AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 623 productos para "AChR".
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Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Fórmula:C20H24N·CH3O4SPureza:98% - 99.27%Forma y color:White SolidPeso molecular:389.51Dequalinium chloride
CAS:Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.Fórmula:C30H40Cl2N4Pureza:99.79% - 99.9%Forma y color:SolidPeso molecular:527.59Valethamate bromide
CAS:Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.Fórmula:C19H32BrNO2Pureza:99.97%Forma y color:SolidPeso molecular:386.37Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Fórmula:C12H14N2O2Pureza:99.9% - 99.91%Forma y color:SolidPeso molecular:218.25Methscopolamine
CAS:Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.Fórmula:C18H24BrNO4Pureza:99.12% - ≥98%Forma y color:White SolidPeso molecular:398.29Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:SolidPeso molecular:424.32Dicyclomine hydrochloride
CAS:Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.Fórmula:C19H36ClNO2Pureza:99.81%Forma y color:SolidPeso molecular:345.958-Aminoadenine
CAS:8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.Fórmula:C5H6N6Pureza:99.82%Forma y color:SolidPeso molecular:150.14Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Fórmula:C21H28ClNOPureza:99.15% - 99.38%Forma y color:White SolidPeso molecular:345.91Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Fórmula:C7H17N2O2·ClPureza:95% - 99.98%Forma y color:White SolidPeso molecular:196.68Lysipressin acetate(50-57-7(fb_acetate))
CAS:Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.Fórmula:C48H69N13O14S2Pureza:98.08%Forma y color:SolidPeso molecular:1116.28Oxybutynin chloride
CAS:Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.Fórmula:C22H32ClNO3Pureza:99.27% - >99.99%Forma y color:White SolidPeso molecular:393.96Otilonium bromide
CAS:Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.Fórmula:C29H43BrN2O4Pureza:99.78% - 99.88%Forma y color:SolidPeso molecular:563.57MK-7622
CAS:MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.48TAK-071
CAS:TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).Fórmula:C24H24FN3O3Pureza:98.02% - 99.82%Forma y color:SolidPeso molecular:421.46Pyrantel tartrate
CAS:Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Fórmula:C15H20N2O6SPureza:99.96%Forma y color:White CrystalsPeso molecular:356.39Hexamethonium Bromide
CAS:Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.Fórmula:C12H30Br2N2Pureza:99.76% - 99.95%Forma y color:White SolidPeso molecular:362.19(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Fórmula:C9H15Cl2N3Pureza:98.72%Forma y color:SolidPeso molecular:236.142Propantheline bromide
CAS:Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscleFórmula:C23H30BrNO3Pureza:97.11% - 98%Forma y color:White SolidPeso molecular:448.4
