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Receptor de opioides

Receptor de opioides

Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.

Se han encontrado 353 productos para "Receptor de opioides".

productos por página.
  • Matrine

    CAS:
    Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
    Fórmula:C15H24N2O
    Pureza:99.77% - >99.99%
    Forma y color:White Solid
    Peso molecular:248.3639
  • Naltrexone hydrochloride

    CAS:
    Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.
    Fórmula:C20H24ClNO4
    Pureza:98.72% - 99.65%
    Forma y color:Solid
    Peso molecular:377.862
  • Alvimopan

    CAS:
    Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
    Fórmula:C25H32N2O4
    Pureza:99.47% - 99.78%
    Forma y color:Solid
    Peso molecular:424.5326
  • Apitegromab

    CAS:
    Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including
    Pureza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)
    Forma y color:Liquid
    Peso molecular:145.06 kDa (Predicted)
  • Loperamide hydrochloride

    CAS:
    Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
    Fórmula:C29H34Cl2N2O2
    Pureza:99.91% - >99.99%
    Forma y color:White Solid
    Peso molecular:513.498
  • LY2940094

    CAS:
    LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
    Fórmula:C22H23ClF2N4O2S
    Pureza:99.4%
    Forma y color:White Solid
    Peso molecular:480.958
  • Samidorphan HCl

    CAS:
    Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.
    Fórmula:C21H27ClN2O4
    Pureza:96.79% - 97.85%
    Forma y color:Solid
    Peso molecular:406.9
  • ZT 52656A hydrochloride

    CAS:
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Fórmula:C19H26ClF3N2O
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:390.871
  • Moguisteine

    CAS:
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Fórmula:C16H21NO5S
    Pureza:99.98%
    Forma y color:White Solid
    Peso molecular:339.41
  • BTRX-335140

    CAS:
    BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.
    Fórmula:C25H32FN5O2
    Pureza:98% - 99.89%
    Forma y color:White Solid
    Peso molecular:453.5523
  • Meptazinol hydrochloride

    CAS:
    Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
    Fórmula:C15H23NO·HCl
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:269.81
  • CP 866087

    CAS:
    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
    Fórmula:C24H30N2O3S
    Pureza:99.22% - 99.74%
    Forma y color:Solid
    Peso molecular:426.57
  • Trimebutine maleate

    CAS:
    Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.
    Fórmula:C26H33NO9
    Pureza:99.89% - 99.98%
    Forma y color:White Solid
    Peso molecular:503.55
  • Sinomenine hydrochloride

    CAS:
    Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
    Fórmula:C19H24ClNO4
    Pureza:99.43%
    Forma y color:White Solid
    Peso molecular:365.85
  • SNC 80

    CAS:
    SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.
    Fórmula:C28H39N3O2
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:449.63
  • Dermorphin

    CAS:
    Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
    Fórmula:C40H50N8O10
    Pureza:98.82%
    Forma y color:White Solid
    Peso molecular:802.8726
  • KOR agonist 6


    KOR agonist 6 is a KOR agonist with a Ki value of 0.25 pM. In CHO cells, it exhibits agonistic activity on MOR and DOR and inhibits forskolin-stimulated cAMP accumulation. The compound stimulates KOR-mediated [35S]GTPγS binding in HEK293 cells expressing KOR and effectively suppresses cAMP accumulation as a potent agonist, showing lower β-arrestin recruitment efficacy. Additionally, KOR agonist 6 demonstrates analgesic effects in mice and can be employed in the study of analgesics with reduced central nervous system (CNS) side effects.
    Forma y color:Odour Solid
  • Dynorphin (2-17), amide, porcine


    Dynorphin (2-17), amide, porcine is a C-terminally amidated KOR agonist with enhanced protease resistance.
    Fórmula:C90H147N31O20
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1983.33
  • μ/κ/δ opioid receptor agonist 1


    μ/κ/δopioid receptor agonist1 is an agonist for the μ opioid receptor (MOR), κ opioid receptor (KOR), and δ opioid receptor (DOR). It produces potent and long-lasting analgesic effects in the tail flick test through peripheral MOR and KOR activation.
    Fórmula:C35H45FN8O8
    Forma y color:Solid
    Peso molecular:724.33444
  • Dynorphin (2-17), porcine acetate


    Dynorphin (2-17), porcine acetate is a porcine dynorphin fragment that acts as a potent KOR agonist.
    Fórmula:C92H150N30O23
    Pureza:98.19%
    Peso molecular:2044.40