1-(4-Fluorophenyl)-4-[4-(3-isoquinolyl)-1-piperazinyl]butan-1-one hydrochloride
CAS: 82117-52-0
Ref. 3D-FF100458
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Informação sobre produto
- 1-Butanone, 1-(4-fluorophenyl)-4-(4-(3-isoquinolinyl)-1-piperazinyl)-, monohydrochloride
- 3-(4-(3-(4-Fluorobenzoyl)propyl)-1-piperazinyl)isoquinoline hcl
4-Fluorophenylbutanoyl is a δ-opioid agonist that binds to the δ-opioid receptor with a binding affinity of 1.2 nM. It has been shown to be a constant, with an EC50 of 0.05 nM when tested in binding experiments on human erythrocytes, and an ED50 of 0.5 mg/kg in mice when given intraperitoneally. 4-Fluorophenylbutanoyl has also been shown to be degradable by cytochrome P-450 enzymes and is metabolized via CYP3A4 and CYP2D6 pathways. These properties make it a potential nootropic agent for use in patients suffering from schizophrenic disorders or other inflammatory diseases that are associated with dopamine release.
Propriedades químicas
Consulta técnica sobre: 3D-FF100458 1-(4-Fluorophenyl)-4-[4-(3-isoquinolyl)-1-piperazinyl]butan-1-one hydrochloride
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