
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 443 productos de "Receptor de dopamina"
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Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Fórmula:C21H29ClN2O5Pureza:99.52%Forma y color:SolidPeso molecular:424.92Bromocriptine mesylate
CAS:Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Fórmula:C33H44BrN5O8SPureza:99.85% - 99.96%Forma y color:White SolidPeso molecular:750.7PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Fórmula:C24H26N4O5Pureza:99.13%Forma y color:SolidPeso molecular:450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Fórmula:C17H25N3O5SPureza:99.65%Forma y color:SolidPeso molecular:383.46Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Fórmula:C18H19ClN4OPureza:98.65% - 99.94%Forma y color:SolidPeso molecular:342.82Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Fórmula:C23H31ClN4O2SPureza:99.37%Forma y color:White SolidPeso molecular:463SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Fórmula:C17H19Cl2NOPureza:98% - 99.83%Forma y color:SolidPeso molecular:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€A-381393
CAS:A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Fórmula:C20H24N4Pureza:99.00%Forma y color:SolidPeso molecular:320.43Ref: TM-T5397
1mg40,00€5mg80,00€10mg117,00€25mg210,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)88,00€Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Fórmula:C24H23ClF3NPureza:99.99%Forma y color:SolidPeso molecular:417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Forma y color:SolidPeso molecular:463.87Pridopidine
CAS:Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Fórmula:C15H23NO2SPureza:95.2% - 99.89%Forma y color:SolidPeso molecular:281.41lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Forma y color:SolidPeso molecular:565.7Ropinirole hydrochloride
CAS:Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Fórmula:C16H24N2O·HClPureza:99.87% - 99.98%Forma y color:Off-White SolidPeso molecular:296.84(-)-Isocorypalmine
CAS:(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine), a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.Fórmula:C20H23NO4Pureza:98.18% - 99.97%Forma y color:SolidPeso molecular:341.4Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Fórmula:C11H16ClNO4Pureza:95.00%Forma y color:SolidPeso molecular:261.7Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Fórmula:C14H25Cl2N3O3Pureza:99.33%Forma y color:SolidPeso molecular:354.27MPTP hydrochloride
CAS:MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.Fórmula:C12H16ClNPureza:96.35% - >99.99%Forma y color:SolidPeso molecular:209.72Ref: TM-T4081
5mg35,00€10mg50,00€25mg85,00€50mg138,00€100mg187,00€200mg298,00€500mg472,00€1mL*10mM (DMSO)52,00€Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Fórmula:C8H12N2Pureza:98%Forma y color:LiquidPeso molecular:136.19Ref: TM-T9540
5mgA consultar10mgA consultar25mgA consultar50mgA consultar100mgA consultar200mgA consultar500mgA consultarZatebradine
CAS:Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Fórmula:C26H36N2O5Pureza:98%Forma y color:SolidPeso molecular:456.57Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Fórmula:C10H17N3SPureza:99.78%Forma y color:SolidPeso molecular:211.33
