Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Bupivacaine hydrochloride
CAS:<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Fórmula:C18H28N2O·HClPureza:99.9% - >99.99%Cor e Forma:SolidPeso molecular:324.89Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Cor e Forma:White SolidPeso molecular:332.87Topotecan hydrochloride
CAS:<p>Topotecan hydrochloride (NSC609699) is an antineoplastic agent used to treat ovarian cancer.</p>Fórmula:C23H24ClN3O5Pureza:97.88% - 99.41%Cor e Forma:White Crystalline SolidPeso molecular:457.92Praziquantel
CAS:<p>Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.</p>Fórmula:C19H24N2O2Pureza:99.67% - 99.69%Cor e Forma:SolidPeso molecular:312.41Sarafloxacin hydrochloride
CAS:<p>Sarafloxacin hydrochloride (A-56620 (hydrochloride)), a quinolone antibiotic drug, is a hydrochloride salt form of sarafloxacin.</p>Fórmula:C20H18ClF2N3O3Pureza:97.33% - 97.44%Cor e Forma:White To Yellow Crystalline SolidPeso molecular:421.83Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:383.51Mirodenafil
CAS:<p>Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>Fórmula:C26H37N5O5SPureza:99.89%Cor e Forma:SolidPeso molecular:531.67Elexacaftor
CAS:<p>Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.</p>Fórmula:C26H34F3N7O4SPureza:98.87% - 99.87%Cor e Forma:SolidPeso molecular:597.65Spirodiclofen
CAS:<p>Spirodiclofen (BAJ-2740), a selective acaricide from tetronic acid, resists cross-resistance, has insecticidal properties.</p>Fórmula:C21H24Cl2O4Pureza:99.94%Cor e Forma:White PowerPeso molecular:411.32Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:463.79Prazosin hydrochloride
CAS:<p>Prazosin HCl, a synthetic antiadrenergic, treats hypertension, heart failure, and more by relaxing blood vessels with an unclear mechanism.</p>Fórmula:C19H22ClN5O4Pureza:99.88% - >99.99%Cor e Forma:White To Tan Powder Off-White To Yellow PowderPeso molecular:419.86Gabapentin
CAS:<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Fórmula:C9H17NO2Pureza:99.55% - 99.91%Cor e Forma:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidPeso molecular:171.24Altretamine
CAS:<p>Altretamine (ENT-50852) is an alkylating agent with antineoplastic activity.</p>Fórmula:C9H18N6Pureza:99.54%Cor e Forma:Less Crystalline Solid Insoluble In Water (Ntp 1992) Physical Description Colorless Crystalline Solid Insoluble In Water (Ntp 1992)Peso molecular:210.28STL127705
CAS:<p>STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.</p>Fórmula:C22H20FN5O4Pureza:99.53% - 99.81%Cor e Forma:SolidPeso molecular:437.42Pyrimethamine
CAS:<p>Pyrimethamine (Pirimecidan) is a competitive inhibitor of dihydrofolate reductase (DHFR), used as an antimalarial drug.</p>Fórmula:C12H13ClN4Pureza:99.67%Cor e Forma:CrystalsPeso molecular:248.71Copanlisib dihydrochloride
CAS:<p>Copanlisib dihydrochloride: ATP-competitive PI3K inhibitor, potent for PI3Kα/δ/β/γ, antitumor, 2000x selectivity over other kinases except mTOR.</p>Fórmula:C23H30Cl2N8O4Pureza:99.05% - 99.16%Cor e Forma:SolidPeso molecular:553.44Niclosamide
CAS:<p>Niclosamide (Niclocide)(BAY2353) is used to treat most tapeworm infections by inhibiting DNA replication.</p>Fórmula:C13H8Cl2N2O4Pureza:98.47% - 99.1%Cor e Forma:Pale Yellow Crystals SolidPeso molecular:327.12Rupatadine Fumarate
CAS:<p>Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.</p>Fórmula:C26H26ClN3·C4H4O4Pureza:99.86%Cor e Forma:White Or Almost-White PowderPeso molecular:532.03Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Cor e Forma:Off-White SolidPeso molecular:406.86Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Fórmula:C17H22ClNOPureza:99.86%Cor e Forma:White SolidPeso molecular:291.82Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Cor e Forma:SolidPeso molecular:296.79Ranolazine dihydrochloride
CAS:<p>Ranolazine 2HCl, an antianginal, treats arrhythmia by inhibiting sodium current without changing blood pressure or heart rate.</p>Fórmula:C24H35Cl2N3O4Pureza:99.30% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:500.46Losartan potassium
CAS:<p>Losartan potassium (DuP-753 potassium) , an Angiotensin II Receptor Blocker, selectively and competitively blocks the binding of angiotensin II to the</p>Fórmula:C22H22ClKN6OPureza:99.9% - >99.99%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:461.01Chloramphenicol
CAS:<p>Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.</p>Fórmula:C11H12Cl2N2O5Pureza:99.6% - 99.84%Cor e Forma:Needles Or Elongated Plates From Water Or Ethylene Dichloride SolidPeso molecular:323.13Imrecoxib
CAS:<p>Imrecoxib (BAP-909) is a novel and selective cyclooxygenase 2 (COX-2) inhibitor (IC50: 18 nM).</p>Fórmula:C21H23NO3SPureza:99.87%Cor e Forma:SolidPeso molecular:369.48Incyclinide
CAS:<p>Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.</p>Fórmula:C19H17NO7Pureza:97.99%Cor e Forma:SolidPeso molecular:371.34Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Fórmula:C26H28Cl2F2N2Pureza:99.53% - 99.89%Cor e Forma:White Crystalline Powder Odorless And TastelessPeso molecular:477.42Meclofenoxate hydrochloride
CAS:<p>Meclofenoxate HCl (Lucidril) boosts memory and cognition; it's a DIMETHYLAMINOETHANOL and p-chlorophenoxyacetic acid ester.</p>Fórmula:C12H16ClNO3·HClPureza:97.05%Cor e Forma:White Crystal PowderPeso molecular:294.17Deferiprone
CAS:<p>Deferiprone (Deferidone) is an Iron Chelator. The mechanism of action of deferiprone is as an Iron Chelating Activity.</p>Fórmula:C7H9NO2Pureza:99.58% - ≥95%Cor e Forma:White NeedlesPeso molecular:139.15Labetalol hydrochloride
CAS:<p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>Fórmula:C19H25ClN2O3Pureza:99.54% - 99.85%Cor e Forma:SolidPeso molecular:364.87Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Fórmula:C26H35NO7Pureza:98.53% - 99.43%Cor e Forma:CoaPeso molecular:473.57Benzocaine
CAS:<p>Benzocaine is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.</p>Fórmula:C9H11NO2Pureza:99.16% - 99.88%Cor e Forma:Rhombohedra From Ether DrypowderPeso molecular:165.19Ribociclib succinate
CAS:<p>Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).</p>Fórmula:C27H36N8O5Pureza:99.9%Cor e Forma:SolidPeso molecular:552.63Diminazene Aceturate
CAS:<p>Diminazene is a trypanocidal agent.</p>Fórmula:C22H29N9O6Pureza:96.86% - 99.58%Cor e Forma:SolidPeso molecular:515.52Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55Sunitinib
CAS:<p>Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).</p>Fórmula:C22H27FN4O2Pureza:98% - 99.67%Cor e Forma:Yellow SolidPeso molecular:398.47Prochlorperazine Maleate
CAS:<p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>Fórmula:C28H32ClN3O8SPureza:99.78%Cor e Forma:Off-White PowderPeso molecular:606.09Nevirapine
CAS:<p>Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C15H14N4OPureza:99.58% - 99.59%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:266.3Tizanidine hydrochloride
CAS:<p>Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.</p>Fórmula:C9H9Cl2N5SPureza:99.96%Cor e Forma:Solid WhitePeso molecular:290.17Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Fórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:434.41Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Fórmula:C18H23Cl2NOPureza:98.04% - >99.99%Cor e Forma:Antihypertensive DrugPeso molecular:340.3Mefloquine
CAS:<p>Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor.</p>Fórmula:C17H16F6N2OPureza:99.89%Cor e Forma:SolidPeso molecular:378.31Opicapone
CAS:<p>Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).</p>Fórmula:C15H10Cl2N4O6Pureza:98.17% - 99.36%Cor e Forma:SolidPeso molecular:413.17Lomustine
CAS:<p>Lomustine (NSC-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.</p>Fórmula:C9H16ClN3O2Pureza:98.36% - 99.44%Cor e Forma:Solid SolidPeso molecular:233.7Phenothiazine
CAS:<p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>Fórmula:C12H9NSPureza:99.95%Cor e Forma:Yellow Solid PelletsPeso molecular:199.27Azelastine hydrochloride
CAS:<p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>Fórmula:C22H24ClN3O·HClPureza:98% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:418.36Phenformin
CAS:<p>Phenformin: a biguanide with anti-cancer, anti-glycemic effects, inhibits skin tumors, enhances keratinocyte differentiation/apoptosis.</p>Fórmula:C10H15N5Pureza:99.72%Cor e Forma:SolidPeso molecular:205.26Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Fórmula:C17H18F3NOPureza:99.07% - 99.28%Cor e Forma:SolidPeso molecular:309.33Pazopanib
CAS:<p>Pazopanib (GW786034) is an inhibitor of protein tyrosine kinases that inhibits VEGFR1/2/3. Pazopanib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C21H23N7O2SPureza:98.78% - 99.85%Cor e Forma:White PowderPeso molecular:437.52Clidinium bromide
CAS:<p>Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.</p>Fórmula:C22H26BrNO3Pureza:98.89% - 99.86%Cor e Forma:White Crystalline SolidPeso molecular:432.35
