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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 441 productos de "Receptor de dopamina"

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  • PD168,077

    CAS:
    PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.
    Fórmula:C20H22N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:334.41
  • Savoxepin mesylate

    CAS:
    Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.
    Fórmula:C26H30N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:466.59
  • Nafadotride

    CAS:
    Nafadotride is a dopamine D3 receptor antagonist.
    Fórmula:C22H27N3O2
    Forma y color:Solid
    Peso molecular:365.47
  • WAY-260022

    CAS:
    WAY-260022 is the norepinephrine transporter inhibitor.
    Fórmula:C21H31F3N2O2
    Pureza:97.61% - 99.41%
    Forma y color:Solid
    Peso molecular:400.48
  • (R)-PF-06256142

    CAS:
    (R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.
    Fórmula:C21H16N4O2
    Forma y color:Solid
    Peso molecular:356.38
  • L 741742 hydrochloride

    CAS:
    L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.
    Fórmula:C23H26Cl2N2O
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:417.37
  • Org-10490

    CAS:
    Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.
    Fórmula:C17H19NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:253.34
  • ST-836

    CAS:
    ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .
    Fórmula:C23H34N4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:414.61
  • GBR 12783

    CAS:
    GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.
    Fórmula:C28H32N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:412.57
  • Foscarbidopa

    CAS:
    Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
    Fórmula:C10H15N2O7P
    Pureza:96.17% - 97.27%
    Forma y color:Solid
    Peso molecular:306.21
  • Talipexole

    CAS:
    Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.
    Fórmula:C10H15N3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:209.31
  • UNC9975

    CAS:
    <p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>
    Fórmula:C23H28Cl2N4O2
    Pureza:98.78% - 98.78%
    Forma y color:Solid
    Peso molecular:463.4
  • Dicarbine

    CAS:
    Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.
    Fórmula:C13H18N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:202.3
  • PD 120697

    CAS:
    PD 120697 is a dopamine antagonist with central dopamine agonist properties.
    Fórmula:C11H15N3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:221.32
  • Acetophenazine

    CAS:
    Acetophenazine is an anxiolytic compound that is used in the study of depression.
    Fórmula:C23H29N3O2S
    Pureza:99.30%
    Forma y color:Soild
    Peso molecular:411.56
  • L-750,667 Trihydrochloride

    CAS:
    L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.
    Fórmula:C18H22Cl3IN4
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:527.66
  • Tesofensine

    CAS:
    Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.
    Fórmula:C17H23Cl2NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:328.28
  • 6-Chloromelatonin

    CAS:
    6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
    Fórmula:C13H15ClN2O2
    Pureza:97.26% - 99.25%
    Forma y color:Solid
    Peso molecular:266.72
  • CP-226269

    CAS:
    <p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>
    Fórmula:C18H19FN4
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:310.37
  • (-)-GSK598809

    CAS:
    (-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.
    Fórmula:C22H23F4N5OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.51