
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 435 productos de "Receptor de dopamina"
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Dopamine D2 receptor agonist-2
CAS:<p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>Fórmula:C25H31Cl2N5OSPureza:98.93%Forma y color:SoildPeso molecular:520.52A 77636 hydrochloride
CAS:<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Fórmula:C20H28ClNO3Pureza:99.57%Forma y color:SolidPeso molecular:365.89ADTN hydrobromide
CAS:<p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>Fórmula:C10H14BrNO2Forma y color:SolidPeso molecular:260.13Amisulpride hydrochloride
CAS:<p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>Fórmula:C17H28ClN3O4SForma y color:SolidPeso molecular:405.94MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71LE 300
CAS:<p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>Fórmula:C20H22N2Pureza:97.91% - 98.79%Forma y color:SolidPeso molecular:290.4S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Fórmula:C29H29N3O2Pureza:98%Forma y color:SolidPeso molecular:451.56PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Forma y color:White Crystalline SolidPeso molecular:451.6(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Fórmula:C159H252N40O58Pureza:98%Forma y color:SolidPeso molecular:3651.95ADTN
CAS:ADTN is an agonist of the dopamine receptor.Fórmula:C10H13NO2Pureza:98%Forma y color:SolidPeso molecular:179.22Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Quinelorane
CAS:Quinelorane is dextrorotary isomer.Fórmula:C14H22N4Forma y color:SolidPeso molecular:246.35Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Fórmula:C22H26F3N3OSForma y color:SolidPeso molecular:437.52Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Fórmula:C22H26ClNO4SForma y color:SolidPeso molecular:435.96N-0500 HCl
CAS:<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Fórmula:C15H22ClNO2Pureza:98.85% - 99.54%Forma y color:SolidPeso molecular:283.79Moperone
CAS:Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Fórmula:C22H26FNO2Forma y color:SolidPeso molecular:355.45

