
Canal de sodio
Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.
Se han encontrado 258 productos de "Canal de sodio"
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Nav1.7 inhibitor
CAS:Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.Fórmula:C15H11Cl3FNO4SPureza:97.52%Forma y color:SolidPeso molecular:426.68Ref: TM-T12184
1mg42,00€2mg55,00€5mg89,00€10mg135,00€25mg264,00€50mg423,00€100mg677,00€1mL*10mM (DMSO)87,00€GX-936
CAS:GX-936, Selective Nav1.7 inhibitor, binds activated VSD4 to oppose inactivation, for pain perception research.Fórmula:C24H20F3N7O3S2Pureza:98.04%Forma y color:SolidPeso molecular:575.59ATX-II TFA
ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).Pureza:98%Forma y color:Odour SolidNav1.1 activator 1
CAS:Nav1.1 activator 1, Selective Nav1.1 agonist, BBB permeable, increases current decay time, for central nervous system disorder research.Fórmula:C24H23F3N4OPureza:99.99%Forma y color:SolidPeso molecular:440.46Ref: TM-T12179
1mg99,00€5mg249,00€10mg386,00€25mg758,00€50mg1.180,00€100mg1.848,00€1mL*10mM (DMSO)272,00€Relutrigine
CAS:Relutrigine, Oral sodium current inhibitor, suppresses sustained INa (SCN8A mutations), reduces neuronal excitability, for anticonvulsant therapy.Fórmula:C15H11F6N5O2Pureza:99.68%Forma y color:SolidPeso molecular:407.27Ref: TM-T69652
1mg260,00€5mg650,00€10mg1.009,00€25mg1.504,00€50mg1.963,00€100mg2.520,00€1mL*10mM (DMSO)583,00€KR-32568
CAS:KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).Fórmula:C13H12FN3O2Pureza:99.91%Forma y color:SolidPeso molecular:261.25NaV1.2/1.6 channel blocker-1
CAS:NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.Fórmula:C14H14N2OSPureza:99.54%Forma y color:SolidPeso molecular:258.34Ralitoline
CAS:Ralitoline (Ralitolinum) is an anticonvulsant with anticancer activity and sodium channel blocking activity.Fórmula:C13H13ClN2O2SPureza:98.45%Forma y color:SolidPeso molecular:296.77Elpetrigine
CAS:Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used to study epilepsy.Fórmula:C10H7Cl3N4Pureza:99.04% - 99.43%Forma y color:SolidPeso molecular:289.55Silperisone HCl
CAS:Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.Fórmula:C15H25ClFNSiPureza:99.97%Forma y color:SolidPeso molecular:301.9Nisoxetine hydrochloride
CAS:Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitorFórmula:C17H21NO2·HClPureza:99.21%Forma y color:White SolidPeso molecular:307.82TC-N 1752
CAS:TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.Fórmula:C25H27F3N6O3Pureza:99.71%Forma y color:SolidPeso molecular:516.52Ref: TM-T23439
1mg34,00€5mg75,00€10mg111,00€25mg245,00€50mg363,00€100mg515,00€200mg702,00€1mL*10mM (DMSO)84,00€NHE3-IN-1
CAS:NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。Fórmula:C12H10ClN3SPureza:99.93%Forma y color:SolidPeso molecular:263.75GDC-0310
CAS:GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.Fórmula:C25H29Cl2FN2O4SPureza:99.877%Forma y color:SolidPeso molecular:543.486-Iodoamiloride
CAS:6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.Fórmula:C6H8IN7OPureza:98%Forma y color:SolidPeso molecular:321.08Sodium Channel inhibitor 4
CAS:Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].Fórmula:C19H18ClN3O4S2Pureza:98%Forma y color:SolidPeso molecular:451.95(Rac)-AMG8379
CAS:(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.Fórmula:C25H16ClF2N3O5SPureza:99.6%Forma y color:SolidPeso molecular:543.93Ref: TM-T12655
1mg175,00€2mg264,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€1mL*10mM (DMSO)512,00€Aneratrigine
CAS:Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].Fórmula:C19H20ClF2N5O2S2Pureza:98%Forma y color:SolidPeso molecular:487.97PF 04531083
CAS:PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.Fórmula:C17H16ClN5O2Pureza:99.85%Forma y color:SolidPeso molecular:357.79SLC13A5-IN-1
CAS:SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).Fórmula:C19H19Cl3N2O3SPureza:99.67%Forma y color:SolidPeso molecular:461.79Ref: TM-T12931
1mg48,00€5mg92,00€10mg152,00€25mg268,00€50mg447,00€100mg623,00€200mg883,00€500mg1.305,00€1mL*10mM (DMSO)114,00€

