
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 441 productos de "Receptor de dopamina"
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Protein deglycase DJ-1 against-1
CAS:Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Fórmula:C24H23N3O4Pureza:97.23%Forma y color:SolidPeso molecular:417.46(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS:(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H14D5Cl2N3SForma y color:SolidPeso molecular:289.28L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Fórmula:C18H19ClN4Pureza:98%Forma y color:SolidPeso molecular:326.82Ropinirole
CAS:Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Fórmula:C16H24N2OPureza:99.68%Forma y color:SolidPeso molecular:260.38Dopamine D4 receptor ligand 2
CAS:Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Fórmula:C20H24ClN3O2Forma y color:SolidPeso molecular:373.88Vanoxerine
CAS:Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).Fórmula:C28H32F2N2OPureza:98%Forma y color:SolidPeso molecular:450.56Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Fórmula:C12H15N3O2Pureza:98%Forma y color:SolidPeso molecular:233.27A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Fórmula:C22H24ClNPureza:98%Forma y color:SolidPeso molecular:337.89Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Fórmula:C18H22ClN3O3SForma y color:SolidPeso molecular:395.9Bromperidol decanoate
CAS:Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.Fórmula:C31H41BrFNO3Forma y color:SolidPeso molecular:574.56LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Fórmula:C17H14O5Pureza:98%Forma y color:SolidPeso molecular:298.29Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Fórmula:C22H25NO6Pureza:98%Forma y color:SolidPeso molecular:399.44Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Fórmula:C24H28ClN3OSPureza:95.51%Forma y color:SolidPeso molecular:442.02CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Fórmula:C12H17N5Pureza:98%Forma y color:SolidPeso molecular:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Fórmula:C34H35F2N3O6Pureza:98%Forma y color:SolidPeso molecular:619.66NGB 2904 hydrochloride
CAS:dopamine D3 receptor antagonistFórmula:C28H30Cl3N3OPureza:98%Forma y color:SolidPeso molecular:530.92Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Fórmula:C25H31NOPureza:98%Forma y color:SolidPeso molecular:361.52PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Fórmula:C11H17N3SPureza:98%Forma y color:SolidPeso molecular:223.34U-101958 Maleate
CAS:U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.Fórmula:C25H33N3O5Pureza:98%Forma y color:SolidPeso molecular:455.55Roxindole hydrochloride
CAS:Dopamine D2 autoreceptor agonistFórmula:C23H27ClN2OPureza:98%Forma y color:SolidPeso molecular:382.93
