Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Se han encontrado 217 productos de "Receptor de cannabinoides"
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ANEB-001
CAS:ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.Fórmula:C22H24ClF3N2O2Forma y color:SolidPeso molecular:440.89CB1R Allosteric modulator 4
CAS:Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.Fórmula:C20H17N3O2SForma y color:SolidPeso molecular:363.43PGN36
CAS:PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).Fórmula:C21H23N3O3Forma y color:SolidPeso molecular:365.43CB1R Allosteric modulator 2
CAS:Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.Fórmula:C19H15ClFN3OForma y color:SolidPeso molecular:355.79GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Fórmula:C22H18N2O2Forma y color:SolidPeso molecular:342.39CB1-IN-2
CAS:CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.Fórmula:C17H19Cl2N5OForma y color:SolidPeso molecular:380.27COR167
CAS:COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.Fórmula:C28H38N2O2Forma y color:SolidPeso molecular:434.61UCM 707
CAS:endocannabinoid transport inhibitorFórmula:C25H37NO2Pureza:98%Forma y color:SolidPeso molecular:383.57SMM-189
CAS:SMM-189 is a potent and selective CB2 inverse agonist.Fórmula:C19H12Cl2O3Forma y color:SolidPeso molecular:359.2CAY10412
CAS:Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.Fórmula:C25H36O2SForma y color:SolidPeso molecular:400.62(S)-SLV 319
CAS:Ibipinabant (SLV319), a potent CB1 antagonist, K i = 7.8 nM, >1000x selective over CB2, for obesity and diabetic research.Fórmula:C23H20Cl2N4O2SForma y color:SolidPeso molecular:487.4LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Fórmula:C23H25FN4O4SPureza:98%Forma y color:SolidPeso molecular:472.53Palmitoyl serinol
CAS:Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.Fórmula:C19H39NO3Forma y color:SolidPeso molecular:329.52ZCZ011
CAS:ZCZ011 enhances CB1 receptor effects, crosses blood-brain barrier, and potentiates cannabimimetic behaviors in mice.Fórmula:C21H18N2O2SPureza:98%Forma y color:SolidPeso molecular:362.44KLS-13019
CAS:KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).Fórmula:C22H29NO3Pureza:>99.99% - >99.99%Forma y color:SolidPeso molecular:355.47Virodhamine trifluoroacetate
CAS:Virodhamine trifluoroacetate: full GPR55 & CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.Fórmula:C24H38F3NO4Pureza:98%Forma y color:SolidPeso molecular:461.56OMDM-6
CAS:OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.Fórmula:C28H42N2O3Pureza:99.66%Forma y color:SolidPeso molecular:454.64Ref: TM-T12307
1mg85,00€5mg170,00€10mg250,00€25mg371,00€50mg522,00€100mg712,00€200mg954,00€1mL*10mM (DMSO)187,00€LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Fórmula:C23H29ClN6O3Forma y color:SolidPeso molecular:472.97N-Arachidonyldopamine
CAS:N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1Fórmula:C28H41NO3Pureza:97.65%Forma y color:SolidPeso molecular:439.632-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFórmula:C23H38O4Pureza:95%Forma y color:LiquidPeso molecular:378.55
