB pathways.</p>
    Fórmula:C25H34N2O2
    Cor e Forma:Solid
    Peso molecular:394.55
  • Pyrromycin

    CAS:
    <p>Pyrromycin is a monosaccharide anthracycline which can be used to inhibit cellular RNA synthesis.</p>
    Fórmula:C30H35NO11
    Cor e Forma:Solid
    Peso molecular:585.60
  • BXL0124

    CAS:
    <p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>
    Fórmula:C32H44F6O4
    Cor e Forma:Solid
    Peso molecular:606.68
  • PTP1B-IN-16


    <p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>
    Fórmula:C26H18ClN3O4S
    Cor e Forma:Solid
    Peso molecular:503.96
  • Cilobamine (free base)

    CAS:
    <p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>
    Fórmula:C17H23Cl2NO
    Cor e Forma:Solid
    Peso molecular:328.28
  • 11-Deoxy-13-dihydrodaunorubicin

    CAS:
    <p>11-Deoxy-13-dihydrodaunorubicin is an anthracycline antibiotic with activity against Gram-positive bacteria, Gram-negative bacteria, and tumors.</p>
    Fórmula:C27H31NO9
    Cor e Forma:Solid
    Peso molecular:513.536
  • CEP-7055

    CAS:
    <p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>
    Fórmula:C32H35N3O4
    Cor e Forma:Solid
    Peso molecular:525.64
  • Npc 12626

    CAS:
    <p>Npc 12626 is a N-methyl-D-aspartate receptor antagonist; NPC 17742, the (2R,4R,5S)-isomer, is the most potent isomer in the mixture NPC 12626.</p>
    Fórmula:C11H22NO5P
    Cor e Forma:Solid
    Peso molecular:279.27
  • Calphostin B

    CAS:
    <p>Calphostins, PKC inhibitors from Cladosporium fungus, include A, B, C, D, I; C is most potent.</p>
    Fórmula:C37H34O11
    Cor e Forma:Solid
    Peso molecular:654.66
  • GSK-1264

    CAS:
    <p>GSK-1264: allosteric HIV integrase inhibitor, halts viral replication &amp; abnormal protein multimerization.</p>
    Fórmula:C26H28FNO5
    Cor e Forma:Solid
    Peso molecular:453.5
  • Melithiazole C

    CAS:
    <p>Melithiazol C is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA) with antifungal properties.</p>
    Fórmula:C16H21NO5S
    Cor e Forma:Solid
    Peso molecular:339.407
  • Emimycin

    CAS:
    <p>Emimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as fungi like Saccharomyces cerevisiae (brewer's yeast).</p>
    Fórmula:C4H4N2O2
    Cor e Forma:Solid
    Peso molecular:112.087
  • Sdz 210-096

    CAS:
    <p>Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.</p>
    Fórmula:C27H31NO2
    Cor e Forma:Solid
    Peso molecular:401.54
  • PD-1/PD-L1-IN-30

    CAS:
    <p>PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.</p>
    Fórmula:C29H28F3NO5
    Cor e Forma:Solid
    Peso molecular:527.53
  • 5(S),6(S)-DiHETE

    CAS:
    <p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>
    Fórmula:C20H32O4
    Cor e Forma:Solid
    Peso molecular:336.47
  • Purine phosphoribosyltransferase-IN-2


    <p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>
    Fórmula:C11H15N5Na4O10P2
    Cor e Forma:Solid
    Peso molecular:531.17
  • TCMDC-125431


    <p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>
    Fórmula:C25H27N3O2S
    Cor e Forma:Solid
    Peso molecular:433.57
  • PPO-IN-1


    <p>PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).</p>
    Fórmula:C18H10F3N3O4S
    Cor e Forma:Solid
    Peso molecular:421.35
  • Sekdel sequence

    CAS:
    Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.
    Fórmula:C29H49N7O14
    Cor e Forma:Solid
    Peso molecular:719.74
  • BGC-638

    CAS:
    <p>BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.</p>
    Fórmula:C32H33N5O9
    Cor e Forma:Solid
    Peso molecular:631.63
  • MRS2179 tetrasodium hydrate


    <p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>
    Fórmula:C11H15N5Na4O10P2
    Cor e Forma:Solid
    Peso molecular:576.21
  • VU0463271 quarterhydrate


    <p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>
    Fórmula:C19H20N4O2S2
    Cor e Forma:Solid
    Peso molecular:387
  • Plasma kallikrein-IN-2


    <p>Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.</p>
    Fórmula:C28H24ClF3N8O3
    Cor e Forma:Solid
    Peso molecular:612.99
  • PTP1B-IN-3 diammonium


    <p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>
    Fórmula:C12H13BrF2N3O3P
    Cor e Forma:Solid
    Peso molecular:396.12
  • Eupenoxide

    CAS:
    <p>Eupenoxide is an antibiotic with antifungal properties, derived from fungi belonging to the Eupenicillium genus.</p>
    Fórmula:C14H22O4
    Cor e Forma:Solid
    Peso molecular:254.322
  • Seldomycin factor 3

    CAS:
    <p>Seldomycin factor 3 (XK 88-3) is an aminoglycoside antibiotic with broad-spectrum antibacterial activity.</p>
    Fórmula:C17H35N5O9
    Cor e Forma:Solid
    Peso molecular:453.488
  • VEGFR-2-IN-5 hydrochloride


    <p>VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.</p>
    Fórmula:C19H25ClN8
    Cor e Forma:Solid
    Peso molecular:400.91
  • Piperazinomycin

    CAS:
    <p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>
    Fórmula:C18H20N2O2
    Cor e Forma:Solid
    Peso molecular:296.36
  • PDE4B/7A-IN-1

    CAS:
    <p>5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.</p>
    Fórmula:C25H35N3O3
    Cor e Forma:Solid
    Peso molecular:425.56
  • 2-Hydroxymethylclavam

    CAS:
    <p>2-Hydroxymethylclavam is a β-lactam antibiotic with antifungal properties, particularly effective against plant pathogenic fungi.</p>
    Fórmula:C6H9NO3
    Cor e Forma:Solid
    Peso molecular:143.141
  • Clecarmycin C

    CAS:
    <p>Clecarmycin C is an antitumor antibiotic that demonstrates cytotoxic and antitumor properties. Additionally, Clecarmycin C exhibits antibacterial activity.</p>
    Fórmula:C29H26O11
    Cor e Forma:Solid
    Peso molecular:550.51
  • Citreamicin γ

    CAS:
    <p>Citreamicin γ demonstrates activity against aerobic and anaerobic Gram-positive bacteria.</p>
    Fórmula:C33H25NO12
    Cor e Forma:Solid
    Peso molecular:627.551
  • PARP7-IN-12

    CAS:
    <p>PARP7-IN-12, a potent inhibitor targeting PARP7, exhibits an IC50 of 7.836 nM. This compound is applicable in cancer research.</p>
    Fórmula:C23H27ClF3N5O5
    Cor e Forma:Solid
    Peso molecular:545.94
  • BMS-681

    CAS:
    <p>BMS-681 is a CCR2 antagonist blocking chemokine binding, aiding control of inflammatory and neurodegenerative diseases.</p>
    Fórmula:C26H36F3N5O
    Cor e Forma:Solid
    Peso molecular:491.59
  • Polyoxin E

    CAS:
    <p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>
    Fórmula:C17H23N5O13
    Cor e Forma:Solid
    Peso molecular:505.39
  • Antiviral agent 7


    <p>Antiviral agent 7 is a peptide-based coating that kills viruses.</p>
    Fórmula:C29H31F2N3O6
    Cor e Forma:Solid
    Peso molecular:555.57
  • 16(S)-Iloprost

    CAS:
    <p>Iloprost, a potent prostacyclin analog, binds to human IP &amp; EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>
    Fórmula:C22H32O4
    Cor e Forma:Solid
    Peso molecular:360.49
  • PTP1B-IN-21


    <p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>
    Fórmula:C22H22O11
    Cor e Forma:Solid
    Peso molecular:462.4
  • Fluperolone acetate

    CAS:
    <p>Fluperolone acetate is a Glucocorticoid/Adrenal Cortex Hormone.</p>
    Fórmula:C24H31FO6
    Cor e Forma:Solid
    Peso molecular:434.50
  • Coriolin B

    CAS:
    <p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Fórmula:C23H36O6
    Cor e Forma:Solid
    Peso molecular:408.528
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Fórmula:C20H24N2O2
    Cor e Forma:Solid
    Peso molecular:324.42
  • Anticancer agent 78


    <p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>
    Fórmula:C19H14BrNO4
    Cor e Forma:Solid
    Peso molecular:400.22
  • Lipohexin

    CAS:
    <p>Lipohexin is a peptide antibiotic that exhibits activity against Gram-positive bacteria. It competitively inhibits human placental proline endopeptidase (proline endopeptidase) with an IC50 of 3.5 μM. Additionally, Lipohexin inhibits proline endopeptidase from Flavobacterium meningosepticum, with an IC50 of 25 μM.</p>
    Fórmula:C39H68N6O9
    Cor e Forma:Solid
    Peso molecular:764.992
  • Naltrindole

    CAS:
    <p>Naltrindole is a delta opioid receptor antagonist.</p>
    Fórmula:C26H26N2O3
    Cor e Forma:Solid
    Peso molecular:414.5
  • NAZ2329

    CAS:
    <p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) &amp; hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>
    Fórmula:C21H18F3NO4S3
    Cor e Forma:Soild
    Peso molecular:501.56
  • CPX-351

    CAS:
    <p>CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.</p>
    Fórmula:C36H42N4O15
    Pureza:98.95% - 99.763%
    Cor e Forma:Solid
    Peso molecular:770.74
  • Salfredin C1

    CAS:
    <p>Salfredin C1 is an inhibitor of aldose reductase.</p>
    Fórmula:C13H11NO6
    Cor e Forma:Solid
    Peso molecular:277.229
  • Plumbemycin B

    CAS:
    <p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>
    Fórmula:C12H21N4O8P
    Cor e Forma:Solid
    Peso molecular:380.29
  • Antileishmanial agent-5


    <p>Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.</p>
    Fórmula:C17H17ClN4O4
    Cor e Forma:Solid
    Peso molecular:376.79
  • Hypoglycemic agent 1

    CAS:
    <p>Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.</p>
    Fórmula:C25H24FN5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:477.49
  • Antibiotic LL Z1640-2

    CAS:
    <p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>
    Fórmula:C19H22O7
    Cor e Forma:Solid
    Peso molecular:362.38
  • SAR107375

    CAS:
    <p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>
    Fórmula:C24H30ClN5O5S2
    Cor e Forma:Solid
    Peso molecular:568.11
  • NCATS-SM4487

    CAS:
    <p>NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).</p>
    Fórmula:C25H24ClFN8O2
    Cor e Forma:Solid
    Peso molecular:522.96
  • Sinulatumolin E

    CAS:
    <p>Sinulatumolin E, a terpenoid, inhibits TNF-α (IC 50: 3.6 μM); has anti-inflammatory properties.</p>
    Fórmula:C15H22O2
    Cor e Forma:Solid
    Peso molecular:234.33
  • SP inhibitor 1


    <p>SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250&lt;5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.</p>
    Fórmula:C36H38N2O2
    Cor e Forma:Solid
    Peso molecular:530.7
  • ZK159222

    CAS:
    <p>ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.</p>
    Fórmula:C32H48O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:512.72
  • GP-1681

    CAS:
    <p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>
    Fórmula:C24H30NaO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:421.48
  • MEIS-IN-1

    CAS:
    <p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>
    Fórmula:C24H21F3N2O4
    Cor e Forma:Solid
    Peso molecular:458.43
  • PF1070A

    CAS:
    <p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>
    Fórmula:C31H44N4O6
    Cor e Forma:Solid
    Peso molecular:568.7
  • AS2575959

    CAS:
    <p>AS2575959 is a novel GPR40 agonist, exhibiting glucose metabolism improvement and synergistic effect with sitagliptin on insulin and incretin secretion.</p>
    Fórmula:C32H35NaO7
    Cor e Forma:Solid
    Peso molecular:554.6148
  • (S)-Butaprost free acid

    CAS:
    <p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>
    Fórmula:C23H38O5
    Cor e Forma:Solid
    Peso molecular:394.54
  • Hymenidin

    CAS:
    <p>Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.</p>
    Fórmula:C11H12BrN5O
    Pureza:96.85% - 99.52%
    Cor e Forma:Solid
    Peso molecular:310.15
  • TP-030-1

    CAS:
    <p>TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.</p>
    Fórmula:C23H22N4O3
    Cor e Forma:Solid
    Peso molecular:402.45
  • mPGES-1-IN-1


    <p>MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.</p>
    Fórmula:C21H14N4O2S
    Cor e Forma:Solid
    Peso molecular:386.43
  • AVE-1330A sodium

    CAS:
    <p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>
    Fórmula:C7H10N3NaO6S
    Cor e Forma:Solid
    Peso molecular:287.23
  • THR-β agonist 5

    CAS:
    <p>THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of &lt;50 nM [1].</p>
    Fórmula:C22H23N5O2
    Cor e Forma:Solid
    Peso molecular:389.45
  • Steroid sulfatase/17β-HSD1-IN-1


    <p>Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities,</p>
    Fórmula:C19H18N2O5S
    Cor e Forma:Solid
    Peso molecular:386.42
  • Anti-inflammatory agent 13


    <p>Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.</p>
    Fórmula:C30H48O4
    Cor e Forma:Solid
    Peso molecular:472.7
  • Anti-inflammatory agent 18


    <p>Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.</p>
    Fórmula:C30H50O6
    Cor e Forma:Solid
    Peso molecular:506.71
  • Glycotriosyl glutamine

    CAS:
    <p>Glycotriosyl glutamine is a nephritogenoside analog.</p>
    Fórmula:C23H40N2O18
    Cor e Forma:Solid
    Peso molecular:632.57
  • MurB-IN-1


    <p>MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.</p>
    Fórmula:C12H7Cl2F3N2O2
    Cor e Forma:Solid
    Peso molecular:339.1
  • P2X7 receptor antagonist-1


    <p>P2X7 receptor antagonist-1 is a purinergic P2X7 receptor antagonist with anti-neuroinflammatory effects.</p>
    Fórmula:C22H20F4N2O3
    Cor e Forma:Solid
    Peso molecular:436.4
  • LPA5 antagonist 2


    <p>LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.</p>
    Fórmula:C26H25FN2O4S
    Cor e Forma:Solid
    Peso molecular:480.55
  • 12(S)-HEPE

    CAS:
    <p>12(S)-HEPE, made from EPA by 12-LO, is an anti-inflammatory ω-3 derivative affecting leukotriene formation.</p>
    Fórmula:C20H30O3
    Cor e Forma:Solid
    Peso molecular:318.45
  • Dihydrobisdechlorogeodin

    CAS:
    <p>Dihydrobisdechlorogeodin, produced by the fungus strain [FO-4712] of the genus Acremonium, serves as a herbicide.</p>
    Fórmula:C17H16O7
    Cor e Forma:Solid
    Peso molecular:332.31
  • AEP-IN-1


    <p>APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.</p>
    Fórmula:C18H27N3O3
    Cor e Forma:Solid
    Peso molecular:333.43
  • ZIKV-IN-4


    <p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>
    Fórmula:C33H37NO4
    Cor e Forma:Solid
    Peso molecular:511.65
  • Neuraminidase-IN-7


    <p>Neuraminidase-IN-7, a thiophene, inhibits neuraminidase (IC50 0.03 μM), showing promise for flu research.</p>
    Fórmula:C21H20N2O6S
    Cor e Forma:Solid
    Peso molecular:428.46
  • Pyruvate Carboxylase-IN-2

    CAS:
    <p>Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.</p>
    Fórmula:C21H22O8
    Cor e Forma:Solid
    Peso molecular:402.39
  • O4

    CAS:
    <p>O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.</p>
    Fórmula:C24H15NO7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:429.38
  • AS-1940477 hydrobromide

    CAS:
    <p>AS-1940477 hydrobromide is a p38 mitogen-activated protein kinase (MAPK) inhibitor.</p>
    Fórmula:C24H23BrFN5O2
    Cor e Forma:Solid
    Peso molecular:512.38
  • L 731735

    CAS:
    <p>L 731735 is a farnesyltransferase inhibitor.</p>
    Fórmula:C19H40N4O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:420.61
  • PI4KIIIbeta-IN-11

    CAS:
    <p>PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.</p>
    Fórmula:C33H39N7O3
    Cor e Forma:Solid
    Peso molecular:581.71
  • PDE4-IN-5


    <p>PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.</p>
    Fórmula:C21H28N2O3
    Cor e Forma:Solid
    Peso molecular:356.46
  • Esorubicin

    CAS:
    <p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>
    Fórmula:C27H29NO10
    Cor e Forma:Solid
    Peso molecular:527.52
  • Mf 268

    CAS:
    <p>Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.</p>
    Fórmula:C28H46N4O3
    Cor e Forma:Solid
    Peso molecular:486.69
  • Harziphilone

    CAS:
    <p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>
    Fórmula:C15H18O4
    Cor e Forma:Solid
    Peso molecular:262.301
  • Epicillin

    CAS:
    <p>Epicillin possesses antibacterial activity.</p>
    Fórmula:C16H21N3O4S
    Cor e Forma:Solid
    Peso molecular:351.421
  • Hsp90-IN-16


    <p>Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.</p>
    Fórmula:C30H26FN3O6
    Cor e Forma:Solid
    Peso molecular:543.54
  • AFP-07 free acid

    CAS:
    <p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>
    Fórmula:C22H30F2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:412.47
  • Pentenocin A

    CAS:
    <p>Pentenocin A exhibits a relatively weak inhibitory effect on IL-1 and β-glucuronidase (ICE) activity.</p>
    Fórmula:C7H10O5
    Cor e Forma:Solid
    Peso molecular:174.151
  • Dehydelone

    CAS:
    <p>Dehydelone(KOS-1584, R-1645, SK-10088) is a microtubule stabilizer that may be used in the treatment of non-small cell lung cancer.</p>
    Fórmula:C27H39NO5S
    Cor e Forma:Solid
    Peso molecular:489.67
  • Pralatrexate, (R)-

    CAS:
    <p>Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.</p>
    Fórmula:C23H23N7O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:477.47
  • GNTI TFA

    CAS:
    <p>GNTI TFA is a selective kappa opioid receptor antagonist.</p>
    Fórmula:C31H31F6N5O7
    Cor e Forma:Solid
    Peso molecular:699.60
  • Bcl-2-IN-8


    <p>Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.</p>
    Fórmula:C36H44O6
    Cor e Forma:Solid
    Peso molecular:572.73
  • BMS-824

    CAS:
    <p>BMS-824: potent HCV NS5A inhibitor, IC50 ~5 nM, therapeutic index &gt;10,000, specific to HCV.</p>
    Fórmula:C27H25F3N4O5
    Cor e Forma:Solid
    Peso molecular:542.51
  • Ataprost

    CAS:
    <p>Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.</p>
    Fórmula:C21H32O4
    Cor e Forma:Solid
    Peso molecular:348.48
  • PD-1/PD-L1-IN-23

    CAS:
    <p>PD-1/PD-L1-IN-23: potent, oral PD-1/PD-L1 inhibitor; L7's ester prodrug; exhibits strong antitumor effects.</p>
    Fórmula:C32H30BrCl2N3O6
    Cor e Forma:Solid
    Peso molecular:703.41
  • SHR902275

    CAS:
    <p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>
    Fórmula:C26H23F3N4O4
    Cor e Forma:Solid
    Peso molecular:512.48
  • KFA1982

    CAS:
    <p>KFA1982 is a novel and potent factor Xa inhibitor.</p>
    Fórmula:C28H34ClN3O9S2
    Cor e Forma:Solid
    Peso molecular:656.17
  • Fandosentan

    CAS:
    <p>Fandosentan is an endothelin receptor antagonist.</p>
    Fórmula:C25H18F3NO6S
    Cor e Forma:Solid
    Peso molecular:517.47
  • ROPA

    CAS:
    <p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>
    Fórmula:C28H32O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:464.55
  • TRK-IN-19


    <p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) &amp; TRKAG595R (5.3 nM), promising for cancer research.</p>
    Fórmula:C22H26FN5O2
    Cor e Forma:Solid
    Peso molecular:411.47
  • PKG1α activator 3


    <p>PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).</p>
    Fórmula:C27H26Cl2N2O6
    Cor e Forma:Solid
    Peso molecular:545.41
  • AZD2353

    CAS:
    <p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>
    Fórmula:C22H19ClFN3O3
    Cor e Forma:Solid
    Peso molecular:427.86
  • CHNQD-01255

    CAS:
    <p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>
    Fórmula:C23H29NO6
    Cor e Forma:Solid
    Peso molecular:415.48
  • Utrophin modulator 1


    <p>UM1 upregulates utrophin, has EC50 of 0.11 μM, useful in DMD research.</p>
    Fórmula:C22H18N6O
    Cor e Forma:Solid
    Peso molecular:382.42
  • AL-6556

    CAS:
    <p>AL-6556 is a prostaglandin DP receptor agonist.</p>
    Fórmula:C20H33ClO5
    Cor e Forma:Solid
    Peso molecular:388.93
  • UNC9426

    CAS:
    <p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>
    Fórmula:C32H34F6N6O
    Pureza:98.051%
    Cor e Forma:Solid
    Peso molecular:632.642
  • Indinavir monohydrate

    CAS:
    <p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>
    Fórmula:C36H49N5O5
    Cor e Forma:Solid
    Peso molecular:631.82
  • Squalestatin 2

    CAS:
    <p>Squalestatin 2 is an inhibitor of squalene synthase.</p>
    Fórmula:C33H44O13
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:648.69
  • MB-07344 sodium


    <p>"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."</p>
    Fórmula:C19H25NaO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:387.36
  • TrxR-IN-5


    <p>TrxR-IN-5 (compound 4f) is an effective inhibitor of thioredoxin reductase (TrxR) with an IC₅₀ of 0.16 μM. anti-proliferative and anti-metastatic.</p>
    Fórmula:C26H22O3
    Cor e Forma:Solid
    Peso molecular:382.46
  • Cystothiazole A

    CAS:
    <p>Cystothiazole A exhibits antifungal properties, effectively inhibiting Candida albicans, Saccharomyces cerevisiae, and Aspergillus fumigatus with minimum inhibitory concentrations (MIC) of 0.4 μg/mL, 0.1 μg/mL, and 1.6 μg/mL, respectively. It also demonstrates inhibitory activity against human tumor cells such as HPT-116 and K562, with MIC values of 130 ng/mL and 110 ng/mL. However, it shows no antibacterial activity.</p>
    Fórmula:C20H26N2O4S2
    Cor e Forma:Solid
    Peso molecular:422.561
  • 5-cis Carbaprostacyclin

    CAS:
    <p>5-cis Carbaprostacyclin: a PGI2 stable analog; poor human platelet aggregation inhibitor (IC50: 2.8 μM); weakens rabbit artery relaxation (EC50: 104 μM).</p>
    Fórmula:C21H34O4
    Cor e Forma:Solid
    Peso molecular:350.49
  • EP-7041 HCl

    CAS:
    <p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>
    Fórmula:C19H27ClN4O4
    Cor e Forma:Solid
    Peso molecular:410.89
  • Emd 52297

    CAS:
    <p>Emd 52297 is an inhibitor of renin.</p>
    Fórmula:C39H59N11O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:793.96
  • MetRS-IN-1

    CAS:
    <p>MetRS-IN-1 (Compound 27) is an inhibitor of E. coli methionyl-tRNA synthetase (MetRS) with an IC50 value of 237 nM [1].</p>
    Fórmula:C15H13N3O4S
    Cor e Forma:Solid
    Peso molecular:331.35
  • Dersimelagon phosphate

    CAS:
    <p>Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.</p>
    Fórmula:C36H48F4N3O9P
    Cor e Forma:Solid
    Peso molecular:773.75
  • KT2-962

    CAS:
    <p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>
    Fórmula:C23H27ClNNaO5S2
    Cor e Forma:Solid
    Peso molecular:520.04
  • 17β-HSD1-IN-1


    <p>17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.</p>
    Fórmula:C21H21NO3
    Cor e Forma:Solid
    Peso molecular:335.4
  • OXS007417


    <p>OXS007417 induces AML cell differentiation at 48 nM EC50 and shows potent in vivo antitumor effects.</p>
    Fórmula:C20H14F3N3O
    Cor e Forma:Solid
    Peso molecular:369.34
  • CI 922

    CAS:
    <p>CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.</p>
    Fórmula:C26H30N10O6
    Cor e Forma:Solid
    Peso molecular:578.58
  • KNI 10033

    CAS:
    <p>KNI 10033 is a potent inhibitor of HIV protease</p>
    Fórmula:C40H45N5O7S2
    Cor e Forma:Solid
    Peso molecular:771.95
  • Sannamycin J

    CAS:
    <p>Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C14H30N4O4
    Cor e Forma:Solid
    Peso molecular:318.41
  • MDL-27210

    CAS:
    <p>MDL-27210 is the ethyl ester prodrug of a potent angiotensin-converting enzyme inhibitor, MDL-27088.</p>
    Fórmula:C27H32N2O5
    Cor e Forma:Solid
    Peso molecular:464.55
  • Annonin VI

    CAS:
    <p>Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.</p>
    Fórmula:C37H66O7
    Cor e Forma:Solid
    Peso molecular:622.92
  • Tuvatidine

    CAS:
    <p>Tuvatidine is a histamine 2 receptor antagonist.</p>
    Fórmula:C10H17N9O2S3
    Cor e Forma:Solid
    Peso molecular:391.5
  • Cryptopleurine

    CAS:
    <p>Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.</p>
    Fórmula:C24H27NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:377.48
  • Nolpitantium Free Base

    CAS:
    <p>Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.</p>
    Fórmula:C37H45Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:620.67
  • 15(R)-Lipoxin A4

    CAS:
    <p>Lipid-derived lipoxins are produced at the site of vascular and mucosal inflammation where they down-regulate polymorphonuclear leukocyte recruitment and</p>
    Fórmula:C20H32O5
    Cor e Forma:Solid
    Peso molecular:352.47
  • EBOV-GP-IN-1


    <p>EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).</p>
    Fórmula:C25H40ClN3O2
    Cor e Forma:Solid
    Peso molecular:450.06
  • CJ-887

    CAS:
    <p>CJ-887 is a STAT3 inhibitor.</p>
    Fórmula:C34H45N6O10P
    Cor e Forma:Solid
    Peso molecular:728.73
  • LY 190388

    CAS:
    <p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>
    Fórmula:C30H41N5O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:615.74
  • GR-71251

    CAS:
    <p>GR-71251 is a Tachykinin receptor antagonist.</p>
    Fórmula:C74H105N19O13
    Cor e Forma:Solid
    Peso molecular:1468.74
  • VEGFR-2-IN-10


    <p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>
    Fórmula:C20H21N3O2
    Cor e Forma:Solid
    Peso molecular:335.4
  • iMDK quarterhydrate


    <p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>
    Fórmula:C21H15FN2O3S
    Cor e Forma:Solid
    Peso molecular:380.91
  • Bacithrocin C

    CAS:
    <p>Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.</p>
    Fórmula:C18H27N5O3
    Cor e Forma:Solid
    Peso molecular:361.439
  • Oberadilol

    CAS:
    <p>Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action</p>
    Fórmula:C25H30ClN5O3
    Cor e Forma:Solid
    Peso molecular:483.99
  • NVP-CFC218

    CAS:
    <p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>
    Fórmula:C37H45ClN4O4
    Cor e Forma:Solid
    Peso molecular:645.23
  • TLN-232

    CAS:
    <p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>
    Fórmula:C36H49N9O7S2
    Cor e Forma:Solid
    Peso molecular:783.96
  • Anti-inflammatory agent 19


    <p>Anti-inflammatory agent 19: NO inhibitor (IC50: 36μM), blocks HMGB1, for late-stage inflammation, relevant for COVID-19, sepsis.</p>
    Fórmula:C30H50O7
    Cor e Forma:Solid
    Peso molecular:522.71
  • Carbacyclin

    CAS:
    <p>Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.</p>
    Fórmula:C21H34O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:350.49
  • NNTA

    CAS:
    <p>NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.</p>
    Fórmula:C31H32N2O4
    Cor e Forma:Solid
    Peso molecular:496.60
  • Monorden diacetate

    CAS:
    <p>Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.</p>
    Fórmula:C22H21ClO8
    Cor e Forma:Solid
    Peso molecular:448.85
  • NCI-006

    CAS:
    <p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>
    Fórmula:C31H24F2N4O4S3
    Cor e Forma:Solid
    Peso molecular:650.74
  • Rhamnitol

    CAS:
    <p>Rhamnitol, the reduction product of L-rhamnose, can be observed during the metabolism of rhamnose in the body. Rhamnitol is promising for use in assessing intestinal permeability and studying carbohydrate metabolism.</p>
    Fórmula:C6H14O5
    Cor e Forma:Solid
    Peso molecular:166.17
  • Imolamine hydrochloride

    CAS:
    <p>Imolamine hydrochloride is a blood platelet aggregation antagonist.</p>
    Fórmula:C14H21ClN4O
    Cor e Forma:Solid
    Peso molecular:296.80