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Termina em 31 de dez.( faltam 11 dias )
LYRM03
CAS:<p>LYRM03, a ubenimex derivative and aminopeptidase inhibitor, suppresses TLR4 to treat LPS-induced ALI in mice.</p>Fórmula:C21H33N3O5Cor e Forma:SolidPeso molecular:407.510-Oxononadecanedioic acid
CAS:<p>10-Oxononadecanedioic acid: a long-chain linker with two carboxylic ends, forms stable amides with amines using activators like EDC/HATU.</p>Fórmula:C19H34O5Cor e Forma:SolidPeso molecular:342.47Fipravirimat
CAS:<p>Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.</p>Fórmula:C43H67FN2O4SCor e Forma:SolidPeso molecular:727.07CDK8-IN-4k
CAS:<p>CDK8-IN-4k is a potent and highly selective CDK8 inhibitor, with no apparent potential for time-dependent CYP3A4 inhibition.</p>Fórmula:C24H23F2N5OCor e Forma:SolidPeso molecular:435.47PomCapstafin
CAS:<p>PomCapstafin is a prodrug of Capstafin, acting as a potent, selective STAT5b inhibitor.</p>Fórmula:C41H69NO17P2Cor e Forma:SolidPeso molecular:909.93Vps34-IN-1
CAS:<p>Vps34-IN-1: potent, selective Vps34 inhibitor, 25 nM IC50, spares class I/II PI3Ks.</p>Fórmula:C21H24ClN7OPureza:97.04%Cor e Forma:SolidPeso molecular:425.91Capstafin
CAS:<p>Capstafin is a highly potent and selective inhibitor of STAT5b.</p>Fórmula:C17H29NO9P2Cor e Forma:SolidPeso molecular:453.36MeTC7
CAS:<p>MeTC7 is a VDR antagonist with antitumor activity that inhibits PD-L1 and may inhibit the growth of xenografts and transgenic tumors in vivo.</p>Fórmula:C32H48BrN3O4Pureza:99.69%Cor e Forma:SolidPeso molecular:618.65Miransertib mesylate
CAS:<p>Miransertib mesylate inhibits AKT non-competitively, potentially reducing tumor growth and triggering apoptosis.</p>Fórmula:C29H32N6O6S2Cor e Forma:SolidPeso molecular:624.73Pipoxolan hydrochloride
CAS:<p>Pipoxolan is an antispasmodic treating GI tract, gallbladder, urogenital, and menstrual cramps, with emerging anticancer properties.</p>Fórmula:C22H26ClNO3Cor e Forma:SolidPeso molecular:387.9041-Hydroxyvaldecoxib
CAS:<p>1-Hydroxyvaldecoxib is a COX-2 inhibitor.</p>Fórmula:C16H14N2O4SCor e Forma:SolidPeso molecular:330.36Fenoldopam hydrochloride
CAS:<p>Fenoldopam HCl: D1 dopamine receptor agonist, vasodilator, doesn't cross blood-brain barrier, α2-adrenoceptor antagonist.</p>Fórmula:C16H17Cl2NO3Cor e Forma:SolidPeso molecular:342.22K-5a2
CAS:<p>K-5a2 is a novel human immunodeficiency virus type 1 (HIV-1) non-nucleoside reverse transcriptase inhibitor (NNRTI).</p>Fórmula:C27H28N6O3S2Cor e Forma:SolidPeso molecular:548.68GGTI-297
CAS:<p>GGTI-297 is a potent, cell-permeable, and selective peptidomimetic inhibitor of GGTase I compared to Farnesyl Transferase (FTase).</p>Fórmula:C26H31N3O3SCor e Forma:SolidPeso molecular:465.61UniPR1331
CAS:<p>UniPR1331 is a novel selective antagonist of the Eph-ephrin system.</p>Fórmula:C35H48N2O4Cor e Forma:SolidPeso molecular:560.77VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Fórmula:C19H16ClN5O6SPureza:98.99% - 99.22%Cor e Forma:SolidPeso molecular:477.88PF-06427878
CAS:<p>PF-06427878 is an orally active, potent and selective diacylglycerol acyltransferase 2 inhibitor.</p>Fórmula:C26H28N4O5Cor e Forma:SolidPeso molecular:476.52Berotralstat HCl
CAS:<p>Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.</p>Fórmula:C30H28Cl2F4N6OCor e Forma:SolidPeso molecular:635.4886GPA512
CAS:<p>GPA512 is a prodrug of aliellalactone, inhibiting STAT3 and preventing the transcription of STAT3 regulated genes.</p>Fórmula:C17H25NO6SCor e Forma:SolidPeso molecular:371.45Bizine dihydrochloride
CAS:<p>Bizine dihydrochloride is a potent LSD1 inhibitor in vitro, being selective versus monoamine oxidases A/B and the LSD1 homologue, LSD2.</p>Fórmula:C18H25Cl2N3OCor e Forma:SolidPeso molecular:370.32LASSBio-1829 HCl
CAS:<p>LASSBio-1829 HCl is an orally active IKK2 inhibitor.</p>Fórmula:C25H19ClN4OCor e Forma:SolidPeso molecular:426.9V-125
CAS:<p>V-125 is an agonist of retinoid X receptors.</p>Fórmula:C23H30N2O2Cor e Forma:SolidPeso molecular:366.5Indinavir monohydrate
CAS:<p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>Fórmula:C36H49N5O5Cor e Forma:SolidPeso molecular:631.82BP-5-087
CAS:<p>BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.</p>Fórmula:C36H30F8N2O6SCor e Forma:SolidPeso molecular:770.69Tofacitinib HCl
CAS:<p>Tofacitinib (tasocitinib, CP-690550) is a JAK inhibitor impacting phosphorylation/activation of STATs with varied IC50 values.</p>Fórmula:C16H21ClN6OCor e Forma:SolidPeso molecular:348.835UAWJ-247
CAS:<p>UAWJ-247 is a SARS-CoV-2 Main Protease inhibitor (IC50 = 45 nM).</p>Fórmula:C24H28N3NaO8SCor e Forma:SolidPeso molecular:541.55WNK463
CAS:<p>WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).</p>Fórmula:C21H24F3N7O2Pureza:>99.99% - ≥95%Cor e Forma:SolidPeso molecular:463.46Milvexian TFA
CAS:<p>Milvexian (BMS-986177/JNJ-70033093) is a factor XIa inhibitor with Ki=44 nM for kallikrein, Ki=35 nM for chymotrypsin, 32% bioavailability.</p>Fórmula:C30H26Cl2F5N9O4Cor e Forma:SolidPeso molecular:742.49GSK1379767A
CAS:<p>GSK1379767A is a dual inhibitor of BPTF and Brd4.</p>Fórmula:C26H30N6O6Cor e Forma:SolidPeso molecular:522.55NY0173
CAS:<p>NY0173 is a potent exchange protein activated by cAMP antagonists.</p>Fórmula:C18H15Cl3N4O2Cor e Forma:SolidPeso molecular:425.7NY0123
CAS:<p>NY0123 is an active EPAC antagonist with low micromolar inhibitory activity.</p>Fórmula:C16H13Cl3N4O2Cor e Forma:SolidPeso molecular:399.66Fadaltran
CAS:<p>Fadaltran is an α2-adrenoreceptor antagonist.</p>Fórmula:C24H29N5O2Cor e Forma:SolidPeso molecular:419.52P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Fórmula:C21H16F3N9Cor e Forma:SolidPeso molecular:451.42OAT-177
CAS:<p>OAT-177 is a potent, selective, orally active acidic mammalian chitinase (AMCase) inhibitor.</p>Fórmula:C19H29ClN6Cor e Forma:SolidPeso molecular:376.93Sonidegib metabolite M25
CAS:<p>Sonidegib metabolite M25 is a smoothened (SMO) antagonist.</p>Fórmula:C26H26F3N3O4Cor e Forma:SolidPeso molecular:501.5THIQ-40
CAS:<p>THIQ-40: potent ERα antagonist, oral SERD with antitumor effects.</p>Fórmula:C28H29NO3Cor e Forma:SolidPeso molecular:427.53WZB117
CAS:<p>WZB117 inhibits GLUT1; IC50 ~10μM slows A549 lung & MCF7 breast cancer cell growth.</p>Fórmula:C20H13FO6Pureza:99.03% - 99.18%Cor e Forma:SolidPeso molecular:368.31LFS-829
CAS:<p>LFS-829: small molecule, inhibits exportin-1, low nanomolar activity, orally reverses colitis in mice, low toxicity, promising for clinical trials.</p>Fórmula:C13H9F6NOS2Cor e Forma:SolidPeso molecular:373.34FFA3-Antagonist-6
CAS:<p>FFA3-Antagonist-6 is a PAM-antagonist of the function of C3 at FFA3.</p>Fórmula:C30H28N2O3Cor e Forma:SolidPeso molecular:464.55NVP-BHS345
CAS:<p>NVP-BHS345 is a dual inhibitor of TORC1 and TORC2.</p>Fórmula:C25H20N6OCor e Forma:SolidPeso molecular:420.47Eptapirone fumarate
CAS:<p>Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.</p>Fórmula:C20H27N7O6Cor e Forma:SolidPeso molecular:461.479YM-60828 dihydrochloride
CAS:<p>YM-60828 dihydrochloride is a Factor Xa (FXa) inhibitor and anticoagulant used in the treatment of venous thromboembolic disease.</p>Fórmula:C27H33Cl2N5O5SCor e Forma:SolidPeso molecular:610.55Desmethyl atenolol
CAS:<p>Desmethyl atenolol is an impurity of Atenolol -- a selective β1 receptor antagonist.</p>Fórmula:C13H20N2O3Cor e Forma:SolidPeso molecular:252.31Methazolamide-d6
CAS:<p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>Fórmula:C5H2D6N4O3S2Cor e Forma:SolidPeso molecular:242.31NPC-18915
CAS:<p>NPC-18915 is a benzofuran compound, inhibitor of neutophil activation.</p>Fórmula:C23H16O3Cor e Forma:SolidPeso molecular:340.37ER-34122
CAS:<p>ER-34122, a novel orally available dual 5-lipoxygenase/cyclooxygenase inhibitor with potent anti-inflammatory activity.</p>Fórmula:C27H26ClN3O5Pureza:>99.99%Cor e Forma:SolidPeso molecular:507.96Navoximod phosphate
CAS:<p>Navoximod phosphate is an indoleamine 2,3-dioxygenase (IDO) inhibitor, immunomodulator and antineoplastic.</p>Fórmula:C18H24FN2O6PCor e Forma:SolidPeso molecular:414.37Z-IETD-FMK
CAS:<p>Z-IETD-FMK (Z-IE(OMe)TD(OMe)-FMK) is a selective caspase 8 inhibitor, which has cell permeable.</p>Fórmula:C30H43FN4O11Pureza:95% - 99.81%Cor e Forma:SolidPeso molecular:654.68Tinostamustine HCl
CAS:<p>Tinostamustine (EDO-S101) is an alkylating HDACi fusion molecule, enhancing potency and overcoming drug resistance.</p>Fórmula:C19H29Cl3N4O2Cor e Forma:SolidPeso molecular:451.82GI261520A
CAS:<p>GI261520A is a potent egfr/erbb2 dual inhibitor</p>Fórmula:C22H19N3O2Cor e Forma:SolidPeso molecular:357.41
