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Outros inibidores

Outros inibidores

Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.

Foram encontrados 37926 produtos de "Outros inibidores"

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  • SARS-CoV-2 nsp14-IN-2


    <p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>
    Fórmula:C21H21N5O5S
    Cor e Forma:Solid
    Peso molecular:455.49
  • GNTI TFA

    CAS:
    <p>GNTI TFA is a selective kappa opioid receptor antagonist.</p>
    Fórmula:C31H31F6N5O7
    Cor e Forma:Solid
    Peso molecular:699.60
  • Trk-IN-8


    <p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>
    Fórmula:C18H16F2N6O2
    Cor e Forma:Solid
    Peso molecular:386.36
  • Acetoxycycloheximide

    CAS:
    <p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>
    Fórmula:C17H25NO6
    Cor e Forma:Solid
    Peso molecular:339.38
  • ROS1-IN-1


    <p>ROS1-IN-1, a potent ROS1 kinase inhibitor, has an IC50 of 0.097 μM.</p>
    Fórmula:C17H15ClN6S
    Cor e Forma:Solid
    Peso molecular:370.86
  • PTP1B-IN-18


    <p>PTP1B-IN-18 is an orally active, fully mixed protein tyrosine phosphatase 1B (PTP1B) inhibitor (Ki: 35.2 μM).PTP1B-IN-18 can be used to study type 2 diabetes.</p>
    Fórmula:C26H19N3O4S
    Cor e Forma:Solid
    Peso molecular:469.51
  • CGS 22652

    CAS:
    <p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>
    Fórmula:C22H29ClN2O4S
    Cor e Forma:Solid
    Peso molecular:452.99
  • Dexnebivolol

    CAS:
    <p>Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.</p>
    Fórmula:C22H25F2NO4
    Cor e Forma:Solid
    Peso molecular:405.43
  • ZK-Thiazolidinone

    CAS:
    <p>ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.</p>
    Fórmula:C23H26F3N5O2S
    Cor e Forma:Solid
    Peso molecular:493.55
  • Anti-inflammatory agent 23


    <p>Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.</p>
    Fórmula:C34H49NO6
    Cor e Forma:Solid
    Peso molecular:567.76
  • SARS 3CLpro-IN-1

    CAS:
    <p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>
    Fórmula:C22H38N4O2
    Cor e Forma:Solid
    Peso molecular:390.56
  • ER Thermo Yellow

    CAS:
    <p>ER Thermo Yellow is a high-sensitivity (3.9%/°C) fluorescent probe designed for temperature visualization specifically targeting the endoplasmic reticulum.</p>
    Fórmula:C27H20BClF5N3O3
    Peso molecular:575.72
  • Tezampanel hydrate

    CAS:
    <p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>
    Fórmula:C13H23N5O3
    Cor e Forma:Solid
    Peso molecular:297.35
  • FCE-24379

    CAS:
    <p>FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.</p>
    Fórmula:C20H22N4O2
    Cor e Forma:Solid
    Peso molecular:350.41
  • UNC7467

    CAS:
    <p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>
    Fórmula:C20H13NO3
    Pureza:98.28% - 98.64%
    Cor e Forma:Soild
    Peso molecular:315.32
  • Antitumor agent-65

    CAS:
    <p>Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.</p>
    Fórmula:C18H17NO10
    Cor e Forma:Solid
    Peso molecular:407.33
  • Gentamicin C1

    CAS:
    <p>Gentamicin C1 is a broad-spectrum aminoglycoside antibiotic with antibacterial activity.</p>
    Fórmula:C21H43N5O7
    Cor e Forma:Solid
    Peso molecular:477.595
  • Naphthablin

    CAS:
    <p>Naphthablin is a naphthoquinone compound that inhibits the function of the Abl oncogene. It prevents the morphological transformation of v-ablts-NIH3T3 cells induced by Abl and also suppresses RNA synthesis.</p>
    Fórmula:C29H36O8
    Cor e Forma:Solid
    Peso molecular:512.591
  • Isoleucyl tRNA synthetase-IN-1

    CAS:
    <p>Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>
    Fórmula:C23H35N5O7S
    Cor e Forma:Solid
    Peso molecular:525.62
  • Sannamycin K

    CAS:
    <p>Sannamycin K is an aminoglycoside antibiotic with weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C13H26N4O4
    Cor e Forma:Solid
    Peso molecular:302.37
  • MCTR2

    CAS:
    <p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>
    Fórmula:C27H40N2O6S
    Cor e Forma:Solid
    Peso molecular:520.68
  • FTI-2153 TFA


    <p>FTI-2153 TFA inhibits farnesyltransferase with high selectivity (IC50: 1.4 nM), over 3000x more than Rap1A processing.</p>
    Fórmula:C27H31F3N4O5S
    Cor e Forma:Solid
    Peso molecular:580.62
  • Vicanicin

    CAS:
    <p>Vicanicin is an aryl phenol ether compound found in lichens. It inhibits the expression of Hsp70, modulates intracellular redox-sensitive mechanisms, increases reactive oxygen species (ROS) in cancer cells, alters the Bax/Bcl-2 ratio, activates caspase-3, and induces apoptosis. Vicanicin suppresses cell growth and promotes apoptosis in androgen-sensitive (LNCaP) and androgen-insensitive (DU-145) human prostate cancer cells. It holds potential for prostate cancer research.</p>
    Fórmula:C18H16Cl2O5
    Cor e Forma:Solid
    Peso molecular:383.223
  • DN-F01


    <p>DN-F01 exhibits a potent calcium-dependent inhibitory effect on cardiac myofibrillar ATPase activity, with an IC50 of 11 ± 4 nmol/L.</p>
    Fórmula:C22H16N2O2
    Cor e Forma:Solid
    Peso molecular:340.37
  • Tandutinib (MLN518) HCl


    <p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>
    Fórmula:C31H43ClN6O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:599.16
  • Monamycin H2

    CAS:
    <p>Monamycin H2 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.</p>
    Fórmula:C34H56ClN7O8
    Peso molecular:726.30
  • De-N-methylpamamycin-593A

    CAS:
    <p>De-N-methylpamamycin-593A is a 16-membered macrocyclic dilactone known for its ability to induce aerial mycelium formation.</p>
    Fórmula:C34H59NO7
    Peso molecular:593.84
  • TT15

    CAS:
    <p>TT15 is an agonist of the GLP-1R.</p>
    Fórmula:C51H44Cl2N4O6
    Cor e Forma:Solid
    Peso molecular:879.82
  • Formadicin C

    CAS:
    <p>Formadicin C exhibits the strongest activity among all components against certain strains of Pseudomonas, Proteus, and Alcaligenes.</p>
    Fórmula:C24H26N4O10
    Peso molecular:530.48
  • Cuevaene A

    CAS:
    <p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>
    Fórmula:C21H22O5
    Cor e Forma:Solid
    Peso molecular:354.396
  • Griseorhodin G

    CAS:
    <p>Griseorhodin G is a quinone antibiotic with antitumor activity.</p>
    Fórmula:C25H18O12
    Peso molecular:510.40
  • 20-HEDE

    CAS:
    <p>20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.</p>
    Fórmula:C20H36O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:324.50
  • HS-731

    CAS:
    <p>HS-731 is a μ-Opioid Receptor Agonist.</p>
    Fórmula:C20H26N2O5
    Cor e Forma:Solid
    Peso molecular:374.43
  • SCP1-IN-1

    CAS:
    <p>SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.</p>
    Fórmula:C20H19F3N2O7S2
    Pureza:99.53%
    Cor e Forma:Soild
    Peso molecular:520.5
  • Maltophilin

    CAS:
    <p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>
    Fórmula:C29H38N2O6
    Peso molecular:510.62
  • Polyoxin J

    CAS:
    <p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>
    Fórmula:C17H25N5O12
    Peso molecular:491.41
  • Antiplatelet agent 3

    CAS:
    <p>Antiplatelet agent 3 (Compound K-10) is a compound with antiplatelet aggregation activity, exhibiting IC50 values of 2.55, 3.22, and 2.09 mg/mL for platelet aggregation induced by ADP, AA, and COL, respectively. It holds potential for research in cardiovascular diseases.</p>
    Fórmula:C38H32N2O5
    Cor e Forma:Solid
    Peso molecular:596.671
  • 5,6-Dihydro-4-methoxy-2H-pyran-2-one

    CAS:
    <p>5,6-Dihydro-4-methoxy-2H-pyran-2-one is produced by the Penicillium italicum strain MRC 1360.</p>
    Fórmula:C6H8O3
    Peso molecular:128.13
  • Monamycin G1

    CAS:
    <p>Monamycin G1 is an ester-peptide antibiotic [esterpeptid]. It shows activity against Gram-positive bacteria.</p>
    Fórmula:C33H54ClN7O8
    Peso molecular:712.28
  • Annonin VI

    CAS:
    <p>Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.</p>
    Fórmula:C37H66O7
    Cor e Forma:Solid
    Peso molecular:622.92
  • Glaucarubin

    CAS:
    <p>Glaucarubin is a bitter lactone naturally found in the fruits of Simaruba glauca. It is employed as an anti-amebic agent in research focused on amebiasis. The compound exhibits good tolerability, with a median lethal dose (LD50) of 1,600 mg/kg in mice and 6,400 mg/kg in rats.</p>
    Fórmula:C25H36O10
    Peso molecular:496.55
  • Oryzoxymycin

    CAS:
    <p>Oryzoxymycin is an aromatic derivative antibiotic with activity against Gram-negative bacteria.</p>
    Fórmula:C10H13NO5
    Peso molecular:227.21
  • Dihydropergillin

    CAS:
    <p>Dihydropergillin is produced by the Aspergillus terreus strain (ATCC 38849) and has the ability to inhibit plant growth.</p>
    Fórmula:C15H18O4
    Peso molecular:262.30
  • Lucilactaene

    CAS:
    <p>Lucilactaene exhibits potent antimalarial activity and functions as a P53-transfected tumor cell cycle inhibitor. It effectively halts the cell cycle progression of H1299/TSP53 cells at the G1 phase.</p>
    Fórmula:C22H27NO6
    Peso molecular:401.45
  • MRS2279

    CAS:
    <p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>
    Fórmula:C13H18ClN5O8P2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:469.71
  • Milbemycin α13

    CAS:
    <p>Milbemycin α13 (Meilingmycin B) is an antibiotic that is effective against nematodes and mites.</p>
    Fórmula:C37H52O9
    Peso molecular:640.80
  • Polyoxin K

    CAS:
    <p>Polyoxin K is a nucleoside antifungal antibiotic that exhibits significant effectiveness against rice sheath blight.</p>
    Fórmula:C22H30N6O13
    Peso molecular:586.51
  • JTE 151A

    CAS:
    <p>JTE-151 is a novel RORγ inverse agonist.</p>
    Fórmula:C26H30ClN3O5
    Cor e Forma:Solid
    Peso molecular:499.99
  • Papyracon D

    CAS:
    <p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>
    Fórmula:C14H18O5
    Peso molecular:266.29
  • PI3K-IN-23


    <p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>
    Fórmula:C24H33NO4S
    Cor e Forma:Solid
    Peso molecular:431.59
  • Melanoxazal

    CAS:
    <p>Melanoxazal is an inhibitor of melanin biosynthesis, effectively suppressing melanin formation in silkworm larva hemolymph with an IC50 of 30.1 μg/mL, and it also exhibits strong inhibitory effects on mushroom tyrosinase (IC50 of 4.2 μg/mL), while lacking antibacterial activity.</p>
    Fórmula:C8H9NO3
    Peso molecular:167.16
  • Hispidospermidin

    CAS:
    <p>Hispidospermidin is a phospholipase C inhibitor.</p>
    Fórmula:C25H47N3O
    Cor e Forma:Solid
    Peso molecular:405.66
  • iMDK quarterhydrate


    <p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>
    Fórmula:C21H15FN2O3S
    Cor e Forma:Solid
    Peso molecular:380.91
  • Norplicacetin

    CAS:
    <p>Norplicacetin exhibits activity against Gram-positive bacteria and mycobacteria.</p>
    Fórmula:C24H33N5O7
    Peso molecular:503.55
  • Amidinomycin

    CAS:
    <p>Amidinomycin primarily acts against Gram-positive bacteria.</p>
    Fórmula:C9H18N4O
    Peso molecular:198.27
  • Demycarosyl platenomycin

    CAS:
    <p>Demycarosylplatenomycin (DM-PLM) is an antibiotic that exhibits mild activity against Gram-positive bacteria.</p>
    Fórmula:C31H51NO11
    Peso molecular:613.74
  • Polyoxin L

    CAS:
    <p>Polyoxin L is a nucleoside-type antifungal antibiotic that is notably effective against rice sheath blight.</p>
    Fórmula:C16H23N5O12
    Peso molecular:477.38
  • Monamycin D1

    CAS:
    <p>Monamycin D1 is a lipopeptide antibiotic with activity against Gram-positive bacteria.</p>
    Fórmula:C34H57N7O8
    Peso molecular:691.86
  • Methylenomycin A

    CAS:
    <p>Methylenomycin A is a cyclopentanone-derived antibiotic effective against both Gram-negative and Gram-positive bacteria.</p>
    Fórmula:C9H10O4
    Cor e Forma:Solid
    Peso molecular:182.173
  • Danavorexton

    CAS:
    <p>Danavorexton is an orexin receptor agonist.</p>
    Fórmula:C21H32N2O5S
    Cor e Forma:Solid
    Peso molecular:424.55
  • Azonafide-PEABA

    CAS:
    <p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>
    Fórmula:C32H33N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:551.64
  • MB725

    CAS:
    <p>MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.</p>
    Fórmula:C18H21IN4O2S
    Cor e Forma:Solid
    Peso molecular:484.35
  • Glucosylceramide synthase-IN-3


    <p>Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.</p>
    Fórmula:C21H20FN3O3
    Cor e Forma:Solid
    Peso molecular:381.4
  • Falecalcitriol

    CAS:
    <p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>
    Fórmula:C27H38F6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:524.58
  • GLS1 Inhibitor-5


    <p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>
    Cor e Forma:Solid
  • NTPDase-IN-1


    <p>NTPDase-IN-1 selectively inhibits NTPDases 1, 2, 8 with IC50 of 0.05, 0.23, 0.54 μM. Non-competitive, K m 21 μM, used in cancer, immune, infection research.</p>
    Fórmula:C18H25N3OS2
    Cor e Forma:Solid
    Peso molecular:363.54
  • Z57346765

    CAS:
    <p>Z57346765 is a specific PGK1 inhibitor that inhibits PGK1-dependent cell proliferation by decreasing the metabolic enzyme activity of PGK1 during glycolysis.</p>
    Fórmula:C17H18N4O
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:294.35
  • Napsagatran hydrate

    CAS:
    <p>Napsagatran hydrate is a novel and specific inhibitor of thrombin.</p>
    Fórmula:C26H36N6O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:576.66
  • Hazimycin 6

    CAS:
    Hazimycin 6 exhibits weak activity against gram-negative bacteria, yeast, and dermatophytes.
    Fórmula:C20H18N4O4
    Cor e Forma:Solid
    Peso molecular:378.381
  • Griseolutein A

    CAS:
    <p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C17H14N2O6
    Cor e Forma:Solid
    Peso molecular:342.303
  • Herbicidin B

    CAS:
    <p>Herbicidin B exhibits herbicidal properties and activity against Gram-positive bacteria.</p>
    Fórmula:C18H23N5O9
    Cor e Forma:Solid
    Peso molecular:453.403
  • 6-Hydroxytetrangulol

    CAS:
    <p>6-Hydroxytetrangulol is an inducer of CPP32 protease found in Streptomyces.</p>
    Fórmula:C19H12O5
    Cor e Forma:Solid
    Peso molecular:320.30
  • Pelagiomicin C

    CAS:
    <p>Pelagiomicin C exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C17H15N3O5
    Cor e Forma:Solid
    Peso molecular:341.318
  • Pentenocin A

    CAS:
    <p>Pentenocin A exhibits a relatively weak inhibitory effect on IL-1 and β-glucuronidase (ICE) activity.</p>
    Fórmula:C7H10O5
    Cor e Forma:Solid
    Peso molecular:174.151
  • Saframycin Mx2

    CAS:
    <p>Saframycin Mx2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C29H38N4O8
    Cor e Forma:Solid
    Peso molecular:570.634
  • GW311616 hydrochloride

    CAS:
    <p>GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>
    Fórmula:C19H32ClN3O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.99
  • Epicillin

    CAS:
    <p>Epicillin possesses antibacterial activity.</p>
    Fórmula:C16H21N3O4S
    Cor e Forma:Solid
    Peso molecular:351.421
  • Fleephilone

    CAS:
    <p>Fleephilone is a fungal metabolite isolated from Trichoderma harzianum. It acts as an HIV REV/RRE binding inhibitor, hindering the interaction between REV protein and RRE RNA with an IC50 of 7.6 μM.</p>
    Fórmula:C24H27NO7
    Cor e Forma:Solid
    Peso molecular:441.474
  • Harziphilone

    CAS:
    <p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>
    Fórmula:C15H18O4
    Cor e Forma:Solid
    Peso molecular:262.301
  • Nemotin

    CAS:
    <p>Nemotin exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while its effectiveness against Gram-negative bacteria is present but relatively weaker.</p>
    Fórmula:C11H8O2
    Cor e Forma:Solid
    Peso molecular:172.18
  • Kahweol linoleate

    CAS:
    <p>Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.</p>
    Fórmula:C38H56O4
    Cor e Forma:Solid
    Peso molecular:576.85
  • Dihydrobisdechlorogeodin

    CAS:
    <p>Dihydrobisdechlorogeodin, produced by the fungus strain [FO-4712] of the genus Acremonium, serves as a herbicide.</p>
    Fórmula:C17H16O7
    Cor e Forma:Solid
    Peso molecular:332.31
  • ODN 2088

    CAS:
    <p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>
    Cor e Forma:Solid
  • Hypercalin B

    CAS:
    <p>Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.</p>
    Fórmula:C33H42O5
    Cor e Forma:Solid
    Peso molecular:518.684
  • 3,4-Dimethoxytropolone

    CAS:
    <p>3,4-Dimethoxytropolone can be isolated from the fermentation broth of Streptoverticillium hadanonense, and it shows activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C9H10O4
    Cor e Forma:Solid
    Peso molecular:182.173
  • Imolamine hydrochloride

    CAS:
    <p>Imolamine hydrochloride is a blood platelet aggregation antagonist.</p>
    Fórmula:C14H21ClN4O
    Cor e Forma:Solid
    Peso molecular:296.80
  • Oiligodendrocyte differentiation promoter 1

    CAS:
    <p>Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .</p>
    Fórmula:C25H25Cl2NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:490.38
  • Difeterol

    CAS:
    <p>Difeterol is a biochemical.</p>
    Fórmula:C25H29NO2
    Cor e Forma:Solid
    Peso molecular:375.50
  • SPR7


    <p>SPR7 is a potent and selective rhodesain inhibitor (Ki: 0.51 nM). SPR7 exhibited antiparasitic effects against T. b. brucei (EC50: 1.65 μM).</p>
    Fórmula:C30H32ClN3O3
    Cor e Forma:Solid
    Peso molecular:518.05
  • Luffolide

    CAS:
    <p>Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.</p>
    Fórmula:C27H40O6
    Cor e Forma:Solid
    Peso molecular:460.60
  • 23-De(mycinosyloxy)tylosin

    CAS:
    <p>23-De(mycinosyloxy)tylosin is a macrolide antibiotic exhibiting activity against Gram-positive bacteria, with limited efficacy against Gram-negative bacteria and mycoplasma.</p>
    Fórmula:C38H63NO12
    Cor e Forma:Solid
    Peso molecular:725.91
  • GC 14

    CAS:
    <p>GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.</p>
    Fórmula:C26H27NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:449.5
  • ONO-AE1-259 lysine

    CAS:
    <p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>
    Fórmula:C28H49ClN2O6
    Cor e Forma:Solid
    Peso molecular:545.15
  • Mycinamicin Ⅵ

    CAS:
    <p>Mycinamicin VI is a macrolide antibiotic with antibacterial activity against Gram-positive bacteria.</p>
    Fórmula:C35H57NO11
    Cor e Forma:Solid
    Peso molecular:667.83
  • Megovalicin G

    CAS:
    <p>Megovalicin G is effective against Bacillus subtilis and Escherichia coli, and it also acts on Pseudomonas aeruginosa.</p>
    Fórmula:C35H61NO7
    Cor e Forma:Solid
    Peso molecular:607.86
  • Monamycin B

    CAS:
    <p>Monamycin B is an ester peptide antibiotic with activity against Gram-positive bacteria.</p>
    Fórmula:C33H55N7O8
    Cor e Forma:Solid
    Peso molecular:677.83
  • FR-900482

    CAS:
    <p>FR-900482 exhibits high sensitivity to Thermoactinomyces calidolactis strain C 953 and demonstrates activity against cell lines such as P388, B16, EL4, FM3A, L1210, BHK-21, among others.</p>
    Fórmula:C14H15N3O6
    Cor e Forma:Solid
    Peso molecular:321.29
  • 9-Hydroxycrisamicin

    CAS:
    <p>9-Hydroxycrisamicin exhibits moderate activity against Gram-positive bacteria with a minimum inhibitory concentration (MIC) ranging from 6.25 to 25 μg/mL. Additionally, 9-Hydroxycrisamicin demonstrates significant growth inhibition towards various human tumor cell lines.</p>
    Fórmula:C32H22O13
    Cor e Forma:Solid
    Peso molecular:614.51
  • Dictyopanine A

    CAS:
    <p>Dictyopanine A exhibits a relatively narrow antibacterial spectrum, demonstrating moderate antimicrobial activity only against certain filamentous fungi and Gram-positive bacteria.</p>
    Fórmula:C25H34O5
    Cor e Forma:Solid
    Peso molecular:414.53
  • Monamycin I

    CAS:
    <p>Monamycin I is an ester peptide antibiotic with activity against Gram-positive bacteria.</p>
    Fórmula:C35H58ClN7O8
    Cor e Forma:Solid
    Peso molecular:740.33
  • RIP1 kinase inhibitor 1

    CAS:
    <p>RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.</p>
    Fórmula:C24H20ClN5O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:461.9
  • Chitinase-IN-4


    <p>Chitinase-IN-4 (compound 8f) is a potent and selective inhibitor of OfChi-h with an IC50 value of 0.1 μM and good insecticidal activity.</p>
    Fórmula:C21H24ClN7
    Cor e Forma:Solid
    Peso molecular:409.92
  • 5-Deoxygentamicin C1

    CAS:
    <p>5-Deoxygentamicin C1 exhibits activity against both gram-positive and gram-negative bacteria.</p>
    Fórmula:C21H43N5O6
    Cor e Forma:Solid
    Peso molecular:461.60
  • TAM&Met-IN-1

    CAS:
    <p>TAM&amp;Met-IN-1 inhibits AXL, MER, TYRO3 with IC50s 6.1, 13.2, 21.6 nM, respectively, for cancer research.</p>
    Fórmula:C29H27F2N7O5
    Cor e Forma:Solid
    Peso molecular:591.57
  • Anticancer agent 26


    <p>Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.</p>
    Fórmula:C28H33NO5
    Cor e Forma:Solid
    Peso molecular:463.57
  • DWN-12088 HCl

    CAS:
    <p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>
    Fórmula:C15H21Cl4N3O
    Cor e Forma:Solid
    Peso molecular:401.15
  • Mepixetil


    <p>Mepixetil is a potent angiotensin II receptor antagonist[1].</p>
    Fórmula:C12H18N2O3
    Cor e Forma:Solid
    Peso molecular:238.28
  • ErSO-DFP


    <p>ErSO-DFP activates a-UPR, targets ERα+ cancer cells with high selectivity, and effectively reduces MCF-7 tumours.</p>
    Fórmula:C20H17F5N2O2
    Cor e Forma:Solid
    Peso molecular:412.35
  • Pefcalcitol

    CAS:
    <p>Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.</p>
    Fórmula:C26H34F5NO4
    Cor e Forma:Solid
    Peso molecular:519.54
  • Rimegepant sulfate hydrate

    CAS:
    <p>Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.</p>
    Fórmula:C56H64F4N12O13S
    Cor e Forma:Solid
    Peso molecular:1221.2526
  • Retezorogant

    CAS:
    <p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>
    Fórmula:C23H33ClN2O3
    Cor e Forma:Solid
    Peso molecular:420.97
  • Pyrisulfoxin B

    CAS:
    <p>Pyrisulfoxin B is an antibiotic produced by the bacterium Streptomyces (BS-75).</p>
    Fórmula:C13H11N3O2S
    Cor e Forma:Solid
    Peso molecular:273.31
  • AZ0108

    CAS:
    <p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>
    Fórmula:C24H20F4N6O2
    Cor e Forma:Solid
    Peso molecular:500.45
  • AVE 0991

    CAS:
    <p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>
    Fórmula:C29H32N4O5S2
    Pureza:98.69%
    Cor e Forma:Solid
    Peso molecular:580.72
  • Enpp-1-IN-12


    <p>ENPP1-IN-12 is a potent, oral ENPP1 inhibitor with a Ki of 41 nM and anti-tumor properties.</p>
    Fórmula:C17H19N5O3S
    Cor e Forma:Solid
    Peso molecular:373.43
  • Keap1-Nrf2-IN-1 TFA


    <p>Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.</p>
    Fórmula:C26H25F3N2O9S
    Cor e Forma:Solid
    Peso molecular:598.54
  • P2X receptor-1


    <p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>
    Fórmula:C14H14ClN3O3S2
    Cor e Forma:Solid
    Peso molecular:371.86
  • ZK824859 hydrochloride (2271122-53-1 free base)


    <p>ZK824859 hydrochloride: oral, selective uPA inhibitor, IC50s: 79 nM (uPA), 1580 nM (tPA), 1330 nM (plasmin).</p>
    Fórmula:C23H23ClF2N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:464.89
  • PCSK9-IN-16

    CAS:
    <p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>
    Fórmula:C16H20N6O2S3
    Cor e Forma:Solid
    Peso molecular:424.56
  • Aplysin

    CAS:
    <p>Aplysin suppresses breast cancer cells and protects liver cells by blocking PI3K/AKT/FOXO3a and preventing oxidative damage.</p>
    Fórmula:C15H19BrO
    Cor e Forma:Solid
    Peso molecular:295.21
  • Zetomipzomib

    CAS:
    <p>KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) &amp; LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.</p>
    Fórmula:C30H42N4O8
    Cor e Forma:Solid
    Peso molecular:586.68
  • 20-Deoxynarasin

    CAS:
    <p>20-Deoxynarasin exhibits activity against Gram-positive bacteria, mycoplasma, coccidia, and viruses, and it also promotes growth.</p>
    Fórmula:C43H72O10
    Cor e Forma:Solid
    Peso molecular:749.03
  • SPR-00305

    CAS:
    <p>SPR-00305 is a novel potent inhibitor of the mvfr pathway</p>
    Fórmula:C24H19ClN2O3
    Cor e Forma:Solid
    Peso molecular:418.87
  • GSK1820795A

    CAS:
    <p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>
    Fórmula:C35H34N8
    Cor e Forma:Solid
    Peso molecular:566.7
  • Domitroban

    CAS:
    <p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>
    Fórmula:C20H27NO4S
    Cor e Forma:Solid
    Peso molecular:377.5
  • Kigamicin B

    CAS:
    <p>Kigamicin B exhibits activity against gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>
    Fórmula:C40H45NO15
    Cor e Forma:Solid
    Peso molecular:779.78
  • Phenazostatin B

    CAS:
    <p>Phenazostatin B is a phenazine derivative known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. It inhibits glutamate toxicity in N18-RE-105 cells, with an EC50 of 0.33 μg/mL.</p>
    Fórmula:C32H26N4O4
    Cor e Forma:Solid
    Peso molecular:530.57
  • PEN-866

    CAS:
    <p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>
    Fórmula:C49H49N7O9
    Cor e Forma:Solid
    Peso molecular:879.95
  • Oberadilol

    CAS:
    <p>Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action</p>
    Fórmula:C25H30ClN5O3
    Cor e Forma:Solid
    Peso molecular:483.99
  • hTrkA-IN-2


    <p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>
    Fórmula:C24H22F3N5O3
    Cor e Forma:Solid
    Peso molecular:485.46
  • THR-β agonist 4

    CAS:
    <p>THR-β agonist 4 is a potent agonist of THR-β.</p>
    Fórmula:C16H11Cl2F2N5O6S
    Cor e Forma:Solid
    Peso molecular:510.26
  • Oral antiplatelet agent 1

    CAS:
    <p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>
    Fórmula:C23H24N4O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:468.53
  • Cinnatriacetin A

    CAS:
    <p>Cinnatriacetin A exhibits activity against Gram-positive bacteria.</p>
    Fórmula:C23H20O5
    Cor e Forma:Solid
    Peso molecular:376.402
  • Coriolin A

    CAS:
    <p>Coriolin A exhibits activity against gram-positive bacteria, weakly against gram-negative bacteria, as well as yeasts and Trichomonas vaginalis. At a concentration of 5 μg/mL, it inhibits 61.6% of the growth of Yoshida sarcoma, but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Fórmula:C15H20O5
    Cor e Forma:Solid
    Peso molecular:280.316
  • Lipohexin

    CAS:
    <p>Lipohexin is a peptide antibiotic that exhibits activity against Gram-positive bacteria. It competitively inhibits human placental proline endopeptidase (proline endopeptidase) with an IC50 of 3.5 μM. Additionally, Lipohexin inhibits proline endopeptidase from Flavobacterium meningosepticum, with an IC50 of 25 μM.</p>
    Fórmula:C39H68N6O9
    Cor e Forma:Solid
    Peso molecular:764.992
  • Leucomycin A6

    CAS:
    <p>Leucomycin A6 effectively combats Gram-positive bacteria.</p>
    Fórmula:C41H67NO14
    Cor e Forma:Solid
    Peso molecular:797.969
  • CB-7646

    CAS:
    <p>CB-7646 is a stable trimelamol (TM) analogue, which is an antitumor agent.</p>
    Fórmula:C8H16N6O2
    Cor e Forma:Solid
    Peso molecular:228.25
  • Coriolin B

    CAS:
    <p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Fórmula:C23H36O6
    Cor e Forma:Solid
    Peso molecular:408.528
  • Salfredin C3

    CAS:
    <p>Salfredin C3 is an inhibitor of aldose reductase (aldose reductase).</p>
    Fórmula:C16H15NO8
    Cor e Forma:Solid
    Peso molecular:349.292
  • Griseolic acid C

    CAS:
    <p>Griseolic acid C (Dihydrodeoxygriseolic acid) is an antibiotic found in the Streptomyces griseoaurantiacus SANK43894 strain. This compound is a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase [EC 3.1.4.17], with an IC50 of 0.12 μM (enzyme sourced from rat brain tissue).</p>
    Fórmula:C14H15N5O7
    Cor e Forma:Solid
    Peso molecular:365.298
  • Hcyb1


    <p>Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.</p>
    Fórmula:C24H20N4O
    Cor e Forma:Solid
    Peso molecular:380.44
  • MU1656

    CAS:
    <p>MU1656 is a selective inhibitor of histone methyltransferase DOT1L, which significantly inhibits cancer cell proliferation in hematological malignancies.</p>
    Fórmula:C32H45N7O2
    Pureza:96.92%
    Cor e Forma:Solid
    Peso molecular:559.75
  • Rhodomycin B

    CAS:
    <p>Rhodomycin B exhibits activity against Gram-positive bacteria, while its effects on Gram-negative bacteria and fungi are relatively weak.</p>
    Fórmula:C28H33NO10
    Cor e Forma:Solid
    Peso molecular:543.562
  • Saframycin B

    CAS:
    <p>Saframycin B exhibits activity against Gram-positive bacteria and has weaker efficacy against mycobacteria.</p>
    Fórmula:C28H31N3O8
    Cor e Forma:Solid
    Peso molecular:537.561
  • Azicemicin A

    CAS:
    <p>Azicemicin A exhibits mild antibacterial activity and shows no acute toxicity when administered via intraperitoneal injection to mice at a dosage of 150 mg/kg.</p>
    Fórmula:C23H25NO9
    Cor e Forma:Solid
    Peso molecular:459.446
  • Kynapcin-28

    CAS:
    <p>Kynapcin-28 is a non-competitive inhibitor of prolyl endopeptidase (PEP) with an IC50 of 76.80 μM and exhibits weak inhibitory effects on other serine proteases.</p>
    Fórmula:C19H12O10
    Cor e Forma:Solid
    Peso molecular:400.293
  • Deoxyradicinin

    CAS:
    <p>Deoxyradicinin is a biosynthetic precursor of Radicinin. It can inhibit Xylella fastidiosa and Liberibacter crescens, with a minimum inhibitory concentration (MIC) of 3.5 μg/mL against Liberibacter crescens. Deoxyradicinin is applicable for research on controlling plant diseases caused by these pathogens.</p>
    Fórmula:C12H12O4
    Cor e Forma:Solid
    Peso molecular:220.221
  • Cremeomycin

    CAS:
    <p>Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.</p>
    Fórmula:C8H6N2O4
    Cor e Forma:Solid
    Peso molecular:194.144
  • Polyozellin

    CAS:
    <p>Polyozellin is a prolyl endopeptidase inhibitor with properties effective against inflammation, cancer, and diseases related to oxidative stress.</p>
    Fórmula:C22H14O10
    Cor e Forma:Solid
    Peso molecular:438.341
  • Salfredin C1

    CAS:
    <p>Salfredin C1 is an inhibitor of aldose reductase.</p>
    Fórmula:C13H11NO6
    Cor e Forma:Solid
    Peso molecular:277.229
  • Phencomycin

    CAS:
    <p>Phencomycin exhibits mild activity against Gram-positive bacteria and inhibits physiologically important enzymes such as renin, with an IC50 of 440 μg/mL.</p>
    Fórmula:C15H10N2O4
    Cor e Forma:Solid
    Peso molecular:282.251
  • Diatretyne Ⅰ

    CAS:
    Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.
    Fórmula:C8H5NO3
    Cor e Forma:Solid
    Peso molecular:163.13
  • XR8-89

    CAS:
    <p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>
    Fórmula:C29H36N4O2S
    Cor e Forma:Solid
    Peso molecular:504.69
  • Crotocin

    CAS:
    <p>Crotocin exhibits bactericidal activity against Cryptococcus neoformans, Candida albicans, and Saccharomyces cerevisiae (brewer’s yeast), but it can be inactivated by blood.</p>
    Fórmula:C19H24O5
    Cor e Forma:Solid
    Peso molecular:332.391
  • SAR107375

    CAS:
    <p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>
    Fórmula:C24H30ClN5O5S2
    Cor e Forma:Solid
    Peso molecular:568.11
  • Enactin Ia

    CAS:
    <p>Enactin Ia is found in Streptomyces roseoviridis and exhibits mild antibacterial activity.</p>
    Fórmula:C20H38N2O6
    Cor e Forma:Solid
    Peso molecular:402.526
  • Kurasoin A

    CAS:
    <p>Kurasoin A is an inhibitor of the enzyme farnesyltransferase.</p>
    Fórmula:C16H16O3
    Cor e Forma:Solid
    Peso molecular:256.296
  • Piloquinone

    CAS:
    <p>Piloquinone is a type of phenanthrene compound that exhibits mild inhibitory effects on mycobacteria and protozoa.</p>
    Fórmula:C21H20O5
    Cor e Forma:Solid
    Peso molecular:352.38
  • Azirinomycin

    CAS:
    <p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C4H5NO2
    Cor e Forma:Solid
    Peso molecular:99.088
  • ZK159222

    CAS:
    <p>ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.</p>
    Fórmula:C32H48O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:512.72
  • 1-Deamino-1-hydroxysagamicin

    CAS:
    <p>1-Deamino-1-hydroxysagamicin (AntibioticSUM-3) is an aminoglycoside antibiotic that is effective against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C20H40N4O8
    Cor e Forma:Solid
    Peso molecular:464.554
  • Symplostatin 1

    CAS:
    <p>Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.</p>
    Fórmula:C43H70N6O6S
    Cor e Forma:Solid
    Peso molecular:799.12
  • GNE-616

    CAS:
    <p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>
    Fórmula:C24H23F4N5O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:537.53
  • Pyrrolomycin A

    CAS:
    <p>Pyrrolomycin A is a pyrrole antibiotic that exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>
    Fórmula:C4H2Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:180.977
  • NSC 357754

    CAS:
    <p>NSC 357754 is an inhibitor of Claudin. It can enhance transepithelial electrical resistance and reduce specific cation permeability. NSC 357754 is useful for research involving Claudin-2 and/or Claudin-15 mediated intestinal disorders.</p>
    Fórmula:C26H20N4O2
    Cor e Forma:Solid
    Peso molecular:420.463
  • DMP-728 free base

    CAS:
    <p>DMP-728 free base is a highly potent and selective GPIIbDIIa antagonist</p>
    Fórmula:C25H36N8O7
    Cor e Forma:Solid
    Peso molecular:560.60
  • O-Desmethyl Midostaurin

    CAS:
    <p>O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.</p>
    Fórmula:C34H28N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:556.61
  • Miyakamide A2

    CAS:
    <p>Miyakamide A2 is an antibiotic with insecticidal properties. It inhibits the growth of brine shrimp and exhibits weak activity against Xanthomonas species. The IC50 for inhibiting P388 cells is 12.2 μg/mL.</p>
    Fórmula:C31H32N4O3
    Cor e Forma:Solid
    Peso molecular:508.611
  • Fluoropolyoxin L

    CAS:
    <p>Fluoropolyoxin L exhibits inhibitory activity against Escherichia coli and Enterococcus faecalis.</p>
    Fórmula:C16H22FN5O12
    Cor e Forma:Solid
    Peso molecular:495.371
  • NTPDase-IN-2

    CAS:
    <p>NTPDase-IN-2 inhibits h-NTPDase-2/-8 (IC50: 0.04, 2.27 µM), non-competitive for h-NTPDase-1/-2 (Km: 74 µM); useful in cancer, immune, bacterial research.</p>
    Fórmula:C24H20FN3OS2
    Cor e Forma:Solid
    Peso molecular:449.56
  • Dephostatin

    CAS:
    <p>Dephostatin is a competitive protein tyrosine phosphatase (PTP) inhibitor isolated from Streptomyces spp., exhibiting activity within the micromolar range.</p>
    Fórmula:C7H8N2O3
    Cor e Forma:Solid
    Peso molecular:168.15
  • 3HKT-IN-1

    CAS:
    <p>3HKT-IN-1 (Compound 17122279) is an inhibitor of Anopheles gambiae 3-hydroxykynurenine transaminase (3HKT) and is utilized in malaria research.</p>
    Fórmula:C12H11BrN2O3
    Cor e Forma:Solid
    Peso molecular:311.131
  • Peptaibolin

    CAS:
    <p>Peptaibolin exhibits activity against Gram-positive bacteria and yeast. The minimum inhibitory concentration (MIC) for its effect on Bacillus subtilis [ATCC 6633] and Candida albicans is 100 μg/mL.</p>
    Fórmula:C31H51N5O6
    Cor e Forma:Solid
    Peso molecular:589.77
  • Tzc 5665

    CAS:
    <p>Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.</p>
    Fórmula:C31H38ClN5O7
    Cor e Forma:Solid
    Peso molecular:628.12
  • PCTR1

    CAS:
    <p>PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.</p>
    Fórmula:C32H47N3O9S
    Cor e Forma:Solid
    Peso molecular:649.8
  • Megovalicin A

    CAS:
    <p>Megovalicin A is effective against Bacillus subtilis and Escherichia coli.</p>
    Fórmula:C35H63NO8
    Cor e Forma:Solid
    Peso molecular:625.88
  • 20-Deoxysalinomycin

    CAS:
    <p>20-Deoxysalinomycin primarily targets Gram-positive bacteria, with a particular effectiveness against poultry coccidia.</p>
    Fórmula:C42H70O10
    Cor e Forma:Solid
    Peso molecular:735.00
  • VU6028418


    <p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>
    Cor e Forma:Liquid
  • Pradimicin B

    CAS:
    <p>Pradimicin B is an antibiotic with potent antifungal and anti-yeast activities.</p>
    Fórmula:C35H36N2O14
    Cor e Forma:Solid
    Peso molecular:708.665
  • Calphostin D

    CAS:
    <p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>
    Fórmula:C30H30O10
    Cor e Forma:Solid
    Peso molecular:550.55
  • BSc5367

    CAS:
    <p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>
    Fórmula:C20H15N3O2
    Cor e Forma:Soild
    Peso molecular:329.35
  • Exfoliazone

    CAS:
    <p>Exfoliazone is a phenazinic antibiotic with activity against Trichoderma viride, exhibiting an ED50 for inhibiting mycelial growth of 70 μg/mL.</p>
    Fórmula:C15H12N2O4
    Cor e Forma:Solid
    Peso molecular:284.267
  • Dynemicin Q

    CAS:
    <p>Dynemicin Q is an antibiotic that demonstrates potent activity against Gram-positive bacteria.</p>
    Fórmula:C28H19NO9
    Cor e Forma:Solid
    Peso molecular:513.45
  • Hydrolyzed Fumonisin B2

    CAS:
    <p>Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.</p>
    Fórmula:C22H47NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.61
  • AN-12-H5

    CAS:
    <p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>
    Fórmula:C24H23N3O4S3
    Cor e Forma:Solid
    Peso molecular:513.65
  • Sulprostone

    CAS:
    <p>EP3 and EP1 receptor agonist</p>
    Fórmula:C23H31NO7S
    Pureza:98%
    Cor e Forma:White To Off-White Solid
    Peso molecular:465.56
  • Prohibitin ligand 1


    <p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>
    Fórmula:C20H22N2O
    Cor e Forma:Solid
    Peso molecular:306.4
  • Pyridoxatin

    CAS:
    <p>Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.</p>
    Fórmula:C15H21NO3
    Cor e Forma:Solid
    Peso molecular:263.33
  • Celesticetin B

    CAS:
    <p>Celesticetin B is an antibiotic primarily exhibiting antibacterial activity against Gram-positive microorganisms.</p>
    Fórmula:C21H38N2O8S
    Cor e Forma:Solid
    Peso molecular:478.6
  • (1R,3S)-THCCA-Asn


    <p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>
    Fórmula:C24H24N4O6
    Cor e Forma:Solid
    Peso molecular:464.47
  • Leucomycin U

    CAS:
    <p>Leucomycin U is a macrolide antibiotic. It demonstrates significant activity against Gram-positive bacteria and also exhibits effects on spirochetes, rickettsiae, and chlamydiae.</p>
    Fórmula:C37H61NO14
    Cor e Forma:Solid
    Peso molecular:743.878
  • Gilvusmycin

    CAS:
    <p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>
    Fórmula:C38H34N6O8
    Cor e Forma:Solid
    Peso molecular:702.712
  • Unoprostone

    CAS:
    <p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>
    Fórmula:C22H38O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:382.53
  • Atiratecan

    CAS:
    <p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>
    Fórmula:C31H34N6O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:586.64
  • Thielavin B

    CAS:
    <p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>
    Fórmula:C31H34O10
    Cor e Forma:Solid
    Peso molecular:566.6
  • PRN694

    CAS:
    <p>PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.</p>
    Fórmula:C28H35F2N5O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:543.67
  • SSTR5 antagonist 2 TFA

    CAS:
    <p>Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.</p>
    Fórmula:C34H36F4N2O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:660.65
  • MK-8970


    <p>MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.</p>
    Fórmula:C25H29FN6O8
    Cor e Forma:Solid
    Peso molecular:560.54
  • 2-Hydroxy-5-iminoazacyclopent-3-ene

    CAS:
    <p>2-Hydroxy-5-iminoazacyclopent-3-ene is a pyrroline-class antibiotic with mild activity against both Gram-positive and Gram-negative bacteria.</p>
    Fórmula:C4H6N2O
    Cor e Forma:Solid
    Peso molecular:98.103
  • AMPK Activator SC4

    CAS:
    <p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>
    Fórmula:C26H18ClN3O4
    Cor e Forma:Solid
    Peso molecular:471.89