Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 693 produtos de "Moduladores enzimáticos"
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Teriflunomide
CAS:Produto Controlado<p>Inhibitor of dihydroorotate dehydrogenase; anti-inflammatory; immunomodulatory</p>Fórmula:C12H9F3N2O2Pureza:Min. 98 Area-%Cor e Forma:White PowderPeso molecular:270.21 g/molCX 4945
CAS:<p>Inhibitor of CK2 protein kinase; anti-proliferative</p>Fórmula:C19H12ClN3O2Pureza:Min. 98 Area-%Cor e Forma:SolidPeso molecular:349.0618BAY 607550
CAS:<p>A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.</p>Fórmula:C27H32N4O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:476.24236Vildagliptin - Bio-X ™
CAS:<p>Vildagliptin is an antihyperglycemic agent that is used for the management of type 2 diabetes mellitus. This drug is a dipeptidyl peptidase 4 inhibitor and prevents the degradation of glucagon-like peptide 1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP). This leads to improved glycemic control.</p>Fórmula:C17H25N3O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:303.4 g/molMK 886 - Bio-X ™
CAS:<p>MK 886 is a leukotriene antagonist that has been studied for use in treating atherosclerosis. This drug inhibits the 5-lipoxygenase activating protein thus inhibiting 5-lipoxygenase.</p>Fórmula:C27H34ClNO2SPureza:Min. 95%Cor e Forma:PowderPeso molecular:472.08 g/molSCH 772984
CAS:<p>Inhibitor of ERK1 and ERK2 serine/threonine kinases</p>Fórmula:C33H33N9O2Pureza:Min. 95%Cor e Forma:Light (Or Pale) Yellow To Yellow SolidPeso molecular:587.67 g/molSB 431542
CAS:<p>Inhibitor of activin receptor-like kinases (ALK4, ALK5 and ALK7), members of TGFβ type I receptor family. Blocks activin- and TGFβ-mediated signaling and phosphorylation of Smad2 downstream. Suppresses tumor-promoting and tumor-suppressing effects of TGFβ. Promotes differentiation of human embryonic stem cells (hESCs), whilst sustaining mouse ESCs in the undifferentiated state.</p>Fórmula:C22H16N4O3Pureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:384.4 g/moleCF506
CAS:<p>Selective inhibitor of the Src kinase family with subnanomolar IC50 values and good selectivity over c-Abl, PDGFRα and c-Kit kinases. The compound is effective in inhibiting growth in drug resistant cancer cell lines. In a recent study, it inhibited the growth of HER2-positive breast cancer cell lines which were resistant to pan-HER family kinase inhibitors such as lapatinib.</p>Fórmula:C26H38N8O3Pureza:Min. 95%Cor e Forma:SolidPeso molecular:510.63 g/molBLU 667
CAS:<p>RET receptor tyroine kinase inhibitor</p>Fórmula:C27H32FN9O2Pureza:Min. 95%Cor e Forma:White/Off-White SolidPeso molecular:533.6 g/molRigosertib sodium
CAS:<p>Rigosertib sodium is an experimental chemotherapeutic agent that is a derivative of benzyl styryl sulfone. It is synthesized chemically and functions primarily by inhibiting key signaling pathways involved in cancer cell proliferation. Specifically, Rigosertib targets the RAS signaling pathway along with the phosphatidylinositol-3-kinase/AKT and polo-like kinase 1 (Plk1) pathways, impeding the progression of the cell cycle and inducing apoptosis in malignant cells.</p>Fórmula:C21H24NNaO8SPureza:Min. 95%Cor e Forma:White PowderPeso molecular:473.47 g/molAbemaciclib
CAS:<p>Inhibitor of cyclin-dependent kinases CDK4 and CDK6</p>Fórmula:C27H32F2N8Pureza:Min. 95%Peso molecular:506.59 g/molLarotrectinib
CAS:<p>A potent ATP-competitive inhibitor of tropomyosin-related kinases (TRK1, TRK2 and TRK3), members of the receptor tyrosine kinase family of neurotrophin receptors. Tumors with oncogenic TRK fusions are sensitive to larotrectinib, leading to reduced proliferation and tumor growth in patients with soft tissue sarcoma, triple-negative breast cancer and lung cancer.</p>Fórmula:C21H22F2N6O2Pureza:Min. 98 Area-%Cor e Forma:Yellow PowderPeso molecular:428.44 g/molSulindac - Bio-X ™
CAS:<p>Sulindac is a non-steroidal anti-inflammatory drug that has anti-inflammatory and analgesic properties. It is used to relieve the pain of osteoarthritis and rheumatoid arthritis by reducing inflammation and inhibiting the production of prostaglandins, which are chemicals that cause inflammation.</p>Fórmula:C20H17FO3SPureza:Min. 95%Cor e Forma:PowderPeso molecular:356.41 g/molAxitinib
CAS:<p>Inhibits VEGFR1, VEGFR2, VEGFR3, c-kit and PDGFR tyrosine kinases</p>Fórmula:C22H18N4OSPureza:Min. 98 Area-%Cor e Forma:White Yellow PowderPeso molecular:386.47 g/molCZC 25146
CAS:<p>Inhibitor of leucine-rich repeat kinase LRRK2Â</p>Fórmula:C22H25FN6O4SPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:488.54 g/molMethocarbamol
CAS:<p>Inhibitor of carbonic anhydrase; muscle relaxant</p>Fórmula:C11H15NO5Pureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:241.24 g/molLovastatin - Bio-X ™
CAS:<p>Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.</p>Fórmula:C24H36O5Pureza:Min. 95%Cor e Forma:PowderPeso molecular:404.54 g/molPF 06447475
CAS:<p>Inhibitor of LRRK2 kinase</p>Fórmula:C17H15N5OPureza:Min. 95%Cor e Forma:White To Off-White To Pink SolidPeso molecular:305.33 g/molBetrixaban
CAS:<p>Inhibitor of factor Xa</p>Fórmula:C23H22ClN5O3Pureza:Min. 95%Cor e Forma:Off-White PowderPeso molecular:451.91 g/molIbuprofen - Bio-X ™
CAS:<p>Ibuprofen is a non-steroidal anti-inflammatory drug (NSAID) used to reduce inflammation, relieve pain and reduce fever. The mechanism of action of ibuprofen has not been fully elucidated, but it may be due to inhibiting the enzyme cyclooxygenase and thus decreasing the synthesis of prostaglandins allowing a reduction of pain and inflammation.</p>Fórmula:C13H18O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:206.28 g/mol
