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Caseína quinasa

Caseína quinasa

Las caseína quinasas son una familia de quinasas de proteínas serina/treonina que regulan varios procesos celulares, incluyendo la reparación del ADN, los ritmos circadianos y la transducción de señales. Estas quinasas están involucradas en la fosforilación de numerosas proteínas y están implicadas en enfermedades como el cáncer, los trastornos neurodegenerativos y los síndromes metabólicos. En CymitQuimica, ofrecemos una selección de inhibidores de caseína quinasa para apoyar su investigación en transducción de señales, regulación del ciclo celular y desarrollo terapéutico.

Se han encontrado 130 productos de "Caseína quinasa"

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  • Casein Kinase II Inhibitor IV Hydrochloride

    CAS:
    <p>Casein Kinase II Inhibitor IV HCl promotes keratinocyte differentiation, potential for skin disorder therapy.</p>
    Fórmula:C24H24ClN5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:465.93
  • CK2-IN-3


    <p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>
    Fórmula:C22H26N4O7
    Forma y color:Solid
    Peso molecular:458.46
  • Casein kinase 1δ-IN-19

    CAS:
    <p>Casein kinase1δ-IN-19 (compound 492) is a potent inhibitor of casein kinase 1δ. It is utilized in research related to neurodegenerative disorders, such as Alzheimer's disease.</p>
    Fórmula:C21H19N5O3
    Forma y color:Solid
    Peso molecular:389.407
  • Casein kinase 1δ-IN-23

    CAS:
    <p>Casein kinase1δ-IN-23 (compound 423) is an effective inhibitor of casein kinase1δ. It is applicable in research related to neurodegenerative diseases such as Alzheimer's disease.</p>
    Fórmula:C19H15N3O3S
    Forma y color:Solid
    Peso molecular:365.406
  • Casein kinase 1δ-IN-25

    CAS:
    <p>Casein kinase1δ-IN-25 (compound 487) is a potent inhibitor of casein kinase1δ. It is applicable in research on neurodegenerative diseases such as Alzheimer's disease.</p>
    Fórmula:C20H14FN3O4S2
    Forma y color:Solid
    Peso molecular:443.471
  • CK1δ-IN-3

    CAS:
    <p>CK1δ-IN-3 (compound 376) is a CK1δ (casein kinase 1δ) inhibitor that can be used to study neurodegenerative diseases such as Alzheimer's disease.</p>
    Fórmula:C24H19N3O2S
    Pureza:99.27%
    Forma y color:Solid
    Peso molecular:413.49
  • TMX-4113


    <p>TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].</p>
    Fórmula:C12H12N4O2S2
    Forma y color:Solid
    Peso molecular:308.38
  • Casein kinase 1δ-IN-17

    CAS:
    <p>Casein kinase1δ-IN-17 (compound 753) is an inhibitor of casein kinase 1δ (CK1δ). It is applicable in research related to neurodegenerative diseases.</p>
    Fórmula:C14H14N4S
    Forma y color:Solid
    Peso molecular:270.353
  • TMX-4116

    CAS:
    <p>TMX-4116 is a CK1α degrader targeting multiple cell lines with DC50s below 200 nM, used in multiple myeloma research and protein degradation strategy studies.</p>
    Fórmula:C17H19N5O4S
    Forma y color:Solid
    Peso molecular:389.43
  • CK2 inhibitor 2

    CAS:
    <p>CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.</p>
    Fórmula:C21H17ClN4O2
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:392.84