AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 625 productos para "AChR".
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PTI-125 HCl
PTI-125 HCl (Simufilamum HCl) binds and reverses an altered conformation of the scaffolding protein filamin A found in Alzheimer's disease brain.Fórmula:C15H22ClN3OPureza:99.64%Peso molecular:295.81Perindoprilat
CAS:Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.Fórmula:C17H28N2O5Pureza:99.21%Forma y color:White SolidPeso molecular:340.41Methylatropine (nitrate)
CAS:Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.Fórmula:C18H26N2O6Forma y color:SolidPeso molecular:366.414nAChR modulator-1
CAS:nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .Fórmula:C12H8ClN3O2Forma y color:SolidPeso molecular:261.66ANQ-9040
CAS:ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92(S)-OPC-51803
CAS:(S)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.Fórmula:C19H16N2O2Pureza:98.73% - 99.59%Forma y color:White SolidPeso molecular:304.3425Lu AE51090
CAS:Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.Fórmula:C24H29N3O3Pureza:99.57%Forma y color:White SolidPeso molecular:407.51(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS:(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.Fórmula:C22H32ClNO2Forma y color:SolidPeso molecular:377.95AC1-IN-1
CAS:AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).Fórmula:C18H18FN5O2Pureza:99.89%Forma y color:White SolidPeso molecular:355.3662Muscarine
CAS:Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.Fórmula:C9H20NO2Pureza:98%Forma y color:SolidPeso molecular:174.26Rivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.Fórmula:C10H16Cl2N2Pureza:99.4%Forma y color:SoildPeso molecular:235.15TC-2559 difumarate
CAS:TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.Fórmula:C20H26N2O9Forma y color:SolidPeso molecular:438.43α-Bungarotoxin
CAS:Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).Fórmula:C338H529N97O105S11Pureza:98%Forma y color:SolidPeso molecular:7984.14(R)-Dinotefuran
CAS:(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.Fórmula:C7H14N4O3Forma y color:SolidPeso molecular:202.21M1/M4 muscarinic agonist 1
M1/M4 muscarinic agonist 1 (Compound 41) is a selective muscarinic M4/M1 agonist with EC50 values of 14 nM for M4 receptors and 55 nM for M1 receptors. This compound is utilized in research related to psychiatric disorders, including schizophrenia and delusional disorders.Fórmula:C23H34N2O2Peso molecular:370.26203M4 mAChR agonist-1
CAS:M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).Fórmula:C14H18N4OSPureza:99.14%Forma y color:SolidPeso molecular:290.384G-Protein antagonist peptide
CAS:Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.Fórmula:C57H64N12O9SPureza:98%Forma y color:SolidPeso molecular:1093.27trans-Cevimeline hydrochloride
CAS:AF 102A hydrochloride is a biochemical.Fórmula:C10H18ClNOSForma y color:SolidPeso molecular:235.77Atracurium
CAS:Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.Fórmula:C53H72N2O122Forma y color:SolidPeso molecular:929.14(R)-(+)-Anatabine
CAS:(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.Fórmula:C10H12N2Pureza:98%Forma y color:SolidPeso molecular:160.22
