
Receptores acoplados a G-proteína e Receptores 7-TM
Os receptores acoplados à proteína G (GPCRs) e os receptores de 7-transmembrana (7-TM) são uma grande família de proteínas de membrana que desempenham papéis fundamentais na comunicação celular e na transdução de sinais. Esses receptores estão envolvidos em uma ampla gama de processos fisiológicos, incluindo percepção sensorial, resposta imunológica e regulação hormonal. Os GPCRs são alvos principais na descoberta de medicamentos, tornando-os essenciais para a pesquisa em farmacologia e medicina. Na CymitQuimica, oferecemos uma ampla seleção de reagentes e compostos de alta qualidade relacionados a GPCRs e receptores 7-TM para apoiar sua pesquisa e esforços de desenvolvimento de medicamentos.
Foram encontrados 6050 produtos para "Receptores acoplados a G-proteína e Receptores 7-TM".
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Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:384.9Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Fórmula:C31H33N3O4Pureza:99.66%Cor e Forma:SolidPeso molecular:511.6114Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFórmula:C17H20ClN3Pureza:98% - 99.53%Cor e Forma:White SolidPeso molecular:301.814Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Fórmula:C19H26ClNO2Pureza:99.35%Cor e Forma:White SolidPeso molecular:335.87Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White SolidPeso molecular:463.787Cefaclor monohydrate
CAS:Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.Fórmula:C15H16ClN3O5SPureza:97.36% - 99.9%Cor e Forma:White SolidPeso molecular:385.823Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Cor e Forma:White SolidPeso molecular:448.385(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H10FNO2Pureza:97.82%Cor e Forma:SolidPeso molecular:195.1903Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Cor e Forma:SolidPeso molecular:408.33Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Fórmula:C14H15Cl2NSPureza:99.83% - 99.97%Cor e Forma:White PowderPeso molecular:300.247Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Fórmula:C23H30FN3Pureza:99.85% - 99.99%Cor e Forma:SolidPeso molecular:367.50Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:SolidPeso molecular:522.55AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Fórmula:C17H14O5Pureza:97.07%Cor e Forma:SolidPeso molecular:298.29Ref: TM-T14148
1mg34,00€5mg63,00€1mL*10mM (DMSO)67,00€10mg92,00€25mg165,00€50mg250,00€100mg401,00€200mg580,00€Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Cor e Forma:White SolidPeso molecular:434.41Ref: TM-T1077
1mL*10mM (DMSO)35,00€10mg49,00€25mg65,00€50mg80,00€100mg109,00€200mg161,00€500mg263,00€Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Fórmula:C25H37NO4Pureza:99.2% - 99.9%Cor e Forma:SolidPeso molecular:415.5656Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White SolidPeso molecular:341.43Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Fórmula:C22H23N3O2Pureza:99.29% - 99.97%Cor e Forma:White SolidPeso molecular:361.4369Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H11ClFNO2Pureza:99.98%Cor e Forma:SolidPeso molecular:231.651Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Cor e Forma:SolidPeso molecular:307.3895Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Cor e Forma:SolidPeso molecular:266.55
