
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 441 productos de "Receptor de dopamina"
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Lenperone HCl
CAS:Lenperone HCl is a dopamine antagonist and an antipsychotic agent.Fórmula:C22H24ClF2NO2Pureza:98%Forma y color:SolidPeso molecular:407.88Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Fórmula:C20H29FN2O3Pureza:98.97% - >99.99%Forma y color:SolidPeso molecular:364.45A-77636
CAS:A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Fórmula:C20H27NO3Pureza:98%Forma y color:SolidPeso molecular:329.43Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Fórmula:C22H26ClNPureza:98%Forma y color:SolidPeso molecular:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Fórmula:C20H25BrN4OForma y color:SolidPeso molecular:417.34SKF-104557
CAS:N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.Fórmula:C13H18N2OForma y color:SolidPeso molecular:218.29A 68930 hydrochloride
CAS:A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].Fórmula:C16H18ClNO3Forma y color:Off-White SolidPeso molecular:307.77SB269652
CAS:SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.Fórmula:C27H30N4OPureza:98%Forma y color:SolidPeso molecular:426.55SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Fórmula:C19H22BrNO2Pureza:98%Forma y color:SolidPeso molecular:376.29Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Fórmula:C28H37N5O2SForma y color:SolidPeso molecular:507.69GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Fórmula:C28H32Cl2F2N2OPureza:98%Forma y color:SolidPeso molecular:521.47DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Fórmula:C11H11Cl2NPureza:96.7%Forma y color:SolidPeso molecular:228.12D4R agonist-1
CAS:D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.Fórmula:C19H22N4SPureza:98.44%Forma y color:SolidPeso molecular:338.47Octoclothepin maleate salt
CAS:Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.Fórmula:C23H25ClN2O4SForma y color:SolidPeso molecular:460.97RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Fórmula:C24H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:429.38SV-156
CAS:SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).Fórmula:C21H23BrN2O2Forma y color:SolidPeso molecular:415.32SKF-75670 Hydrobromide
CAS:SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.Fórmula:C17H20BrNO2Forma y color:SolidPeso molecular:350.25FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Fórmula:C11H14N4OForma y color:SolidPeso molecular:218.26S-3608
CAS:S-3608 is an atypical dopamine agonist.Fórmula:C16H20ClN3OSForma y color:SolidPeso molecular:337.87UNC9995
CAS:UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).Fórmula:C20H21Cl2N3OSPureza:98%Forma y color:SolidPeso molecular:422.37
