CymitQuimica logo
Integrin

Integrin

Los inhibidores de integrinas se dirigen a las integrinas, una familia de receptores en la superficie celular que desempeñan un papel crucial en la adhesión celular, la migración y la transducción de señales. Las integrinas están involucradas en la regulación del ciclo celular, particularmente en procesos como la división y la diferenciación celular. Inhibir las integrinas puede interrumpir estos procesos, lo que lleva al arresto del ciclo celular y la apoptosis, lo que hace que estos inhibidores sean valiosos en la investigación del cáncer y el estudio de la metástasis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de integrinas de alta calidad para apoyar su investigación en la regulación del ciclo celular, la biología del cáncer y el desarrollo terapéutico.

Se han encontrado 224 productos de "Integrin"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • A-205804

    CAS:
    <p>A-205804 is a specific and effective inhibitor of E-selectin( IC50=20 nM ) and ICAM-1(IC50=25 nM) expression.</p>
    Fórmula:C15H12N2OS2
    Pureza:98.07% - 98.52%
    Forma y color:Solid
    Peso molecular:300.4
  • Cyclo(-RGDfK)

    CAS:
    <p>Cyclo(-RGDfK) is a selective and potent inhibitor of integrin αvβ3 with an IC50 value of 0.94 nM.Cost-effective and quality-assured.</p>
    Fórmula:C27H41N9O7
    Pureza:95.29% - >99.99%
    Forma y color:Solid
    Peso molecular:603.67
  • PND-1186

    CAS:
    <p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>
    Fórmula:C25H26F3N5O3
    Pureza:99.14% - 99.75%
    Forma y color:Solid
    Peso molecular:501.5
  • GLPG0187

    CAS:
    <p>GLPG0187, a broad spectrum integrin receptor antagonist, inhibits αvβ1-integrin (IC50: 1.3 nM).</p>
    Fórmula:C29H37N7O5S
    Pureza:99.4% - 99.70%
    Forma y color:Solid
    Peso molecular:595.71
  • OSU-T315

    CAS:
    <p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>
    Fórmula:C30H30F3N5O
    Pureza:98.69%
    Forma y color:Solid
    Peso molecular:533.59
  • Arginine-glycine-aspartic acid

    CAS:
    <p>RGD (RGD (Arg-Gly-Asp) Peptides) (Arg-Gly-Asp) Peptides is a cell adhesion motif which can mimic cell adhesion proteins and bind to integrins.</p>
    Fórmula:C12H22N6O6
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:346.34
  • Cyclo(RADfK)

    CAS:
    <p>Cyclo(RADfK) is a selective α(v)β(3) integrin ligand used in neoangiogenesis research, therapy, and diagnostics; it's a control for RGD peptides.</p>
    Fórmula:C28H43N9O7
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:617.7
  • Cyclo(-RGDfK) TFA

    CAS:
    <p>Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).</p>
    Fórmula:C29H42F3N9O9
    Pureza:98.99% - 99.54%
    Forma y color:Solid
    Peso molecular:717.69
  • CWHM-12

    CAS:
    <p>CWHM-12 is a potent inhibitor of αV integrins (IC50s of 0.2/0.8/1.5/1.8 nM for αvβ8/αvβ3/αvβ6/αvβ1).</p>
    Fórmula:C26H32BrN5O6
    Pureza:98.05% - 99.83%
    Forma y color:Solid
    Peso molecular:590.47
  • H-Gly-Arg-Gly-Asp-Asn-Pro-OH

    CAS:
    <p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>
    Fórmula:C23H38N10O10
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:614.61
  • iRGD peptide

    CAS:
    <p>iRGD peptide: 9-amino acid cyclic compound (CRGDKGPDC), found through phage display in mice with tumors.</p>
    Fórmula:C35H57N13O14S2
    Pureza:98.77%
    Forma y color:Solid
    Peso molecular:948.04
  • Leukadherin-1

    CAS:
    <p>Leukadherin-1 boosts CD11b/CD18 adhesion, lowers leukocyte movement, cuts inflammation.</p>
    Fórmula:C22H15NO4S2
    Pureza:98.49% - 98.93%
    Forma y color:Solid
    Peso molecular:421.49
  • Pyrintegrin

    CAS:
    <p>Pyrintegrin: β1-integrin agonist, boosts embryonic stem cell survival, and podocyte protection, improves cell-matrix adhesion.</p>
    Fórmula:C23H25N5O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:451.54
  • Orbofiban

    CAS:
    <p>Orbofiban, an orally administered antagonist of the platelet GPIIb/IIIa receptor, effectively inhibits platelet aggregation.</p>
    Fórmula:C17H23N5O4
    Forma y color:Solid
    Peso molecular:361.4
  • Cucurbitacin B

    CAS:
    <p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>
    Fórmula:C32H46O8
    Pureza:97.1% - 99.33%
    Forma y color:Solid
    Peso molecular:558.7
  • ILK-IN-2

    CAS:
    <p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>
    Fórmula:C30H30F3N5O
    Pureza:99.30%
    Forma y color:Solid
    Peso molecular:533.59
  • A-286982

    CAS:
    <p>A 286982 blocks the LFA-1 and ICAM-1 integrin-ligand interaction.</p>
    Fórmula:C24H27N3O4S
    Pureza:97.81%
    Forma y color:Solid
    Peso molecular:453.55
  • Arg-Gly-Asp TFA (99896-85-2(free base))


    <p>Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.</p>
    Fórmula:C14H23F3N6O8
    Pureza:99.2% - ≥98%
    Forma y color:Solid
    Peso molecular:460.36
  • roxifiban

    CAS:
    <p>Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.</p>
    Fórmula:C21H29N5O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:447.48
  • LXW7

    CAS:
    <p>LXW7 is an octamer disulfide cyclic peptide and αvβ3 integrin ligand, acts as a potent and specific endothelial progenitor cells (EPCs) and endothelial cells (</p>
    Fórmula:C29H48N12O12S2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:820.89