Receptor de bradicinina
Los receptores de bradicinina son GPCR que median los efectos de la bradicinina, un péptido involucrado en las respuestas inflamatorias, la sensación de dolor y la regulación de la presión arterial. Hay dos tipos principales de receptores de bradicinina, B1 y B2, cada uno con roles distintos en procesos fisiopatológicos. Los antagonistas de los receptores de bradicinina se utilizan en el tratamiento de afecciones como el angioedema hereditario, el dolor crónico y la hipertensión. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de bradicinina de alta calidad para apoyar su investigación en inflamación, manejo del dolor y biología cardiovascular.
Se han encontrado 59 productos de "Receptor de bradicinina"
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Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.58%Forma y color:SoildPeso molecular:784.58Bradykinin (1-7)
CAS:<p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>Fórmula:C35H52N10O9Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:756.85FR167344 free base
CAS:<p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>Fórmula:C30H28BrCl2N5O4Pureza:98%Forma y color:SolidPeso molecular:673.38Bradykinin (1-6)
CAS:<p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>Fórmula:C30H45N9O8Pureza:98%Forma y color:SolidPeso molecular:659.73Labradimil
CAS:<p>Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.</p>Fórmula:C49H75N15O12SPureza:98%Forma y color:SolidPeso molecular:1098.29MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Fórmula:C60H90N20O11SPureza:98%Forma y color:SolidPeso molecular:1299.56Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Fórmula:C16H28N6O4Pureza:98%Forma y color:SolidPeso molecular:368.43[Des-Arg9]-Bradykinin
CAS:<p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>Fórmula:C44H61N11O10Pureza:98%Forma y color:SolidPeso molecular:904.02Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:<p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>Fórmula:C47H66N12O11Pureza:98%Forma y color:SolidPeso molecular:975.11Icatibant
CAS:<p>Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).</p>Fórmula:C59H89N19O13SPureza:98%Forma y color:White SolidPeso molecular:1304.52Lys-[Des-Arg9]Bradykinin
CAS:<p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>Fórmula:C50H73N13O11Pureza:98%Forma y color:SolidPeso molecular:1032.21[Des-Arg10]-HOE I40 TFA
<p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>Fórmula:C53H77N15O12S·xC2HF3O2Forma y color:SolidBombinakinin M
CAS:<p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>Fórmula:C100H159N31O24Pureza:98%Forma y color:SolidPeso molecular:2179.55[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:<p>Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.</p>Fórmula:C50H75N15O10Pureza:98%Forma y color:SolidPeso molecular:1046.23Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Fórmula:C36H49Cl3N6O6SForma y color:SolidPeso molecular:800.23NPC 567
CAS:<p>NPC 567 is an antagonist of the bradykinin receptor.</p>Fórmula:C60H87N19O13Pureza:98%Forma y color:SolidPeso molecular:1282.48Fasitibant chloride hydrochloride
CAS:<p>Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.</p>Fórmula:C36H50Cl4N6O6SForma y color:SolidPeso molecular:836.7Lys-Bradykinin
CAS:<p>Endogenous bradykinin receptor agonist</p>Fórmula:C56H85N17O12Pureza:98%Forma y color:SolidPeso molecular:1188.38Zoliprofen
CAS:<p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>Fórmula:C12H11NO3SPureza:99.62%Forma y color:SolidPeso molecular:249.29Retrobradykinin
CAS:<p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>Fórmula:C50H73N15O11Forma y color:SolidPeso molecular:1060.228
![[Des-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT7645.webp&w=3840&q=75)
![Sar-[D-Phe8]-des-Arg9-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1917.webp&w=3840&q=75)
![Lys-[Des-Arg9]Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1918.webp&w=3840&q=75)
![[Phe8Ψ(CH-NH)-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2076.webp&w=3840&q=75)
