Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65924 productos de "Derivados de Quinazolina y Quinolina"
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5-(4-chlorophthalazin-1-yl)-N,2-dimethylbenzenesulfonamide
CAS:Pureza:95.0%Peso molecular:347.82000732421875Dothiepin
CAS:Producto controlado<p>Applications A tricyclic antidepressant.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Metysova, J., et al.: Arzneim.-Forsch., 13, 1039 (1963), Maguire, K.P., et al.: Br. J. Clin. Pharmacol., 12, 405 (1981), Donovan, S., et al.: Prog. Neuro-Psychopharmacol. Biol. Psychiatry, 18, 1143 (1994),<br></p>Fórmula:C19H21NSForma y color:Light Yellow Solid With A Low Melting PointPeso molecular:295.44(D,L)-threo-α-Phenyl-2-piperidineacetamide
CAS:Producto controlado<p>Applications Intermediate in the preparation of D-threo-Methylphenidate (Ritalin)<br></p>Fórmula:C13H18N2OForma y color:White To BeigePeso molecular:218.29[2-[(2-Amino-4-chlorophenyl)amino]phenyl](4-methyl-1-piperazinyl)methanone
CAS:<p>Impurity Clozapine EP Impurity D<br>Applications [2-[(2-Amino-4-chlorophenyl)amino]phenyl](4-methyl-1-piperazinyl)methanone (Clozapine EP Impurity D) is used in the synthesis of substituted dibenzodiazepines. Also an impurity in the synthesis of Clozepine (C587500), an antipsychotic.<br>References Stille, et al: Farnaco, Ed. Prat., 26, 603 (1971), Hane, J.M., et al.: Psychopharmacol. Bull., 24, 62 (1988), Meltzer, H.Y.: J. Clin. Psychiatry, 55, Suppl. B, 47 (1994)<br></p>Fórmula:C18H21ClN4OForma y color:Light Red To RedPeso molecular:344.84MMP 8-I
CAS:Producto controlado<p>Applications MMP 8-I is a matrix metalloproteinase 8 inhibitor. Matrix metalloproteinases are involved with tight junction protein degradation in endothelial cells.<br>References Kumar, H., et al.: Mol Neurobiol. (2017)<br></p>Fórmula:C13H12N4O2SForma y color:NeatPeso molecular:288.325Dihydro Dutasteride
CAS:<p>Applications Dihydro Dutasteride is an impurity arose during the process development of Dutasteride (D735000).<br>References Solomons, W., et al.: J. Pharma. Sci., 63, 19 (1974), Rasmusson, G., et al.: J. Med. Chem., 29, 2298 (1986),<br></p>Fórmula:C27H32F6N2O2Forma y color:NeatPeso molecular:530.55Thiamethoxam-d4
CAS:Producto controlado<p>Stability Light Sensitive<br>Applications Labelled Thiamethoxam (T344180). A neonicotinoid insecticide. Reports show that when exposed to neonicotinid pesticides honeybees have probelms returnign home after foraging and bumblebee colonies grow poorly and produce fewer queens. Used in Cannabis testing.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Oliver, J., et al.: J. Environ. Horticult., 28, 135 (2010), Ghosh, A., et al.: J. Entomol. Res., 34, 35 (2010), Chem. and Eng. News 90: 10 (2012)<br></p>Fórmula:C82H4H6ClN5O3SForma y color:ColourlessPeso molecular:295.742-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)acetohydrazide
CAS:Pureza:95.0%Peso molecular:253.61000061035156Hydroxydehydro Nifedipine Carboxylate
CAS:Producto controladoFórmula:C16H14N2O7Forma y color:NeatPeso molecular:346.292-[(2-Azidoethoxy)methyl]-4-(2-chlorophenyl)-3-ethoxycarbonyl-5-methoxycarbonyl)-6-methyl-1,4-dihydropyridine
CAS:Producto controladoFórmula:C20H23ClN4O5Forma y color:NeatPeso molecular:434.872-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-3-bromopropan-2-ol
CAS:Producto controlado<p>Impurity Fluconazole EP Impurity H<br>Applications 2-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-3-bromopropan-2-ol (Fluconazole EP Impurity H) is an impurity of the antifungal agent Fluconazole (F421000).<br>References Bourichi, H., et al.: STP Pharma Pratiques, 18, 285 (2008); Richard, K. et al.: Antimicrob. Ag. Chemother., 27, 832 (1985)<br></p>Fórmula:C11H10BrF2N3OForma y color:Off-WhitePeso molecular:318.12(S)-(-)-3-Acetylthio-2-methylpropionic Acid
CAS:Producto controlado<p>Applications S-Acetylthio-2-methylpropionic Acid (S-AMPA) is a key chiral intermediate for Captopril (C175750) and other hypertension drugs.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Cushman, D., et al.: Biochem., 16, 5484 (1977), Ondetti, M., et al.: J. Med. Chem., 24, 355 (1981), Tseng, T., et al.: Cancer Lett., 62, 233 (1992),<br></p>Fórmula:C6H10O3SForma y color:ColourlessPeso molecular:162.21Iso Rizatriptan
CAS:Producto controlado<p>Impurity Rizatriptan EP Impurity C<br>Applications Iso Rizatriptan (Rizatriptan EP Impurity C) is a potential impurity of Rizatriptan. A regioisomer of Rizatriptan.<br>References Dill, K., et al.: J. Phys. Chem., 91, 1980 (1987), Cole, L., et al.: Anal. Chem., 64, 1317 (1992), Street, L., et al.: J. Med. Chem., 1995, 38, 1799<br></p>Fórmula:C15H19N5Forma y color:NeatPeso molecular:269.346-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)butoxy]-1-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butyl]-3,4-dihydro-2(1H)-quinolinone
CAS:Producto controlado<p>Impurity Cilostazol USP Related Compound C<br>Applications 6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)butoxy]-1-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butyl]-3,4-dihydro-2(1H)-quinolinone, is an impurity of Cilostazol (C441500), a potent phosphodiesterase III A (PDE3A) inhibitor (IC50=0.2uM) and inhibitor of adenosine uptake.<br>References Suri, A., et al.: J. Clin. Pharmacol., 38, 144 (1998), Park, S.-W., et al.: Am. J. Cardiol., 84, 511 (1999), Tsuchikane, E., et al.: Circulation, 100, 21 (1999);<br></p>Fórmula:C31H45N9O2Forma y color:NeatPeso molecular:575.75(S)-5-Bromo Naproxen
CAS:Producto controladoFórmula:C14H13BrO3Forma y color:NeatPeso molecular:309.166-Methyl Risperidone
CAS:Producto controlado<p>Impurity Risperidone EP Impurity E<br>Applications 6-Methyl Risperidone (Risperidone EP Impurity E) is a Risperidone (R525000) impurity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Fórmula:C24H29FN4O2Forma y color:Light YellowPeso molecular:424.51Vioxx-d5 (Major)
CAS:Producto controlado<p>Applications A selective labelled cyclooxygenase-2 (COX-2) inhibitor. Use as an anti-inflammatory, analgesic.<br>References Catalla-Lawson, F., et al.: J. Pharmacol. Exp. Ther., 289, 735 (1999), Ehrich, E.W., et al.: Clin. Pharmacol. Ther., 65, 336 (1999), Langman, M.J., et al.: J. Am. Med. Assoc., 282, 1929 (1999),<br></p>Fórmula:C172H5H9O4SForma y color:NeatPeso molecular:319.3871-Isopropyl-6-(6-(4-isopropylpiperazin-1-yl)pyridin-3-yl)-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-1H-indazole-4-carboxamide
CAS:Pureza:98%Forma y color:SolidPeso molecular:569.754028320313O-Ethyl Albuterol
CAS:Producto controlado<p>Impurity Levalbuterol USP Related Compound E<br>Applications O-Ethyl Albuterol is an analog of Albuterol (A514500). A β2-adrenoceptor agonist. Bronchodilator; tocolytic. Levalbuterol USP Related Compound E.<br>References Han, et al.: Bioorg. Med. Chem., 14, 6043 (2006), Liyou, H., et al.: Biochem., 46, 1432 (2007), Agrawal, D., et al.: J. Allergy Clin. Immunol., 113, 503 (2004),<br></p>Fórmula:C15H25NO3Forma y color:NeatPeso molecular:267.36cis-Ambroxol Hydrochloride
CAS:<p>Stability Hygroscopic<br>Applications cis-Ambroxol Hydrochloride is a cis isomer of Ambroxol Hydrochloride (A575900 ), a metabolite of Bromohexine. Ambroxol Hydrochloride is a bronchosecretolytic drug.<br>References Jauch, R., et al.: Arzneim-Forsch., 13, 474 (1963)<br></p>Fórmula:C13H18Br2N2O·x(HCl)Forma y color:NeatPeso molecular:378.10 + x(36.46)4-(4,6-Bis(2,4-dimethylphenyl)-1,3,5-triazin-2-yl)benzene-1,3-diol
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:397.4779968261719Mavoglurant
CAS:Producto controlado<p>Applications Mavoglurant is a non-competitive metabotropic glutamate receptor 5 (mGlu5) receptor antagonist.<br>References Vranesic, I., et al.; Bioorg. Med. Chem., 22, 5790 (2014); Kubas, H., et al.: Bioorg. Med. Chem. Lett., 23, 6370 (2013)<br></p>Fórmula:C19H23NO3Forma y color:NeatPeso molecular:313.39METHYL 1-CHLORO-4-HYDROXY-7-PHENOXYISOQUINOLINE-3-CARBOXYLATE
CAS:Pureza:90.0%Peso molecular:329.7399902343751-(4-Methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:309.3210144042969Vemurafenib
CAS:Producto controlado<p>Applications Vemurafenib selective BRAFV600E kinase inhibitor; an antitumor agent. Vemurafenib functions by inhibiting the proliferation and mitogen-activated protein/extracellular signal-regulated kinase (ERK) kinase and ERK phosphorylation in a panel of tumor cell lines, including melanoma cell lines expressing BRAFV600E or other mutant BRAF proteins altered at codon 600. Potent B-Raf inhibitor<br>References Halaban, R. et al.: Pigm. Cell. Melonoma Res., 23, 190 (2010); Yang, H. et al.: Cancer Res., 70, 5518 (2010); Comin-Anduix, B. et al.: Clin. Cancer Res., 16, 6040 (2010);<br></p>Fórmula:C23H18ClF2N3O3SForma y color:NeatPeso molecular:489.92Ebastine
CAS:<p>Applications A nonsedating type histamine H1-receptor antagonist. Antihistaminic.<br>References Fliri, A., et al.: J. Med. Chem., 52, 8038 (2009), Inomata, N., et al.: J. Dermatol., 36, 224 (2009), Carvajal, A., et al.: Clin. Pharmacol. Ther., 85, 481 (2009), Yamashita, S., et al.: Mol. Pharm., 6, 48 (2009),<br></p>Fórmula:C32H39NO2Forma y color:White To Off-WhitePeso molecular:469.66Etomidate Hydrochloride
CAS:Producto controlado<p>Applications (cas# 53188-20-8) is a useful research chemical.<br></p>Fórmula:C14H17ClN2O2Forma y color:NeatPeso molecular:280.758-methyl-4-(thiophene-2-carbonyl)-1-oxa-4,8-diazaspiro[4.5]decane-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:310.3699951171875Dibenzyloxy Tezacaftor-D4
Producto controladoFórmula:C40H35D4F3N2O6Forma y color:NeatPeso molecular:704.782-Oxazolidinone
CAS:Producto controlado<p>Applications An oxazole derivative used as an antibiotic. It is also used in the preparation of compounds with antitumor activity. A metabolite of Furazolidone (F864100).<br>References Miyahara, M. et al.: CHem. Pharmac. Bull., 29, 2366 (1981); Hunder, G. et al.: Arch. Toxicol., 61, 161 (1987); Roloff, T. et al.: Med. Monat. Pharrm., 22, 370 (1999);<br></p>Fórmula:C3H5NO2Forma y color:NeatPeso molecular:87.08Loratadine N-Oxide
CAS:Producto controlado<p>Applications Loratadine N-oxide nonsedating-type histamine.<br></p>Fórmula:C22H23ClN2O3Forma y color:NeatPeso molecular:398.8842-O-tert-Butyldimethylsilyloxyethyl Rapamycin
CAS:<p>Stability Hygroscopic<br>Applications 42-O-tert-Butyldimethylsilyloxyethyl Rapamycin is a useful synthetic intermediate in the synthesis of Everolimus (E945400); an immunosuppressant macrolide and analog of the parent drug Rapamycin (R124000). Everolimus inhibits cytokine-mediated lymphocyte proliferation.<br>References Dumont, F.J., et al.: Curr. Opin. Invest. Drugs, 2, 1220 (2001); Kovarik, J. M., et al.: Clin. Pharmacol. Ther., 69, 48 (2001); Nashan, B., et al.: Ther. Drug Monit., 24, 53 (2002); Venkata, S.P., et al.: PCT Int. Appl. WO 2012066502 A1 20120524. May 24, 2012<br></p>Fórmula:C59H97NO14SiForma y color:NeatPeso molecular:1072.485-(1,3-Dioxolan-2-yl)-2-(4-hexyloxybenzoyl)thiophene
CAS:Pureza:97.0%Peso molecular:360.47000122070317-Hydroxy Loxapine-D8
CAS:Producto controlado<p>Applications 7-Hydroxy Loxapine-D8 is a labelled analogue of 7-Hydroxy Loxapine (H943790).<br>References Kapur, S., et al.: Am. J. Psychiatry, 154, 1525 (1997); Rivers-Bulkeley, N. & Hollender, M.: Am. J. Psychiat., 139, 1345 (1982)<br></p>Fórmula:C18H10D8ClN3O2Forma y color:Dark YellowPeso molecular:351.866-methyl-2-(3-methylphenyl)quinoline-4-carboxylic acid
CAS:Pureza:95.0%Peso molecular:277.3229980468752-(3-Aminophenyl)-quinoline-4-carboxylic acid
CAS:Pureza:97%Forma y color:SolidPeso molecular:264.283996582031255-(2,6-DIMETHOXYPHENYL)-1-(4-FLUOROPHENYL)-1H-PYRAZOLE-3-CARBOXYLIC ACID
Pureza:90.0%Peso molecular:342.32598876953125Levofloxacin-d8
CAS:Producto controlado<p>Applications Labelled S-(-)-Form of Ofloxacin. An antibiotic used against gram-negative organisms.<br>References Kato, M., et al.: Arzneim.-Forsch., 42, 365 (1992), North, D.S., et al.: Pharmacotherapy, 18, 915 (1998), Hwang, D.G., et al.: Br. J. Ophthalmol., 87, 1004 (2003),<br></p>Fórmula:C18H12D8FN3O4Forma y color:Light Yellow SolidPeso molecular:369.428-tert-butyl-4-(pyridine-3-carbonyl)-1-oxa-4-azaspiro[4.5]decane-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:346.427001953125Brigatinib
CAS:Producto controlado<p>Applications Brigatinib is a tyrosine kinase receptor Mer (MERTK) inhibitor and can be used in combination with epidermal growth factor receptor (EGFR) inhibitors for the treatment of cancer.<br>References Yan, D.; et al.: U.S. Pat. Appl. Publ. 48 pp. Patent 2017 CODEN:USXXCO<br></p>Fórmula:C29H39ClN7O2PForma y color:NeatPeso molecular:584.094-Hydroxy Phenobarbital-d5
CAS:Producto controladoFórmula:C122H5H7N2O4Forma y color:NeatPeso molecular:253.27Aripiprazole-d8
CAS:Producto controlado<p>Applications Aripiprazole-d8 is a deuterated version of Aripiprazole (A771000), a selective dopamine D2-receptor antagonist with dopamine autoreceptor agonist activity.<br>References Canive, J.M., et al.: Psychopharmacol. Bull., 34, 101 (1998), Oshiro, Y., et al.: J. Med. Chem., 41, 658 (1998),<br></p>Fórmula:C232H8H19Cl2N3O2Forma y color:Off White SolidPeso molecular:456.4310H-Phenothiazine 5-Oxide
CAS:<p>Applications 10H-Phenothiazine 5-Oxide is a by-product in the synthesis of Phenothiazine S,S-Dioxide (P297600). Phenothiazine S,S-Dioxide is a derivative of Phenothiazine (P318040), a key component of antipsychotic and antihistaminic drugs.<br>References Bansode, T., et al.: Eur. J. Med. Chem., 44, 5094 (2009); Baell, J., et al.: J. Med. Chem., 53, 2719 (2010); Howard, P., et al.: Environ. Sci. Technol., 44, 2277 (2010); Koren, J., et al.: J. Biol. Chem., 285, 2498 (2010); Amobi, N., et al.: Eur. J. Pharmacol., 627, 285 (2010)<br></p>Fórmula:C12H9NOSForma y color:Light Beige To Light BrownPeso molecular:215.27Levosimendan Cyanoacetamide Hydrazone Impurity
CAS:Producto controlado<p>Applications Levosimendan Cyanoacetamide Hydrazone Impurity is an impurity of Levosimendan (L378000) which is a bioactive enantiomer of racemate, Simendan. It is a positive inotropic agent with vasodilating activity and also cardiotonic.<br>References Sandell, E.-P., et al.: J. Cardiovasc. Pharmacol., 26, S57 (1995); Pagel, P.S., et al.: Cardiovasc. Drug Rev., 14, 286 (1996)<br></p>Fórmula:C14H14N6O2Forma y color:Off-White To Dark OrangePeso molecular:298.3Pyrazinamide-15N,d3
CAS:Producto controlado<p>Applications Antibacterial (tuberculostatic).<br>References Weiner, I.M., et al.: J. Pharmacol. Exp. Ther., 180, 411 (1972), Feldner, E., et al.: Anal. Profiles Drug Subs., 12, 433 (1983)<br></p>Fórmula:C5H2D3N215NOForma y color:White Crystalline PowderPeso molecular:127.122-Chloromethyl-3-methyl-4-(2,2,2-trifluoroethoxy)pyridine, Hydrochloride
CAS:Producto controladoFórmula:C9H9ClF3NO·ClHForma y color:NeatPeso molecular:276.083-Methyl-1-(3-methylphenyl)-1H-pyrazol-5-amine hydrochloride
CAS:Pureza:97%Peso molecular:223.6999969482422Loratadine Epoxide
CAS:Producto controladoFórmula:C22H23ClN2O3Forma y color:White To Off-WhitePeso molecular:398.882-Mercapto-N-methyl-benzamide
CAS:Producto controlado<p>Stability Air Sensitive<br>Applications 2-Mercapto-N-methyl-benzamide is an intermediate used to prepare axitinib (A794650) which is a tyrosine kinase inhibitor. Axitinib is used in cancer therapy.<br>References Wasser, K., et al.: Eur. Radiol., 13, 80 (2003), Park, J., et al.: Clin. Cancer Res., 8, 1172 (2002), Bergers, G., et al.: J. Clin. Invest., 111, 1287 (2003),<br></p>Fórmula:C8H9NOSForma y color:BeigePeso molecular:167.228Cyanuric Acid-13C3
CAS:<p>Applications Useful for diagnostic determination of Melamine and related compounds in kidney tissue.<br>References Mast, R., et al.: Food Chem. Toxicol., 21, 807 (1983), Yokley, R., et al.: J. Agric. Food Chem., 48, 3352 (2000), Ehling, S., et al.: Food Addit. Contam., 24, 1319 (2007), Vail, T., et al.: J. Anal. Toxicol., 31, 304 (2007),<br></p>Fórmula:C3H3N3O3Forma y color:NeatPeso molecular:132.053-(1-METHYL-1H-PYRAZOL-4-YL)QUINOLINE-6-CARBOXYLIC ACID
CAS:Pureza:95.0%Peso molecular:253.26100158691406Simendan
CAS:Producto controlado<p>Applications Simendan is the racemic mixture of Levosimendan (L378000) which is a positive inotropic agent with vasodilating activity.<br>References Sandell, E.-P., et al.: J. Cardiovasc. Pharmacol., 26, S57 (1995); Pagel, P.S., et al.: Cardiovasc. Drug Rev., 14, 286 (1996)<br></p>Fórmula:C14H12N6OForma y color:Yellow SolidPeso molecular:280.28(2R)-Vildagliptin
CAS:<p>Applications (2R)-Vildagliptin is an oral anti-hyperglycemic agent that inhibit dipeptidyl peptidase 4 (DPP-4) which can act as a serine exopeptidase. Aside from there use in type 2 diabetes, gliptins have positive cardiovascular and anti-inflammtatory effects. Antidiabetic.<br>References Ahren, B., et al.: J. Clin. Endocrinol. Metab., 89, 2078 (2004), Ahren, B., et al.: Diabetes Care, 27, 2874 (2004), Barlocco, D., et al.: Curr. Opin. Invest. Drugs, 5, 1094 (2004),<br></p>Fórmula:C17H25N3O2Forma y color:Off-White To Light BeigePeso molecular:303.403-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one Hydrochloride
CAS:Producto controlado<p>Applications Risperidone (R525000) metabolite.<br>References Meuldermans, W. et al.; Drug Metab. Dispos. 22, 129 (1994); Mannens, G. et al.; Drug Metab. Dispos. 21, 1134 (1993)<br></p>Fórmula:C23H28FN3O3·HClForma y color:NeatPeso molecular:449.9466-Amino-1,3-dimethyluracil
CAS:Producto controlado<p>Applications 6-Amino-1,3-dimethyluracil is used as a reagent in the synthesis of new pyrimidine and caffeine derivatives that display highly potential antitumor activity. It is also used as a starting material in the synthesis of fused pyrido-pyrimidines.<br>References Abu-Hashem, A., et al.: Lett. Drug. Des. Discov., 12, 471 (2015); Azev, Y., et al.: Mendeleev Commun., 25, 310 (2015)<br></p>Fórmula:C6H9N3O2Forma y color:Light YellowPeso molecular:155.155-(4-cyclohexylphenyl)-1H-pyrazole-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:270.33200073242194-{[(5Z)-3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}-2-methoxyphenyl thiophene-2-carboxylate
CAS:Peso molecular:541.6500244140625Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Fórmula:C20H13F6N3O2SPureza:99.83%Forma y color:White PowderPeso molecular:473.399’-Desmethyl Granisetron
CAS:Producto controlado<p>Impurity Granisetron EP Impurity C<br>Applications An impurity in the synthesis of Granisetron Hydrochloride.<br>References Nishikawa, M., et al.: Drug Metab. Pharmacokin., 19, 280 (2004), Firkusny, L., et al.: Biochem. Pharmacol., 49, 1777 (1995), Sanwald, P., et al.: Drug Metab. Dispos., 24, 602 (1996), Vanderstreene, et al.: J. Labelled Comp. Radiopharm., XLI, 3, 71 (1997),<br></p>Fórmula:C17H22N4OForma y color:White To Light YellowPeso molecular:298.38N’-(1-Methylazepan-4-yl)benzohydrazine Monohydrochloride Salt
CAS:Producto controlado<p>Impurity Azelastine EP Impurity B/Azelastine USP Related Compound B<br>Stability Hygroscopic<br>Applications An intermediate in the preparation of Azelastine (A808250(P)), which is an orally active H1-hystamine receptor antagonist and an antihistaminic.<br>References Scheffler, G. et al.: Arch. Pharm., 321, 205 (1988); Tasaka, K., et al.: Arzneim.-Forsch., 29, 488 (1979); Chand, N., et al.: Int. J. Immunopharmacol., 7, 833 (1985)<br></p>Fórmula:C14H21N3O·ClHForma y color:Light Yellow To Dark YellowPeso molecular:283.80Xanthurenic Acid
CAS:<p>Applications Excreted by pyridoxine-deficient animals after the ingestion of tryptophan.<br>References Aquilina, J., et al.: Biochemistry, 39, 16176 (2000), Roberts, J., et al.: Photochem. Photobiol., 74, 740 (2001),<br></p>Fórmula:C10H7NO4Forma y color:NeatPeso molecular:205.172-[3-(4-nitrophenyl)-1-phenyl-1h-pyrazol-4-yl]acetic acid
CAS:Pureza:97%Peso molecular:323.30801391601563,4-Dehydro Cilostazol
CAS:Producto controlado<p>Impurity Cilostazol USP Related Compound B<br>Applications A metabolite of Cilostazol.<br></p>Fórmula:C20H25N5O2Forma y color:Off WhitePeso molecular:367.44N-Nitro-1,2,3,4-tetradehydro Argatroban Ethyl Ester
CAS:<p>Applications N-Nitro-1,2,3,4-tetradehydro Argatroban Ethyl Ester is an intermediate in the preparation of Argatroban (A769000).<br></p>Fórmula:C25H35N7O7SForma y color:Off White SolidPeso molecular:577.655-chloro-2-(1H-pyrazol-5-yl)aniline
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:193.63000488281251-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazine
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:242.3260040283203Pyrimethamine
CAS:Producto controlado<p>Applications Dihydrofolate reductase inhibitor; generally used in combination with other antimicrobial agents. Antiprotozoal (Toxoplasma); antimalarial.<br>References Loutfy, M.A., et al.: Anal. Profiles Drug Subs., 12, 463 (1983), Leport, C., et al.: Am. J. Med., 84, 94 (1988), McIntosh, H.M., et al.: Ann. Trop. Med., Parasitol., 93, 265 (1998), Plowe, C.V., et al.: Br. Med. J., 328, 545 (2004),<br></p>Fórmula:C12H13ClN4Forma y color:White To Off-WhitePeso molecular:248.711,1'-(1,3-Phenylene)bis-1H-1,2,4-triazole
CAS:Producto controlado<p>Impurity Fluconazole EP Impurity C / Fluconazole USP Related Compound C<br>Stability Light Sensitive<br>Applications 1,1'-(1,3-Phenylene)bis-1H-1,2,4-triazole (Fluconazole EP Impurity C) is a Fluconazole (F421000) impurity.<br>References Bauer, M., et al.: Eur. J. Pharma. Sci., 6, 331 (1998), Dongre, V., et al.: J. Pharma. Biomed. Anal., 42, 334 (2006),<br></p>Fórmula:C10H8N6Forma y color:BeigePeso molecular:212.21tert-Butyl (R)-3-Aminopiperidine-1-carboxylate
CAS:Producto controlado<p>Applications tert-Butyl (R)-3-Aminopiperidine-1-carboxylate, is an heterocyclic building block used for the synthesis of more complex pharmaceutical compounds. It is also found to act as a γ-secretase modulators, and a potent structure for lowering Aβ42 production in both in vitro and in vivo.<br>References Kobayashi, T., et al.: Bioorg. Med. Chem. Lett., 24, 378 (2014);<br></p>Fórmula:C10H20N2O2Forma y color:NeatPeso molecular:200.284-(3-Aminophenyl)-3-morpholinone
CAS:Producto controlado<p>Applications 4-(3-Aminophenyl)-3-morpholinone is an intermediate during the preparation of imidazothiazoles as protein kinase inhibitors for treating cancers.<br>References Bamaung, N., et al.: PCT Int. Appl. (2009), WO 2009070516 A1 20090604.<br></p>Fórmula:C10H12N2O2Forma y color:NeatPeso molecular:192.2142-((2R,3R)-4-(Anthracen-9-yl)-3-(tert-butyl)-2,3-dihydrobenzo[d][1,3]oxaphosphol-2-yl)pyridine
CAS:Pureza:97%Peso molecular:447.51800537109375Desfluoro Risperidone
CAS:Producto controlado<p>Impurity Risperidone EP Impurity K<br>Applications Desfluoro Risperidone (Risperidone EP Impurity K) is a Risperidone (R525000) impurity, as antipsychotics.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Fórmula:C23H28N4O2Forma y color:NeatPeso molecular:392.49Adrafinil
CAS:Producto controladoFórmula:C15H15NO3SForma y color:Off-White Light Orange ColourPeso molecular:289.35N-Desmethyl Deferiprone
CAS:Producto controladoFórmula:C6H7NO2Forma y color:NeatPeso molecular:125.13(Z,Z)-5-(2-Methyl-3-phenyl-propenylidene)-4-oxo-2-thioxo-3-thiazolidineacetic Acid
CAS:Producto controlado<p>Stability Light Sensitive<br>Applications (Z,Z)-5-(2-Methyl-3-phenyl-propenylidene)-4-oxo-2-thioxo-3-thiazolidineacetic Acid is a stereoisomer of Epalrestat (E565300), an aldose reductase inhibitor. Used in the treatment of diabetic neuropathy.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Terashima, H., et al.: J. Pharmacol. Exp. Ther., 229, 226 (1983), Kikkawa, R., et al.: Diabetologia, 24, 290 (1983), Kojima, K., et al.: Jpn. J. Ophthalmol., 29, 99 (1985), Qi, M. et al.: J. Beij, Inst. Tech., 13, 445 (2004);<br></p>Fórmula:C15H13NO3S2Forma y color:Yellow-Red SolidPeso molecular:319.410H-Phenothiazine-2-carbonitrile
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:224.27999877929688
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