AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 623 productos para "AChR".
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Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56VU 0365114
CAS:VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).Fórmula:C22H14F3NO3Pureza:99.86%Forma y color:Red SolidPeso molecular:397.35Ref: TM-T13325
2mg35,00€5mg55,00€1mL*10mM (DMSO)62,00€10mg78,00€25mg130,00€50mg212,00€100mg318,00€200mg444,00€Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:SolidPeso molecular:424.328-Aminoadenine
CAS:8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.Fórmula:C5H6N6Pureza:99.82%Forma y color:SolidPeso molecular:150.14Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Fórmula:C7H17N2O2·ClPureza:95% - 99.98%Forma y color:White SolidPeso molecular:196.68Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Fórmula:C17H20N2S·HClPureza:99.85%Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Atropine methyl bromide
CAS:Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.Fórmula:C18H26BrNO3Pureza:99.7%Forma y color:White SolidPeso molecular:384.308Ref: TM-T14345
1mg34,00€5mg63,00€1mL*10mM (DMSO)70,00€10mg95,00€25mg167,00€50mg248,00€100mg363,00€200mg528,00€Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Fórmula:C9H15Cl2N3Pureza:98.72%Forma y color:SolidPeso molecular:236.142Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Fórmula:C12H14N2O2Pureza:99.9% - 99.91%Forma y color:SolidPeso molecular:218.25Adiphenine hydrochloride
CAS:Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.Fórmula:C20H26ClNO2Pureza:97.76% - 99.53%Forma y color:White Or Almost White PowderPeso molecular:347.879Acetamiprid
CAS:Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.Fórmula:C10H11ClN4Pureza:99.66% - 99.89%Forma y color:White PowderPeso molecular:222.67Lysipressin acetate(50-57-7(fb_acetate))
CAS:Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.Fórmula:C48H69N13O14S2Pureza:98.08%Forma y color:SolidPeso molecular:1116.28Rocuronium bromide
CAS:Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.Fórmula:C32H53BrN2O4Pureza:99.77% - >99.99%Forma y color:SolidPeso molecular:609.68Benzethonium chloride
CAS:Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.Fórmula:C27H42ClNO2Pureza:99.91%Forma y color:White SolidPeso molecular:448.081Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Fórmula:C12H17ClN2OPureza:99.42%Forma y color:SolidPeso molecular:240.729Carbachol
CAS:Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.Fórmula:C6H15ClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:182.65TAK-071
CAS:TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).Fórmula:C24H24FN3O3Pureza:98.02% - 99.82%Forma y color:SolidPeso molecular:421.46bPiDDB
CAS:bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.Fórmula:C24H38Br2N2Pureza:99.71%Forma y color:White SolidPeso molecular:514.38Dibucaine
CAS:Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.Fórmula:C20H29N3O2Pureza:99.69% - 99.88%Forma y color:White SolidPeso molecular:343.46
