Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
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Benserazide
CAS:<p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>Fórmula:C10H15N3O5Cor e Forma:SolidPeso molecular:257.24Fidarestat
CAS:<p>Fidarestat (SNK 860),Aldose reductase inhibitor (IC50=26 nM). Targets AKR1B10 (33 μM) and V301L AKR1B10 (1.8 μM). Potential diabetes treatment.</p>Fórmula:C12H10FN3O4Pureza:98%Cor e Forma:SolidPeso molecular:279.22Quinfamide
CAS:<p>Quinfamide is a compound with the potential to treat tropical parasitic infections such as Amoebiasis and Helminthiasis.</p>Fórmula:C16H13Cl2NO4Pureza:99.92%Cor e Forma:SolidPeso molecular:354.18Diethyl pyimDC
CAS:<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Fórmula:C14H15N3O4Cor e Forma:SolidPeso molecular:289.29Quoromycin
CAS:<p>Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.</p>Fórmula:C12H8N2O2SCor e Forma:SolidPeso molecular:244.27Distigmine Bromide
CAS:<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Fórmula:C22H32BrN4O4Pureza:98%Cor e Forma:SolidPeso molecular:496.42Carisbamate
CAS:<p>CarisbAMate (JNJ-10234094, RWJ 333369, YKP-509) is an antiepileptic drug candidate.</p>Fórmula:C9H10ClNO3Cor e Forma:SolidPeso molecular:215.63CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Fórmula:C12H14ClN3OPureza:98%Cor e Forma:SolidPeso molecular:251.71Isothipendyl
CAS:Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.Fórmula:C16H19N3SCor e Forma:SolidPeso molecular:285.41BR351 precursor
CAS:<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C27H32N2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:576.68Vandetanib Fumarate
CAS:<p>Oral tyrosine kinase inhibitor Vandetanib Fumarate targets RET, VEGFRs, EGFR in thyroid cancer.</p>Fórmula:C26H28BrFN4O6Pureza:98%Cor e Forma:SolidPeso molecular:591.43Moricizine
CAS:<p>Moricizine is an antiarrhythmia agent which is used primarily for ventricular rhythm disturbances.</p>Fórmula:C22H25N3O4SPureza:98%Cor e Forma:SolidPeso molecular:427.52Levomepromazine Maleate
CAS:<p>Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.</p>Fórmula:C23H28N2O5SCor e Forma:SolidPeso molecular:444.546Arasertaconazole
CAS:<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Fórmula:C20H15Cl3N2OSCor e Forma:SolidPeso molecular:437.77Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Cor e Forma:SolidPeso molecular:481.56Atomoxetine
CAS:<p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>Fórmula:C17H21NOPureza:98%Cor e Forma:SolidPeso molecular:255.35PTIQ
CAS:<p>MMP-3 expression inhibitor</p>Fórmula:C13H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:235.28Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Cor e Forma:SolidPeso molecular:264.36Pridinol
CAS:<p>Pridinol is an antispasmodic and muscle relaxant.</p>Fórmula:C20H25NOPureza:98%Cor e Forma:Crystals SolidPeso molecular:295.42(S)-Terazosin
CAS:<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43RS-104966
CAS:<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Fórmula:C19H21NO6SPureza:98%Cor e Forma:SolidPeso molecular:391.44TAPI-1
CAS:<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Fórmula:C26H37N5O5Pureza:≥95%Cor e Forma:SolidPeso molecular:499.6ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Fórmula:C15H16ClNO3S2Pureza:99.49%Cor e Forma:SolidPeso molecular:357.88Evogliptin HCl
CAS:<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Fórmula:C19H27ClF3N3O3Cor e Forma:SolidPeso molecular:437.88Safironil
CAS:<p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>Fórmula:C15H23N3O4Pureza:99.83%Cor e Forma:SolidPeso molecular:309.36Cycloguanil
CAS:<p>Cycloguanil is an antimalarial.</p>Fórmula:C11H14ClN5Pureza:98%Cor e Forma:SolidPeso molecular:251.72Lorbamate
CAS:<p>Carbamate is a type of carbamate that has been studied as a muscle relaxant and sedative.</p>Fórmula:C12H22N2O4Cor e Forma:SolidPeso molecular:258.31(R)-Praziquantel
CAS:<p>(R)-Praziquantel is an active enantiomer of praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:312.41AZD5248
CAS:<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Fórmula:C22H22N4O2Cor e Forma:SolidPeso molecular:374.44Otamixaban
CAS:<p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>Fórmula:C25H26N4O4Pureza:98.08%Cor e Forma:SolidPeso molecular:446.5Phenindamine Tartrate
CAS:<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Fórmula:C23H25NO6Cor e Forma:SolidPeso molecular:411.454Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Fórmula:C23H31N3NaO4S2Pureza:98%Cor e Forma:SolidPeso molecular:500.63Gemigliptin Tartrate(911637-19-9 free base)
CAS:<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Fórmula:C22H25F8N5O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:639.45Ketotifen
CAS:<p>Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.</p>Fórmula:C19H19NOSCor e Forma:SolidPeso molecular:309.43Indisetron Dihydrochloride
CAS:<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Fórmula:C17H24ClN5OCor e Forma:SolidPeso molecular:349.86Ivabradine
CAS:<p>Ivabradine: oral HCN blocker, lowers heart rate without affecting blood pressure, has anticonvulsant and anti-anginal properties.</p>Fórmula:C27H36N2O5Cor e Forma:SolidPeso molecular:468.59Selatinib
CAS:<p>Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer activity that inhibits the growth of NCI-N87 tumor cells.</p>Fórmula:C29H26ClFN4O3SPureza:98.00%Cor e Forma:SolidPeso molecular:565.06Vasicinone
CAS:<p>Vasicinone may act as a hepatoprotective agent.</p>Fórmula:C11H10N2O2Pureza:98.06%Cor e Forma:SolidPeso molecular:202.21Rolapitant
CAS:<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Fórmula:C25H26F6N2O2Pureza:99.86%Cor e Forma:SolidPeso molecular:500.48Protriptyline
CAS:<p>Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.</p>Fórmula:C19H21NCor e Forma:SolidPeso molecular:263.38BR351
CAS:<p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C20H25FN2O5SPureza:98%Cor e Forma:SolidPeso molecular:424.49(S)-Propafenone
CAS:<p>(S)-Propafenone, or (S)-SA-79, is an S-enantiomer with beta-blocking effects and sodium channel blocking class 1 antiarrhythmic properties.</p>Fórmula:C21H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:341.44Lanicemine
CAS:<p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>Fórmula:C13H14N2Pureza:98%Cor e Forma:SolidPeso molecular:198.26Ingavirin
CAS:<p>Ingavirin, a novel inhibitor of the influenza virus reproduction, inhubits the formation of the virus specific hemagglutinin.</p>Fórmula:C10H15N3O3Pureza:98%Cor e Forma:SolidPeso molecular:225.24NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Fórmula:C13H20N2O5SPureza:98.41%Cor e Forma:SolidPeso molecular:316.37Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Fórmula:C23H19ClO3SPureza:98%Cor e Forma:SolidPeso molecular:410.91Daltroban
CAS:<p>Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist.</p>Fórmula:C16H16ClNO4SPureza:99.74%Cor e Forma:SolidPeso molecular:353.82WAY 629
CAS:<p>WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.</p>Fórmula:C15H18N2Cor e Forma:SolidPeso molecular:226.32cis-Tadalafil
CAS:<p>Cis-Tadalafil is a potent inhibitor of phosphodiesterase 5, which is used to treat erectile dysfunction (ED) and primary pulmonary hypertension (PPH). It works by increasing blood flow to the penis, allowing men with ED to achieve and maintain an erection. Cis-Tadalafil is also used to treat symptoms of prostatic hyperplasia (enlarged prostate) in men. This drug has been shown to be effective in treating PPH by reducing pulmonary arterial pressure and improving exercise capacity. Cis-Tadalafil belongs to the carboline class of drugs and is a phosphodiesterase 5 inhibitor that selectively inhibits cGMP-specific phosphodiesterase type 5 (PDE5). This drug has been shown to be highly effective in treating both ED and PPH with minimal side effects.</p>Fórmula:C22H19N3O4Pureza:Min. 95%Cor e Forma:White/Off-White SolidPeso molecular:389.4 g/molNifekalant hydrochloride
CAS:<p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>Fórmula:C19H28ClN5O5Pureza:99.91%Cor e Forma:SolidPeso molecular:441.91Hemustine
CAS:<p>Hemustine is an inhibitor of human glutathione reductase and widely used as an anti-tumor agent.</p>Fórmula:C5H10ClN3O3Cor e Forma:SolidPeso molecular:195.6PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Cor e Forma:SolidPeso molecular:464.96Indenolol
CAS:<p>Indenolol is a blocker of beta-adrenergic.</p>Fórmula:C15H21NO2Pureza:98%Cor e Forma:SolidPeso molecular:247.33Tropatepine
CAS:<p>Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.</p>Fórmula:C22H23NSCor e Forma:SolidPeso molecular:333.49Ivaltinostat
CAS:<p>CG-200745 is a potent inhibitor of HDAC. CG200745 induces apoptosis and also inhibits the deacetylation of histone H3 and tubulin.</p>Fórmula:C24H33N3O4Pureza:98%Cor e Forma:SolidPeso molecular:427.54Metaproterenol
CAS:<p>Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).</p>Fórmula:C11H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:211.26(R)-Carvedilol
CAS:<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:SolidPeso molecular:406.47(S)-Hydroxychloroquine
CAS:(S)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine shows efficiently inhibits SARS-CoV-2 infection in vitro.Fórmula:C18H26ClN3OPureza:98%Cor e Forma:SolidPeso molecular:335.87Oxolamine
CAS:<p>Oxolamine is an agent of a cough suppressant.</p>Fórmula:C14H19N3OPureza:98%Cor e Forma:SolidPeso molecular:245.32Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Fórmula:C22H24ClF4NO2Cor e Forma:SolidPeso molecular:445.88Hexazinone
CAS:<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Fórmula:C12H20N4O2Pureza:99.99%Cor e Forma:SolidPeso molecular:252.31Clencyclohexerol
CAS:<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:319.23Piribedil dihydrochloride
CAS:<p>dopamine agonist</p>Fórmula:C16H20Cl2N4O2Pureza:98%Cor e Forma:SolidPeso molecular:371.26Bornaprine
CAS:<p>Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.</p>Fórmula:C21H31NO2Cor e Forma:SolidPeso molecular:329.48Afacifenacin
CAS:<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Fórmula:C27H26F3N3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:481.51Robenidine
CAS:<p>Robenidine, an anticoccidial guanidine, is used as an additive in rabbit fodder.</p>Fórmula:C15H13Cl2N5Pureza:98%Cor e Forma:SolidPeso molecular:334.2Esreboxetine
CAS:<p>Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.</p>Fórmula:C19H23NO3Cor e Forma:SolidPeso molecular:313.39Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Cor e Forma:White To Pink PowderPeso molecular:291.39Procarbazine free base
CAS:<p>Procarbazine: chemo drug for Hodgkin's, brain cancer; liver-activated; MAO inhibitor.</p>Fórmula:C12H19N3OPureza:98%Cor e Forma:SolidPeso molecular:221.3Mesopram
CAS:<p>PDE4 inhibitor, orally active</p>Fórmula:C14H19NO4Pureza:98%Cor e Forma:SolidPeso molecular:265.3Amorolfine
CAS:<p>Amorolfine is available in the nail lacquer and can be used to treat fungal nail infections.</p>Fórmula:C21H35NOCor e Forma:White To Off-White Crystalline PowderPeso molecular:317.517ND-336
CAS:<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Fórmula:C16H18ClNO3S2Cor e Forma:SolidPeso molecular:371.9(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Cor e Forma:SolidPeso molecular:398.34Sarafloxacin
CAS:<p>Sarafloxacin (A56620) has antibacterial activities against Gram-positive and Gram-negative bacteria.</p>Fórmula:C20H17F2N3O3Pureza:98.07% - 98.94%Cor e Forma:SolidPeso molecular:385.36Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Fórmula:C21H25NOPureza:98%Cor e Forma:SolidPeso molecular:307.43TAK-875 Hemihydrate
CAS:<p>TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.</p>Fórmula:C29H32O7SH2OPureza:98%Cor e Forma:SolidPeso molecular:533.63U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Cor e Forma:SolidPeso molecular:448.56Niclosamide monohydrate
CAS:<p>Niclosamide Monohydrate is used for the treatment of most tapeworm infections by inhibiting DNA replication.</p>Fórmula:C13H10Cl2N2O5Pureza:98%Cor e Forma:SolidPeso molecular:345.14Anitrazafen
CAS:<p>Anitrazafen is a locally effective anti-inflammatory agent that has been shown to have COX-2 inhibitor activity.</p>Fórmula:C18H17N3O2Pureza:98%Cor e Forma:SolidPeso molecular:307.35Propiomazine
CAS:<p>Propiomazine is an orally active antihistamine compound with sedative properties, useful for controlling insomnia in neurological disorders.</p>Fórmula:C20H24N2OSPureza:98.5%Cor e Forma:SolidPeso molecular:340.48Bifeprunox
CAS:<p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>Fórmula:C24H23N3O2Pureza:98%Cor e Forma:SolidPeso molecular:385.46Eltenac
CAS:<p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>Fórmula:C12H9Cl2NO2SPureza:98.53%Cor e Forma:SolidPeso molecular:302.18(R,R)-Montelukast bis-sulfide
CAS:<p>(R,R)-Montelukast bis-sulfide is a drug product that is used in the analytical and research and development of drugs. It is also used as an impurity standard for HPLC. (R,R)-Montelukast bis-sulfide has been shown to have niche applications in drug development and research, as well as being a high purity API.</p>Fórmula:C41H46ClNO5S2Pureza:90%MinPeso molecular:732.39 g/mol(S)-Rabeprazole sodium
CAS:<p>(S)-Rabeprazole sodium is an anticancer drug that acts as a kinase inhibitor. It is an analog of Rabeprazole and has been shown to inhibit the growth of cancer cells in vitro and in vivo. (S)-Rabeprazole sodium inhibits the activity of kinases, which are enzymes that play a key role in cell signaling pathways. This inhibition leads to apoptosis, or programmed cell death, in cancer cells. (S)-Rabeprazole sodium has been tested against various types of cancer, including Chinese hamster ovary cells and tumor xenografts in mice. It has also been shown to inhibit elastin degradation, which is important for preventing metastasis of cancer cells. (S)-Rabeprazole sodium may be a promising candidate for the development of new anticancer drugs that target specific kinases and proteins involved in cancer cell growth and survival.</p>Fórmula:C18H21N3O3S•NaPureza:Min. 95%Peso molecular:382.43 g/molCyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Cor e Forma:SolidPeso molecular:323.46Moveltipril
CAS:<p>Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action.</p>Fórmula:C19H30N2O5SPureza:97.55% - 98.28%Cor e Forma:SolidPeso molecular:398.52Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Cor e Forma:SolidPeso molecular:381.44UNC0321
CAS:<p>UNC0321 is an effective inhibitor of histone methyltransferase G9a with a Ki of 63 pM and with IC50s 9 nM and 6 nM in ECSD and CLOT assays.</p>Fórmula:C27H45N7O3Pureza:99.80%Cor e Forma:SolidPeso molecular:515.69Gemigliptin
CAS:<p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>Fórmula:C18H19F8N5O2Pureza:99.72%Cor e Forma:SolidPeso molecular:489.363-Trifluoroacetylamino linagliptin
CAS:<p>Please enquire for more information about 3-Trifluoroacetylamino linagliptin including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C27H27F3N8O3Pureza:Min. 95%Peso molecular:568.55 g/molEzetimibe ketone
CAS:<p>Ezetimibe ketone is a lipid-lowering agent that inhibits cholesterol absorption through the inhibition of Niemann-Pick C1-like 1 (NPC1L1). Ezetimibe ketone is used to reduce the levels of low-density lipoprotein cholesterol (LDL-C) in patients with primary hypercholesterolemia, sitosterolemia, and familial combined hyperlipidemia. Ezetimibe ketone has been shown to be bioequivalent to ezetimibe, which is an oral drug that inhibits cholesterol absorption by blocking NPC1L1. The drug binds to the NPC1L1 receptor in the brush border membrane of enterocytes and prevents cholesterol uptake. Ezetimibe ketone has a high solubility in organic solvents such as dichloromethane or chloroform. It also has a high melting point, which makes it suitable for use on chromatographic columns.</p>Fórmula:C24H19F2NO3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:407.41 g/molPG-116800
CAS:<p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>Fórmula:C24H27N3O7SPureza:98.03% - 99.66%Cor e Forma:SolidPeso molecular:501.55Vildagliptin carboxylic acid methyl ester
CAS:<p>Please enquire for more information about Vildagliptin carboxylic acid methyl ester including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C18H28N2O4Pureza:Min. 95%Peso molecular:336.43 g/molAGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Fórmula:C18H17F2N3O2Pureza:98.92%Cor e Forma:SolidPeso molecular:345.34Roflumilast Impurity A
CAS:<p>Roflumilast impurity A is a metabolite of roflumilast. It is a drug product that is used as an analytical standard for the determination of roflumilast in HPLC analysis. Roflumilast impurity A is not natural and is synthetic. It has been shown to be a substrate for CYP1A2, CYP2C8, CYP2C9, and CYP3A4 enzymes. Studies have shown that it may be involved in the metabolism of roflumilast through hydroxylation and deamination.</p>Fórmula:C16H14Cl2N2O3Pureza:Min. 95%Peso molecular:353.2 g/molGallopamil
CAS:<p>Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.</p>Fórmula:C28H40N2O5Pureza:99.85%Cor e Forma:SolidPeso molecular:484.63Givinostat hydrochloride
CAS:<p>Givinostat HCl (ITF2357 HCl) inhibits HDAC1/3 (IC50: 198/157 nM) with anti-inflammatory, anti-angiogenic, and antineoplastic properties.</p>Fórmula:C24H28ClN3O4Pureza:99.39%Cor e Forma:SolidPeso molecular:457.95Ephedrine Hydrochloride
CAS:Produto ControladoEphedrine and its saltsFórmula:C10H15NO·HClCor e Forma:White Off-White PowderPeso molecular:201.09204DB04760
CAS:<p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>Fórmula:C22H20F2N4O2Pureza:99.93% - 99.99%Cor e Forma:SolidPeso molecular:410.42Fenoverine
CAS:<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Fórmula:C26H25N3O3SPureza:98.34%Cor e Forma:SolidPeso molecular:459.56
