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AChR

AChR

Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.

Se han encontrado 625 productos para "AChR".

productos por página.
  • Gallamine triethiodide

    CAS:
    Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.
    Fórmula:C30H60I3N3O3
    Pureza:98.90%
    Forma y color:White Amorphous Powder Solid
    Peso molecular:891.5291
  • Promethazine hydrochloride

    CAS:
    Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
    Fórmula:C17H20N2S·HCl
    Pureza:99.85%
    Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Peso molecular:320.88
  • Nebracetam hydrochloride

    CAS:
    Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.
    Fórmula:C12H17ClN2O
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:240.729
  • bPiDDB

    CAS:
    bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.
    Fórmula:C24H38Br2N2
    Pureza:99.71%
    Forma y color:White Solid
    Peso molecular:514.38
  • Valethamate bromide

    CAS:
    Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.
    Fórmula:C19H32BrNO2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:386.367
  • Primidone

    CAS:
    Primidone (NCI-C56360) is a potent anticonvulsant agent.
    Fórmula:C12H14N2O2
    Pureza:99.9% - 99.91%
    Forma y color:Solid
    Peso molecular:218.25
  • Meclofenoxate hydrochloride

    CAS:
    Meclofenoxate HCl (Lucidril) boosts memory and cognition; it's a DIMETHYLAMINOETHANOL and p-chlorophenoxyacetic acid ester.
    Fórmula:C12H17Cl2NO3
    Pureza:97.05%
    Forma y color:White Crystal Powder
    Peso molecular:294.174
  • Orphenadrine Citrate

    CAS:
    Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.
    Fórmula:C24H31NO8
    Pureza:99.58%
    Forma y color:White Solid
    Peso molecular:461.5048
  • Disopyramide

    CAS:
    Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.
    Fórmula:C21H29N3O
    Pureza:99.62%
    Forma y color:White Solid
    Peso molecular:339.4745
  • MN58b

    CAS:
    MN58b is a selective inhibitor of choline kinase α (CHKα).
    Fórmula:C32H40Br2N4
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:640.495
  • Diphenmanil methylsulfate

    CAS:
    Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.
    Fórmula:C21H27NO4S
    Pureza:98% - 99.27%
    Forma y color:White Solid
    Peso molecular:389.508
  • Solifenacin succinate

    CAS:
    Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.
    Fórmula:C23H26N2O2·C4H6O4
    Pureza:99.85% - 99.98%
    Forma y color:Solid
    Peso molecular:480.56
  • PF-4348235 2HCl


    PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.
    Fórmula:C36H51Cl3N4O7S
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:790.24
  • Procainamide hydrochloride

    CAS:
    Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog
    Fórmula:C13H22ClN3O
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:271.786
  • Hexamethonium Bromide

    CAS:
    Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.
    Fórmula:C12H30Br2N2
    Pureza:99.76% - 99.95%
    Forma y color:White Solid
    Peso molecular:362.19
  • Clidinium bromide

    CAS:
    Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.
    Fórmula:C22H26BrNO3
    Pureza:98.89% - 99.86%
    Forma y color:Solid
    Peso molecular:432.35
  • MK-7622

    CAS:
    MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.
    Fórmula:C25H25N3O2
    Pureza:99.77% - 99.8%
    Forma y color:Solid
    Peso molecular:399.4849
  • Lysipressin acetate(50-57-7(fb_acetate))

    CAS:
    Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.
    Fórmula:C48H69N13O14S2
    Pureza:98.08%
    Forma y color:Solid
    Peso molecular:1116.27
  • Pirenzepine dihydrochloride

    CAS:
    Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
    Fórmula:C19H21N5O2·2HCl
    Pureza:99.48% - 99.62%
    Forma y color:Solid
    Peso molecular:424.32
  • Tolterodine tartrate

    CAS:
    Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.
    Fórmula:C22H31NO·C4H6O6
    Pureza:99.95%
    Forma y color:White-To-Off-White Crystalline Powder
    Peso molecular:475.58