Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 693 produtos de "Moduladores enzimáticos"
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Crenolanib
CAS:<p>Inhibits type III tyrosine kinases (PDGFRα, PDGFRβ, FLT3)</p>Fórmula:C26H29N5O2Pureza:Min. 95%Cor e Forma:White To Yellow SolidPeso molecular:443.54 g/molBMS 754807
CAS:<p>A reversible inhibitor of IGF-1R kinase and insulin receptor. Has anti-growth effects in mesenchymal, epithelial and hematopoietic tumor types. Synergistic with other cytotoxic, hormonal and targeted anti-cancer therapy.</p>Fórmula:C23H24FN9OPureza:Min. 95%Cor e Forma:PowderPeso molecular:461.49 g/molAceclofenac - Bio-X ™
CAS:<p>Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.</p>Fórmula:C16H13Cl2NO4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:354.18 g/molSivelestat
CAS:<p>Inhibitor of human neutrophil elastase</p>Fórmula:C20H22N2O7SPureza:Min. 95%Peso molecular:434.46 g/molMGCD 265
CAS:<p>Inhibits MET, VEGFR1-3, Tie and Ron tyrosine kinases; antineoplastic</p>Fórmula:C26H20FN5O2S2Pureza:Min. 95%Peso molecular:517.60 g/molThioglycosyl Naphthalimide
CAS:<p>Thioglycosyl Naphthalimide is a highly potent human O-GlcNAcase (hOGA) inhibitor with good selectivity against human β-N-acetylhexosaminidase B (HsHexB).</p>Fórmula:C30H40N4O7SPureza:Min. 95%Peso molecular:600.73 g/molXMU MP 2
CAS:<p>BRK tyrosine kinase (PTK6) inhibitor; anti-proliferative in breast cancer cells</p>Fórmula:C32H33F3N8O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:618.65 g/molCZC 25146
CAS:<p>Inhibitor of leucine-rich repeat kinase LRRK2Â</p>Fórmula:C22H25FN6O4SPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:488.54 g/molMRK 560
CAS:<p>γ-secretase inhibitor; reduces amyloid-β in brainÂ</p>Fórmula:C19H17ClF5NO4S2Pureza:Min. 95%Peso molecular:517.92 g/molGNE 6776
CAS:<p>Specific inhibitor of the ubiquitin specific protease-7 (USP7), which is a validated deubiquitinase of the E3 ubiquitin-protein ligase MDM2. The compound inhibits the USP7 deubiquitinase activity by binding to acidic amino acid residues important for the interaction with ubiquitin. Induces tumor cell death and enhances cytotoxicity of chemotherapeutic agents.</p>Fórmula:C20H20N4O2Pureza:Min. 95%Peso molecular:348.4 g/molIdelalisib
CAS:<p>Idelalisib is a pharmaceutical drug that functions as a PI3Kδ inhibitor, developed through synthetic chemical processes. Its mode of action involves selectively targeting and inhibiting phosphatidylinositol 3-kinase delta (PI3Kδ), a lipid kinase that plays a crucial role in the signaling pathways responsible for cell proliferation, survival, and differentiation. By inhibiting this enzyme, Idelalisib effectively impedes pathways that are often hyperactivated in certain hematologic malignancies, thereby exerting antitumor effects.</p>Fórmula:C22H18FN7OPureza:Min. 95%Cor e Forma:PowderPeso molecular:415.42 g/molSRT1720 hydrochloride
CAS:<p>SIRT1 activator</p>Fórmula:C25H23N7OS·xHClPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:469.56 g/molAG 221
CAS:<p>Inhibitor of isocitrate dehydrogenase 2</p>Fórmula:C19H17F6N7OPureza:Min. 95%Cor e Forma:PowderPeso molecular:473.38 g/molDCC 2036
CAS:<p>Inhibits multiple tyrosine kinases (Abl1, Src family kinases, Tie-2 and VEGFR-2)</p>Fórmula:C30H28FN7O3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:553.59 g/molPeiminine
CAS:<p>Inhibitor of TGF-α, CTGF, ERK1/2, NF-κB and FasL; anti-inflammatory</p>Fórmula:C27H43NO3Pureza:Min. 98 Area-%Peso molecular:429.64 g/molSGC AAK1 1
CAS:<p>Dual inhibitor of the adaptor protein 2-associated kinase 1 (AAK1) and BMP2-inducible kinase (BMP2K) with IC50 values of 270 nM and 1 μM, respectively. In a recent study, SGC AAK1 1 stabilised β-catenin, inhibited phosphorylation of the AP2 complex subunit mu protein (AP2M1) and activated Wnt signalling in in vitro experiments._x000D_</p>Fórmula:C21H25N5O3SPureza:Min. 95%Cor e Forma:SolidPeso molecular:427.52 g/molEbselen
CAS:<p>Ebselen is a non-toxic organoselenium compound with antioxidant, anti-inflammatory and cytoprotective properties. Ebselen is an inhibitor of lipoxygenases, nitric oxide (NO) synthases, protein kinase C, H+/K+-ATPase, thioredoxin reductase and NADPH oxidase. Recently, ebselen has been identified by several studies as a covalent inhibitor of the main protease Mpro from coronaviruses. For the SARS-CoV-2 main protease Mpro, the IC50 value is 0.67 μM and EC50 is 4.57 μM.</p>Fórmula:C13H9NOSePureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:274.18 g/molMinaprine dihydrochloride
CAS:Produto Controlado<p>Short acting monoamine oxidase inhibitor</p>Fórmula:C17H22N4O•(HCl)2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:371.3 g/molLY 2886721
CAS:<p>Inhibitor of BACE1 protease</p>Fórmula:C18H16F2N4O2SPureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:390.41 g/molTacrolimus - Bio-X ™
CAS:<p>Tacrolimus is a calcineurin inhibitor drug that is used for the prevention of rejection after an organ transplant. This drug can also be used in the treatment of severe atopic dermatitis. Tacrolimus’ mechanism of action is not well known however it is understood that this drug inhibits T-lymphocyte activation by binding to an intracellular protein called FKBP-12. This drug also has anti-inflammatory properties.</p>Fórmula:C44H69NO12Pureza:Min. 95%Cor e Forma:White Off-White PowderPeso molecular:804.02 g/mol
