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Canal de sodio

Canal de sodio

Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.

Se han encontrado 258 productos de "Canal de sodio"

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  • Nav1.7 inhibitor

    CAS:
    Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.
    Fórmula:C15H11Cl3FNO4S
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:426.68

    Ref: TM-T12184

    1mg
    42,00€
    2mg
    55,00€
    5mg
    89,00€
    10mg
    135,00€
    25mg
    264,00€
    50mg
    423,00€
    100mg
    677,00€
    1mL*10mM (DMSO)
    87,00€
  • GX-936

    CAS:
    GX-936, Selective Nav1.7 inhibitor, binds activated VSD4 to oppose inactivation, for pain perception research.
    Fórmula:C24H20F3N7O3S2
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:575.59

    Ref: TM-T27521

    25mg
    1.908,00€
    50mg
    A consultar
    100mg
    A consultar
  • ATX-II TFA


    ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).
    Pureza:98%
    Forma y color:Odour Solid

    Ref: TM-T82936

    1mg
    1.035,00€
    5mg
    2.277,00€
    10mg
    3.420,00€
    25mg
    5.814,00€
  • Nav1.1 activator 1

    CAS:
    Nav1.1 activator 1, Selective Nav1.1 agonist, BBB permeable, increases current decay time, for central nervous system disorder research.
    Fórmula:C24H23F3N4O
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:440.46

    Ref: TM-T12179

    1mg
    99,00€
    5mg
    249,00€
    10mg
    386,00€
    25mg
    758,00€
    50mg
    1.180,00€
    100mg
    1.848,00€
    1mL*10mM (DMSO)
    272,00€
  • Relutrigine

    CAS:
    Relutrigine, Oral sodium current inhibitor, suppresses sustained INa (SCN8A mutations), reduces neuronal excitability, for anticonvulsant therapy.
    Fórmula:C15H11F6N5O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:407.27

    Ref: TM-T69652

    1mg
    260,00€
    5mg
    650,00€
    10mg
    1.009,00€
    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
    1mL*10mM (DMSO)
    583,00€
  • KR-32568

    CAS:
    KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).
    Fórmula:C13H12FN3O2
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:261.25

    Ref: TM-T36569

    5mg
    39,00€
    10mg
    55,00€
    25mg
    101,00€
    50mg
    152,00€
    100mg
    222,00€
    1mL*10mM (DMSO)
    46,00€
  • NaV1.2/1.6 channel blocker-1

    CAS:
    NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.
    Fórmula:C14H14N2OS
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:258.34

    Ref: TM-T72170

    1mg
    38,00€
    5mg
    81,00€
    10mg
    111,00€
    25mg
    215,00€
    50mg
    319,00€
    100mg
    475,00€
  • Ralitoline

    CAS:
    Ralitoline (Ralitolinum) is an anticonvulsant with anticancer activity and sodium channel blocking activity.
    Fórmula:C13H13ClN2O2S
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:296.77

    Ref: TM-T28503

    1mg
    81,00€
    5mg
    172,00€
    10mg
    259,00€
    25mg
    424,00€
    50mg
    620,00€
    100mg
    884,00€
  • Elpetrigine

    CAS:
    Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used to study epilepsy.
    Fórmula:C10H7Cl3N4
    Pureza:99.04% - 99.43%
    Forma y color:Solid
    Peso molecular:289.55

    Ref: TM-T31614

    1mg
    264,00€
    5mg
    650,00€
    10mg
    888,00€
    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Silperisone HCl

    CAS:
    Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.
    Fórmula:C15H25ClFNSi
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:301.9

    Ref: TM-T28778

    1mg
    84,00€
    5mg
    172,00€
    10mg
    259,00€
    25mg
    424,00€
    50mg
    583,00€
    100mg
    800,00€
    200mg
    1.071,00€
  • Nisoxetine hydrochloride

    CAS:
    Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor
    Fórmula:C17H21NO2·HCl
    Pureza:99.21%
    Forma y color:White Solid
    Peso molecular:307.82

    Ref: TM-T23070

    5mg
    66,00€
    10mg
    90,00€
    25mg
    166,00€
    50mg
    259,00€
    100mg
    411,00€
  • TC-N 1752

    CAS:
    TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.
    Fórmula:C25H27F3N6O3
    Pureza:99.71%
    Forma y color:Solid
    Peso molecular:516.52

    Ref: TM-T23439

    1mg
    34,00€
    5mg
    75,00€
    10mg
    111,00€
    25mg
    245,00€
    50mg
    363,00€
    100mg
    515,00€
    200mg
    702,00€
    1mL*10mM (DMSO)
    84,00€
  • NHE3-IN-1

    CAS:
    NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。
    Fórmula:C12H10ClN3S
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:263.75

    Ref: TM-T12219

    25mg
    52,00€
    50mg
    88,00€
  • GDC-0310

    CAS:
    GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.
    Fórmula:C25H29Cl2FN2O4S
    Pureza:99.877%
    Forma y color:Solid
    Peso molecular:543.48

    Ref: TM-T39208

    1mg
    154,00€
    5mg
    371,00€
    10mg
    590,00€
    25mg
    888,00€
    50mg
    1.251,00€
    100mg
    1.693,00€
  • 6-Iodoamiloride

    CAS:
    6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.
    Fórmula:C6H8IN7O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:321.08

    Ref: TM-T79246

    5mg
    A consultar
    50mg
    A consultar
  • Sodium Channel inhibitor 4

    CAS:
    Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].
    Fórmula:C19H18ClN3O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:451.95

    Ref: TM-T81134

    5mg
    A consultar
    50mg
    A consultar
  • (Rac)-AMG8379

    CAS:
    (Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.
    Fórmula:C25H16ClF2N3O5S
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:543.93

    Ref: TM-T12655

    1mg
    175,00€
    2mg
    264,00€
    5mg
    404,00€
    10mg
    592,00€
    25mg
    888,00€
    50mg
    1.243,00€
    100mg
    1.701,00€
    500mg
    3.402,00€
    1mL*10mM (DMSO)
    512,00€
  • Aneratrigine

    CAS:
    Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].
    Fórmula:C19H20ClF2N5O2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:487.97

    Ref: TM-T79834

    5mg
    A consultar
    50mg
    A consultar
  • PF 04531083

    CAS:
    PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.
    Fórmula:C17H16ClN5O2
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:357.79

    Ref: TM-T16514

    1mg
    38,00€
    5mg
    84,00€
    10mg
    137,00€
    25mg
    205,00€
    50mg
    313,00€
    1mL*10mM (DMSO)
    93,00€
  • SLC13A5-IN-1

    CAS:
    SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).
    Fórmula:C19H19Cl3N2O3S
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:461.79

    Ref: TM-T12931

    1mg
    48,00€
    5mg
    92,00€
    10mg
    152,00€
    25mg
    268,00€
    50mg
    447,00€
    100mg
    623,00€
    200mg
    883,00€
    500mg
    1.305,00€
    1mL*10mM (DMSO)
    114,00€