
Canal de sodio
Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.
Se han encontrado 273 productos para "Canal de sodio".
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Tocainide
CAS:Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.Fórmula:C11H16N2OPureza:99.84%Forma y color:SolidPeso molecular:192.26Phenytoin
CAS:Phenytoin: a non-sedative hydantoin, antiepileptic with anticonvulsant effects, stabilizes neurons, prevents seizure spread, and relaxes muscles.Fórmula:C15H12N2O2Pureza:99.95%Forma y color:White SolidPeso molecular:252.27Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Fórmula:C21H29N3OPureza:99.62%Forma y color:White SolidPeso molecular:339.47NaV1.7 inhibitor-1
CAS:NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Fórmula:C23H30FNO4SPureza:99.89%Forma y color:SolidPeso molecular:435.55Ref: TM-T12181
1mg99,00€5mg241,00€1mL*10mM (DMSO)265,00€10mg385,00€25mg663,00€50mg888,00€100mg1.305,00€Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Fórmula:C12H14N2O2Pureza:99.91%Forma y color:SolidPeso molecular:218.25Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Fórmula:C21H28ClNOPureza:99.15% - 99.38%Forma y color:White SolidPeso molecular:345.91Lidocaine
CAS:Lidocaine, an amide local anesthetic, reduces pain and inflammation by dampening ICAM-1, cytokines, and neutrophil influx.Fórmula:C14H22N2OPureza:99.88% - >99.99%Forma y color:White SolidPeso molecular:234.34Tocainide hydrochloride
CAS:Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.Fórmula:C11H17ClN2OPureza:97%Forma y color:SolidPeso molecular:228.72Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Fórmula:C18H28N2O·HClPureza:99.89% - 99.9%Forma y color:White SolidPeso molecular:324.89Lamotrigine
CAS:Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Fórmula:C9H7Cl2N5Pureza:99.76% - 99.95%Forma y color:White SolidPeso molecular:256.09Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Forma y color:Crystal PowderPeso molecular:435.31Butamben
CAS:Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Fórmula:C11H15NO2Pureza:99.43%Forma y color:SolidPeso molecular:193.24Ropivacaine
CAS:Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.Fórmula:C17H26N2OPureza:97.75% - >99.99%Forma y color:SolidPeso molecular:274.40DSP-2230
CAS:DSP-2230 is a selective blocker of Nav1.7/Nav1.8.Fórmula:C20H20F3N5O2Pureza:97.14%Forma y color:SolidPeso molecular:419.4Ref: TM-T15174
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg99,00€25mg205,00€50mg334,00€100mg537,00€200mg762,00€QX-314 chloride
CAS:QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.Fórmula:C16H27ClN2OPureza:99.73%Forma y color:SolidPeso molecular:298.85Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Fórmula:C21H17ClF3N3O3Pureza:99.86%Forma y color:SolidPeso molecular:451.83Ref: TM-T15207
1mg58,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg166,00€25mg268,00€50mg403,00€100mg532,00€200mg705,00€PF-04885614
CAS:PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.Fórmula:C13H14F3N3OPureza:98.02%Forma y color:SolidPeso molecular:285.27Ref: TM-T12421
2mg39,00€5mg60,00€1mL*10mM (DMSO)60,00€10mg96,00€25mg166,00€50mg299,00€100mg424,00€200mg595,00€Articaine hydrochloride
CAS:Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.Fórmula:C13H21ClN2O3SPureza:99.76%Forma y color:SolidPeso molecular:320.84Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24Nefopam hydrochloride
CAS:Nefopam hydrochloride (Nefopam HCl) is the hydrochloride salt form of nefopam, a centrally-acting, non-opioid benzoxazocine with analgesic activity.Fórmula:C17H20ClNOPureza:99.32% - 99.85%Forma y color:SolidPeso molecular:289.8
