Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 693 produtos de "Moduladores enzimáticos"
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Seratrodast - Bio-X ™
CAS:Seratrodast is a thromboxane receptor antagonist that is used to treat asthma. However, this drug does not affect thrombus formation as other thromboxane synthase inhibitors do such as ozagrel.Fórmula:C22H26O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:354.44 g/molRebamipide - Bio-X ™
CAS:Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.Fórmula:C19H15ClN2O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:370.79 g/molAminopterin
CAS:Aminopterin is an antineoplastic agent and antifolate, which is a synthetic derivative of pteroylglutamic acid. It functions as a chemotherapeutic agent by inhibiting dihydrofolate reductase, an enzyme crucial in the folic acid pathway, thereby preventing the conversion of dihydrofolate to tetrahydrofolate. This disruption leads to impaired synthesis of purine nucleotides and thymidylate, which are essential for DNA synthesis and cell division.Fórmula:C19H20N8O5Pureza:Min. 97 Area-%Cor e Forma:Slightly Yellow PowderPeso molecular:440.41 g/molFluvastatin sodium
CAS:Fluvastatin is a statin that lowers blood cholesterol and triglycerides by inhibiting HMG-CoA reductase, an enzyme that plays a critical role in the synthesis of cholesterol. Fluvastatin has also been shown to reduce the incidence of myocardial infarction, and to reduce atherosclerotic lesions in animal models, reducing the incidence of cardiovascular disease. Fluvastatin also has been shown to inhibit the activation of toll-like receptor 4 (TLR4) by lipopolysaccharide (LPS), which may be related to its anti-inflammatory effects. Furthermore, through lowering blood cholesterol, Fluvastatin also inhibits tubulointerstitial injury and prevents renal damage caused by high concentrations of the lipid.
Fórmula:C24H25FNNaO4Pureza:Min. 98%Cor e Forma:Off-White PowderPeso molecular:433.45 g/molApixaban - Bio-X ™
CAS:Apixaban is an anticoagulant agent used for the prophylaxis of stroke and deep vein thrombosis leading to pulmonary embolism. This drug is an inhibitor of factor Xa and prothrominase. As a result, this prevents the formation of a thrombus.Fórmula:C25H25N5O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:459.5 g/molRosuvastatin calcium - Bio-X ™
CAS:Rosuvastatin is a drug that belongs to the group of statins. It is used for the treatment of high cholesterol and as an adjunct therapy for patients with coronary heart disease. Rosuvastatin reduces serum cholesterol by inhibiting HMG-CoA reductase, which is the rate-limiting enzyme in the production of cholesterol. Furthermore, this drug has been shown to have anti-inflammatory properties, which may be due to its ability to inhibit prostaglandin synthesis.Fórmula:C22H27FN3O6SCaPureza:(%) Min. 95%Cor e Forma:PowderPeso molecular:500.57 g/molMethotrexate sodium
CAS:Inhibitor of folate synthesis; folic acid analogueFórmula:C20H22N8O5•NaxPureza:Min. 95%Peso molecular:476.42 g/molAfatinib - Bio-X ™
CAS:Afatinib is a small molecule that inhibits the activity of cellular kinases that are involved in the progression of cancer. It is an Irreversible inhibitor of three members of the ErbB family. This molecule binds covalently to cysteine 797 residue in HER2 and blocks downstream cellular signalling which inhibits cellular growth and promotes apoptosis. It has been researched for the treatment of non-small cell lung cancer (NSCLC), breast cancer, pancreatic cancer and colorectal cancer.Fórmula:C24H25ClFN5O3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:485.94 g/molTenatoprazole
CAS:H+/K+ ATPase inhibitorFórmula:C16H18N4O3SPureza:Min. 95%Cor e Forma:PowderPeso molecular:346.41 g/molCamostat mesylate - Bio-X ™
CAS:Camostat is a serine protease inhibitor that is used for the treatment of chronic pancreatitis. This drug has shown to reduce inflammation and pain. Studies have shown that Camostat has also inhibited the entry of SARS-CoV-2 in lung cells by inhibiting the priming process of S-protein, necessary for the viral entry into host cells.Fórmula:C20H22N4O5•CH4O3SPureza:Min. 95%Cor e Forma:PowderPeso molecular:494.52 g/molPentoxifylline
CAS:Produto ControladoPhosphodiesterase inhibitorFórmula:C13H18N4O3Pureza:Min. 95%Cor e Forma:White PowderPeso molecular:278.31 g/mol3-(4-Phenylbutyl)-4-propyloxetan-2-one
CAS:Cis/trans-form of GK 563 [2351820-19-2]Fórmula:C16H22O2Pureza:Min. 95%Cor e Forma:SolidPeso molecular:246.34 g/molMK 4827
CAS:Inhibitor of PARP1 and PARP2 enzymes
Fórmula:C19H20N4OPureza:Min. 96 Area-%Cor e Forma:White PowderPeso molecular:320.39 g/molRucaparib camsylate
CAS:Inhibitor of poly (ADP-ribose) polymerase enzyme; antineoplasticFórmula:C19H18FN3O•C10H16O4SPureza:Min. 95%Cor e Forma:Off-White To Yellow SolidPeso molecular:555.66 g/molDiacerein - Bio-X ™
CAS:Diacerein is a slow-onset anthraquinone IL-1 inhibitor that is used in the treatment of joint diseases such as osteoarthritis. This drug is also being studied for the treatment of insulin resistance and diabetes mellitus. Diacerein works to decrease inflammation and cartilage destruction by reducing the level of interleukin-1.Fórmula:C19H12O8Pureza:Min. 95%Cor e Forma:PowderPeso molecular:368.29 g/molCetilistat - Bio-X ™
CAS:Cetilistat is a drug that is used to treat obesity. This drug inhibits the enzyme pancreatic lipase and so it prevents triglycerides from being hydrolyzed into absorbable free fatty acids.Fórmula:C25H39NO3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:401.58 g/molBrivanib alaninate
CAS:VEGFR2 a tyrosine kinase receptor inhibitor; antineoplasticFórmula:C22H24FN5O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:441.18123SU 0268
CAS:Inhibitor of 8-oxoguanine DNA glycosylase OGG1 with IC50 of 0.059 μM and excellent specificity over other DNA repair enzymes. OGG1 and its substrate 8-oxoguanine are involved in mutagenesis, genotoxicity, inflammation and cancer. The compound can cause accumulation of 8-oxoguanine in DNA in vitro and is a potent tool for the study of OGG1 biology.Fórmula:C26H25N3O4SPureza:Min. 95%Cor e Forma:White PowderPeso molecular:475.56 g/molArbutin - Synthetic origin
CAS:Inhibitor of tyrosinase in melanocytes: skin whitener
Fórmula:C12H16O7Pureza:Min. 98 Area-%Cor e Forma:White PowderPeso molecular:272.25 g/molAtorvastatin sodium salt - Bio-X ™
CAS:Atorvastatin is an HMG-CoA reductase inhibitor which is used to lower lipid levels and to reduce the risk of cardiovascular disease. This drug belongs to the class of medicines called statins. It lowers abnormal levels of cholesterol and lipids to reduce the risk of cardiovascular disease by inhibiting the enzyme HMG-CoA.Fórmula:C33H35FN2O5•NaPureza:(%) Min. 95%Cor e Forma:PowderPeso molecular:581.63 g/mol
