
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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Benserazide hydrochloride
CAS:Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.Fórmula:C10H15N3O5·HClPureza:98.63% - 99.74%Forma y color:White Crystalline SolidPeso molecular:293.7(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Forma y color:Odour SolidHaloperidol D4
CAS:Haloperidol D4 is deuterium-labeled haloperidol.Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Losulazine
CAS:Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.Fórmula:C27H22F4N4O3SPureza:98.83%Forma y color:SolidPeso molecular:558.55Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;
Forma y color:Odour SolidA 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Fórmula:C22H22ClNForma y color:SolidPeso molecular:335.87MOR agonist-3
MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.Forma y color:Odour SolidAmisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Fórmula:C17H28ClN3O4SForma y color:SolidPeso molecular:405.94S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Fórmula:C29H29N3O2Pureza:98%Forma y color:SolidPeso molecular:451.56N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS:N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Fórmula:C10H16ClNForma y color:SolidPeso molecular:185.69ABT 724 trihydrochloride
CAS:ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Fórmula:C17H22Cl3N5Pureza:99.91%Forma y color:SolidPeso molecular:402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€LE 300
CAS:LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Fórmula:C20H22N2Pureza:97.91% - 98.79%Forma y color:SolidPeso molecular:290.4Quinelorane
CAS:Quinelorane is dextrorotary isomer.Fórmula:C14H22N4Forma y color:SolidPeso molecular:246.35Dopamine D2 receptor agonist-2
CAS:Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Fórmula:C25H31Cl2N5OSPureza:98.93%Forma y color:SoildPeso molecular:520.52A 77636 hydrochloride
CAS:A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).Fórmula:C20H28ClNO3Pureza:99.57%Forma y color:SolidPeso molecular:365.89MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71ADTN hydrobromide
CAS:ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).
Fórmula:C10H14BrNO2Forma y color:SolidPeso molecular:260.13O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18

