AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Pirenzepine dihydrochloride
CAS:<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:White PowderPeso molecular:424.32VU 0365114
CAS:<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Fórmula:C22H14F3NO3Pureza:99.86%Forma y color:SolidPeso molecular:397.35Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Procainamide hydrochloride
CAS:<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Fórmula:C13H21N3O·HClPureza:99.83% - 99.97%Forma y color:White To Slightly Yellow PowderPeso molecular:271.79Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56Pancuronium dibromide
CAS:<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Fórmula:C35H60Br2N2O4Pureza:99.86%Forma y color:solidPeso molecular:732.67Gallamine triethiodide
CAS:<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Fórmula:C30H60I3N3O3Pureza:98.90%Forma y color:White Amorphous Powder SolidPeso molecular:891.53(Rac)-ABT-202 dihydrochloride
CAS:<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Fórmula:C9H15Cl2N3Pureza:97.4%Forma y color:SolidPeso molecular:236.142Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Fórmula:C18H26BrNO3Pureza:99.7%Forma y color:SolidPeso molecular:384.308Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59Acetamiprid
CAS:<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Fórmula:C10H11ClN4Pureza:99.66%Forma y color:White PowderPeso molecular:222.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Fórmula:C32H53BrN2O4Pureza:99.77% - >99.99%Forma y color:White Or Off-White PowderPeso molecular:609.68MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.48Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Fórmula:C20H26ClNO3Pureza:99.03% - 99.94%Forma y color:SolidPeso molecular:363.88Benzethonium chloride
CAS:<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Fórmula:C27H42ClNO2Pureza:99.91%Forma y color:White To Off-White Solid Solid Particulate/PowderPeso molecular:448.09Pyrantel tartrate
CAS:<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Fórmula:C15H20N2O6SPureza:99.96%Forma y color:White CrystalsPeso molecular:356.39Nebracetam hydrochloride
CAS:<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Fórmula:C12H17ClN2OPureza:99.23%Forma y color:SolidPeso molecular:240.729Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Fórmula:C6H15ClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:182.65Bethanechol chloride
CAS:<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Fórmula:C7H17N2O2·ClPureza:95% - 99.73%Forma y color:White CrystallinePeso molecular:196.68Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Fórmula:C22H22FN3O2Pureza:97.16% - 98%Forma y color:SolidPeso molecular:379.43
