Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 644 produtos para "Moduladores enzimáticos".
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Crenolanib
CAS:Inhibits type III tyrosine kinases (PDGFRα, PDGFRβ, FLT3)Fórmula:C26H29N5O2Pureza:Min. 95%Cor e Forma:White To Yellow SolidPeso molecular:443.54 g/molBMS 754807
CAS:A reversible inhibitor of IGF-1R kinase and insulin receptor. Has anti-growth effects in mesenchymal, epithelial and hematopoietic tumor types. Synergistic with other cytotoxic, hormonal and targeted anti-cancer therapy.
Fórmula:C23H24FN9OPureza:Min. 95%Cor e Forma:PowderPeso molecular:461.49 g/molAceclofenac - Bio-X ™
CAS:Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.Fórmula:C16H13Cl2NO4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:354.18 g/molSB 239063
CAS:Inhibits p38 MAP kinase; anti-inflammatory; neuroprotectiveFórmula:C20H21FN4O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:368.4 g/molMGCD 265
CAS:Inhibits MET, VEGFR1-3, Tie and Ron tyrosine kinases; antineoplasticFórmula:C26H20FN5O2S2Pureza:Min. 95%Peso molecular:517.60 g/molXMU MP 2
CAS:BRK tyrosine kinase (PTK6) inhibitor; anti-proliferative in breast cancer cells
Fórmula:C32H33F3N8O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:618.65 g/molSivelestat
CAS:Inhibitor of human neutrophil elastase
Fórmula:C20H22N2O7SPureza:Min. 95%Peso molecular:434.46 g/molGC376 sodium
CAS:GC 376 is an inhibitor of the main protease Mpro (3CLpro) in coronaviruses as well as picornaviruses. This broad-spectrum antiviral compound has been used as investigational veterinary drug for treatment of feline infectious peritonitis virus (FIPV) infections. Recent studies also showed that GC 376 inhibits the main protease Mpro (3CLpro) from SARS-CoV-2 with IC50 of 0.03 μM and EC50 of 3.37 μM.
Fórmula:C21H30N3NaO8SPureza:Min. 95 Area-%Cor e Forma:White PowderPeso molecular:507.53 g/molIdelalisib
CAS:Idelalisib is a pharmaceutical drug that functions as a PI3Kδ inhibitor, developed through synthetic chemical processes. Its mode of action involves selectively targeting and inhibiting phosphatidylinositol 3-kinase delta (PI3Kδ), a lipid kinase that plays a crucial role in the signaling pathways responsible for cell proliferation, survival, and differentiation. By inhibiting this enzyme, Idelalisib effectively impedes pathways that are often hyperactivated in certain hematologic malignancies, thereby exerting antitumor effects.Fórmula:C22H18FN7OPureza:Min. 95%Cor e Forma:PowderPeso molecular:415.42 g/molSRT1720 hydrochloride
CAS:SIRT1 activatorFórmula:C25H23N7OS·xHClPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:469.56 g/molAG 221
CAS:Inhibitor of isocitrate dehydrogenase 2Fórmula:C19H17F6N7OPureza:Min. 95%Cor e Forma:PowderPeso molecular:473.38 g/molDCC 2036
CAS:Inhibits multiple tyrosine kinases (Abl1, Src family kinases, Tie-2 and VEGFR-2)Fórmula:C30H28FN7O3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:553.59 g/molSGC AAK1 1
CAS:Dual inhibitor of the adaptor protein 2-associated kinase 1 (AAK1) and BMP2-inducible kinase (BMP2K) with IC50 values of 270 nM and 1 μM, respectively. In a recent study, SGC AAK1 1 stabilised β-catenin, inhibited phosphorylation of the AP2 complex subunit mu protein (AP2M1) and activated Wnt signalling in in vitro experiments._x000D_Fórmula:C21H25N5O3SPureza:Min. 95%Cor e Forma:SolidPeso molecular:427.52 g/molEbselen
CAS:Ebselen is a non-toxic organoselenium compound with antioxidant, anti-inflammatory and cytoprotective properties. Ebselen is an inhibitor of lipoxygenases, nitric oxide (NO) synthases, protein kinase C, H+/K+-ATPase, thioredoxin reductase and NADPH oxidase. Recently, ebselen has been identified by several studies as a covalent inhibitor of the main protease Mpro from coronaviruses. For the SARS-CoV-2 main protease Mpro, the IC50 value is 0.67 μM and EC50 is 4.57 μM.Fórmula:C13H9NOSePureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:274.18 g/molPD 169316
CAS:Inhibitor of p38 kinase
Fórmula:C20H13FN4O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:360.34 g/molLY 2886721
CAS:Inhibitor of BACE1 proteaseFórmula:C18H16F2N4O2SPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:390.41 g/molZileuton- Bio-X ™
CAS:Zileuton is an inhibitor of the 5-lipoxygenase enzyme, thus preventing the leukotrienes LTE4, LDT4, LTB4 and LTC4 from being formed. This in turn reduces inflammation, bronchoconstriction and mucus secretion in the airways. As a result, Zileuton can be used in the treatment and management of asthma and allergic rhinitis. Studies have shown that Zileuton has the potential to reverse dementia-related brain damage.Fórmula:C11H12N2O2SPureza:(%) Min. 95%Cor e Forma:PowderPeso molecular:236.29 g/molKenpaullone
CAS:Inhibitor of glycogen synthase 3 (GSK-3) and cyclin-dependent kinases CDK1, CDK2 and CDK5. Kenpaullone can substitute transcription factor Klf4 in reprogramming of fibroblast to induced pluripotent stem cells when using the method of ectopic expression of transcriptional factors. In an in vitro model for Alzheimer’s disease, kenpaullone decreased production of amyloid beta peptides Aβ40 and Aβ42.
Fórmula:C16H11BrN2OPureza:Min. 95%Cor e Forma:Yellow To Dark Yellow SolidPeso molecular:326.00548GSK 2606414
CAS:Inhibitor of EIF2AK3/PERK kinasesFórmula:C24H20F3N5OPureza:Min. 95%Cor e Forma:PowderPeso molecular:451.44 g/molA 485
CAS:Histone acetyltransferase inhibitor of p300/CBP; anti-proliferative
Fórmula:C25H24F4N4O5Pureza:Min. 95%Cor e Forma:PowderPeso molecular:536.48 g/mol
