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AChR

AChR

Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.

Se han encontrado 575 productos de "AChR"

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  • Solifenacin succinate

    CAS:
    <p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>
    Fórmula:C23H26N2O2·C4H6O4
    Pureza:99.85% - 99.98%
    Forma y color:Solid
    Peso molecular:480.56
  • Diphenmanil methylsulfate

    CAS:
    <p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>
    Fórmula:C20H24N·CH3O4S
    Pureza:98% - 99.27%
    Forma y color:Solid
    Peso molecular:389.51
  • Pirenzepine dihydrochloride

    CAS:
    <p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>
    Fórmula:C19H21N5O2·2HCl
    Pureza:99.48% - 99.62%
    Forma y color:White Powder
    Peso molecular:424.32
  • Temephos

    CAS:
    <p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>
    Fórmula:C16H20O6P2S3
    Pureza:≥95%
    Forma y color:White Crystalline Solid Or Liquid
    Peso molecular:466.47
  • Carbetapentane citrate

    CAS:
    <p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>
    Fórmula:C20H31NO3·C6H8O7
    Pureza:99.46%
    Forma y color:White To Off-White Solid
    Peso molecular:525.59
  • Zelminemab

    CAS:
    <p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>
    Pureza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)
    Forma y color:Liquid
  • Rivastigmine tartrate

    CAS:
    <p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>
    Fórmula:C14H22N2O2·C4H6O6
    Pureza:98% - 99.66%
    Forma y color:White To Off-White Powder
    Peso molecular:400.43
  • Dequalinium chloride

    CAS:
    <p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>
    Fórmula:C30H40Cl2N4
    Pureza:99.79% - 99.9%
    Forma y color:Solid
    Peso molecular:527.59
  • Cotinine

    CAS:
    <p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>
    Fórmula:C10H12N2O
    Pureza:98% - 99.89%
    Forma y color:Viscous Oil Solid
    Peso molecular:176.22
  • MK-7622

    CAS:
    <p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>
    Fórmula:C25H25N3O2
    Pureza:99.77% - 99.8%
    Forma y color:Solid
    Peso molecular:399.48
  • Dicyclomine hydrochloride

    CAS:
    <p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>
    Fórmula:C19H36ClNO2
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:345.95
  • Benactyzine hydrochloride

    CAS:
    <p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>
    Fórmula:C20H26ClNO3
    Pureza:99.03% - 99.94%
    Forma y color:Solid
    Peso molecular:363.88
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Fórmula:C21H25NO·CH4SO3
    Pureza:98.41% - 99.96%
    Forma y color:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecular:403.53
  • Procainamide hydrochloride

    CAS:
    <p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>
    Fórmula:C13H21N3O·HCl
    Pureza:99.83% - 99.97%
    Forma y color:White To Slightly Yellow Powder
    Peso molecular:271.79
  • VU 0365114

    CAS:
    <p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>
    Fórmula:C22H14F3NO3
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:397.35
  • Fipexide

    CAS:
    <p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>
    Fórmula:C20H21ClN2O4
    Pureza:97.6% - 99.95%
    Forma y color:Solid
    Peso molecular:388.84
  • (Rac)-ABT-202 dihydrochloride

    CAS:
    <p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>
    Fórmula:C9H15Cl2N3
    Pureza:97.4%
    Forma y color:Solid
    Peso molecular:236.142
  • Lysipressin acetate(50-57-7(fb_acetate))

    CAS:
    <p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction &amp; activates adenylate cyclase, is an antidiuretic in pigs &amp; marsupials.</p>
    Fórmula:C48H69N13O14S2
    Pureza:98.08%
    Forma y color:Solid
    Peso molecular:1116.28
  • Nebracetam hydrochloride

    CAS:
    <p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>
    Fórmula:C12H17ClN2O
    Pureza:99.23%
    Forma y color:Solid
    Peso molecular:240.729
  • nAChR agonist 1

    CAS:
    <p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>
    Fórmula:C20H18ClNO3S2
    Pureza:97.59%
    Forma y color:Solid
    Peso molecular:419.94