KD 5170

CAS: 940943-37-3

Ref. 3D-QMB94337

Informação sobre produto

• Nome: KD 5170
• Marca: Biosynth
• Descrição: KD 5170 is a potent and selective inhibitor of histone H3K9 methyltransferases. It has been shown to inhibit the growth of tumor xenografts in mice. KD 5170 also inhibits the acetylation of histone H4K5, which is necessary for the activation of transcription factors that control cell differentiation and proliferation. This drug also induces necrotic cell death by inhibiting mitochondrial membrane potential and oxidative DNA damage. KD 5170 may be clinically effective against cancer, as it has been shown to have an inhibitory effect on tumor xenografts in mice.This drug has natural compounds that are being studied for their effects on cancer cells, specifically those with mutations in genes related to TNF-related apoptosis-inducing ligand (TNFAIP6) or programmed cell death 1 (PDCD1).

Propriedades químicas

• Peso molecular: 451.56 g/mol
• Fórmula: C₂₀H₂₅N₃O₅S₂
• Pureza: Min. 95%