Pirenperone

CAS: 75444-65-4

Ref. TR-P508505

Informação sobre produto

• Nome: Pirenperone
• Sinónimos: 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, R 47465, 3-(2-(4-(p-Fluorobenzoyl)piperidino)ethyl)-2-methyl-4H-pyrido(1,2-a)pyrimidin-4-one, 3-{2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl}-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, 4H-Pyrido(1,2-a)pyrimidin-4-one, 3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-2-methyl-, Pirenperona, Pirenperona [INN-Spanish], Pirenperone [USAN:INN:BAN], Pirenperonum, Pirenperonum [INN-Latin], R-47,465, Unii-Y9Fmc4513X
• CAS: 75444-65-4

Descrição

Applications Pirenperone is a 5-HT2 serotonin receptor antagonist. Pirenperone also increases phosphorylation in human glioma cells by inhibiting cellular gap junctions.
References Warchal, S., et.al.: Bioorganic & Medicinal Chemistry. (2019); Yeo, J.Y., et.al: PLoS One. 14(9), 222-326. (2019)

• Marca: TRC

Propriedades químicas

• Peso molecular: 393.45
• Fórmula: C₂₃H₂₄FN₃O₂
• Cor/forma: Neat
• InChI: InChI=1S/C23H24FN3O2/c1-16-20(23(29)27-12-3-2-4-21(27)25-16)11-15-26-13-9-18(10-14-26)22(28)17-5-7-19(24)8-6-17/h2-8,12,18H,9-11,13-15H2,1H3
• Chave InChI: InChIKey=HXCNRYXBZNHDNE-UHFFFAOYSA-N
• SMILES: Cc1nc2ccccn2c(=O)c1CCN1CCC(C(=O)c2ccc(F)cc2)CC1