
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Fórmula:C23H30FN3Pureza:99.85%Forma y color:SolidPeso molecular:367.50Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Fórmula:C28H32ClN3O8SPureza:99.78%Forma y color:Off-White PowderPeso molecular:606.09Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Fórmula:C21H21ClN4OSPureza:99.55%Forma y color:Tan SolidPeso molecular:412.94Pericyazine
CAS:Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.
Fórmula:C21H23N3OSPureza:99.61%Forma y color:SolidPeso molecular:365.49Ref: TM-T16472
1mg46,00€2mg59,00€5mg93,00€10mg124,00€25mg235,00€50mg389,00€100mg567,00€500mg1.225,00€L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Fórmula:C20H21ClN2OPureza:98.57%Forma y color:SolidPeso molecular:340.85Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Fórmula:C9H15ClNO5PPureza:99.84%Forma y color:SolidPeso molecular:283.65L-DOPA
CAS:L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Fórmula:C9H11NO4Pureza:98.99% - 99.93%Forma y color:Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidPeso molecular:197.19Bromopride
CAS:Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Fórmula:C14H22BrN3O2Pureza:99.95%Forma y color:SolidPeso molecular:344.25Ref: TM-T1175
2mg39,00€5mg58,00€10mg93,00€25mg167,00€50mg260,00€100mg409,00€200mg595,00€1mL*10mM (DMSO)64,00€Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Fórmula:C23H27FN4O2Pureza:99.73%Forma y color:Crystalline SolidPeso molecular:410.48Ref: TM-T0351
10mg48,00€25mg56,00€50mg88,00€100mg122,00€200mg192,00€500mg323,00€1mL*10mM (DMSO)50,00€Pramipexole
CAS:Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.Fórmula:C10H17N3SPureza:98% - 99.96%Forma y color:SolidPeso molecular:211.33Sulpiride
CAS:Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Fórmula:C15H23N3O4SPureza:99.94%Forma y color:White Crystalline PowderPeso molecular:341.43GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Fórmula:C30H35N3O3Pureza:98.94% - 99.29%Forma y color:SolidPeso molecular:485.62Ref: TM-T11463
2mg39,00€5mg58,00€10mg92,00€25mg177,00€50mg289,00€100mg462,00€200mg655,00€1mL*10mM (DMSO)63,00€Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Fórmula:C22H24ClN3O5Pureza:99.69%Forma y color:White To Of-White SolidPeso molecular:445.9Thioridazine hydrochloride
CAS:Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Fórmula:C21H27ClN2S2Pureza:99.55% - 99.957%Forma y color:White To Off-White SolidPeso molecular:407.04Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:99.32% - >99.99%Forma y color:White Crystalline SolidPeso molecular:883.09Oxidopamine hydrobromide
CAS:Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Fórmula:C8H12BrNO3Pureza:98.22% - 99.88%Forma y color:Beige To Brown Fine Crystalline PowderPeso molecular:250.09Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Fórmula:C17H21ClN2SPureza:99.90%Forma y color:SolidPeso molecular:320.88Domperidone
CAS:Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Fórmula:C22H24ClN5O2Pureza:98% - 99.82%Forma y color:SolidPeso molecular:425.91Haloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Fórmula:C21H23ClFNO2Pureza:98.69% - 98.97%Forma y color:Crystals SolidPeso molecular:375.86Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.Fórmula:C20H24Cl2N4O2Pureza:99.01% - 99.40%Forma y color:SoildPeso molecular:423.34
