Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65541 productos de "Derivados de Quinazolina y Quinolina"
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CAS:<p>P2X1 receptor antagonist</p>Fórmula:C18H15N4NaO14PS2Pureza:98%Forma y color:SolidPeso molecular:629.42Licogliflozin
CAS:<p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>Fórmula:C23H28O7Pureza:98%Forma y color:SolidPeso molecular:416.46Propoxur
CAS:<p>Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.</p>Fórmula:C11H15NO3Pureza:99.84% - 99.87%Forma y color:Minute Crystals (Niosh 2016)Peso molecular:209.24Evogliptin HCl
CAS:<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Fórmula:C19H27ClF3N3O3Forma y color:SolidPeso molecular:437.88LPA2 antagonist 1
CAS:<p>LPA2 antagonist 1 is a potent LPA2 antagonist.</p>Fórmula:C20H23Cl2N5O2S2Pureza:99.85%Forma y color:SolidPeso molecular:500.47Evogliptin
CAS:<p>Evogliptin (DA-1229) is an oral DPP4 inhibitor effective in reducing blood sugar and liver inflammation.</p>Fórmula:C19H26F3N3O3Forma y color:SolidPeso molecular:401.42WAY-151693
CAS:<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Fórmula:C21H22ClN3O5SForma y color:SolidPeso molecular:463.93Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Forma y color:SolidPeso molecular:481.56Otamixaban
CAS:<p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>Fórmula:C25H26N4O4Pureza:98.08%Forma y color:SolidPeso molecular:446.5Bornaprine
CAS:<p>Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.</p>Fórmula:C21H31NO2Forma y color:SolidPeso molecular:329.48Midodrine (R-isomer HCl)
CAS:<p>Midodrine is a vasopressor/antihypertensive agent for the treatment of symptomatic postural hypotension.</p>Fórmula:C12H19ClN2O4Forma y color:SolidPeso molecular:290.74(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Forma y color:SolidPeso molecular:398.34Gemigliptin Tartrate(911637-19-9 free base)
CAS:<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Fórmula:C22H25F8N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:639.45Laropiprant
CAS:<p>Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki</p>Fórmula:C21H19ClFNO4SPureza:98.24% - 99.89%Forma y color:SolidPeso molecular:435.9Nifekalant hydrochloride
CAS:<p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>Fórmula:C19H28ClN5O5Pureza:99.91%Forma y color:SolidPeso molecular:441.91MMP13-IN-4
CAS:<p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>Fórmula:C21H17BrN4O5Pureza:98%Forma y color:SolidPeso molecular:485.29Carisbamate
CAS:<p>CarisbAMate (JNJ-10234094, RWJ 333369, YKP-509) is an antiepileptic drug candidate.</p>Fórmula:C9H10ClNO3Forma y color:SolidPeso molecular:215.63Blonanserin HCl
CAS:<p>Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.</p>Fórmula:C23H32Cl2FN3Pureza:98%Forma y color:SolidPeso molecular:440.42Bifeprunox
CAS:<p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>Fórmula:C24H23N3O2Pureza:98%Forma y color:SolidPeso molecular:385.46Pirbuterol
CAS:<p>Pirbuterol, a short-acting β2 adrenoreceptor agonist, has bronchodilating action used in the treatment of asthma.</p>Fórmula:C12H20N2O3Forma y color:SolidPeso molecular:240.3Clonidine
CAS:<p>Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.</p>Fórmula:C9H9Cl2N3Pureza:99.42% - 99.44%Forma y color:Crystals SolidPeso molecular:230.09MMP-2/9-IN-1
CAS:<p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>Fórmula:C14H16IN7SForma y color:SolidPeso molecular:441.29(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SForma y color:SolidPeso molecular:322.47M-25
CAS:<p>M-25 is a Smoothened antagonist and inhibitor of the Hedgehog pathway.</p>Fórmula:C23H29N3O2Forma y color:SolidPeso molecular:379.5Robenidine
CAS:<p>Robenidine, an anticoccidial guanidine, is used as an additive in rabbit fodder.</p>Fórmula:C15H13Cl2N5Pureza:98%Forma y color:SolidPeso molecular:334.2(R)-Afatinib
CAS:<p>(R)-Afatinib: oral ErbB inhibitor (EGFR/HER2), IC50 ≤14 nM. For ESCC, NSCLC, gastric cancer research.</p>Fórmula:C24H25ClFN5O3Forma y color:SolidPeso molecular:485.94MMP2-IN-2
CAS:<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Fórmula:C13H8N4O4Pureza:98.09%Forma y color:SolidPeso molecular:284.23TAK-875 Hemihydrate
CAS:<p>TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.</p>Fórmula:C29H32O7SH2OPureza:98%Forma y color:SolidPeso molecular:533.63U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Forma y color:SolidPeso molecular:448.56Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Fórmula:C19H24N2OPureza:98%Forma y color:SolidPeso molecular:296.41Ketotifen
CAS:<p>Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.</p>Fórmula:C19H19NOSForma y color:SolidPeso molecular:309.43Isothipendyl
CAS:<p>Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.</p>Fórmula:C16H19N3SForma y color:SolidPeso molecular:285.41PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Forma y color:SolidPeso molecular:464.96Mesopram
CAS:<p>PDE4 inhibitor, orally active</p>Fórmula:C14H19NO4Pureza:98%Forma y color:SolidPeso molecular:265.3Selatinib
CAS:<p>Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer activity that inhibits the growth of NCI-N87 tumor cells.</p>Fórmula:C29H26ClFN4O3SPureza:98.00%Forma y color:SolidPeso molecular:565.06Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Fórmula:C12H14N4OSPureza:98%Forma y color:SolidPeso molecular:262.33Alimemazine
CAS:<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Fórmula:C18H22N2SPureza:98%Forma y color:Crystals SolidPeso molecular:298.45CP-471474
CAS:<p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>Fórmula:C16H17FN2O5SPureza:98%Forma y color:SolidPeso molecular:368.38Propentofylline
CAS:<p>Propentofylline (Hextol) has neuroprotective, antiproliferative and anti-inflammatory activities and can be used in the study of Alzheimer's disease.</p>Fórmula:C15H22N4O3Pureza:99.76% - 99.86%Forma y color:Off-White SolidPeso molecular:306.36RS-104966
CAS:<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Fórmula:C19H21NO6SPureza:98%Forma y color:SolidPeso molecular:391.44Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Fórmula:C23H31N3NaO4S2Pureza:98%Forma y color:SolidPeso molecular:500.63(R)-Azelastine
CAS:<p>(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Fórmula:C22H24ClN3OForma y color:SolidPeso molecular:381.9Quoromycin
CAS:<p>Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.</p>Fórmula:C12H8N2O2SForma y color:SolidPeso molecular:244.27Cycloguanil
CAS:<p>Cycloguanil is an antimalarial.</p>Fórmula:C11H14ClN5Pureza:98%Forma y color:SolidPeso molecular:251.72Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Fórmula:C24H27Cl2FN6OPureza:98%Forma y color:SolidPeso molecular:505.42Piperaquine
CAS:<p>Piperaquine is a bisquinoline antimalarial compound and a companion compound to artemisinin.</p>Fórmula:C29H32Cl2N6Pureza:98%Forma y color:SolidPeso molecular:535.51Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Fórmula:C20H24N2O5Forma y color:SolidPeso molecular:372.42(S)-Pomalidomide
CAS:<p>(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.</p>Fórmula:C13H11N3O4Forma y color:SolidPeso molecular:273.24Zuclopenthixol decanoate
CAS:<p>Zuclopenthixol decanoate is an anti-schizophrenia drug.</p>Fórmula:C32H43ClN2O2SPureza:98%Forma y color:SolidPeso molecular:555.21Metaproterenol
CAS:<p>Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).</p>Fórmula:C11H17NO3Pureza:98%Forma y color:SolidPeso molecular:211.26Fidarestat
CAS:<p>Fidarestat (SNK 860),Aldose reductase inhibitor (IC50=26 nM). Targets AKR1B10 (33 μM) and V301L AKR1B10 (1.8 μM). Potential diabetes treatment.</p>Fórmula:C12H10FN3O4Pureza:98%Forma y color:SolidPeso molecular:279.22Levomepromazine Maleate
CAS:<p>Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.</p>Fórmula:C23H28N2O5SForma y color:SolidPeso molecular:444.546Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Forma y color:White To Pink PowderPeso molecular:291.39(R)-Carvedilol
CAS:<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Forma y color:SolidPeso molecular:406.47Bromhexine
CAS:<p>Bromhexine is an expectorant/mucolytic agent which can be used in the treatment of respiratory disorders associated with excessive mucus or viscid.</p>Fórmula:C14H20Br2N2Pureza:98%Forma y color:SolidPeso molecular:376.13Vapendavir diphosphate
CAS:<p>Vapendavir diphosphate binds enterovirus capsids, inhibiting EV71 replication effectively (EC50: 0.5-1.4 μM).</p>Fórmula:C21H32N4O11P2Pureza:98.75% - 98.75%Forma y color:SolidPeso molecular:578.45BR351
CAS:<p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C20H25FN2O5SPureza:98%Forma y color:SolidPeso molecular:424.49CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Fórmula:C12H14ClN3OPureza:98%Forma y color:SolidPeso molecular:251.71Deterenol Free Base
CAS:<p>Deterenol Free Base is a beta-adrenoceptor agonist.</p>Fórmula:C11H17NO2Forma y color:SolidPeso molecular:195.26Niclosamide monohydrate
CAS:<p>Niclosamide Monohydrate is used for the treatment of most tapeworm infections by inhibiting DNA replication.</p>Fórmula:C13H10Cl2N2O5Pureza:98%Forma y color:SolidPeso molecular:345.14(S)-Carvedilol
CAS:<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Forma y color:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47Clofedanol
CAS:<p>Clofedanol, also known as chlophedianol or antitussin, is used in the treatment of pediatric pertussis.</p>Fórmula:C17H20ClNOPureza:98%Forma y color:SolidPeso molecular:289.8(S)-Azelastine
CAS:<p>(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.</p>Fórmula:C22H24ClN3OForma y color:SolidPeso molecular:381.9Vandetanib Fumarate
CAS:<p>Oral tyrosine kinase inhibitor Vandetanib Fumarate targets RET, VEGFRs, EGFR in thyroid cancer.</p>Fórmula:C26H28BrFN4O6Pureza:98%Forma y color:SolidPeso molecular:591.43Procarbazine free base
CAS:<p>Procarbazine: chemo drug for Hodgkin's, brain cancer; liver-activated; MAO inhibitor.</p>Fórmula:C12H19N3OPureza:98%Forma y color:SolidPeso molecular:221.3BP-5-087
CAS:<p>BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.</p>Fórmula:C36H30F8N2O6SForma y color:SolidPeso molecular:770.69Afacifenacin
CAS:<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Fórmula:C27H26F3N3O2Pureza:99.83%Forma y color:SolidPeso molecular:481.51Enadoline (Free Base)
CAS:<p>Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.</p>Fórmula:C24H32N2O3Forma y color:SolidPeso molecular:396.52(R)-Hydroxychloroquine
CAS:<p>(R)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine is an agent of synthetic antimalarial.</p>Fórmula:C18H26ClN3OPureza:98%Forma y color:SolidPeso molecular:335.87Daltroban
CAS:<p>Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist.</p>Fórmula:C16H16ClNO4SPureza:99.74%Forma y color:SolidPeso molecular:353.82Benserazide
CAS:<p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>Fórmula:C10H15N3O5Forma y color:SolidPeso molecular:257.24cis-Tadalafil
CAS:<p>Cis-Tadalafil is a potent inhibitor of phosphodiesterase 5, which is used to treat erectile dysfunction (ED) and primary pulmonary hypertension (PPH). It works by increasing blood flow to the penis, allowing men with ED to achieve and maintain an erection. Cis-Tadalafil is also used to treat symptoms of prostatic hyperplasia (enlarged prostate) in men. This drug has been shown to be effective in treating PPH by reducing pulmonary arterial pressure and improving exercise capacity. Cis-Tadalafil belongs to the carboline class of drugs and is a phosphodiesterase 5 inhibitor that selectively inhibits cGMP-specific phosphodiesterase type 5 (PDE5). This drug has been shown to be highly effective in treating both ED and PPH with minimal side effects.</p>Fórmula:C22H19N3O4Pureza:Min. 95%Forma y color:White/Off-White SolidPeso molecular:389.4 g/molGivinostat hydrochloride monohydrate
CAS:<p>Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.</p>Fórmula:C24H27N3O4·HCl·H2OPureza:97.97% - 99.51%Forma y color:SolidPeso molecular:475.97Pipotiazine
CAS:<p>Pipotiazine treats chronic schizophrenia with less sedation, low hypotension risk, but high extrapyramidal side effects.</p>Fórmula:C24H33N3O3S2Forma y color:SolidPeso molecular:475.67Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Fórmula:C21H25NOPureza:98%Forma y color:SolidPeso molecular:307.43Riodoxol
CAS:<p>Riodoxol is an antiviral agent that effectively affects the reproduction and maturation of viruses.</p>Fórmula:C6H3I3O2Forma y color:SolidPeso molecular:487.8Benproperine
CAS:<p>Benproperine is a bioactive molecule with antineoplastic properties.</p>Fórmula:C21H27NOPureza:98%Forma y color:SolidPeso molecular:309.45NBI-42902
CAS:<p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>Fórmula:C27H24F3N3O3Forma y color:SolidPeso molecular:495.49Rufloxacin hydrochloride
CAS:<p>Rufloxacin HCl (MF-934 HCl): a fluoroquinolone that inhibits topoisomerase and B-cell differentiation.</p>Fórmula:C17H19ClFN3O3SPureza:99.80%Forma y color:SolidPeso molecular:399.867Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Fórmula:C20H21NO5Forma y color:SolidPeso molecular:355.38Lanicemine
CAS:<p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>Fórmula:C13H14N2Pureza:98%Forma y color:SolidPeso molecular:198.26Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Fórmula:C23H19ClO3SPureza:98%Forma y color:SolidPeso molecular:410.91Esreboxetine
CAS:<p>Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.</p>Fórmula:C19H23NO3Forma y color:SolidPeso molecular:313.39Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Forma y color:SolidPeso molecular:264.36Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Fórmula:C22H24ClF4NO2Forma y color:SolidPeso molecular:445.88Protriptyline
CAS:<p>Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.</p>Fórmula:C19H21NForma y color:SolidPeso molecular:263.38Piribedil dihydrochloride
CAS:<p>dopamine agonist</p>Fórmula:C16H20Cl2N4O2Pureza:98%Forma y color:SolidPeso molecular:371.26Azatadine
CAS:<p>Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).</p>Fórmula:C20H22N2Pureza:98%Forma y color:SolidPeso molecular:290.4Indisetron Dihydrochloride
CAS:<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Fórmula:C17H24ClN5OForma y color:SolidPeso molecular:349.86Oxolamine
CAS:<p>Oxolamine is an agent of a cough suppressant.</p>Fórmula:C14H19N3OPureza:98%Forma y color:SolidPeso molecular:245.32Rolapitant
CAS:<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Fórmula:C25H26F6N2O2Pureza:99.86%Forma y color:SolidPeso molecular:500.48Distigmine Bromide
CAS:<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Fórmula:C22H32BrN4O4Pureza:98%Forma y color:SolidPeso molecular:496.42Indenolol
CAS:<p>Indenolol is a blocker of beta-adrenergic.</p>Fórmula:C15H21NO2Pureza:98%Forma y color:SolidPeso molecular:247.33Oxyphenbutazone monohydrate
CAS:<p>Oxyphenbutazone monohydrate: Phenylbutazone derivative, anti-inflammatory, non-selective COX inhibitor, kills dormant M. tuberculosis.</p>Fórmula:C19H22N2O4Forma y color:SolidPeso molecular:342.39Enflicoxib
CAS:<p>Enflicoxib is an effective treatment for canine osteoarthritis pain and inflammation, with faster onset than mavacoxib, improving veterinary outcomes.</p>Fórmula:C16H12F5N3O2SPureza:99.88%Forma y color:SolidPeso molecular:405.34Vernakalant
CAS:<p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>Fórmula:C20H31NO4Pureza:98%Forma y color:SolidPeso molecular:349.46Phenindamine Tartrate
CAS:<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Fórmula:C23H25NO6Forma y color:SolidPeso molecular:411.454Pridinol
CAS:<p>Pridinol is an antispasmodic and muscle relaxant.</p>Fórmula:C20H25NOPureza:98%Forma y color:Crystals SolidPeso molecular:295.42GW-3333
CAS:<p>GW-3333 inhibits matrix metalloproteinases and TNF-Converting Enzyme, showing potential as an antiarthritic therapy.</p>Fórmula:C22H36N4O4Pureza:98%Forma y color:SolidPeso molecular:420.55Moricizine
CAS:<p>Moricizine is an antiarrhythmia agent which is used primarily for ventricular rhythm disturbances.</p>Fórmula:C22H25N3O4SPureza:98%Forma y color:SolidPeso molecular:427.52(S)-Propafenone
CAS:<p>(S)-Propafenone, or (S)-SA-79, is an S-enantiomer with beta-blocking effects and sodium channel blocking class 1 antiarrhythmic properties.</p>Fórmula:C21H27NO3Pureza:98%Forma y color:SolidPeso molecular:341.44ABT-770
CAS:<p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>Fórmula:C22H22F3N3O6Forma y color:SolidPeso molecular:481.42(Rac)-Tanomastat
CAS:<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Fórmula:C23H19ClO3SForma y color:SolidPeso molecular:410.91TAPI-0
CAS:<p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>Fórmula:C24H32N4O5Forma y color:SolidPeso molecular:456.53WAY 629
CAS:<p>WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.</p>Fórmula:C15H18N2Forma y color:SolidPeso molecular:226.32(R)-Praziquantel
CAS:<p>(R)-Praziquantel is an active enantiomer of praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Forma y color:SolidPeso molecular:312.41ND-336
CAS:<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Fórmula:C16H18ClNO3S2Forma y color:SolidPeso molecular:371.9Vildagliptin related compound F
CAS:<p>Vildagliptin related compound F (VRCF) is a drug product that has been custom synthesized. VRCF is a high purity, analytical standard. It is metabolized in the body and can be used as a research and development standard to study the metabolism of vildagliptin. VRCF is a natural metabolite that has been identified as an impurity in the drug product Vildagliptin. VRCF has not been recognized by the USP or EP for use as an impurity standard. CAS no: 1789703-36-1</p>Fórmula:C17H24N2O3Pureza:Min. 95%Forma y color:PowderPeso molecular:304.4 g/molLaduviglusib trihydrochloride
CAS:<p>Laduviglusib trihydrochloride, a GSK-3α/β inhibitor (IC50: 10/6.7 nM), activates Wnt/β-catenin signaling and induces autophagy.</p>Fórmula:C22H20Cl5N8Pureza:99.34%Forma y color:SolidPeso molecular:573.71N-De[2-(methylsulfonyl)ethyl] lapatinib
CAS:<p>Lapatinib is a tyrosine kinase inhibitor that blocks the epidermal growth factor receptor (EGFR) and other tyrosine kinases. It is used in cancer treatment to inhibit tumor growth, with a high success rate. Lapatinib is also used to treat lung cancer and other types of cancer. The drug has been shown to inhibit EGFR phosphorylation in vitro, which leads to inhibition of cell proliferation and induction of apoptosis. Lapatinib also inhibits the expression of EGFR downstream target genes such as b-raf, serine/threonine-protein kinase, and cyp3a5.</p>Fórmula:C26H20ClFN4O2Pureza:Min. 95%Peso molecular:474.91 g/molVildagliptin Related Compound 2
CAS:<p>Vildagliptin Related Compound 2 is a synthetic compound that has been shown to be an inhibitor of DPP-4. It is a white solid that can be synthesized by condensation of vildagliptin with chloroacetyl chloride in the presence of an alkali. The compound was found to have impurities, including 1-(2-chlorophenyl)ethanol and 3-chlorobenzaldehyde.</p>Fórmula:C17H25N3O2Pureza:Min. 95%Peso molecular:303.4 g/molAmlodipine EP Impurity E maleate
CAS:<p>Amlodipine EP Impurity E maleate is a high purity and analytical grade chemical. It is a metabolite of Amlodipine, which is used in the treatment of hypertension. This chemical has been shown to be a natural product that is produced by the human body. It also has been shown to have pharmacological properties, such as anti-inflammatory and vasodilatory effects. The impurity standard for this compound is available from Sigma-Aldrich.br>br></p>Fórmula:C21H27ClN2O5•C4H4O4Pureza:Min. 95%Peso molecular:538.98 g/molN-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methyloxirane-2-carboxamide
CAS:<p>N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methyloxirane-2-carboxamide (NUOX) is a potential anticancer agent that has been shown to have an acidic pKa of 5.8 and to be active against cancer cells in the same way as bicalutamide, which is a known antiandrogen. NUOX has been shown to increase the number of cavities in polybenzimidazole (PBI) films by enhancing the rate of oxidation. NUOX also inhibits the growth of human cancer cells by binding sulfide groups on proteins and DNA, inhibiting cellular respiration. NUOX is not water soluble, so it must be dissolved in solvents such as acetonitrile or chloroform before administration.</p>Fórmula:C12H9F3N2O2Pureza:Min. 95%Forma y color:White PowderPeso molecular:270.21 g/molEzetimibe ketone
CAS:<p>Ezetimibe ketone is a lipid-lowering agent that inhibits cholesterol absorption through the inhibition of Niemann-Pick C1-like 1 (NPC1L1). Ezetimibe ketone is used to reduce the levels of low-density lipoprotein cholesterol (LDL-C) in patients with primary hypercholesterolemia, sitosterolemia, and familial combined hyperlipidemia. Ezetimibe ketone has been shown to be bioequivalent to ezetimibe, which is an oral drug that inhibits cholesterol absorption by blocking NPC1L1. The drug binds to the NPC1L1 receptor in the brush border membrane of enterocytes and prevents cholesterol uptake. Ezetimibe ketone has a high solubility in organic solvents such as dichloromethane or chloroform. It also has a high melting point, which makes it suitable for use on chromatographic columns.</p>Fórmula:C24H19F2NO3Pureza:Min. 95%Forma y color:PowderPeso molecular:407.41 g/mol3-Trifluoroacetylamino linagliptin
CAS:<p>Please enquire for more information about 3-Trifluoroacetylamino linagliptin including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C27H27F3N8O3Pureza:Min. 95%Peso molecular:568.55 g/mol(S)-Rabeprazole sodium
CAS:<p>(S)-Rabeprazole sodium is an anticancer drug that acts as a kinase inhibitor. It is an analog of Rabeprazole and has been shown to inhibit the growth of cancer cells in vitro and in vivo. (S)-Rabeprazole sodium inhibits the activity of kinases, which are enzymes that play a key role in cell signaling pathways. This inhibition leads to apoptosis, or programmed cell death, in cancer cells. (S)-Rabeprazole sodium has been tested against various types of cancer, including Chinese hamster ovary cells and tumor xenografts in mice. It has also been shown to inhibit elastin degradation, which is important for preventing metastasis of cancer cells. (S)-Rabeprazole sodium may be a promising candidate for the development of new anticancer drugs that target specific kinases and proteins involved in cancer cell growth and survival.</p>Fórmula:C18H21N3O3S•NaPureza:Min. 95%Peso molecular:382.43 g/molImipramine
CAS:<p>Imipramine (Dimipressin) is a Fascin1 inhibitor with antitumor activity and induces apoptosis.</p>Fórmula:C19H24N2Pureza:99.4%Forma y color:White To Off-White /Hydrochloride/ SolidPeso molecular:280.41Amiodarone impurity E
CAS:<p>Amiodarone impurity E is a nucleophilic compound that is synthesized by the acylation of a diazonium salt with an amine. It has been shown to be active against staphylococci, but not against subtilis. The reaction may be catalyzed by acid or chloride. Amiodarone impurity E is also demethylated and dehydrated to form the final product, amiodarone.</p>Fórmula:C19H18O3Pureza:Min. 95%Forma y color:PowderPeso molecular:294.34 g/mol(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Fórmula:C23H29N3O2S2Pureza:99.21%Forma y color:Yellow To Yellow With A Tan Cast PowderPeso molecular:443.63Pantoprazole sulphide
CAS:<p>Pantoprazole sulphide is a benzimidazole derivative that has been synthesized in an asymmetric synthesis. The purified compound was characterized by its nmr spectra, which showed the presence of the carboethoxy group and the chromatographic method. The compound belongs to a family of inhibitors known as benzimidazole derivatives and has shown inhibitory activity against a number of bacterial species including Staphylococcus aureus, Clostridium perfringens, and Mycobacterium tuberculosis. Pantoprazole sulphide has been used as an inhibitor to treat gastric acid pump disorders such as Zollinger-Ellison syndrome. It is also used for treating pathological conditions such as duodenal ulcers or gastroesophageal reflux disease.</p>Fórmula:C16H15F2N3O3SPureza:Min. 95%Forma y color:PowderPeso molecular:367.37 g/molGivinostat hydrochloride
CAS:<p>Givinostat HCl (ITF2357 HCl) inhibits HDAC1/3 (IC50: 198/157 nM) with anti-inflammatory, anti-angiogenic, and antineoplastic properties.</p>Fórmula:C24H28ClN3O4Pureza:99.39%Forma y color:SolidPeso molecular:457.95Arimoclomol
CAS:<p>Arimoclomol (BRX-220 free base) is a co-inducer of heat shock proteins (HSP) and can be used in studies about the treatment of amyotrophic lateral sclerosis (</p>Fórmula:C14H20ClN3O3Pureza:99.15%Forma y color:SolidPeso molecular:313.78Eltenac
CAS:<p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>Fórmula:C12H9Cl2NO2SPureza:98.53%Forma y color:SolidPeso molecular:302.18Edoxaban
CAS:<p>Edoxaban: potent, selective FXa inhibitor; Ki 0.561 nM. Used as an oral anticoagulant for stroke prevention, also inhibits thrombin and FIXa.</p>Fórmula:C24H30ClN7O4SPureza:97.67% - 99.71%Forma y color:SolidPeso molecular:548.06DB04760
CAS:<p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>Fórmula:C22H20F2N4O2Pureza:99.93% - 99.99%Forma y color:SolidPeso molecular:410.42ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
CAS:<p>Please enquire for more information about ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C22H22N4O4Pureza:Min. 95%Peso molecular:406.43 g/molStepronin
CAS:<p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>Fórmula:C10H11NO4S2Pureza:99.59%Forma y color:White Or Off White CrystallinePeso molecular:273.33Pitavastatin N-oxide
CAS:<p>Pitavastatin N-oxide is a drug product that is an analytical standard and natural API impurity. It is used in the synthesis of other drugs, such as pitavastatin, which is a statin drug used to lower cholesterol levels. Pitavastatin N-oxide has been shown to be a potent inhibitor of HMG-CoA reductase, the enzyme that catalyzes the conversion of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) to mevalonate. This inhibits cholesterol production and lowers levels of low density lipoprotein (LDL) cholesterol in the blood.</p>Fórmula:C25H24FNO5Pureza:Min. 95%Peso molecular:437.46 g/mol(R,R)-Montelukast bis-sulfide
CAS:<p>(R,R)-Montelukast bis-sulfide is a drug product that is used in the analytical and research and development of drugs. It is also used as an impurity standard for HPLC. (R,R)-Montelukast bis-sulfide has been shown to have niche applications in drug development and research, as well as being a high purity API.</p>Fórmula:C41H46ClNO5S2Pureza:90%MinPeso molecular:732.39 g/molMMP2-IN-3
CAS:<p>MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).</p>Fórmula:C23H21N3OPureza:99.38%Forma y color:SolidPeso molecular:355.43Amlodipine EP Impurity F maleate
CAS:<p>Amlodipine EP Impurity F maleate is an impurity of amlodipine, a drug product. It is a natural substance that has been classified as an API impurity in the United States Pharmacopeia (USP). The chemical name for this drug is 3-(2-chlorophenyl)-1-methyl-5-(o-tolyloxy)-2,4-dihydro-6H-[1,3]thiazolo[3,2-a]pyrimidin-7-one. Amlodipine EP Impurity F maleate has the following properties: C12H9ClNO2S and a melting point of 210°C with a purity of 99.5%. This compound was synthesized by custom synthesis and is used as an analytical standard for HPLC. This compound was also used during the development of amlodipine to determine its metabolism studies.</p>Fórmula:C19H23ClN2O5•C4H4O4Pureza:Min. 95%Peso molecular:510.92 g/molMMP-2/MMP-9 Inhibitor I
CAS:<p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>Fórmula:C21H19NO4SPureza:99.74%Forma y color:SolidPeso molecular:381.44Pramipexole EP Impurity C
CAS:<p>Pramipexole EP Impurity C is a synthetic impurity that is used as an impurity standard in the manufacture of Pramipexole EP. It is also used as a research and development tool for drug product, custom synthesis, CAS No. 1973461-14-1, and analytical studies. This compound has been shown to be a metabolite of Pramipexole EP and may have pharmacological properties. Pramipexole EP Impurity C has been found to inhibit the growth of certain bacteria, such as methicillin-resistant Staphylococcus aureus (MRSA) isolates.</p>Fórmula:C20H32N6S2Pureza:Min. 95%Moveltipril
CAS:<p>Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action.</p>Fórmula:C19H30N2O5SPureza:97.55% - 98.28%Forma y color:SolidPeso molecular:398.52Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Forma y color:SolidPeso molecular:323.461-Oxo mirtazapine
CAS:<p>1-Oxo mirtazapine is a metabolite of mirtazapine. It is a synthetic compound and is not found in nature. This product is a research and development impurity standard for the preparation of drug product, which has been synthesized to be highly pure. The material is used for drug development, including pharmacopoeia requirements for analytical studies and metabolism studies. 1-Oxo mirtazapine has been shown to have niche applications in pharmacopoeia and as an HPLC standard.</p>Fórmula:C17H17N3OPureza:Min. 95%Peso molecular:279.34 g/molCP-544439
CAS:<p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>Fórmula:C18H19FN2O6SPureza:95.02% - 98.66%Forma y color:SolidPeso molecular:410.42Gallopamil
CAS:<p>Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.</p>Fórmula:C28H40N2O5Pureza:99.85%Forma y color:SolidPeso molecular:484.631-Fluoronaphthalene
CAS:<p>1-Fluoronaphthalene is a polyunsaturated compound that is used in analytical chemistry for the determination of test samples. It is an inhibitor of the enzyme IDO1, which plays an important role in the regulation of immune function, and has been shown to have anti-inflammatory properties. 1-Fluoronaphthalene can be synthesized by reacting n-dimethyl formamide with hydrogen fluoride and then adding a diazonium salt and hydrochloric acid. The UV absorption spectrum of 1-fluoronaphthalene displays a maximum at 248 nm. This compound binds to cation channels on cells, causing hyperpolarization.</p>Fórmula:C10H7FPureza:Min. 95%Peso molecular:146.16 g/mol2,3,4,5-Tetradehydro alfuzosin hydrochloride
CAS:<p>Alfuzosin is a potent, selective, and long-acting α1A-adrenergic receptor antagonist. It is used to treat benign prostatic hyperplasia (BPH) in males. Alfuzosin is also used as an antihypertensive agent, for the treatment of pheochromocytoma, and for the treatment of benign prostatic hyperplasia in males. The hydrogenation of 2,3,4,5-tetradehydroalfuzosin to alfuzosin hydrochloride is performed by liquid hydrogenation or by hydrogenation on a palladium catalyst in a mixture of dimethylformamide and hexamethylphosphoramide. This process minimizes the formation of impurities such as 2,3,4-trimethoxy alfuzosin.</p>Fórmula:C19H24ClN5O4Pureza:Min. 95%Forma y color:White PowderPeso molecular:421.88 g/molEphedrine Hydrochloride
CAS:Producto controladoEphedrine and its saltsFórmula:C10H15NO·HClForma y color:White Off-White PowderPeso molecular:201.09204Apixaban Impurity 1
CAS:<p>Apixaban Impurity 1 is an impurity found in Apixaban, a drug used for the prevention of stroke. It is produced by condensation of 2-aminopyridine and 3-hydroxybenzaldehyde in ethanol with sodium hydroxide as a catalyst. The reaction proceeds via amination of the pyridine ring followed by transesterification. The yield of this impurity is low at about 4%.</p>Pureza:Min. 95%UNC0321
CAS:<p>UNC0321 is an effective inhibitor of histone methyltransferase G9a with a Ki of 63 pM and with IC50s 9 nM and 6 nM in ECSD and CLOT assays.</p>Fórmula:C27H45N7O3Pureza:99.80%Forma y color:SolidPeso molecular:515.69Brivaracetam CV
CAS:Producto controladoLactams, nesoiFórmula:C11H20N2O2Forma y color:White Off-White SolidPeso molecular:212.15248AGPS-IN-2i
CAS:<p>AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.</p>Fórmula:C18H17F2N3O2Pureza:98.92%Forma y color:SolidPeso molecular:345.34Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Fórmula:C13H19NO3Pureza:99.67%Forma y color:SolidPeso molecular:237.29Apixaban Impurity 6
CAS:<p>Please enquire for more information about Apixaban Impurity 6 including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C26H26N4O5Pureza:Min. 95%Peso molecular:474.51 g/molEmpagliflozin S-furanose
CAS:<p>Empagliflozin S-furanose is a Custom synthesis drug product. It is an analytical standard with CAS No. 1620758-32-8, and it is used in research and development of new drugs. Empagliflozin S-furanose has been found to be a metabolite of empagliflozin, a drug that is used to treat type 2 diabetes mellitus. It is also used as an impurity standard for HPLC analysis of empagliflozin because it does not have any biological activity.</p>Fórmula:C23H27ClO7Pureza:Min. 95%Forma y color:PowderPeso molecular:450.91 g/mol(R)-Zanubrutinib
CAS:<p>(R)-Zanubrutinib ((R)-BGB-3111) is a selective inhibitor of Bruton tyrosine kinase (BTK).</p>Fórmula:C27H29N5O3Pureza:99.55%Forma y color:SolidPeso molecular:471.55Desfluoro ezetimibe
CAS:<p>Desfluoro ezetimibe is a synthetic cholesterol-lowering drug that inhibits intestinal cholesterol absorption. It is chemically synthesized, and the process includes the introduction of fluorine at the 3-position of the C-ring. Desfluoro ezetimibe is not metabolized in humans, but it may be subject to oxidative degradation. The product is also subject to oxidation by light and air, which may result in formation of impurities. The drug substance has been validated as well as its isomers and efficiencies in mass spectrometry detection.</p>Fórmula:C24H22FNO3Pureza:Min. 95%Forma y color:White To Off-White SolidPeso molecular:391.43 g/molFenoverine
CAS:<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Fórmula:C26H25N3O3SPureza:98.34%Forma y color:SolidPeso molecular:459.56Gemigliptin
CAS:<p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>Fórmula:C18H19F8N5O2Pureza:99.72%Forma y color:SolidPeso molecular:489.36Roflumilast Impurity A
CAS:<p>Roflumilast impurity A is a metabolite of roflumilast. It is a drug product that is used as an analytical standard for the determination of roflumilast in HPLC analysis. Roflumilast impurity A is not natural and is synthetic. It has been shown to be a substrate for CYP1A2, CYP2C8, CYP2C9, and CYP3A4 enzymes. Studies have shown that it may be involved in the metabolism of roflumilast through hydroxylation and deamination.</p>Fórmula:C16H14Cl2N2O3Pureza:Min. 95%Peso molecular:353.2 g/molLinagliptin impurity G
CAS:<p>Linagliptin impurity G is an impurity in the drug product Linagliptin. It is a natural substance and its CAS number is 668270-11-9. Impurity G can be synthesized from L-phenylalanine and cyclohexane carboxaldehyde in a two step process. The first step involves the reaction of L-phenylalanine with cyclohexane carboxaldehyde to yield methylcyclohexanecarboxylate, which then undergoes hydrolysis to give phenylcyclohexanol. In the second step, phenylcyclohexanol reacts with hydrochloric acid to produce phenylcyclohexanone, which is then oxidized with hydrogen peroxide to yield impurity G. Impurity G can also be found in the pharmacopoeia as a high purity HPLC standard for linagliptin.</p>Fórmula:C25H28N8O2Pureza:Min. 95%Forma y color:PowderPeso molecular:472.54 g/molSovaprevir
CAS:<p>Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.</p>Fórmula:C43H53N5O8SPureza:99.11%Forma y color:SolidPeso molecular:799.97Pitolisant
CAS:<p>Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C17H26ClNOPureza:99.84%Forma y color:SolidPeso molecular:295.85Vildagliptin carboxylic acid methyl ester
CAS:<p>Please enquire for more information about Vildagliptin carboxylic acid methyl ester including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C18H28N2O4Pureza:Min. 95%Peso molecular:336.43 g/molPG-116800
CAS:<p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>Fórmula:C24H27N3O7SPureza:98.03% - 99.66%Forma y color:SolidPeso molecular:501.55Ecopipam
CAS:<p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>Fórmula:C19H20ClNOPureza:99.68%Forma y color:SolidPeso molecular:313.82Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Forma y color:SolidPeso molecular:381.44Dimethindene
CAS:<p>Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.</p>Fórmula:C20H24N2Pureza:98.3% - 98.99%Forma y color:SolidPeso molecular:292.42Ritodrine
CAS:<p>Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].</p>Fórmula:C17H21NO3Forma y color:SolidPeso molecular:287.35Pirtobrutinib
CAS:<p>Pirtobrutinib: a selective, non-covalent BTK inhibitor effective against BTK C481 mutations, causing tumor regression in lymphoma models.</p>Fórmula:C22H21F4N5O3Pureza:99.76% - 99.94%Forma y color:SolidPeso molecular:479.43(Rac)-Lonafarnib
CAS:<p>(Rac)-Lonafarnib is a racemic FTase inhibitor, effective against H-ras, K-ras, N-ras (IC50: 1.9, 5.2, 2.8 nM), and has anti-HDV properties.</p>Fórmula:C27H31Br2ClN4O2Forma y color:SolidPeso molecular:638.82MMP-7-IN-3
CAS:<p>MMP-7-IN-3 (compound 15) is a potent and selective MMP-7 inhibitor, inhibiting renal fibrosis in a unilateral ureteral obstruction mouse model.</p>Fórmula:C34H43ClF3N7O9SPureza:99.915%Forma y color:SolidPeso molecular:818.26XL-784
CAS:<p>XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.</p>Fórmula:C42H42Cl2F4MgN6O16S2Pureza:98%Forma y color:SolidPeso molecular:1122.15Frovatriptan
CAS:<p>Frovatriptan, potent 5-HT 1B/D agonist, shows high cerebroselectivity and efficacy for migraine with aura.</p>Fórmula:C14H17N3OForma y color:SolidPeso molecular:243.3Inz-1
CAS:<p>Inz-1 is an effective and fungal-selective inhibitor of mitochondrial cytochrome bc1 with IC50s of 8.092 and 45.320 μM for yeast and human.</p>Fórmula:C16H14N2O2Pureza:99.55% - 99.88%Forma y color:SolidPeso molecular:266.29Bufuralol (hydrochloride)
CAS:<p>Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.</p>Fórmula:C16H24ClNO2Forma y color:SolidPeso molecular:297.82Mefenidil
CAS:<p>Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.</p>Fórmula:C12H11N3Pureza:98.27%Forma y color:SolidPeso molecular:197.24MMP3 inhibitor 1
CAS:<p>MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).</p>Fórmula:C23H31N3O6SPureza:98%Forma y color:SolidPeso molecular:477.57Cipemastat
CAS:<p>Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).</p>Fórmula:C22H36N4O5Pureza:98%Forma y color:SolidPeso molecular:436.55Collagen proline hydroxylase inhibitor
CAS:<p>Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.</p>Fórmula:C18H18N4O4Pureza:98%Forma y color:SolidPeso molecular:354.36XL-784 free base
CAS:<p>XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).</p>Fórmula:C21H22ClF2N3O8SPureza:98%Forma y color:SolidPeso molecular:549.93Quizalofop
CAS:<p>Quizalofop (Xylafop) is a reagent of biochemical.</p>Fórmula:C17H13ClN2O4Pureza:97.14%Forma y color:SolidPeso molecular:344.75Celiprolol hydrochloride
CAS:<p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>Fórmula:C20H33N3O4·HClForma y color:White Crystalline SolidPeso molecular:415.96Cobimetinib racemate
CAS:<p>Cobimetinib racemate (Cobimetinib (racemate)) (GDC-0973 racemate) is a selective inhibitor of MEK.Cobimetinib racemate is also known as a mitogen-activated</p>Fórmula:C21H21F3IN3O2Pureza:98.00% - 99.71%Forma y color:SolidPeso molecular:531.31RU 58668
CAS:<p>Pure antiestrogen that downregulates estrogen receptor expression</p>Fórmula:C34H43F5O5SPureza:98%Forma y color:SolidPeso molecular:658.76Bufuralol
CAS:<p>Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.</p>Fórmula:C16H23NO2Pureza:98.26%Forma y color:SolidPeso molecular:261.36Zandelisib
CAS:<p>Zandelisib is an inhibitor of phosphatidylinositol 3-kinase (PI3K)(p110δ, IC50 of 3.5 nM), and with antineoplastic activity.</p>Fórmula:C31H38F2N8OPureza:99.88%Forma y color:SolidPeso molecular:576.68Tianagliflozin
CAS:<p>Tianagliflozin, a sodium/glucose cotransporter 2 (SGLT-2) inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Fórmula:C21H25ClO5Pureza:98%Forma y color:SolidPeso molecular:392.87Carmoxirole hydrochloride
CAS:<p>Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity in vivo.</p>Fórmula:C24H27ClN2O2Pureza:99.37% - 99.62%Forma y color:SolidPeso molecular:410.94Z-PDLDA-NHOH
CAS:<p>Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].</p>Fórmula:C22H32N4O6Forma y color:SolidPeso molecular:448.51MMP-7-IN-2
CAS:<p>MMP-7-IN-2 acts as a selective and potent MMP7 inhibitor and can be used to study inflammatory responses and vascular-related diseases.</p>Fórmula:C28H40ClF3N6O9SPureza:97.82%Forma y color:SolidPeso molecular:729.17ONO 4817
CAS:<p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>Fórmula:C22H28N2O6Forma y color:SolidPeso molecular:416.47Dibenamine hydrochloride
CAS:<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Fórmula:C16H19Cl2NPureza:96.43%Forma y color:Oily Liquid SolidPeso molecular:296.23Ubrogepant
CAS:<p>Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.</p>Fórmula:C29H26F3N5O3Pureza:99.452% - 99.78%Forma y color:SolidPeso molecular:549.54Ro 31-9790
CAS:<p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>Fórmula:C15H29N3O4Pureza:98%Forma y color:SolidPeso molecular:315.41ROCK2-IN-7
CAS:<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Fórmula:C26H28FN5OPureza:98%Forma y color:SolidPeso molecular:445.53Fluvalinate
CAS:<p>Fluvalinate is a synthetic chemical compound and can be commonly used to control varroa mites in honey bee colonies.</p>Fórmula:C26H22ClF3N2O3Forma y color:SolidPeso molecular:502.91Gisadenafil
CAS:<p>Gisadenafil (UK-369003) is a selective inhibitor of phosphodiesterase 5 (PDE5) with an IC50 of 3.6 nM and prevents degradation of cGMP.</p>Fórmula:C23H33N7O5SPureza:98.82% - 99.50%Forma y color:SolidPeso molecular:519.62KB-R7785
CAS:<p>KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.</p>Fórmula:C18H27N3O4Forma y color:SolidPeso molecular:349.42Dothiepin
CAS:<p>Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing</p>Fórmula:C19H21NSPureza:98%Forma y color:SolidPeso molecular:295.44Brilaroxazine
CAS:<p>Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.</p>Fórmula:C22H25Cl2N3O3Pureza:99.36%Forma y color:SolidPeso molecular:450.36PIM447
CAS:<p>PIM447 (LGH447) is a pan-PIM kinase inhibitor with anti-tumor and bone protective effects. PIM447 reduces the viability, and motility of HuH6 cell.</p>Fórmula:C24H23F3N4OPureza:98.97%Forma y color:SolidPeso molecular:440.46Caroverine
CAS:<p>Caroverine is a potential chemotherapeutical agent in HNSCC cell lines.</p>Fórmula:C22H27N3O2Forma y color:SolidPeso molecular:365.47Etidocaine Hydrochloride
CAS:<p>Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.</p>Fórmula:C17H29ClN2OPureza:99.86%Forma y color:SolidPeso molecular:312.88ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Fórmula:C23H26Cl2N2O4Forma y color:SolidPeso molecular:465.37ND-378
CAS:<p>ND-378 is a potent and selective inhibitor of MMP-2 with no inhibition on MMP-9 and MMP-14.</p>Fórmula:C18H19NO4S2Pureza:98%Forma y color:SolidPeso molecular:377.48Saredutant
CAS:<p>Saredutant (SR 48968) is a selective neurokinin-2 (NK2) receptor antagonist that inhibits neurokinin A by blocking NK2 receptor, antidepressant and anxiolytic.</p>Fórmula:C31H35Cl2N3O2Pureza:99.12%Forma y color:SolidPeso molecular:552.54
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