Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Se han encontrado 217 productos de "Receptor de cannabinoides"
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O-2093
CAS:anandamide uptake inhibitorFórmula:C34H43Cl2NO3Pureza:98%Forma y color:SolidPeso molecular:584.62CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Fórmula:C23H18FN5O2S2Forma y color:SolidPeso molecular:479.55CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Fórmula:C24H23Cl2N3OForma y color:SolidPeso molecular:440.36TC-C 14G
CAS:CB1 receptor inverse agonistFórmula:C24H17Cl2F2NO4Pureza:98%Forma y color:SolidPeso molecular:492.3(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Fórmula:C23H20Cl2N4O2SForma y color:SolidPeso molecular:487.4Olorinab
CAS:Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Fórmula:C18H23N5O3Pureza:97.67% - 98.47%Forma y color:SolidPeso molecular:357.41CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Fórmula:C24H24N2O5SPureza:98.56%Forma y color:SolidPeso molecular:452.52SR144528
CAS:SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).Fórmula:C29H34ClN3OPureza:99.63%Forma y color:SolidPeso molecular:476.05Nonabine
CAS:Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Fórmula:C25H33NO2Pureza:99.82% - 99.94%Forma y color:SolidPeso molecular:379.54CB1R antagonist 1
CAS:CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Fórmula:C18H23F3N2O3SPureza:99.65%Forma y color:SolidPeso molecular:404.45CB2R PAM
CAS:CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.Fórmula:C21H24BrFN2O2Pureza:99.09%Forma y color:SolidPeso molecular:435.33SCH-336
CAS:SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.Fórmula:C23H25NO8S3Pureza:97.00%Forma y color:SolidPeso molecular:539.64Ref: TM-T24771
5mg49,00€10mg73,00€25mg152,00€50mg213,00€100mg309,00€200mg444,00€1mL*10mM (DMSO)60,00€PSB-CB5
CAS:PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study obesity and metabolic disorders.Fórmula:C20H17ClN2O2SPureza:99.26%Forma y color:SolidPeso molecular:384.88AZD1940
CAS:AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.Fórmula:C20H29F2N3O2SPureza:98.68%Forma y color:SolidPeso molecular:413.52Ref: TM-T30252
1mg130,00€5mg311,00€10mg535,00€25mg847,00€50mg1.169,00€100mg1.586,00€1mL*10mM (DMSO)344,00€JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Fórmula:C24H26N2O6Pureza:99.93%Forma y color:SolidPeso molecular:438.47Ref: TM-T19705
1mg52,00€5mg119,00€10mg177,00€25mg313,00€50mg465,00€100mg662,00€1mL*10mM (DMSO)142,00€AM-1235
CAS:AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.Fórmula:C24H21FN2O3Pureza:99.92%Forma y color:SolidPeso molecular:404.43O-2050
CAS:O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.Fórmula:C23H31NO4SPureza:98%Forma y color:SolidPeso molecular:417.56Heptadecanoyl ethanolamide
CAS:Heptadecanoyl ethanolamide, an endogenous cannabinoid, serves as a synthetic analog of PEA, featuring an odd-numbered (17-carbon) fatty acid chain [1].Fórmula:C19H39NO2Forma y color:SolidPeso molecular:313.52COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Fórmula:C16H16ClNO3SPureza:99.75%Forma y color:SolidPeso molecular:337.82Ref: TM-T36520
1mg38,00€5mg86,00€10mg123,00€25mg215,00€50mg299,00€100mg411,00€200mg560,00€1mL*10mM (DMSO)94,00€PF-03550096
CAS:PF-03550096, an orally active synthetic cannabinoid (CB), selectively binds to peripheral CB2 receptors with a Ki value of 7.9 nM, demonstrating analgesic activity [1].Fórmula:C19H28N4O4Forma y color:SolidPeso molecular:376.45
