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cAMP

cAMP

cAMP es un segundo mensajero importante en muchos procesos biológicos, incluyendo la regulación del metabolismo, la expresión génica y el crecimiento celular. En la vía de señalización MAPK, cAMP puede modular la actividad de varias quinasas, incluida la PKA, que a su vez influye en la cascada MAPK. La desregulación de la señalización de cAMP está implicada en varias enfermedades, incluyendo el cáncer y los trastornos cardiovasculares. En CymitQuimica, ofrecemos una variedad de moduladores de cAMP para apoyar su investigación en transducción de señales, metabolismo y patología de enfermedades.

Se han encontrado 47 productos de "cAMP"

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  • Bucladesine sodium

    CAS:
    <p>Bucladesine sodium (DC2797) is a cAMP analog with cell-permeable properties.</p>
    Fórmula:C18H23N5NaO8P
    Pureza:96.56% - 99.76%
    Forma y color:White Powder
    Peso molecular:491.37
  • HJC0197

    CAS:
    <p>HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.</p>
    Fórmula:C19H21N3OS
    Pureza:98.05%
    Forma y color:Solid
    Peso molecular:339.45
  • MR-L2

    CAS:
    <p>MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).</p>
    Fórmula:C19H16Cl3FN4O
    Pureza:98.09% - 98.94%
    Forma y color:Solid
    Peso molecular:441.71
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Fórmula:C11H19N5
    Pureza:98.33% - 99.62%
    Forma y color:Solid
    Peso molecular:221.3
  • A-3 hydrochloride

    CAS:
    <p>A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.</p>
    Fórmula:C12H14Cl2N2O2S
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:321.22
  • CE3F4

    CAS:
    <p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>
    Fórmula:C11H10Br2FNO
    Pureza:97.15% - 98.06%
    Forma y color:Solid
    Peso molecular:351.01
  • ESI-05

    CAS:
    <p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>
    Fórmula:C16H18O2S
    Pureza:97.22%
    Forma y color:Solid
    Peso molecular:274.38
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Fórmula:C21H24N4O2S
    Pureza:99.64%
    Forma y color:Light Yellow To Yellow Solid
    Peso molecular:396.51
  • Bithionol

    CAS:
    <p>Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential to</p>
    Fórmula:C12H6Cl4O2S
    Pureza:99.04%
    Forma y color:White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)
    Peso molecular:356.05
  • MRS-1706

    CAS:
    <p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>
    Fórmula:C27H29N5O5
    Pureza:99.00%
    Forma y color:Solid
    Peso molecular:503.55
  • OX04528

    CAS:
    <p>OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.</p>
    Fórmula:C16H13F6NO2
    Pureza:99.74%
    Forma y color:Soild
    Peso molecular:365.27
  • BC 11-38

    CAS:
    <p>BC 11-38 is a potent, selective PDE biodepressant which is mainly effective against PDE11 (IC50 : 0.28 μM).</p>
    Fórmula:C15H16N2OS2
    Pureza:98.95% - 99.28%
    Forma y color:Solid
    Peso molecular:304.43
  • 2-PCCA hydrochloride

    CAS:
    <p>2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of GPR88-mediated cAMP production in HEK293 cells with an</p>
    Fórmula:C30H39Cl2N3O
    Pureza:97.54% - 99.36%
    Forma y color:Soild
    Peso molecular:528.56
  • Adenosine 3'-monophosphate (sodium salt hydrate)


    <p>Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.</p>
    Fórmula:C10H15N5NaO8P
    Forma y color:Solid
    Peso molecular:387.22
  • Anti-Cathelicidin/Camp Polyclonal Antibody


    <p>Antibody Type: Rabbit Polyclonal&lt;br&gt;<br>Application: IHC-P,IHC-Fr,ICC/IF,IF,ELISA&lt;br&gt;<br>Reactivity: (predicted:Mouse,Rat)</p>
    Forma y color:Liquid
    Peso molecular:Theoretical: 19 kDa.
  • GLP-1R modulator L7-028

    CAS:
    <p>GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.</p>
    Fórmula:C24H28N2O3
    Pureza:98.76% - >99.99%
    Forma y color:Solid
    Peso molecular:392.49
  • Pinoresinol 4-O-β-D-glucopyranoside

    CAS:
    <p>(+)-Pinoresinol-β-D-glucoside, also known as (+)-pinor, is a major active lignan furanoid found in Forsythia.</p>
    Fórmula:C26H32O11
    Pureza:99.32% - >99.99%
    Forma y color:Solid
    Peso molecular:520.53
  • Ro 20-1724

    CAS:
    <p>Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) is a widely used inhibitor of cyclic nucleotide phosphodiesterase with IC50 of 2.0 μM and Ki of 3.1</p>
    Fórmula:C15H22N2O3
    Pureza:98.82% - 99.79%
    Forma y color:Solid
    Peso molecular:278.35
  • SAX-187

    CAS:
    <p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>
    Fórmula:C15H13ClN4O2S2
    Pureza:97.82% - 98%
    Forma y color:Solid
    Peso molecular:380.87
  • RS-25344 hydrochloride

    CAS:
    <p>RS 25344 hydrochloride is a phosphodiesterase (PDE) 4 inhibitor</p>
    Fórmula:C19H14ClN5O4
    Pureza:99.25%
    Forma y color:Solid
    Peso molecular:411.8