
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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Clothixamide
CAS:<p>Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.</p>Fórmula:C24H28ClN3OSPureza:95.51%Forma y color:SolidPeso molecular:442.02CI-943
CAS:<p>CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.</p>Fórmula:C12H17N5Pureza:98%Forma y color:SolidPeso molecular:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Fórmula:C34H35F2N3O6Pureza:98%Forma y color:SolidPeso molecular:619.66Butaclamol free base
CAS:<p>Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.</p>Fórmula:C25H31NOPureza:98%Forma y color:SolidPeso molecular:361.52PD 118440
CAS:<p>PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.</p>Fórmula:C11H17N3SPureza:98%Forma y color:SolidPeso molecular:223.34Sch 24518
CAS:<p>Sc h24518 is an antagonist of D1 receptor.</p>Fórmula:C16H17BrClNOPureza:98%Forma y color:SolidPeso molecular:354.67Dicarbine
CAS:<p>Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.</p>Fórmula:C13H18N2Pureza:98%Forma y color:SolidPeso molecular:202.3L-750,667 Trihydrochloride
CAS:<p>L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.</p>Fórmula:C18H22Cl3IN4Pureza:99.63%Forma y color:SolidPeso molecular:527.666-Chloromelatonin
CAS:<p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>Fórmula:C13H15ClN2O2Pureza:98.01% - 99.25%Forma y color:SolidPeso molecular:266.72A-77636
CAS:<p>A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50</p>Fórmula:C20H27NO3Pureza:98%Forma y color:SolidPeso molecular:329.43D4R agonist-1
CAS:<p>D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.</p>Fórmula:C19H22N4SPureza:98.44%Forma y color:SolidPeso molecular:338.47PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Forma y color:SolidPeso molecular:554.34SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Forma y color:SolidPeso molecular:317.81WAY-260022
CAS:<p>WAY-260022 is the norepinephrine transporter inhibitor.</p>Fórmula:C21H31F3N2O2Pureza:97.61% - 99.41%Forma y color:SolidPeso molecular:400.48UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C23H28Cl2N4O2Pureza:98.78% - 98.78%Forma y color:SolidPeso molecular:463.4Medifoxamine
CAS:<p>Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine</p>Fórmula:C16H19NO2Pureza:97.14%Forma y color:SolidPeso molecular:257.33Halopemide
CAS:<p>Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).</p>Fórmula:C21H22ClFN4O2Pureza:96.57%Forma y color:SolidPeso molecular:416.88Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Forma y color:SolidPeso molecular:381.44SB-277011
CAS:<p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).</p>Fórmula:C28H30N4OPureza:99.39%Forma y color:SolidPeso molecular:438.56Milenperone
CAS:<p>Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.</p>Fórmula:C22H23ClFN3O2Pureza:98.09% - 99.84%Forma y color:SolidPeso molecular:415.89
