Entre as marcas dos nossos mais de 25 parceiros, destaca-se a TargetMol
We have reached an agreement with TargetMol: CymitQuimica clients will benefit for a 20% discount on all TargetMol products until the end of the year.On our website you can find the products offered by this partner, which has become one of the world's most recognised compound libraries and small molecule inhibitors supplier. TargetMol offers approximately 120 compound libraries and a wide range of chemical products and kits for life sciences.
Termina em 31 de dez.( faltam 8 dias )
PF-06862309
CAS:PF-06862309 is a PI3K inhibitorFórmula:C20H26F3N8O7PCor e Forma:SolidPeso molecular:578.44CGP-78608
CAS:CGP-78608 is a glycine site-specific N-methyl-D-aspartate receptor antagonist prevents activation of the NMDA/NO/CGMP pathway by ammonia.Fórmula:C11H13BrN3O5PCor e Forma:SolidPeso molecular:378.12Ochromycinone
CAS:<p>Ochromycinone (STA 21) is a selective STAT3 inhibitor.</p>Fórmula:C19H14O4Pureza:99.21%Cor e Forma:SolidPeso molecular:306.31Delgocitinib EtOH
CAS:Delgocitinib (LEO-124249/JTE052) is a selective JAK inhibitor used for reducing skin inflammation and treating chronic dermatitis.Fórmula:C18H24N6O2Cor e Forma:SolidPeso molecular:356.43BiBET
CAS:BiBET is a potent, selective, bivalent inhibitor of BET bromodomains.Fórmula:C26H30N10O3Cor e Forma:SolidPeso molecular:530.58MK-8666 Tris
CAS:<p>MK-8666, a partial GPCR agonist, targets GPR40 to enhance insulin secretion, potentially treating type 2 diabetes without adverse effects.</p>Fórmula:C33H42N2O9SCor e Forma:SolidPeso molecular:642.764Fasoracetam monohydrate
CAS:Fasoracetam monohydrate: synthetic, activates glutamate receptors, trialed in Phases I-III for vascular dementia.Fórmula:C11H21N3O5Cor e Forma:SolidPeso molecular:275.31JPI-547 HCl
CAS:JPI-547 (NOV 1402) is an oral anti-cancer drug targeting PARP 1/2 and Tankyrase 1/2, effective alone or with chemo and immunotherapies.Fórmula:C23H26Cl2N6OCor e Forma:SolidPeso molecular:473.402KR30031
CAS:KR30031 is a novel verapamil-like P-glycoprotein inhibitor with fewer heart side-effects, potentially boosting paclitaxel's efficacy.Fórmula:C26H34N2O4Cor e Forma:SolidPeso molecular:438.56Quoromycin
CAS:Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.Fórmula:C12H8N2O2SCor e Forma:SolidPeso molecular:244.27Tofacitinib maleate
CAS:<p>Tofacitinib (tasocitinib, CP-690550) is a JAK inhibitor blocking cytokine signaling and STAT activation.</p>Fórmula:C16H20N6O·xC4H4O4Cor e Forma:SolidPeso molecular:428.449NAS-181 free base
CAS:NAS-181 free base is a 5-HT(1B) receptor antagonist.Fórmula:C19H26N2O4Cor e Forma:SolidPeso molecular:346.42SU 5402
CAS:SU 5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, FGFR1, and PDGF-Rβ, respectively.Fórmula:C17H16N2O3Pureza:98.91% - 99.64%Cor e Forma:Yellow-Green SolidPeso molecular:296.32CJ-15161 hydrochloride
CAS:CJ-15161 hydrochloride is the salt form of CJ-15161 (free base), an opioid κ-receptor agonist, is undergoing development with Pfizer as an analgesic agent.Fórmula:C23H32ClN3O2Cor e Forma:SolidPeso molecular:417.978CJ-15161 (free base)
CAS:<p>CJ-15161 (free base), an opioid κ-receptor agonist, is undergoing development with Pfizer as an analgesic agent.</p>Fórmula:C23H31N3O2Cor e Forma:SolidPeso molecular:381.51IDN-1965
CAS:IDN-1965: potent, irreversible caspase inhibitor; blocks Fas-induced apoptosis; varied administration; promising for liver injury treatment.Fórmula:C21H26FN3O5Cor e Forma:SolidPeso molecular:419.45Bornaprine
CAS:Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.Fórmula:C21H31NO2Cor e Forma:SolidPeso molecular:329.48TP1287
CAS:TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.Fórmula:C21H21ClNO8PCor e Forma:SolidPeso molecular:481.82Laropiprant analog
CAS:Laropiprant analog is an antagonist of the prostaglandin PGD2 receptor DP1.Fórmula:C20H18ClFN2O4SCor e Forma:SolidPeso molecular:436.88ML416
CAS:<p>ML416 is an inhibitor of HIV-1.</p>Fórmula:C14H15FN2OS2Cor e Forma:SolidPeso molecular:310.41RWJ-60475
CAS:RWJ-60475 is a novel CD45 phosphatase inhibitor.Fórmula:C13H11BrNO7PCor e Forma:SolidPeso molecular:404.11SU6656
CAS:SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, 20 nM, 130 nM, and 170 nM for Src, Yes, Lyn, and Fyn, respectively.Fórmula:C19H21N3O3SPureza:98.21% - 98.73%Cor e Forma:SolidPeso molecular:371.45AZD5718
CAS:AZD5718: potent FLAP inhibitor (IC50=2.0 nM), treats Coronary Artery Disease, >90% leukotriene suppression, safe in animal studies, in phase 2a trial.Fórmula:C29H34N6O4Cor e Forma:SolidPeso molecular:530.62GNF7156
CAS:GNF7156 is a potent and selective DYRK1A inhibitor.Fórmula:C22H22N6O3Cor e Forma:SolidPeso molecular:418.45ONL-1204
CAS:ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Fórmula:C71H100N18O16Cor e Forma:SolidPeso molecular:1461.66PF-04363467 HCl
CAS:<p>PF-04363467 HCl is a selective dopamine D3/D2 receptor antagonist.</p>Fórmula:C22H30N2O3SCor e Forma:SolidPeso molecular:402.55Phenamil
CAS:Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.Fórmula:C12H12ClN7OPureza:99.07%Cor e Forma:SolidPeso molecular:305.72Istaroxime oxalate
CAS:<p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>Fórmula:C23H34N2O7Cor e Forma:SolidPeso molecular:450.53WS-691
CAS:<p>WS-691: potent oral ABCB1 modulator; lowers PTX IC50 to 22.02 nM in SW620/Ad300 cells; raises [3H]-PTX uptake; non-toxic in vivo.</p>Fórmula:C20H16FN7SCor e Forma:SolidPeso molecular:405.45BC-1485
CAS:<p>BC-1485 is a small molecule inhibitor of FIEL1 that inhibits the degradation of PIAS4 and ameliorates fibrosis in a mouse model.</p>Fórmula:C19H21N5O5SPureza:97.03% - 97.15%Cor e Forma:SolidPeso molecular:431.47Brostallicin HCl
CAS:Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.Fórmula:C30H36BrClN12O5Cor e Forma:SolidPeso molecular:760.04Risvodetinib
CAS:Risvodetinib: potent inhibitor of protein tyrosine kinases c-Abl1, c-Abl2, and c-kit.Fórmula:C33H34N8O2Cor e Forma:SolidPeso molecular:574.68Tedizolid Phosphate
CAS:Tedizolid Phosphate (TR-701FA) is an oxazolidinone-class antibiotic. Tedizolid phosphate is a phosphate ester prodrug of the active compound tedizolid.Fórmula:C17H16FN6O6PPureza:97.96%Cor e Forma:SolidPeso molecular:450.32XMU-MP-2
CAS:<p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>Fórmula:C32H33F3N8O2Pureza:99.29%Cor e Forma:SolidPeso molecular:618.65CRM-51005
CAS:<p>CRM-51005 is a new phospholipase C inhibitor produced by unidentified fungal strain MT51005</p>Fórmula:C15H20O3Cor e Forma:SolidPeso molecular:248.32VPC-16606
CAS:VPC-16606 inhibits ERα cell growth & gene expression, blocking ERα-LBD & SRC-3 binding dose-dependently.Fórmula:C17H13ClN2O2SCor e Forma:SolidPeso molecular:344.82Ixazomib citrate EtOH
CAS:Ixazomib citrate (MLN9708), a prodrug of Ixazomib, is an oral, next-gen proteasome inhibitor with enhanced anti-cancer properties.Fórmula:C22H29BCl2N2O10Cor e Forma:SolidPeso molecular:563.188Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Fórmula:C14H20ClN3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:313.78Lifirafenib HCl
CAS:Lifirafenib (Beigene-283/BGB-283): a potent, selective RAF/EGFR inhibitor effective against B-RAF mutated colorectal cancers.Fórmula:C26H19ClF3N3O3Cor e Forma:SolidPeso molecular:513.9012BMS-955176 HCl
CAS:<p>GSK-3532795: a broader-spectrum HIV-1 maturation inhibitor than bevirimat, effective in vitro and clinically.</p>Fórmula:C42H62N2O4SCor e Forma:SolidPeso molecular:727.486AMG2504
CAS:AMG2504 is a TRPA1 inhibitor.Fórmula:C15H10Cl4N2O3SCor e Forma:SolidPeso molecular:440.13Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Fórmula:C20H24N2S2Cor e Forma:SolidPeso molecular:356.55(S)-Pomalidomide
CAS:(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.Fórmula:C13H11N3O4Cor e Forma:SolidPeso molecular:273.24Teneligliptin hydrobromide
CAS:Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.Fórmula:C22H30N6OSBrHPureza:97.83% - 99.92%Cor e Forma:SolidPeso molecular:628.86Ruboxistaurin mesylate monohydrate
CAS:<p>Ruboxistaurin mesylate monohydrate, a PKC beta inhibitor, may treat diabetic nephropathy and macular edema, reducing oxidative stress and neovascularization.</p>Fórmula:C29H34N4O7SCor e Forma:SolidPeso molecular:582.67Difenamizole HCl
CAS:Difenamizole HCl, a pyrazolone NSAID with analgesic effects, modulates dopamine and inhibits monoamine oxidase.Fórmula:C20H23ClN4OCor e Forma:SolidPeso molecular:370.88Glutathione sodium
CAS:<p>Glutathione sodium, a water-soluble form of PAO, blocks blood vessel formation and cancer growth.</p>Fórmula:C10H16N3NaO6SCor e Forma:SolidPeso molecular:329.3BIM-46068
CAS:<p>BIM-46068 is a potent inhibitor of human farnesyltransferase with a unique anti-proliferative profile.</p>Fórmula:C21H42N4O3S3Cor e Forma:SolidPeso molecular:494.78BIM-46050
CAS:BIM-46050: potent human farnesyltransferase inhibitor, free acid of BIM-46068, nanomolar IC50, highly selective over GGTase.Fórmula:C20H40N4O3S3Cor e Forma:SolidPeso molecular:480.75
