Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
Y06137
CAS:2226534-49-0
Y06137, selective BET inhibitor, Kd 81 nM for BRD4(1), researched for castration-resistant prostate cancer treatment.
Formula:
C27H32N4O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
444.57
Ref: TM-T13363
| 1mg | 60.00 € | ||
| 2mg | 86.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
FT001
CAS:1778655-51-8
FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.
Formula:
C25H29N3O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
467.58
Ref: TM-T27392
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,052.00 € | ||
| 500mg | 2,103.00 € | ||
| 1mL*10mM (DMSO) | 298.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
LLY-283
CAS:2040291-27-6
LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.
Formula:
C17H18N4O4
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
342.35
Ref: TM-T15767
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
PF-06726304 acetate
CAS:2080306-28-9
PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.
Formula:
C24H25Cl2N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
506.38
Ref: TM-T12428
| 10mg | 513.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
EZM0414
CAS:2411748-50-8
EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM …
Formula:
C22H29FN4O2
Purity:
98.9%
Color and Shape:
Liquid
Molecular weight:
400.49
Ref: TM-T9969
| 1mg | 260.00 € | ||
| 5mg | 642.00 € | ||
| 10mg | 909.00 € | ||
| 25mg | 1,364.00 € | ||
| 50mg | 1,821.00 € | ||
| 100mg | 2,460.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
MM-589
CAS:2097887-20-0
MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) …
Formula:
C28H44N8O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
572.7
Ref: TM-T12091
| 25mg | 2,801.00 € | ||
| 50mg | 3,722.00 € | ||
| 100mg | 5,144.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
PARP1-IN-29
CAS:1567375-93-2
PARP1-IN-29 is an orally active PARP-1 inhibitor with an IC50 of 6.3 nM. When labeled …
Formula:
C18H16FN3O2
Color and Shape:
Liquid
Molecular weight:
325.34
Ref: TM-T200541
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
PARP7-IN-16 free base
CAS:2136325-05-6
PARP7-IN-16 free base is the freebase form of PARP7-IN-16. As a selective oral inhibitor of …
Formula:
C25H27FN4O4
Color and Shape:
Liquid
Molecular weight:
466.51
Ref: TM-T200703
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
W4275
CAS:3051650-00-8
W4275 (Compound 42) is a selective NSD2 inhibitor with oral activity and an IC50 of …
Formula:
C25H36N6O3
Color and Shape:
Liquid
Molecular weight:
468.59
Ref: TM-T200598
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
SMARCA2-IN-2
CAS:2568055-24-1
Compound I-25, also known as SMARCA2-IN-2, is a SMARCA2 inhibitor (IC 50: 101-500 μM) with …
Formula:
C16H17N3
Color and Shape:
Liquid
Molecular weight:
251.33
Ref: TM-T200326
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
JBJ-02-112-05
CAS:2748162-29-8
JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC …
Formula:
C27H20N4O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
464.54
Ref: TM-T11713
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
JDTic dihydrochloride
CAS:785835-79-2
JDTic is a powerful antagonist of kappa-opioid receptors (KOR), effectively inhibiting the antinociceptive effects induced …
Formula:
C28H41Cl2N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.55
Ref: TM-T11721L
| 2mg | 102.00 € | ||
| 25mg | 620.00 € | ||
| 50mg | 813.00 € | ||
| 100mg | 1,208.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
GSK3368715
CAS:1629013-22-4
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases …
Formula:
C20H38N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
366.54
Ref: TM-T11500
| 25mg | 2,523.00 € | ||
| 50mg | 3,348.00 € | ||
| 100mg | 4,583.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
GSK3368715 dihydrochloride
CAS:1628925-77-8
GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study …
Formula:
C20H40Cl2N4O2
Purity:
99.66% - 99.66%
Color and Shape:
Solid
Molecular weight:
439.46
Ref: TM-T11500L
| 1mg | 61.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
Pocenbrodib
CAS:2304372-79-8
Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential …
Formula:
C28H32FN3O6
Purity:
98.44% - 98.48%
Color and Shape:
Liquid
Molecular weight:
525.57
Ref: TM-T69691
| 1mg | 747.00 € | ||
| 5mg | 1,563.00 € | ||
| 25mg | 2,581.00 € | ||
| 50mg | 3,164.00 € | ||
| 100mg | 4,306.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
ITK inhibitor 2
CAS:1309784-09-5
ITK inhibitor 2 is a interleukin-2-inducible T-cell kinase (ITK) inhibitor , with an IC50 of …
Formula:
C25H33N5O2
Color and Shape:
Solid
Molecular weight:
435.56
Ref: TM-T11690
| 50mg | 738.00 € | ||
| 100mg | 1,105.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
SCH-1473759
CAS:1094069-99-4
SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A …
Formula:
C20H26N8OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
426.54
Ref: TM-T16862
| 5mg | 205.00 € | ||
| 50mg | 694.00 € | ||
| 100mg | 1,059.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
INCB054329
CAS:1628607-64-6
INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.
Formula:
C19H16N4O3
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
348.36
Ref: TM-T22345
| 1mg | 45.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
CBP/p300-IN-2
CAS:2158265-96-2
CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and …
Formula:
C27H29F2N7O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
521.56
Ref: TM-T10702
| 25mg | 2,662.00 € | ||
| 50mg | 3,533.00 € | ||
| 100mg | 4,860.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
TY-011
CAS:1389439-77-3
TY-011 is an inhibitor of Aurora A/B kinases. This compound induces DNA damage and cell …
Formula:
C18H16ClN5
Color and Shape:
Liquid
Molecular weight:
337.81
Ref: TM-T89833
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
