
AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 625 productos para "AChR".
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Gallamine triethiodide
CAS:Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.Fórmula:C30H60I3N3O3Pureza:98.90%Forma y color:White Amorphous Powder SolidPeso molecular:891.5291Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Fórmula:C17H20N2S·HClPureza:99.85%Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Fórmula:C12H17ClN2OPureza:99.42%Forma y color:SolidPeso molecular:240.729bPiDDB
CAS:bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.Fórmula:C24H38Br2N2Pureza:99.71%Forma y color:White SolidPeso molecular:514.38Valethamate bromide
CAS:Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.Fórmula:C19H32BrNO2Pureza:99.97%Forma y color:SolidPeso molecular:386.367Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Fórmula:C12H14N2O2Pureza:99.9% - 99.91%Forma y color:SolidPeso molecular:218.25Meclofenoxate hydrochloride
CAS:Meclofenoxate HCl (Lucidril) boosts memory and cognition; it's a DIMETHYLAMINOETHANOL and p-chlorophenoxyacetic acid ester.Fórmula:C12H17Cl2NO3Pureza:97.05%Forma y color:White Crystal PowderPeso molecular:294.174Orphenadrine Citrate
CAS:Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.Fórmula:C24H31NO8Pureza:99.58%Forma y color:White SolidPeso molecular:461.5048Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Fórmula:C21H29N3OPureza:99.62%Forma y color:White SolidPeso molecular:339.4745MN58b
CAS:MN58b is a selective inhibitor of choline kinase α (CHKα).Fórmula:C32H40Br2N4Pureza:97.23%Forma y color:SolidPeso molecular:640.495Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Fórmula:C21H27NO4SPureza:98% - 99.27%Forma y color:White SolidPeso molecular:389.508Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56PF-4348235 2HCl
PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.Fórmula:C36H51Cl3N4O7SPureza:99.85%Forma y color:SolidPeso molecular:790.24Procainamide hydrochloride
CAS:Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analogFórmula:C13H22ClN3OPureza:99.83% - 99.97%Forma y color:SolidPeso molecular:271.786Hexamethonium Bromide
CAS:Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.Fórmula:C12H30Br2N2Pureza:99.76% - 99.95%Forma y color:White SolidPeso molecular:362.19Clidinium bromide
CAS:Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.Fórmula:C22H26BrNO3Pureza:98.89% - 99.86%Forma y color:SolidPeso molecular:432.35MK-7622
CAS:MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.4849Lysipressin acetate(50-57-7(fb_acetate))
CAS:Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.Fórmula:C48H69N13O14S2Pureza:98.08%Forma y color:SolidPeso molecular:1116.27Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:SolidPeso molecular:424.32Tolterodine tartrate
CAS:Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.Fórmula:C22H31NO·C4H6O6Pureza:99.95%Forma y color:White-To-Off-White Crystalline PowderPeso molecular:475.58
