Sais e Derivados de API
Os sais dos Ingredientes Farmacêuticos Ativos (API) são compostos formados pela reação de um ácido com uma base, resultando em um equilíbrio iônico. Esses sais frequentemente melhoram a solubilidade e a estabilidade dos APIs, facilitando sua absorção no organismo. Os derivados de API são variantes químicas de um princípio ativo que podem apresentar propriedades aprimoradas ou modificadas para otimizar a eficácia terapêutica. Os sais de APIs são utilizados na formulação de medicamentos orais, injetáveis e tópicos. Além disso, os derivados de API podem melhorar a farmacocinética dos fármacos, permitindo, por exemplo, a liberação controlada de substâncias ativas.
Na CymitQuimica, oferecemos sais e derivados de APIs com a pureza e qualidade necessárias para pesquisa e desenvolvimento de formulações farmacêuticas.
Foram encontrados 79376 produtos de "Sais e Derivados de API"
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GNE-8324
CAS:<p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>Fórmula:C18H18FN3OSPureza:98.68% - 99.34%Cor e Forma:SolidPeso molecular:343.42Dextromethorphan Related Compound A CI (3-Methoxy-9α,13α,14α-morphinan hydrochloride)
CAS:Produto ControladoCompounds containing a quinoline or isoquinoline ring-system, whether or not hydrogenated, not further fused, excluding drugs and pesticidesFórmula:C17H23NO·HClCor e Forma:White PowderPeso molecular:257.177964-PPBP maleate
CAS:<p>4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.</p>Fórmula:C25H31NO4Pureza:99.88%Cor e Forma:SolidPeso molecular:409.52Cathinone Hydrochloride CI (α-Aminopropiophenone hydrochloride)
CAS:Produto ControladoVegetable alkaloids, natural or reproduced by synthesis, their salts and other derivatives, nesoiFórmula:C9H11NO·HClCor e Forma:White PowderPeso molecular:149.08406Modafinil S-enantiomer CIV ((S)-2-(Benzhydrylsulfinyl)acetamide)
CAS:Produto ControladoOther aromatic organo-sulfur compounds (excluding pesticides)Fórmula:C15H15NO2SCor e Forma:White Off-White SolidPeso molecular:273.08235Aptiganel
CAS:<p>Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.</p>Fórmula:C20H21N3Pureza:98.13% - 98.90%Cor e Forma:SolidPeso molecular:303.4Tropicamide Related Compound D (2-Phenylacetic acid)
CAS:Produto ControladoPhenylacetic acid (alpha-toluic acid) and its saltsFórmula:C8H8O2Cor e Forma:Beige PowderPeso molecular:136.05243Oxacyclohexane open ring tacrolimus
CAS:<p>Please enquire for more information about Oxacyclohexane open ring tacrolimus including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C44H71NO13Pureza:Min. 95%Peso molecular:822.04 g/molDiphenoxylate Related Compound A CI (1-(3-Cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxylic acid)
CAS:Produto ControladoAlfentanil (inn), anileridine (inn), bezitramide (inn), bromazepam (inn), difenoxin (inn), diphenoxylate (inn), dipipanone (inn), fentanyl (inn), etc.Fórmula:C28H28N2O2Cor e Forma:PowderPeso molecular:424.21508Oxandrolone Related Compound B CIII (17 β-hydroxy-17 α-methyl-4-oxa-5 α-androsta-3-one)
CAS:Produto ControladoLactones, nesoiFórmula:C19H30O3Cor e Forma:Off-White Crystalline PowderPeso molecular:306.21949Benzaldehyde
CAS:Produto ControladoBenzaldehydeFórmula:C7H6OCor e Forma:Colorless LiquidPeso molecular:106.04186Morphine Related Compound A CI (7,8-Didehydro-4,5α-epoxy-17-methylmorphinan-3,6α-diol, N-oxide)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereofFórmula:C17H19NO4Cor e Forma:Yellow Tan PowderPeso molecular:301.13141Morphine Related Compound B CII (2,2'-Bimorphine trihydrate)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFórmula:C34H36N2O6·3H2OCor e Forma:White PowderPeso molecular:568.25734Apixaban Impurity 6
CAS:<p>Please enquire for more information about Apixaban Impurity 6 including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C26H26N4O5Pureza:Min. 95%Peso molecular:474.51 g/molOxymorphone Related Compound A CII (4,5α-Epoxy-3,14-dihydroxy-17-methylmorphinan-6-one N-oxide)
CAS:Produto ControladoConcentrates of poppy straw; buprenorphine (inn) codeine, dihydrocodeine (inn), ethylmorphine (inn), etorphine (inn), heroin, hydrococdone (inn), etc.Fórmula:C17H19NO5Cor e Forma:Off-White PowderPeso molecular:317.12632CNS-5161 hydrochloride
CAS:<p>CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.</p>Fórmula:C16H19Cl2N3S2Pureza:99.53%Cor e Forma:SolidPeso molecular:388.38Testosterone Enanthate Related Compound B CIII (Androst-4-en-3-one-17β-yl hexanoate)
CAS:Produto ControladoAdrenal cortical hormones and their derivatives nesoiFórmula:C25H38O3Cor e Forma:White PowderPeso molecular:386.2821Oxycodone Related Compound C CII (codeinone)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereofFórmula:C18H19NO3Cor e Forma:PowderPeso molecular:297.13649Codeine N-Oxide CI
CAS:Produto ControladoConcentrates of poppy straw; buprenorphine (inn) codeine, dihydrocodeine (inn), ethylmorphine (inn), etorphine (inn), heroin, hydrococdone (inn), etc.Fórmula:C18H21NO4Cor e Forma:Brown White PowderPeso molecular:315.14706Edoxaban
CAS:<p>Edoxaban: potent, selective FXa inhibitor; Ki 0.561 nM. Used as an oral anticoagulant for stroke prevention, also inhibits thrombin and FIXa.</p>Fórmula:C24H30ClN7O4SPureza:97.67% - 99.71%Cor e Forma:SolidPeso molecular:548.06Ro 25-6981
CAS:<p>Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.</p>Fórmula:C22H29NO2Pureza:99.88%Cor e Forma:SolidPeso molecular:339.47AMPA receptor antagonist-2
CAS:<p>AMPA receptor antagonist-2 is an AMPA receptor antagonist.</p>Fórmula:C18H17N3O4Pureza:98.76%Cor e Forma:SolidPeso molecular:339.35Apixaban Impurity 1
CAS:<p>Apixaban Impurity 1 is an impurity found in Apixaban, a drug used for the prevention of stroke. It is produced by condensation of 2-aminopyridine and 3-hydroxybenzaldehyde in ethanol with sodium hydroxide as a catalyst. The reaction proceeds via amination of the pyridine ring followed by transesterification. The yield of this impurity is low at about 4%.</p>Pureza:Min. 95%Testosterone Related Compound A CIII (Androst-4-ene-3,17-dione)
CAS:Produto ControladoAdrenal cortical hormones and their derivatives nesoiFórmula:C19H26O2Cor e Forma:PowderPeso molecular:286.19328Delucemine Hydrochloride
CAS:<p>Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.</p>Fórmula:C16H18ClF2NPureza:98.49% - 99.30%Cor e Forma:SolidPeso molecular:297.77Hydromorphone Related Compound A CII (7,8-didehydro-4,5α-epoxy-3-hydroxy-17-methylmorphinan-6-one perchlorate)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFórmula:C17H17NO3·HClO4Cor e Forma:Off-White Light Yellow PowderPeso molecular:383.07718Oxandrolone Related Compound A CIII (17β-hydroxy-17α-methyl-2-oxa-5α-androst-7-en-3-one)
CAS:Produto ControladoLactones nesoiFórmula:C19H28O3Cor e Forma:White Crystalline PowderPeso molecular:304.20384Fentanyl Related Compound E CII (N-Phenyl-1-(2-phenylethyl)-4-piperidinamine)
CAS:Produto Controlado4-anilino-n-phenethylpiperidine (anpp)Fórmula:C19H24N2Cor e Forma:White Light Brown Crystalline PowderPeso molecular:280.19395Dextroamphetamine Related Compound B CII (Phenyl acetone)
CAS:Produto ControladoPhenylacetone (phenylpropan-2-one)Fórmula:C9H10OCor e Forma:Clear Pale Yellow LiquidPeso molecular:134.07316N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide
CAS:<p>N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide is a cavity inhibitor that has inhibitory activity against polymerization. It also reacts with chloride and alkene, which can be used to synthesize an amide. N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide is reactive and has a hydroxyl group, which can react with methyl sulfone in the environment. This agent has been shown to have anticancer activity in cell lines and tumor models.</p>Fórmula:C12H9F3N2OPureza:Min. 95%Peso molecular:254.21 g/molZolpidem Impurities Mixture CIV
Produto ControladoDiagnostic or lab reagents on a backing, prepared diagnostic or lab reagents whether or not on a backing, whether or not in the form of kits, nesoiCor e Forma:Powder2',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine
CAS:<p>2',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine is a cytosine analog that is used as an industrial chemical. It is prepared by the reaction of 5'-deoxycytidine with acetic anhydride in the presence of sodium bicarbonate, followed by a purification procedure. 2',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine reacts with toluene and trifluoromethanesulfonic acid to form 2',3'-di-O-acetyl 5'-deoxyfluorocytidine. This compound can be converted to 5'-deoxyfluorocytosine by heating in the presence of sodium tetrachloride. The yield for this process is high.</p>Fórmula:C13H16FN3O6Pureza:Min. 95%Peso molecular:329.29 g/molBenzphetamine Related Compound A CIII ((R)-N-Benzyl-N-methyl-1-phenylpropan-2-amine hydrochloride)
CAS:Produto Controlado<p>Aromatic monoamines not elsewhere specified or included and their derivatives, salts therof</p>Fórmula:C17H21N·HClCor e Forma:White Off-White PowderPeso molecular:275.14408Selurampanel
CAS:<p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>Fórmula:C16H19N5O4SPureza:99.60% - 99.78%Cor e Forma:SolidPeso molecular:377.42Trospium Chloride Related Compound A (Benzilic Acid)
CAS:Carboxylic acids w/ alcohol function but w/o other oxygen function and their derivatives, nesoiFórmula:C14H12O3Cor e Forma:White PowderPeso molecular:228.07864ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
CAS:<p>Please enquire for more information about ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C22H22N4O4Pureza:Min. 95%Peso molecular:406.43 g/molNeboglamine hydrochloride
CAS:<p>Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.</p>Fórmula:C13H25ClN2O3Pureza:99.19%Cor e Forma:SolidPeso molecular:292.8Testosterone Enanthate Related Compound H CIII (Androst-5-ene-3β,17β-diyl diheptanoate)
CAS:Produto ControladoAdrenal cortical hormones and their derivatives nesoiFórmula:C33H54O4Cor e Forma:White Solid PowderPeso molecular:514.40221Naloxone Related Compound D CII (4,5α-Epoxy-3,14-dihydroxy-17-(prop-2-enyl)morphinan-7-ene-6-one)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFórmula:C19H19NO4Cor e Forma:Light Yellow PowderPeso molecular:325.13141Exemestane Related Compound C CIII (androsta-1,4-diene-3,17-dione)
CAS:Produto ControladoAdrenal cortical hormones and their derivatives nesoiFórmula:C19H24O2Cor e Forma:White PowderPeso molecular:284.17763Hydrocodone Related Compound A CII (4-hydroxy-3-methoxy-17-methylmorphinan-6-one)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereofFórmula:C18H23NO3Cor e Forma:White PowderPeso molecular:301.16779Hydromorphone N-Oxide Hydrochloride CII (4,5α-Epoxy-3-hydroxy-17-methylmorphinan-6-one N-oxide, hydrochloride)
CAS:Produto Controlado<p>Alkaloids of opium and their derivatives, salts thereof</p>Fórmula:C17H19NO4·HClCor e Forma:Off-White PowderPeso molecular:337.79AV-101
CAS:<p>AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.</p>Fórmula:C10H11ClN2O3Pureza:97.78% - 98.27%Cor e Forma:SolidPeso molecular:242.66Noroxymorphone Hydrochloride CII (4,5α-Epoxy-3,14-dihydroxymorphinan-6-one hydrochloride)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFórmula:C16H18NO4ClCor e Forma:Light Brown PowderPeso molecular:323.09244Clopidogrel EP Impurity B hydrochloride
CAS:<p>Please enquire for more information about Clopidogrel EP Impurity B hydrochloride including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C16H16ClNO2S•HClPureza:Min. 95%Peso molecular:358.28 g/molMibampator
CAS:<p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>Fórmula:C21H30N2O4S2Pureza:99.34%Cor e Forma:SolidPeso molecular:438.6TAK-137
CAS:<p>TAK-137 is an AMPA receptor enhancer with antidepressant effects. TAK-137 has the ability to improve cognition and could be used to study schizophrenia.</p>Fórmula:C19H16N2O3SPureza:99.18%Cor e Forma:SolidPeso molecular:352.41Zopiclone R-Isomer CIV ((-)-(5R)-6-(5-Chloropyridin-2-yl)-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-yl 4-methylpiperazine-1-carboxylate)
CAS:Produto ControladoLactams, nesoiFórmula:C17H17ClN6O3Cor e Forma:Light Brown SolidPeso molecular:388.10507Naltrexone Related Compound A CII (17-(But-3-en-1-yl)-4,5α-epoxy-3,14-dihydroxymorphinan-6-one hydrochloride)
CAS:Produto ControladoAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFórmula:C20H23NO4·HClCor e Forma:Off-White PowderPeso molecular:341.16271Fentanyl Related Compound G CI (N-(1-Phenethylpiperidin-4-yl)-N-phenylacetamide)
CAS:Produto Controlado<p>Fentanyls and their derivatives containing an unfused pyrazole ring, whether or not hydrogenated, nesoi</p>Fórmula:C21H26N2OCor e Forma:White PowderPeso molecular:322.45Oxandrolone Related Compound C CIII (17,17-dimethyl-18-nor-2-oxa-5α-androst-13-en-3-one)
Produto ControladoLactones nesoiFórmula:C19H28O2Cor e Forma:PowderPeso molecular:288.42TAK-653
CAS:<p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>Fórmula:C19H23N3O3SPureza:99.89%Cor e Forma:SolidPeso molecular:373.47Minodronic acid
CAS:Minodronic acid (YM-529) is a P2X2/3 antagonist with anticancer properties, inhibiting cell growth and metastasis, and used in osteoporosis research.Fórmula:C9H12N2O7P2Pureza:98.02%Cor e Forma:SolidPeso molecular:322.15PF-4778574
CAS:<p>PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).</p>Fórmula:C19H22N2O3S2Pureza:98%Cor e Forma:SolidPeso molecular:390.52Nevadistinel
CAS:<p>Nevadistinel (NYX-458; NYX-3054) is a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, indicated for mitigating cognitive deficits</p>Fórmula:C15H18N2O3Pureza:98%Cor e Forma:SolidPeso molecular:274.32AMPA receptor modulator-5
CAS:<p>AMPA Receptor Modulator-5 (Example 217) serves as an AMPA receptor modulator, utilized in neurological disease research [1].</p>Fórmula:C20H12F4N6Pureza:98%Cor e Forma:SolidPeso molecular:412.34AMPA receptor modulator-6
CAS:<p>AMPA receptor modulator-6, an AMPA receptor positive allosteric modulator (PAM), is utilized in the research of neurological diseases [1].</p>Fórmula:C24H36N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:480.68Risevistinel
CAS:<p>Risevistinel (NYX-783), a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, may mitigate cognitive deficits in neurodegenerative</p>Fórmula:C14H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:297.35Naspm trihydrochloride
CAS:<p>Naspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride) is a synthetic analogue of Joro spider toxin and is an antagonist of calcium permeable AMPA</p>Fórmula:C22H37Cl3N4OPureza:99.75%Cor e Forma:SolidPeso molecular:479.91AMPA receptor modulator-2
CAS:<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Fórmula:C15H6F6N4OSPureza:99.8%Cor e Forma:SolidPeso molecular:404.29NMDA receptor modulator 4
CAS:<p>NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1].</p>Fórmula:C13H9F3N2O3SCor e Forma:SolidPeso molecular:330.28NPEC-caged-(S)-AMPA
CAS:<p>AMPA receptor agonist</p>Fórmula:C16H17N3O8Pureza:98%Cor e Forma:SolidPeso molecular:379.32p-fin4
CAS:<p>p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.</p>Fórmula:C39H53N8O18PCor e Forma:SolidPeso molecular:952.85AMPA-IN-1
CAS:<p>AMPA-IN-1: Potent AMPA receptor inhibitor; key in regulating brain excitatory transmission and plasticity.</p>Fórmula:C23H12F2N4O2Cor e Forma:SolidPeso molecular:414.36NS1219
CAS:<p>NS1219, an isomer of NS1209, is a selective AMPA antagonist for studying stroke, neuropathic pain, and epilepsy.</p>Fórmula:C24H28N4O7SCor e Forma:SolidPeso molecular:516.57BMT-108908
CAS:<p>BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.</p>Fórmula:C22H25FN2O2Cor e Forma:SolidPeso molecular:368.44GNE-0723
CAS:<p>GNE-0723 is a selective positive allosteric modulator of the NMDA receptor, GluN2A.blood-brain barrier (BBB) and Dravet syndrome and Alzheimer's disease (AD).</p>Fórmula:C16H8ClF6N5OSPureza:97.29% - 99.91%Cor e Forma:SolidPeso molecular:467.78BMS-986169
CAS:<p>BMS-986169 is a high-affinity and selective negative allosteric modulator of the NMDA receptor GluN2B subunit, depression.</p>Fórmula:C23H27FN2O2Pureza:97.61%Cor e Forma:SolidPeso molecular:382.47Dasolampanel etibutil
CAS:<p>Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).</p>Fórmula:C23H32ClN5O3Cor e Forma:SolidPeso molecular:461.98(R)-3,4-DCPG
CAS:<p>AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors</p>Fórmula:C10H9NO6Pureza:98%Cor e Forma:SolidPeso molecular:239.18UBP316
CAS:<p>GluR5-containing kainate receptor antagonist</p>Fórmula:C20H19N3O6SPureza:98%Cor e Forma:SolidPeso molecular:429.45Pregnanolone sulfate (pyridinium)
CAS:<p>Pregnanolone sulfate pyridinium, an endogenous neurosteroid, inhibits NMDA receptors and exhibits neuroprotective properties [1].</p>Fórmula:C26H39NO5SPureza:98%Cor e Forma:SolidPeso molecular:477.66Zelquistinel
CAS:<p>Zelquistinel, an NMDA receptor agonist, aids research on depression, anxiety, and psychiatric disorders.</p>Fórmula:C15H25N3O5Cor e Forma:SolidPeso molecular:327.38TCS 46b
CAS:<p>TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.</p>Fórmula:C22H23N3OPureza:99.78% - 99.78%Cor e Forma:SolidPeso molecular:345.44NMDA receptor modulator 6
CAS:<p>NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders.</p>Fórmula:C20H17FN2O4SCor e Forma:SolidPeso molecular:400.42ADCI
CAS:<p>ADCI inhibits voltage-activated sodium and NMDA channels; boosts dopamine metabolism in prefrontal cortex and nucleus accumbens.</p>Fórmula:C16H14N2OPureza:98%Cor e Forma:SolidPeso molecular:250.3DQP-26
CAS:<p>DQP-26, a potent negative allosteric modulator of NMDA receptors (NMDARs), exhibits IC50 values of 0.77 μM for GluN2C and 0.44 μM for GluN2D subunits,</p>Fórmula:C28H21Cl2N3O4Pureza:98%Cor e Forma:SolidPeso molecular:534.39AMPA receptor antagonist-3
CAS:<p>AMPA receptor antagonist-3 is an AMPA receptor antagonist.</p>Fórmula:C20H19N5O2SPureza:99.79%Cor e Forma:SolidPeso molecular:393.46Rislenemdaz
CAS:<p>Rislenemdaz (CERC-301) (CERC-301) is an antagonist of the N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B).</p>Fórmula:C19H23FN4O2Pureza:98.18%Cor e Forma:SolidPeso molecular:358.41AMPA receptor modulator-1
CAS:<p>AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.</p>Fórmula:C16H11ClF3NO2Pureza:99.93%Cor e Forma:SolidPeso molecular:341.71N1-N2-Di-N-Nitroso methyl (2S,5S)-5-methylpiperazine-2-carboxylate
Fórmula:C7H12N4O4Peso molecular:216.213-O-Desmethyl tacrolimus
CAS:<p>Tacrolimus is a macrolide immunosuppressant that is used to prevent organ rejection in transplant patients. It binds to the cytosolic protein, FKBP-12, which prevents calcineurin from dephosphorylating and activating nuclear factor of activated T cells (NFAT). Tacrolimus inhibits the production of IL-2 and other cytokines by T cells, suppressing proliferation. Tacrolimus has been shown to be bioequivalent when administered orally or intravenously. Bioavailability may be increased when taken with food.</p>Fórmula:C43H67NO12Pureza:90%MinCor e Forma:PowderPeso molecular:789.99 g/mol2,2'-(Thiobis(2-hydroxy-5,1-phenylene))bis(4H-benzo[e][1,3]oxazin-4-one)
CAS:<p>Please enquire for more information about 2,2'-(Thiobis(2-hydroxy-5,1-phenylene))bis(4H-benzo[e][1,3]oxazin-4-one) including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C28H16N2O6SPureza:Min. 95%Peso molecular:508.5 g/molNMDA agonist 1
CAS:<p>NMDA agonist 1 (compound 42d) is a potent NMDA agonist with a Ki value of 96 nM. It acts as a partial agonist of the GluN1/GluN2B complex, exhibiting an EC50 value of 78 nM.</p>Fórmula:C12H13N3O3SCor e Forma:SolidPeso molecular:279.315EMD-95885
CAS:<p>EMD-95885 is a selective antagonist of NMDA receptors containing NR2B subunits, with an IC50 of 3.9 nM. It does not interact with other sites on the NMDA receptor.</p>Fórmula:C22H23FN2O3Cor e Forma:SolidPeso molecular:382.428Macitentan (n-butyl analogue)
CAS:<p>Macitentan n-butyl analogue, an oral ETA/ETB receptor blocker, may treat IPF and PAH.</p>Fórmula:C20H21Br2N5O4SPureza:98%Cor e Forma:SolidPeso molecular:587.29Blixeprodil
CAS:<p>Blixeprodil (GM-1020) is an orally active NMDA receptor antagonist with an affinity of Ki = 3.25 µM in rat cortical tissue. It inhibits NR1/2A-NMDAR-mediated currents in HEK293 cells with an IC50 of 1.192 µM. Blixeprodil demonstrates antidepressant effects in rat models and exhibits blood-brain barrier permeability.</p>Fórmula:C13H16FNOCor e Forma:SolidPeso molecular:221.271NYX-2925
CAS:<p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>Fórmula:C14H23N3O4Cor e Forma:SolidPeso molecular:297.35(RS)-AMPA
CAS:<p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>Fórmula:C7H10N2O4Pureza:98%Cor e Forma:SolidPeso molecular:186.17BMS-986163
CAS:<p>BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).</p>Fórmula:C23H28FN2O5PPureza:98%Cor e Forma:SolidPeso molecular:462.45Caramboxin
CAS:<p>Caramboxin, a neurotoxin, can induce acute kidney injury.</p>Fórmula:C11H13NO6Cor e Forma:SolidPeso molecular:255.22YY-23
CAS:<p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>Fórmula:C33H54O8Cor e Forma:SolidPeso molecular:578.777DL-AP5 lithium
CAS:<p>DL-AP5 (2-APV) lithium is a competitive antagonist of the NMDA (N-Methyl-D-aspartate) receptor. It exhibits notable analgesic activity and specifically blocks channels in the rabbit retina.</p>Fórmula:C5H11LiNO5PCor e Forma:SolidPeso molecular:203.06LY3130481
CAS:<p>LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.</p>Fórmula:C19H18N4O3SCor e Forma:SolidPeso molecular:382.443-Methoxy PCE hydrochloride
CAS:<p>3-Methoxy PCE (3-MEO PCE) hydrochloride is an arylcyclohexylamine compound that functions as an NMDA receptor antagonist with a pKi value of 7.22.</p>Fórmula:C15H24ClNOCor e Forma:SolidPeso molecular:269.81Antidepressant agent 8
CAS:<p>Antidepressant agent 8 (Compound 1f) acts as a selective antagonist for the NMDA receptor GluN1/2A (NMDA receptorGluN1/2A), with an IC50 of 2.94 μmol/L. In a hydrocortisone-induced zebrafish depression model, it demonstrates antidepressant-like effects and shows good blood-brain barrier penetration.</p>Fórmula:C18H23FN4OS2Cor e Forma:SolidPeso molecular:394.53Antidepressant agent 9
CAS:<p>Antidepressant agent 9 (Compound 24) is an orally active inhibitor of NMDAR and SERT, with IC50 values of 3.50 μM and 1044 nM, respectively. It exhibits good metabolic stability and plasma exposure, and demonstrates antidepressant-like effects in the forced swim test in mice.</p>Fórmula:C17H24N2Cor e Forma:SolidPeso molecular:256.386Lu AF90103
CAS:<p>Lu AF90103 (Compound 42e) is the methyl ester prodrug of compound 42d, capable of crossing the blood-brain barrier. Compound 42d acts as a partial agonist of the GluN1/GluN2B complex, with an efficacy of 24% and an EC50 value of 78 nM. Lu AF90103 plays a significant role in neuropsychiatric disorder research.</p>Fórmula:C13H15N3O3SCor e Forma:SolidPeso molecular:293.342LY 235959
CAS:<p>LY 235959 is a NMDA receptor antagonist.</p>Fórmula:C11H20NO5PPureza:98%Cor e Forma:SolidPeso molecular:277.25(3S,6R)-NML
CAS:<p>(3S,6R)-NML is an NMDA receptor antagonist with pIC50 values of 4.8 [GluN1-GluN2A], 4.6 [GluN1-GluN2B], 5.0 [GluN1-GluN2C], and 5.0 [GluN1-GluN2D]. It is applicable in the study of depression.</p>Fórmula:C20H27NOCor e Forma:SolidPeso molecular:297.435Metaphit methylsulfate
CAS:<p>Metaphit methylsulfate is a specific PCP antagonist and an acylating agent for the [3H] phencyclidine binding site in rat brain homogenate. It inhibits PCP-induced motor activity through a presynaptic mechanism.</p>Fórmula:C19H28N2O3S2Cor e Forma:SolidPeso molecular:396.567PDE2 inhibitor 6
CAS:<p>PDE2 inhibitor6 (Compound 1) is an orally active phosphodiesterase (PDE) inhibitor, effectively inhibiting PDE2A, PDE3B, and PDE10A2 with IC50 values of 0.95 nM, 6.17 μM (pIC50=5.21), and 87.1 nM (pIC50=7.06), respectively. It modulates AMPA receptor activity, enhances synaptic plasticity, and improves learning and memory in rat models. Furthermore, PDE2 inhibitor6 possesses blood-brain barrier permeability.</p>Fórmula:C20H22F2N6OCor e Forma:SolidPeso molecular:400.425LY503430
CAS:<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Fórmula:C20H25FN2O3SPureza:98%Cor e Forma:SolidPeso molecular:392.49LY 215490
CAS:<p>LY 215490 is a selective AMPA receptor antagonist with neuroprotective properties in rat ischemia.</p>Fórmula:C13H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:279.34Onfasprodil
CAS:<p>Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)</p>Fórmula:C20H23FN2O3Cor e Forma:SolidPeso molecular:358.41NMDA receptor antagonist-3
<p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>Fórmula:C13H19N3O6Cor e Forma:SolidPeso molecular:313.31(RS)-AMPA hydrobromide
CAS:<p>AMPAR agonist</p>Fórmula:C7H11BrN2O4Pureza:98%Cor e Forma:SolidPeso molecular:267.08EU 1622-240
CAS:<p>EU 1622-240 is an allosteric modulator with a preference for GluN2B, GluN2C, and GluN2D, exhibiting EC50 values of 0.57, 0.82, and 1.1 μM, respectively. It possesses favorable physicochemical properties, along with in vitro stability and permeability.</p>Fórmula:C20H14BrF2N3O2SCor e Forma:SolidPeso molecular:478.31Perfluoroheptanesulfonic acid
CAS:<p>Perfluoroheptanesulfonic acid (1-Perfluoroheptanesulfonic acid; Perfluoroheptanesulphonic acid) is a perfluoroalkyl substance (PFAS). This compound has been detected in landfill leachate and has been shown to induce deformities in zebrafish larvae (EC50=168.1 μM). Exposure to PFHpS in fetuses can lead to reduced birth weight.</p>Fórmula:C7HF15O3SCor e Forma:SolidPeso molecular:450.12Caged MK801
CAS:<p>Caged MK801 (cMK801) is a selective, noncompetitive, and irreversible blocker of the NMDA receptor open channel. The NVOC cage is compatible in neuropharmacology and does not alter the intrinsic activity of the molecule.</p>Fórmula:C26H24N2O6Cor e Forma:SolidPeso molecular:460.48(RS)-AMPA hydrochloride
CAS:<p>(RS)-AMPA ((±)-AMPA) hydrochloride is a glutamate analog and serves as an efficient selective agonist for the excitatory neurotransmitter L-glutamic acid (L-glutamic acid). It does not interfere with the binding sites of alginate or NMDA receptors.</p>Fórmula:C7H11ClN2O4Cor e Forma:SolidPeso molecular:222.63(RS)-AMPA monohydrate
CAS:<p>(RS)-AMPA monohydrate, potent glutamate analogue, selectively activates L-glutamic acid without affecting kainic acid or NMDA receptors.</p>Fórmula:C7H12N2O5Cor e Forma:SolidPeso molecular:204.182Tamitinol
CAS:<p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>Fórmula:C12H20N2OSPureza:98%Cor e Forma:SolidPeso molecular:240.37SDZ 220-040
CAS:<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。</p>Fórmula:C16H16Cl2NO6PPureza:98.13%Cor e Forma:SolidPeso molecular:420.18BDZ-g
CAS:<p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>Fórmula:C21H21N5O2SPureza:99.97%Cor e Forma:SolidPeso molecular:407.49tert-Butyl Hydrogen Tetradecanedioate
CAS:Fórmula:C18H34O4Pureza:>95.0%(GC)(T)Cor e Forma:White to Light yellow powder to crystalPeso molecular:314.47D-2-Phenylglycine
CAS:Fórmula:C8H9NO2Pureza:>99.0%(T)Cor e Forma:White to Almost white powder to crystalPeso molecular:151.17(1E,4E)-1,5-Bis[3,5-bis(methoxymethoxy)phenyl]-1,4-pentadiene-3-one
CAS:Fórmula:C25H30O9Pureza:>97.0%(HPLC)Cor e Forma:White to Yellow to Green powder to crystalPeso molecular:474.514,4'-Diethynylbiphenyl
CAS:Fórmula:C16H10Pureza:>98.0%(GC)Cor e Forma:White to Light yellow to Light orange powder to crystalPeso molecular:202.26
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