CymitQuimica logo
Receptor de estrógeno / progestágeno

Receptor de estrógeno / progestágeno

Los receptores de estrógenos y progestágenos son receptores hormonales nucleares que median los efectos del estrógeno y la progesterona, respectivamente. Estos receptores regulan varios procesos fisiológicos, incluyendo la función reproductiva, la densidad ósea y la salud cardiovascular. Los moduladores de los receptores de estrógenos y progestágenos se estudian extensamente por sus roles en la terapia de reemplazo hormonal, la anticoncepción y el tratamiento de cánceres hormonoresponsivos. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores de estrógenos y progestágenos de alta calidad para apoyar su investigación en endocrinología, salud reproductiva y biología del cáncer.

Se han encontrado 60 productos para "Receptor de estrógeno / progestágeno".

productos por página.
  • SLU-PP-332

    CAS:
    SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,
    Fórmula:C18H14N2O2
    Pureza:97.53% - 98.60%
    Forma y color:Solid
    Peso molecular:290.32
  • Bazedoxifene hydrochloride

    CAS:
    Bazedoxifene hydrochloride (TSE 424 hydrochloride) is an estrogen receptor modulator and an inhibitor of IL-6/GP130 protein interaction.
    Fórmula:C30H35ClN2O3
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:507.064
  • Giredestrant

    CAS:
    Giredestrant (GDC-9545) is a potent oral anti-tumor ER antagonist competing with estradiol.
    Fórmula:C27H31F5N4O
    Pureza:99.12% - 99.56%
    Forma y color:Solid
    Peso molecular:522.5533
  • Clomiphene citrate

    CAS:
    Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.
    Fórmula:C32H36ClNO8
    Pureza:98.67% - >99.99%
    Forma y color:Solid
    Peso molecular:598.083
  • Panomifene TFA


    Panomifene TFA(GYKl13504 TFA) is a antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases.
    Fórmula:C27H25F6NO4
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:541.48
  • CMP8

    CAS:
    CMP8, an estrogen receptor ligand, selectively binds to ERLBD with IC50: 29 nM (MGERα), 41 nM (MGRERα), 1100 nM (hERα), 2200 nM (hERβ).
    Fórmula:C33H34ClNO3
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:528.081
  • 4,4'-Iminodiphenol

    CAS:
    4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.
    Fórmula:C12H11NO2
    Pureza:98.68%
    Forma y color:Yellow Solid
    Peso molecular:201.2212
  • Dienestrol

    CAS:
    Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist.
    Fórmula:C18H18O2
    Pureza:97.07% - 98%
    Forma y color:Solid
    Peso molecular:266.3343
  • Elacestrant

    CAS:
    Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
    Fórmula:C30H38N2O2
    Pureza:99.79% - 99.92%
    Forma y color:White Solid
    Peso molecular:458.6349
  • PROTAC ERRα ligand 1

    CAS:
    PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
    Fórmula:C19H11F3N2O4S
    Pureza:99.02%
    Forma y color:White Solid
    Peso molecular:420.36
  • Amcenestrant

    CAS:
    Amcenestrant (SAR439859) is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER.
    Fórmula:C31H30Cl2FNO3
    Pureza:99%
    Forma y color:White Solid
    Peso molecular:554.479
  • Toremifene

    CAS:
    Toremifene (GTx 006) is a selective estrogen-receptor modulator (SERM).
    Fórmula:C26H28ClNO
    Pureza:99.77% - >99.99%
    Forma y color:Solid
    Peso molecular:405.96
  • (R)-Equol

    CAS:
    (R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.
    Fórmula:C15H14O3
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:242.2699
  • Fulvestrant-3-boronic acid

    CAS:
    Fulvestrant-3-boronic acid (ZB716) is an oral SERD that binds ERα (IC₅₀=4.1 nM) and induces degradation for ER-positive breast cancer research.
    Fórmula:C32H48BF5O4S
    Peso molecular:634.59
  • PROTAC ERRα Degrader-3

    CAS:
    PROTAC ERRα Degrader-3 is a potent, selective VHL-based PROTAC that degrades ERRα by over 80% at 30 nM, with no activity against ERRβ or ERRγ.
    Fórmula:C47H50F6N6O7S
    Forma y color:Solid
    Peso molecular:956.991
  • Methylpiperidino pyrazole

    CAS:
    Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.
    Fórmula:C29H31N3O3
    Pureza:98.84%
    Forma y color:Solid
    Peso molecular:469.57
  • PU-WS13

    CAS:
    PU-WS13 is an active molecule that can be used in life science related research. The CAS number of PU-WS13 is 1454619-14-7.
    Fórmula:C17H20Cl2N6S
    Pureza:99.09%
    Peso molecular:411.35
  • Endoxifen Z-isomer hydrochloride

    CAS:
    Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
    Fórmula:C25H28ClNO2
    Forma y color:Solid
    Peso molecular:409.95
  • Bazedoxifene

    CAS:
    Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.
    Fórmula:C30H34N2O3
    Pureza:98.79%
    Forma y color:Yellow Solid
    Peso molecular:470.61
  • AC-186

    CAS:
    AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.
    Fórmula:C18H17F3O
    Pureza:99.97%
    Forma y color:White Solid
    Peso molecular:306.32