Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Se han encontrado 217 productos de "Receptor de cannabinoides"
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GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Fórmula:C19H16F4N4Forma y color:SolidPeso molecular:376.35AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Fórmula:C26H37NO2Forma y color:SolidPeso molecular:395.58CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Fórmula:C18H19F3N4O2Pureza:99.6%Forma y color:SolidPeso molecular:380.36MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Fórmula:C23H17Cl3N4OPureza:99.63%Forma y color:SolidPeso molecular:471.77CB1/2 agonist 4
CAS:CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.Fórmula:C27H45NO3Forma y color:SolidPeso molecular:431.65CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Fórmula:C24H24ClN3OForma y color:SolidPeso molecular:405.92UCM710
CAS:UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).Fórmula:C19H34O3Pureza:98%Forma y color:SolidPeso molecular:310.47MM-22
CAS:biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamideFórmula:C36H60N4O5SPureza:98%Forma y color:SolidPeso molecular:660.95CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Fórmula:C22H32N2OForma y color:SolidPeso molecular:340.5S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Fórmula:C23H27FN2O4Forma y color:SolidPeso molecular:414.47PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Fórmula:C22H31NO3Forma y color:SolidPeso molecular:357.49AZD-2207
CAS:AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.Fórmula:C25H25Cl2F3N4O4SForma y color:SolidPeso molecular:605.46Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Fórmula:C21H30O2Forma y color:SolidPeso molecular:314.46CB1 inverse agonist 2
CAS:CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.Fórmula:C24H20ClFN2OSForma y color:SolidPeso molecular:438.94GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Fórmula:C22H18N2O2Forma y color:SolidPeso molecular:342.39AM-6538
CAS:AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.Fórmula:C26H25Cl2N5O4Forma y color:SolidPeso molecular:542.41COR 170
CAS:inverse agonist of CB2 receptorsFórmula:C31H36N2O2Pureza:98%Forma y color:SolidPeso molecular:468.63NIDA 41020
CAS:NIDA 41020 is a CB1 receptor antagonist.Fórmula:C23H24Cl2N4O2Pureza:98%Forma y color:SolidPeso molecular:459.37LH 21
CAS:LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.Fórmula:C20H20Cl3N3Forma y color:SolidPeso molecular:408.75CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Fórmula:C24H23N3O4S2Pureza:98%Forma y color:SolidPeso molecular:481.59
