Receptor de vasopresina
Los receptores de vasopresina son una familia de receptores acoplados a proteínas G que median los efectos de la vasopresina, una hormona involucrada en la regulación del equilibrio hídrico, la presión arterial y la función renal. Los agonistas y antagonistas de los receptores de vasopresina se estudian por su papel en el tratamiento de afecciones como la diabetes insípida, la hiponatremia y la insuficiencia cardíaca. Estos receptores también son objetivos importantes en la investigación sobre el equilibrio de líquidos y la salud cardiovascular. En CymitQuimica, ofrecemos una selección de moduladores de receptores de vasopresina de alta calidad para apoyar su investigación en endocrinología, nefrología y biología cardiovascular.
Se han encontrado 48 productos para "Receptor de vasopresina".
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Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Forma y color:SolidPeso molecular:1347.5Nelivaptan
CAS:Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.Fórmula:C30H32ClN3O8SPureza:99.46% - 99.89%Forma y color:SolidPeso molecular:630.11Balovaptan
CAS:Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.Fórmula:C22H24ClN5OPureza:99.88%Forma y color:White SolidPeso molecular:409.91Desmopressin
CAS:Desmopressin (DDAVP)(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin have led to its use in polyuric conditions including primary nocturnal enuresis, nocturia, and diabetes insipidus. Desmopressin works by limiting the amount of water that is eliminated in the urine. Desmopressin binds to V2 receptors in renal collecting ducts, increasing water reabsorption. It also stimulates release of von Willebrand factor from endothelial cells by acting on the V2 receptor.Fórmula:C46H64N14O12S2Pureza:97.45%Peso molecular:1069.22d[Cha4]-AVP
CAS:Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Fórmula:C50H71N13O11S2Pureza:98%Forma y color:SolidPeso molecular:1094.31(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Fórmula:C52H74N14O12S2Pureza:98%Forma y color:SolidPeso molecular:1151.38c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
CAS:c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm: potent, selective V2R agonist; EC50: 0.25 nM (hV2R), 0.05 nM (rV2R).Fórmula:C47H69ClN12O9S2Pureza:98%Forma y color:SolidPeso molecular:1045.71Velmupressin acetate
CAS:Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).Fórmula:C44H64ClN11O10S2Pureza:98%Forma y color:SolidPeso molecular:1006.63d[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Fórmula:C47H67N11O11S2Pureza:98%Forma y color:SolidPeso molecular:1026.2d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Fórmula:C52H72F3N13O13S2Forma y color:SolidPeso molecular:1208.33Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFórmula:C45H63N15O11S2Forma y color:SolidPeso molecular:1054.21[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Fórmula:C48H68N14O12Forma y color:SolidPeso molecular:1033.14(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Fórmula:C44H69N13O13S2Forma y color:SolidPeso molecular:1052.23Selepressin acetate
Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.Fórmula:C48H77N13O13S2Forma y color:SolidPeso molecular:1108.33(Phe2,Orn8)-Oxytocin
CAS:(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.Fórmula:C42H65N13O11S2Forma y color:SolidPeso molecular:992.18Endolide F
Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.Fórmula:C25H32N4O6Forma y color:SolidPeso molecular:484.23218D[LEU4,LYS8]-VP TFA
D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.Fórmula:C49H68F3N11O13S2Forma y color:SolidPeso molecular:1140.25(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.Fórmula:C54H76N14O11Forma y color:SolidPeso molecular:1097.27Ornipressin
CAS:Ornipressin is a vasoconstrictor, haemostatic and renal agent.Fórmula:C45H63N13O12S2Pureza:98%Forma y color:SolidPeso molecular:1042.19Velmupressin
CAS:Peptidic V2R agonist, c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2, with EC50: 0.07 nM (hV2R), 0.02 nM (rV2R); selective, short-acting.Fórmula:C42H60ClN11O8S2Pureza:98%Forma y color:SolidPeso molecular:946.58
![d[Cha4]-AVP](https://static.cymitquimica.com/products/TM/thumb-webp/TP2082.webp)
![d[Leu4,Lys8]-VP](https://static.cymitquimica.com/products/TM/thumb-webp/TP1927.webp)
![[Asu1,6-Arg8]Vasopressin](https://static.cymitquimica.com/products/TM/thumb-webp/T76510.webp)
