CymitQuimica logo
Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 337 productos de "Receptor GABA"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:354.38
  • Tiagabine

    CAS:
    <p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>
    Fórmula:C20H25NO2S2
    Pureza:99.25%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:375.55
  • 2'MeO6MF

    CAS:
    <p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>
    Fórmula:C17H14O3
    Pureza:99.28% - 99.63%
    Forma y color:Solid
    Peso molecular:266.29
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Fórmula:C20H28ClNO3S2
    Forma y color:Solid
    Peso molecular:430.02
  • rac-BHFF

    CAS:
    <p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency &gt;15x, efficacy &gt;149%, has anxiolytic effects, and is orally active.</p>
    Fórmula:C17H21F3O3
    Pureza:99.69% - >99.99%
    Forma y color:Solid
    Peso molecular:330.34
  • Songorine

    CAS:
    <p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>
    Fórmula:C22H31NO3
    Pureza:98% - 99.92%
    Forma y color:Solid
    Peso molecular:357.49
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Forma y color:Light Beige Crystalline Powder
    Peso molecular:109.3
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Fórmula:C16H14O4
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:270.28
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Fórmula:C6H6N2O2
    Pureza:99.94%
    Forma y color:Soild
    Peso molecular:138.1238
  • Loreclezole hydrochloride

    CAS:
    <p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>
    Fórmula:C10H7Cl4N3
    Forma y color:Solid
    Peso molecular:310.99
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Fórmula:C18H21ClF3N3O
    Pureza:99.03% - 99.95%
    Forma y color:Solid
    Peso molecular:387.83
  • Kavain

    CAS:
    <p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>
    Fórmula:C14H14O3
    Pureza:99.93% - ≥95%
    Forma y color:Solid
    Peso molecular:230.26
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Fórmula:C7H6O2
    Pureza:99.05% - 99.86%
    Forma y color:Solid
    Peso molecular:122.12
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Fórmula:C30H18O10
    Pureza:98.21% - 99.22%
    Forma y color:Odourless Whitish Solid
    Peso molecular:538.46
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Fórmula:C6H10ClNO2
    Pureza:98.42%
    Forma y color:Solid
    Peso molecular:163.602
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Fórmula:C4H10N2O2
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:118.13
  • Cyclothiazide

    CAS:
    <p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>
    Fórmula:C14H16ClN3O4S2
    Pureza:98.23% - 99.49%
    Forma y color:Crystals From Dilute Alcohol Solid
    Peso molecular:389.88
  • Isoflurane

    CAS:
    <p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>
    Fórmula:C3H2ClF5O
    Pureza:98%
    Forma y color:Clear Colorless Liquid Liquid
    Peso molecular:184.49
  • Pikamilone

    CAS:
    Pikamilone (Picamilon) is an intelligent medicine.
    Fórmula:C10H12N2O3
    Pureza:99.38%
    Forma y color:White Crystalline Powder
    Peso molecular:208.21
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Fórmula:C10H20CaN2O8S2
    Pureza:98% - 99.93%
    Forma y color:White Odorless Or Nearly Odorless Powder
    Peso molecular:400.48