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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • PF-00217830

    CAS:
    <p>PF-00217830: agonist at serotonin 1A &amp; dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.</p>
    Fórmula:C26H30N4O2
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:430.54
  • U 99194 maleate

    CAS:
    <p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>
    Fórmula:C21H31NO6
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:393.47
  • PD 168568 dihydrochloride

    CAS:
    <p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>
    Fórmula:C22H29Cl2N3O
    Pureza:99.71%
    Forma y color:Solid
    Peso molecular:422.39
  • NGD 94-1

    CAS:
    <p>NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.</p>
    Fórmula:C18H20N6
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:320.39
  • MLS1547

    CAS:
    <p>MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).</p>
    Fórmula:C19H19ClN4O
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:354.83
  • 7-Hydroxy-DPAT hydrobromide

    CAS:
    <p>7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.</p>
    Fórmula:C16H26BrNO
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:328.29
  • GBR 12783 dihydrochloride

    CAS:
    <p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>
    Fórmula:C28H34Cl2N2O
    Pureza:98.08%
    Forma y color:Solid
    Peso molecular:485.49
  • Seridopidine

    CAS:
    <p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>
    Fórmula:C14H20FNO2S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:285.38
  • Ordopidine

    CAS:
    <p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>
    Fórmula:C14H20FNO2S
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:285.38
  • Molindone

    CAS:
    <p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>
    Fórmula:C16H24N2O2
    Pureza:99.37% - 99.46%
    Forma y color:Off-White Solid
    Peso molecular:276.37
  • A-437203

    CAS:
    <p>A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.</p>
    Fórmula:C20H27F3N6OS
    Pureza:98.80%
    Forma y color:Solid
    Peso molecular:456.53
  • BP14979

    CAS:
    <p>BP14979 is D3R-selective partial agonist.</p>
    Fórmula:C23H34N4O2
    Pureza:98.29% - 99.73%
    Forma y color:Solid
    Peso molecular:398.54
  • SK609 HCl

    CAS:
    <p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>
    Fórmula:C10H15Cl2N
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:220.14
  • Remoxipride hydrochloride

    CAS:
    <p>Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-</p>
    Fórmula:C16H24BrClN2O3
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:407.73
  • CyPPA

    CAS:
    <p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>
    Fórmula:C16H23N5
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:285.39
  • Fananserin

    CAS:
    <p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>
    Fórmula:C23H24FN3O2S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:425.52
  • CCG 203769

    CAS:
    <p>CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.</p>
    Fórmula:C8H14N2O2S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:202.27
  • Sonepiprazole

    CAS:
    <p>Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine receptors, exhibiting dissociation</p>
    Fórmula:C21H27N3O3S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:401.52
  • CY 208-243

    CAS:
    <p>CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.</p>
    Fórmula:C19H18N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:274.36
  • Timiperone

    CAS:
    <p>Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it mitigates stereotyped behavior.</p>
    Fórmula:C22H24FN3OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:397.51