
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 441 productos de "Receptor de dopamina"
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PD168,077
CAS:PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.Fórmula:C20H22N4OPureza:98%Forma y color:SolidPeso molecular:334.41Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Fórmula:C26H30N2O4SPureza:98%Forma y color:SolidPeso molecular:466.59Nafadotride
CAS:Nafadotride is a dopamine D3 receptor antagonist.Fórmula:C22H27N3O2Forma y color:SolidPeso molecular:365.47WAY-260022
CAS:WAY-260022 is the norepinephrine transporter inhibitor.Fórmula:C21H31F3N2O2Pureza:97.61% - 99.41%Forma y color:SolidPeso molecular:400.48(R)-PF-06256142
CAS:(R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.Fórmula:C21H16N4O2Forma y color:SolidPeso molecular:356.38L 741742 hydrochloride
CAS:L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.Fórmula:C23H26Cl2N2OPureza:99.9%Forma y color:SolidPeso molecular:417.37Org-10490
CAS:Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.Fórmula:C17H19NOPureza:98%Forma y color:SolidPeso molecular:253.34ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Fórmula:C23H34N4OSPureza:98%Forma y color:SolidPeso molecular:414.61GBR 12783
CAS:GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.Fórmula:C28H32N2OPureza:98%Forma y color:SolidPeso molecular:412.57Foscarbidopa
CAS:Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Forma y color:SolidPeso molecular:306.21Talipexole
CAS:Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.Fórmula:C10H15N3SPureza:98%Forma y color:SolidPeso molecular:209.31UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C23H28Cl2N4O2Pureza:98.78% - 98.78%Forma y color:SolidPeso molecular:463.4Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Fórmula:C13H18N2Pureza:98%Forma y color:SolidPeso molecular:202.3PD 120697
CAS:PD 120697 is a dopamine antagonist with central dopamine agonist properties.Fórmula:C11H15N3SPureza:98%Forma y color:SolidPeso molecular:221.32Acetophenazine
CAS:Acetophenazine is an anxiolytic compound that is used in the study of depression.Fórmula:C23H29N3O2SPureza:99.30%Forma y color:SoildPeso molecular:411.56L-750,667 Trihydrochloride
CAS:L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.Fórmula:C18H22Cl3IN4Pureza:99.63%Forma y color:SolidPeso molecular:527.66Tesofensine
CAS:Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.Fórmula:C17H23Cl2NOPureza:98%Forma y color:SolidPeso molecular:328.286-Chloromelatonin
CAS:6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.Fórmula:C13H15ClN2O2Pureza:97.26% - 99.25%Forma y color:SolidPeso molecular:266.72CP-226269
CAS:<p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>Fórmula:C18H19FN4Pureza:99.08%Forma y color:SolidPeso molecular:310.37(-)-GSK598809
CAS:(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.Fórmula:C22H23F4N5OSPureza:98%Forma y color:SolidPeso molecular:481.51
