
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18Moperone
CAS:Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Fórmula:C22H26FNO2Forma y color:SolidPeso molecular:355.45Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Fórmula:C24H36O2Pureza:98.35%Forma y color:SolidPeso molecular:356.54Trimethobenzamide
CAS:Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.Fórmula:C21H28N2O5Forma y color:SolidPeso molecular:388.46Sumanirole maleate
CAS:Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Fórmula:C15H17N3O5Pureza:98%Forma y color:SolidPeso molecular:319.31ST-836 hydrochloride
CAS:ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Fórmula:C23H35ClN4OSPureza:98%Forma y color:SolidPeso molecular:451.07cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H18ClN3SPureza:98%Forma y color:White Crystalline PowderPeso molecular:247.79PD128907 HCl
CAS:PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.Fórmula:C14H20ClNO3Pureza:98%Forma y color:SolidPeso molecular:285.77Eticlopride hydrochloride
CAS:Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Fórmula:C17H25ClN2O3·HClPureza:98%Forma y color:SolidPeso molecular:377.31UCSF924
CAS:UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Fórmula:C20H22N2O2Pureza:98%Forma y color:SolidPeso molecular:322.4(-)-Apomorphine hydrochloride hydrate
CAS:(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.Fórmula:C17H17NO2HClXH2OForma y color:SolidPeso molecular:303.8Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Fórmula:C15H21D3N2O4SForma y color:SolidPeso molecular:331.45SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Fórmula:C19H21BrClNO2Pureza:98%Forma y color:SolidPeso molecular:410.73GRK2 Inhibitor
CAS:GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).Fórmula:C12H9NO6Forma y color:SolidPeso molecular:263.23-O-Methyldopa-d3
CAS:3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Fórmula:C10H10D3NO4Forma y color:SolidPeso molecular:214.23Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Fórmula:C19H24Cl2N2Forma y color:SolidPeso molecular:354.33ABT-724
CAS:ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Fórmula:C17H19N5Pureza:99.73%Forma y color:SolidPeso molecular:293.37SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Fórmula:C17H18BrNOPureza:95.00% - 99.82%Forma y color:SolidPeso molecular:332.23
