Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65615 productos de "Derivados de Quinazolina y Quinolina"
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Triflusal
CAS:<p>Triflusal (UR1501) is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative.</p>Fórmula:C10H7F3O4Pureza:99.61%Forma y color:SolidPeso molecular:248.16Ritonavir
CAS:<p>Ritonavir (ABT 538) inhibits HIV-1/2 proteases; serum proteins limit it but it enhances other HIV drugs by hindering P450 degradation.</p>Fórmula:C37H48N6O5S2Pureza:99.38% - 99.96%Forma y color:White PowderPeso molecular:720.94Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Fórmula:C12H19NO3H2SO4Pureza:99.47% - 99.94%Forma y color:Crystalline PowderPeso molecular:274.32Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Forma y color:SolidPeso molecular:408.33Levetiracetam
CAS:<p>Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset</p>Fórmula:C8H14N2O2Pureza:99.67% - 99.86%Forma y color:White Crystalline PowderPeso molecular:170.21Orbifloxacin
CAS:<p>Orbifloxacin (CP-104354) is a broad-spectrum fluoroquinolone antibiotic.</p>Fórmula:C19H20F3N3O3Pureza:99.46% - 99.58%Forma y color:SolidPeso molecular:395.38Pyrantel tartrate
CAS:<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Fórmula:C15H20N2O6SPureza:99.96%Forma y color:White CrystalsPeso molecular:356.39Gefitinib
CAS:<p>Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 Del and L858R mutations.</p>Fórmula:C22H24ClFN4O3Pureza:99.92% - >99.99%Forma y color:Light-Yellow Crystalline PowderPeso molecular:446.9Benzbromarone
CAS:<p>Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.</p>Fórmula:C17H12Br2O3Pureza:99.37% - 99.73%Forma y color:SolidPeso molecular:424.08Trelagliptin
CAS:<p>Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.</p>Fórmula:C18H20FN5O2Pureza:98.88%Forma y color:SolidPeso molecular:357.38(S)-(+)-Norepinephrine L-bitartrate
CAS:Fórmula:C12H17NO9Pureza:97%Forma y color:SolidPeso molecular:319.2647Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Fórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Gabapentin
CAS:<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Fórmula:C9H17NO2Pureza:99.55% - 99.91%Forma y color:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidPeso molecular:171.24Tenoxicam
CAS:<p>Tenoxicam (Tilcotil), an antiinflammatory agent with analgesic and antipyretic properties, is used to treat osteoarthritis and control acute pain.</p>Fórmula:C13H11N3O4S2Pureza:99.72% - 99.74%Forma y color:Yellow Crystalline PowderPeso molecular:337.37Mefloquine
CAS:<p>Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor.</p>Fórmula:C17H16F6N2OPureza:99.89%Forma y color:SolidPeso molecular:378.31Phenformin
CAS:<p>Phenformin: a biguanide with anti-cancer, anti-glycemic effects, inhibits skin tumors, enhances keratinocyte differentiation/apoptosis.</p>Fórmula:C10H15N5Pureza:99.72%Forma y color:SolidPeso molecular:205.26Pazopanib
CAS:<p>Pazopanib (GW786034) is an inhibitor of protein tyrosine kinases that inhibits VEGFR1/2/3. Pazopanib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C21H23N7O2SPureza:98.78% - 99.85%Forma y color:White PowderPeso molecular:437.52Enarodustat
CAS:<p>Enarodustat (JTZ-951) is an orally active factor inhibitor of prolyl hydroxylase (EC50: 0.22 μM) and has the potential for renal anemia treatment.</p>Fórmula:C17H16N4O4Pureza:99.73% - 99.75%Forma y color:SolidPeso molecular:340.33Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Fórmula:C21H26ClN3OSPureza:99.3% - 99.99%Forma y color:SolidPeso molecular:403.97Andecaliximab
CAS:<p>Andecaliximab: IgG4 antibody against MMP9, antifibrotic in mice, studies gastric cancer, IPF, dengue.</p>Pureza:> 95%Forma y color:LiquidPeso molecular:150 kDaZileuton
CAS:<p>Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.</p>Fórmula:C11H12N2O2SPureza:98.72% - 99.43%Forma y color:Crystalline SolidPeso molecular:236.29Lomustine
CAS:<p>Lomustine (NSC-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.</p>Fórmula:C9H16ClN3O2Pureza:98.36% - 99.44%Forma y color:Solid SolidPeso molecular:233.7Rofecoxib
CAS:<p>Rofecoxib (MK 966) binds to and inhibits the enzyme cyclooxygenase-2 (COX-2), resulting in an inhibition of the conversion of arachidonic acid to prostaglandins</p>Fórmula:C17H14O4SPureza:99.68% - 99.94%Forma y color:Off-White (Pale Yellow) Crystalline PowderPeso molecular:314.36Dantrolene sodium
CAS:<p>Dantrolene sodium treats spasticity by disrupting muscle contraction; not central in action, grouped with central relaxants.</p>Fórmula:C14H9N4NaO5Pureza:98% - 99.87%Forma y color:CoaPeso molecular:336.23Nisoldipine
CAS:<p>Nisoldipine (BAY-k 5552) is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.</p>Fórmula:C20H24N2O6Pureza:98.79% - 99.57%Forma y color:SolidPeso molecular:388.41STL127705
CAS:<p>STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.</p>Fórmula:C22H20FN5O4Pureza:99.53% - 99.81%Forma y color:SolidPeso molecular:437.42Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Fórmula:C23H23NO5SPureza:99.25% - 99.73%Forma y color:SolidPeso molecular:425.50Naproxen sodium
CAS:<p>Naproxen sodium (Anaprox) is a COX inhibitor for COX-1 and COX-2 with analgesic and antipyretic properties.</p>Fórmula:C14H13NaO3Pureza:99.68% - 99.79%Forma y color:White PowderPeso molecular:252.24Adenine
CAS:<p>Adenine: a purine nucleobase vital for ATP, NAD, FAD production, and DNA/RNA synthesis.</p>Fórmula:C5H5N5Pureza:99.39% - 99.95%Forma y color:SolidPeso molecular:135.13Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Fórmula:C10H16N6SPureza:99.82%Forma y color:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecular:252.34Praziquantel
CAS:<p>Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.</p>Fórmula:C19H24N2O2Pureza:99.67% - 99.69%Forma y color:SolidPeso molecular:312.41Chlormethiazole hydrochloride
CAS:<p>Chlormethiazole hydrochloride is an anticonvulsant and sedative. It also has neuroprotective.</p>Fórmula:C6H9Cl2NSPureza:99.93%Forma y color:SolidPeso molecular:198.11Medrysone
CAS:<p>Medrysone is a synthetic glucocorticoid for topical use with anti-inflammatory and anti-allergic effects, altering gene expression to reduce inflammation.</p>Fórmula:C22H32O3Pureza:97.72% - 99.91%Forma y color:SolidPeso molecular:344.49Menbutone
CAS:<p>Menbutone, a choleretic and oxobutyric acid derivative, peaks in plasma in 1hr, effects last ~10hrs.</p>Fórmula:C15H14O4Pureza:97.48%Forma y color:CoaPeso molecular:258.27Sunitinib
CAS:<p>Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).</p>Fórmula:C22H27FN4O2Pureza:98% - 99.67%Forma y color:Yellow SolidPeso molecular:398.47Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Fórmula:C28H32N2O7Pureza:99.03% - 99.67%Forma y color:SolidPeso molecular:508.56Dipyridamole
CAS:<p>Dipyridamole (Persantin) is a Platelet Aggregation Inhibitor. The physiologic effect of dipyridamole is by means of Decreased Platelet Aggregation.</p>Fórmula:C24H40N8O4Pureza:99.47% - 99.84%Forma y color:SolidPeso molecular:504.63Pranlukast
CAS:<p>Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.</p>Fórmula:C27H23N5O4Pureza:99.41%Forma y color:Off-White SolidPeso molecular:481.52,2-dichloro-N-[(1R,2R)-1,3-dihydroxy-1-(4-methanesulfonylphenyl)propan-2-yl]acetamide
CAS:Fórmula:C12H15Cl2NO5SPureza:98%Forma y color:SolidPeso molecular:356.2222Upamostat
CAS:<p>Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.</p>Fórmula:C32H47N5O6SPureza:99.41%Forma y color:SolidPeso molecular:629.81Procarbazine hydrochloride
CAS:<p>Procarbazine hydrochloride (NSC-77213 HCl) is the hydrochloride salt of a methylhydrazine derivative with antineoplastic and mutagenic activities.</p>Fórmula:C12H19N3O·HClPureza:96.99% - ≥98%Forma y color:(Ntp 1992)Peso molecular:257.76Famotidine
CAS:<p>Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.</p>Fórmula:C8H15N7O2S3Pureza:98.93% - 99.91%Forma y color:White To Off-White Crystalline PowderPeso molecular:337.45Vildagliptin
CAS:<p>Vildagliptin (LAF237), an oral DPP-4 inhibitor with hypoglycemic effects, is metabolized and excreted in urine.</p>Fórmula:C17H25N3O2Pureza:97.81% - >99.99%Forma y color:White Crystalline PowderPeso molecular:303.40Fenofibric acid
CAS:<p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>Fórmula:C17H15ClO4Pureza:99.36%Forma y color:White Or Almost White Crystalline PowderPeso molecular:318.75Sildenafil citrate
CAS:<p>Sildenafil citrate, a PDE5 inhibitor for erectile dysfunction and occasionally pulmonary hypertension.</p>Fórmula:C28H38N6O11SPureza:99.59% - 99.97%Forma y color:White SolidPeso molecular:666.70Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Fórmula:C11H18BrN5O3Pureza:99.84% - >99.99%Forma y color:CoaPeso molecular:348.2Dimenhydrinate
CAS:<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Forma y color:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Fórmula:C17H19ClN4OPureza:99.90%Forma y color:Off-White PowderPeso molecular:330.81Zinc pyrithione
CAS:<p>Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump.</p>Fórmula:C10H8N2O2S2ZnPureza:99.09% - 99.47%Forma y color:Off-White To Tan PowderPeso molecular:317.71Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Forma y color:Off-White SolidPeso molecular:406.86
![2,2-dichloro-N-[(1R,2R)-1,3-dihydroxy-1-(4-methanesulfonylphenyl)propan-2-yl]acetamide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FIN%2Fthumb-webp%2FDA00HY3Z.webp&w=3840&q=75)
