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Angiogenèse

Angiogenèse

Les inhibiteurs de l'angiogenèse sont des composés qui interfèrent avec la formation de nouveaux vaisseaux sanguins, un processus crucial dans la croissance et la métastase des cancers. En inhibant l'angiogenèse, ces composés peuvent restreindre l'apport sanguin aux tumeurs, ralentissant ou arrêtant leur croissance. Les inhibiteurs de l'angiogenèse sont essentiels dans la recherche sur le cancer et le développement thérapeutique, offrant des informations sur les mécanismes de progression tumorale et proposant des traitements potentiels pour le cancer et d'autres maladies liées à l'angiogenèse. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de l'angiogenèse de haute qualité pour soutenir vos recherches en oncologie et biologie vasculaire.

Sous-catégories appartenant à la catégorie "Angiogenèse"

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2387 produits trouvés pour "Angiogenèse"

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  • EGFR-IN-67

    CAS :
    EGFR-IN-67 (Compound 7d) is a potent inhibitor of EGFR with anticancer activity (IC 50 = 0.34 μM) [1].
    Formule :C18H17N3S
    Couleur et forme :Solid
    Masse moléculaire :307.41

    Ref: TM-T60729

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • RO9021

    CAS :
    RO9021 is an orally bioavailable, novel ATP-competitive SYK inhibitor (average IC50: 5.6 nM).
    Formule :C18H25N7O
    Degré de pureté :99.90%
    Couleur et forme :Solid
    Masse moléculaire :355.44

    Ref: TM-T16776

    1mg
    46,00€
    5mg
    92,00€
    10mg
    137,00€
    25mg
    222,00€
    50mg
    319,00€
    100mg
    432,00€
  • BPIQ-II (hydrochloride)

    CAS :
    BPIQ-II, a selective EGFR inhibitor with an IC50 of 8 pM, targets ATP sites and halts EGF signals inside cells.
    Formule :C15H11BrClN5
    Couleur et forme :Solid
    Masse moléculaire :376.64

    Ref: TM-T36783

    500µg
    298,00€
    5mg
    2.070,00€
  • INCB16562

    CAS :
    INCB16562: oral JAK1/2 inhibitor, halts IL-6/STAT3 in myeloma cells, boosts drug efficacy, stunts myeloma in mice.
    Formule :C19H11Cl2N5
    Couleur et forme :Solid
    Masse moléculaire :380.23

    Ref: TM-T68306

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PDGFRα/FLT3-ITD-IN-2

    CAS :
    PDGFRα/FLT3-ITD-IN-2 is a potent inhibitor of PDGFRα (IC50>20 μM) and FLT3 (IC50: 0.004 μM).
    Formule :C28H41N9O
    Couleur et forme :Solid
    Masse moléculaire :519.68

    Ref: TM-T63629

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FIIN-4

    CAS :
    FIIN-4 is a covalent inhibitor of FGFR and can be used in studies about metastatic breast cancer.
    Formule :C35H38N8O4
    Degré de pureté :99.99%
    Couleur et forme :Solid
    Masse moléculaire :634.73

    Ref: TM-T27319

    1mg
    187,00€
    5mg
    455,00€
    10mg
    620,00€
    25mg
    940,00€
    50mg
    1.264,00€
    100mg
    1.663,00€
    200mg
    2.252,00€
  • JAK-IN-20

    CAS :
    JAK-IN-20: potent oral JAK1,2,3 inhibitor with IC50s 7, 5, 14 nM respectively, good pharmacokinetics, anti-inflammatory in vivo.
    Formule :C28H30FN7O2
    Couleur et forme :Solid
    Masse moléculaire :515.58

    Ref: TM-T63581

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Nuvenzepine

    CAS :
    Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.
    Formule :C19H20N4O2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :336.39

    Ref: TM-T16362

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CHMFL-ABL-053

    CAS :
    CHMFL-ABL-053: potent, selective BCR-ABL/SRC/p38 inhibitor (IC50: 70/90/62 nM). Orally available, potential CML drug.
    Formule :C28H26F3N7O2
    Couleur et forme :Solid
    Masse moléculaire :549.55

    Ref: TM-T22067

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Peficitinib hydrochloride

    CAS :
    Peficitinib HCl (ASP015K) is an oral JAK inhibitor with IC50s: JAK1 (3.9 nM), JAK2 (5.0 nM), JAK3 (0.7 nM), Tyk2 (4.8 nM).
    Formule :C18H23ClN4O2
    Couleur et forme :Solid
    Masse moléculaire :362.86

    Ref: TM-T61365

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VEGFR-2-IN-30


    VEGFR-2-IN-30: VEGFR-2 inhibitor, IC50 66 nM; blocks PDGFR, EGFR & FGFR1; halts cancer cell cycle, induces apoptosis.
    Formule :C28H23ClN6O4S2
    Couleur et forme :Solid
    Masse moléculaire :607.1

    Ref: TM-T72890

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BTK inhibitor 10

    CAS :
    BTK inhibitor 10, an oral drug from patent WO2018145525, may treat rheumatoid arthritis.
    Formule :C25H23N5O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :441.48

    Ref: TM-T10627

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • pan-HER-IN-1

    CAS :
    Compound C5: Irreversible, oral pan-HER inhibitor with low IC50s for EGFR/HERs; induces apoptosis and has antitumor effects.
    Formule :C19H14BrN5O
    Couleur et forme :Solid
    Masse moléculaire :408.25

    Ref: TM-T62047

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JAK1-IN-4

    CAS :
    JAK1-IN-4 selectively blocks JAK1 (IC50 = 85 nM) over JAK2/JAK3 and halts STAT3 phosphorylation in NCI-H 1975 cells (IC50 = 227 nM).
    Formule :C26H32FN9O2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :521.59

    Ref: TM-T15606

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Multi-kinase-IN-3

    CAS :
    Multi-kinase-IN-3 (compound 2) is a potent inhibitor of angiokinase and inhibits VEGFR-2 (IC50: 58.3 nM) and PDGFRβ (IC50: 55 nM).
    Formule :C33H33N5O3
    Couleur et forme :Solid
    Masse moléculaire :547.65

    Ref: TM-T63870

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • YF-452

    CAS :
    YF-452 inhibits tumor growth through antiangiogenesis by suppressing VEGF receptor 2 signaling.
    Formule :C24H26BrN3O
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :452.39

    Ref: TM-T29173

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AAE871

    CAS :
    AAE871 is a type I FLT3 inhibitor.
    Formule :C24H34N8O2S
    Couleur et forme :Solid
    Masse moléculaire :498.64

    Ref: TM-T69497

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AG-13958 monohydrochloride

    CAS :
    AG-13958 monohydrochloride, a VEGFA inhibitor, may treat neovascular AMD to prevent rapid vision loss.
    Formule :C26H23ClFN7O
    Couleur et forme :Solid
    Masse moléculaire :503.96

    Ref: TM-T69452

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR/HER2-IN-9

    CAS :
    EGFR/HER2-IN-9, a compound inhibiting both EGFR and HER2, demonstrates potency with IC50 values of 3.2 nM for EGFR, 14 nM for HER2, and 8.3 nM against the EGFR
    Formule :C25H25ClFN5O4
    Couleur et forme :Solid
    Masse moléculaire :513.95

    Ref: TM-T72854

    25mg
    690,00€
    50mg
    895,00€
    100mg
    1.566,00€
  • KRC-108

    CAS :
    KRC-108 is a potent kinase inhibitor targeting Ron, Flt3, TrkA, and c-Met with strong anti-proliferative effects on various cancer cells.
    Formule :C20H20N6O
    Couleur et forme :Solid
    Masse moléculaire :360.41

    Ref: TM-T71382

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Ebselen oxide

    CAS :
    Ebselen oxide (EB-2) is a HER2 inhibitor with antibacterial and antifungal activity and has shown cytoprotective effects against HN2 in vitro.
    Formule :C13H9NO2Se
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :290.18

    Ref: TM-T27235

    1mg
    157,00€
    5mg
    672,00€
    10mg
    1.144,00€
    25mg
    2.565,00€
  • PDGFRα/FLT3-ITD-IN-1

    CAS :
    PDGFRα/FLT3-ITD-IN-1 are potent inhibitors of PDGFRα/FLT3, and their IC50 values are greater than 0.036 and 0.003 μM, respectively.
    Formule :C27H39N9O
    Couleur et forme :Solid
    Masse moléculaire :505.66

    Ref: TM-T63454

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • DPPY

    CAS :
    DPPY inhibits EGFR, BTK, JAK3 (IC50<10 nM), curbs B-cell lymphoma growth, and may be studied for IPF treatment.
    Formule :C25H26ClN7O3
    Couleur et forme :Solid
    Masse moléculaire :507.97

    Ref: TM-T63486

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FGFR4-IN-5

    CAS :
    FGFR4-IN-5: potent, selective FGFR4 inhibitor, IC50 6.5 nM, strong in vivo anti-tumor effect, for liver cancer research.
    Formule :C23H23Cl2N5O5
    Couleur et forme :Solid
    Masse moléculaire :520.37

    Ref: TM-T37425

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • c-ABL-IN-4

    CAS :
    c-ABL-IN-4 is a potent inhibitor of c-Abl.
    Formule :C18H11ClF3N3O3
    Couleur et forme :Solid
    Masse moléculaire :409.75

    Ref: TM-T62065

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BAY 2476568

    CAS :
    BAY 2476568 is a selective and potent EGFR inhibitor that acts on both wild-type EGFR (IC50 <0.2 nM) and mutant EGFR (IC50 <0.2 nM).
    Formule :C24H27FN4O4
    Couleur et forme :Solid
    Masse moléculaire :454.49

    Ref: TM-T62795

    25mg
    1.998,00€
    50mg
    2.602,00€
  • c-ABL-IN-3

    CAS :
    c-ABL-IN-3, from patent WO2021048567A1, is a potent c-Abl inhibitor for researching ALS, PD, and cancer.
    Formule :C17H11F3N4O3
    Couleur et forme :Solid
    Masse moléculaire :376.29

    Ref: TM-T61546

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • EGFR-IN-88

    CAS :
    EGFR-IN-88 (Compound 4i), an EGFR inhibitor with an IC50 of 87 nM, exhibits cytotoxic effects on A549 cells at an IC50 of 3.902 μM and can induce cell apoptosis
    Formule :C22H18Cl2N4O2S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :473.37

    Ref: TM-T79694

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • SMU-B

    CAS :
    SMU-B is a well-tolerated c-Met/ALK dual inhibitor.
    Formule :C26H25Cl2FN4O2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :515.41

    Ref: TM-T24809

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • J-1048

    CAS :
    J-1048, an activin receptor-like kinase 5 (ALK5) inhibitor, effectively suppresses TAA-induced liver fibrosis in mice through specific inhibition of the TGF-β/
    Formule :C23H17FN6S2
    Couleur et forme :Solid
    Masse moléculaire :460.55

    Ref: TM-T78790

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BTK-IN-23

    CAS :
    BTK-IN-23: BTK inhibitor, IC50=12.8 nM; also blocks BLX (35.6 nM), BMX (5.7 nM); better selectivity than Ibrutinib.
    Formule :C27H28N6O2
    Couleur et forme :Solid
    Masse moléculaire :468.55

    Ref: TM-T73276

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • RIPK2-IN-1

    CAS :
    RIPK2-IN-1 (compound 18f) is a potent inhibitor of RIPK2 (IC50: 51 nM) and also inhibits ALK2 (IC50: 5 nM).
    Formule :C23H27N5O3S
    Couleur et forme :Solid
    Masse moléculaire :453.56

    Ref: TM-T62783

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Flonoltinib

    CAS :
    Flonoltinib (JAK2/FLT3-IN-1) is an orally active and efficient JAK2/FLT3 inhibitor with anti-cancer properties.
    Formule :C25H34FN7O
    Degré de pureté :99.52%
    Couleur et forme :Solid
    Masse moléculaire :467.58

    Ref: TM-T11707

    1mg
    71,00€
    5mg
    112,00€
    1mL*10mM (DMSO)
    124,00€
    10mg
    175,00€
    25mg
    279,00€
    50mg
    460,00€
  • TRK II-IN-1

    CAS :
    TRK II-IN-1: potent type II TRK inhibitor; IC50s: TRKA (3.3 nM), TRKB (6.4 nM), TRKC (4.3 nM), TRKA G667C (9.4 nM); also targets FLT3, RET, VEGFR2.
    Formule :C29H31F3N8O
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :564.6

    Ref: TM-T73033

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Lavendustin C6

    CAS :
    Lavendustin C6 is a effective tyrosine kinase inhibitor.
    Formule :C20H25NO5
    Couleur et forme :Solid
    Masse moléculaire :359.42

    Ref: TM-T25644

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • HIV-IN-6

    CAS :
    HIV-IN-6, an anti-HIV agent, blocks replication by targeting SFKs like Hck involved with Nef protein.
    Formule :C20H16N4O3S
    Degré de pureté :97.78%
    Couleur et forme :Solid
    Masse moléculaire :392.43

    Ref: TM-T61793

    10mg
    46,00€
    25mg
    86,00€
    50mg
    124,00€
    100mg
    178,00€
    200mg
    250,00€
  • SJF620

    CAS :
    SJF620 is a potent degrader of PROTAC BTK(DC50 : 7.9 nM).
    Formule :C41H44N8O7
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :760.84

    Ref: TM-T13887

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Tyk2-IN-7

    CAS :
    Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).
    Formule :C18H15D3N6O3S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :401.46

    Ref: TM-T13235

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • UNC-CA359

    CAS :
    UNC-CA359: potent EGFR inhibitor, IC50=18 nM, strong anti-tumor effect, promising for chordoma.
    Formule :C18H14ClN3O2
    Couleur et forme :Solid
    Masse moléculaire :339.78

    Ref: TM-T61077

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MDK5466

    CAS :
    MDK5466 is an Flt3 inhibitor that acts by preventing glutamate-induced cell death.
    Formule :C21H23N3OS
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :365.49

    Ref: TM-T24438

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Nazartinib mesylate

    CAS :
    Nazartinib mesylate is a novel, covalent mutant-selective inhibitor of EGFR (Ki and Kinact: 31 nM and 0.222/min on EGFR(L858R/790M) mutant).
    Formule :C27H35ClN6O5S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :591.12

    Ref: TM-T11156L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • NSC 33994

    CAS :
    NSC 33994 is a selective inhibitor of JAK2 (IC50 = 60 nM). It also shows no effect on Src and TYK2 tyrosine kinase activity at a concentration of 25 μM.
    Formule :C28H42N2O2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :438.65

    Ref: TM-T23091

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JAK3/BTK-IN-6

    CAS :
    JAK3/BTK-IN-6: potent BTK (0.6 nM) & JAK3 (0.4 nM) inhibitor, stable in human liver, for blood/immune research.
    Formule :C21H17BF3N5O3
    Couleur et forme :Solid
    Masse moléculaire :455.2

    Ref: TM-T62813

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-21

    CAS :
    EGFR-IN-21, a potent EGFR inhibitor, exhibits an IC50 of 0.38 nM, demonstrating significant antitumor activity.
    Formule :C36H44BrN10O2P
    Couleur et forme :Solid
    Masse moléculaire :759.68

    Ref: TM-T73103

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • EGFR/CDK2-IN-1

    CAS :
    EGFR/CDK2-IN-1, an inhibitor of both EGFR and CDK2, demonstrates effective cytotoxicity towards MCF7 and HepG2 cells, suggesting its potential application in
    Formule :C19H12BrClO2
    Couleur et forme :Solid
    Masse moléculaire :387.65

    Ref: TM-T72844

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BCR-ABL-IN-6

    CAS :
    BCR-ABL-IN-6, an imatinib derivative, inhibits Bcr-AblWT (4.6 nM IC50) and T315I (277 nM), for chronic myeloid leukemia study.
    Formule :C27H22F3N5O2
    Couleur et forme :Solid
    Masse moléculaire :505.49

    Ref: TM-T63450

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VS 8

    CAS :
    VS 8: potent oral VEGFR-2 inhibitor, anti-angiogenic, induces cancer cell apoptosis & migration, acts on CSCs.
    Formule :C26H20F3N3O3
    Couleur et forme :Solid
    Masse moléculaire :479.45

    Ref: TM-T63147

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR/HER2-IN-2

    CAS :
    EGFR/HER2-IN-2 (Compound ZINC35560729) is a dual EGFR and HER2 inhibitor that acts on both EGFR (IC50: 5.02 μM) and HER2 (IC50: 0.83 μM).
    Formule :C26H23N5O3
    Couleur et forme :Solid
    Masse moléculaire :453.49

    Ref: TM-T62776

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PP2 Analog

    CAS :
    PP2 Analog is an analog of PP2. It also acts as a protein trafficking modulator.
    Formule :C16H17ClN4
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :300.79

    Ref: TM-T6266L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Ficonalkib

    CAS :
    Ficonalkib is a potent antineoplastic agent that inhibits the Anaplastic Lymphoma Kinase (ALK) tyrosine kinase receptor.
    Formule :C29H39N7O3S
    Couleur et forme :Solid
    Masse moléculaire :565.73

    Ref: TM-T73189

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-46

    CAS :
    EGFR-IN-46: Potent EGFR/FAK inhibitor (IC50: 20.17 & 14.25 nM), curbs cancer cell growth, triggers apoptosis.
    Formule :C27H32F3N3O3
    Couleur et forme :Solid
    Masse moléculaire :503.56

    Ref: TM-T63431

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JBJ-09-063 hydrochloride


    JBJ-09-063 hydrochloride: targeted EGFR inhibitor, effective for various mutations and TKI-resistant lung cancer models.
    Formule :C31H30ClFN4O3S
    Couleur et forme :Solid
    Masse moléculaire :593.11

    Ref: TM-T72237

    25mg
    1.179,00€
    50mg
    1.539,00€
    100mg
    2.250,00€
  • EGFR-IN-25

    CAS :
    EGFR-IN-25, an efficacious EGFR inhibitor, demonstrates IC50 values of 9 nM for BaF3 cells (EGFR DEL19/T790M/C797S) and 60 nM for A431 cells (WT), respectively.
    Formule :C34H43N9O2
    Couleur et forme :Solid
    Masse moléculaire :609.76

    Ref: TM-T73101

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CP-690550A

    CAS :
    Cp-690550a is a novel JAK3 inhibitor, which is used to treat rheumatoid arthritis, graft rejection, psoriasis, and other immune-mediated diseases.
    Formule :C15H21N5O2
    Couleur et forme :Solid
    Masse moléculaire :303.36

    Ref: TM-T31074

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-54

    CAS :
    EGFR-IN-54 (Compound 3c) is a potent inhibitor of EGFR (IC50: 1.623 μM) and is toxic to cancer cells.
    Formule :C17H14N4O4S3
    Couleur et forme :Solid
    Masse moléculaire :434.51

    Ref: TM-T62457

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • NSC114792

    CAS :
    NSC114792 is a selective JAK3 inhibitor.
    Formule :C26H32N4O2S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :464.62

    Ref: TM-T24549

    25mg
    1.369,00€
  • EGFR-IN-55

    CAS :
    "EGFR-IN-55 targets EGFRWT (70 nM IC50) & EGFRL858R/T790M (3.9 nM IC50), halts NCI-H1975 cell cycle in G0/G1, showing anticancer properties."
    Formule :C25H25Cl2N7O2
    Couleur et forme :Solid
    Masse moléculaire :526.42

    Ref: TM-T63693

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PD-173956

    CAS :
    PD-173956 is an inhibitor of the Src family tyrosine kinases.
    Formule :C20H13Cl2FN4O
    Couleur et forme :Solid
    Masse moléculaire :415.25

    Ref: TM-T28345

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-52

    CAS :
    EGFR-IN-52, a potent EGFR inhibitor, has IC50s: 0.358 μM (wild-type), 86.02 μM (L858R-TK), 432.67 μM (T790M-TK); induces cancer cell apoptosis.
    Formule :C19H18N4O3S
    Couleur et forme :Solid
    Masse moléculaire :382.44

    Ref: TM-T61646

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • XST-14

    CAS :
    XST-14 is a ULK1 inhibitor.XST-14 induces apoptosis and inhibits the growth of HCC cells.
    Formule :C16H21NO4
    Degré de pureté :99.84% - 99.84%
    Couleur et forme :Solid
    Masse moléculaire :291.34

    Ref: TM-T60604

    1mg
    52,00€
    5mg
    111,00€
    1mL*10mM (DMSO)
    124,00€
    10mg
    169,00€
    25mg
    295,00€
    50mg
    447,00€
  • EGFR/HER2/CDK9-IN-3

    CAS :
    EGFR/HER2/CDK9-IN-3 inhibits EGFR (191.08 nM IC50), HER2 (132.65 nM), CDK9 (113.98 nM); shows anti-tumor effects.
    Formule :C24H21N3O4S2
    Couleur et forme :Solid
    Masse moléculaire :479.57

    Ref: TM-T63161

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • SUN13837

    CAS :
    SUN13837, an oral FGFR modulator, crosses the BBB and shows neuroprotective promise.
    Formule :C21H29N5O2
    Couleur et forme :Solid
    Masse moléculaire :383.49

    Ref: TM-T61666

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Erbstatin

    CAS :
    Erbstatin is a tyrosine-protein kinase inhibitor. When combined with foroxymithine, it has antineoplastic activity against L-1210 leukemia.
    Formule :C9H9NO3
    Couleur et forme :Solid
    Masse moléculaire :179.17

    Ref: TM-T24039

    1mg
    1.108,00€
  • TYK2-IN-11

    CAS :
    TYK2-IN-11 (5B) selectively inhibits TYK2 (IC50: 0.016 nM) and JAK1 (IC50: 0.31 nM), aiding autoimmune and inflammatory disease research.
    Formule :C18H17N5O3S
    Couleur et forme :Solid
    Masse moléculaire :383.42

    Ref: TM-T61658

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR/HER2-IN-3

    CAS :
    EGFR/HER2-IN-3 (Compound ZINC21942954) is a dual EGFR and HER2 inhibitor.
    Formule :C26H23N5O3
    Couleur et forme :Solid
    Masse moléculaire :453.49

    Ref: TM-T62777

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FLT3-IN-18

    CAS :
    FLT3-IN-18: potent, selective FLT3 inhibitor, IC50 0.003 μM, induces apoptosis, G1 arrest, blocks FLT3/STAT5, potential in AML research.
    Formule :C26H36N8O
    Couleur et forme :Solid
    Masse moléculaire :476.62

    Ref: TM-T73142

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • (R)-Elsubrutinib

    CAS :
    (R)-Elsubrutinib ((R)-ABBV-105) is a Btk inhibitor and an isomer of Elsubrutinib, suitable for inflammation research.
    Formule :C17H19N3O2
    Degré de pureté :99.05%
    Couleur et forme :Solid
    Masse moléculaire :297.35

    Ref: TM-T72653

    1mg
    145,00€
    5mg
    250,00€
    10mg
    340,00€
    1mL*10mM (DMSO)
    462,00€
    25mg
    573,00€
    50mg
    879,00€
    100mg
    1.314,00€
  • EGFR-IN-69

    CAS :
    EGFR-IN-69: Potent EGFR inhibitor for NSCLC research; IC50: 4.3-25.6 nM against various EGFR mutations.
    Formule :C31H37Cl2N7O3S
    Couleur et forme :Solid
    Masse moléculaire :658.64

    Ref: TM-T73153

    25mg
    858,00€
    50mg
    1.116,00€
    100mg
    1.791,00€
  • TIE-2/VEGFR-2 kinase-IN-1

    CAS :
    TIE-2/VEGFR-2 kinase-IN-1 synthesizes inhibitors for angiogenesis-related disease research.
    Formule :C13H11N3O2
    Couleur et forme :Solid
    Masse moléculaire :241.25

    Ref: TM-T8817

    25mg
    1.215,00€
    50mg
    1.584,00€
    100mg
    2.412,00€
  • VEGFR2 Kinase Inhibitor II

    CAS :
    VEGFR2 kinase inhibitor II: Reversible, cell-permeable, targets VEGFR2 (IC50=70nM), less effective on PDGFRβ (IC50=920nM). Blocks VEGF/PDGF-stimulated growth.
    Formule :C17H15BrN2O
    Couleur et forme :Solid
    Masse moléculaire :343.22

    Ref: TM-T37079

    500µg
    268,00€
    1mg
    515,00€
  • EGFR-IN-49

    CAS :
    EGFR-IN-49 selectively inhibits EGFR mutations T790M (IC50: 65 nM) & T790M/L858R (IC50: 13.6 nM), triggering apoptosis dose-dependently.
    Formule :C22H15N5O2S
    Couleur et forme :Solid
    Masse moléculaire :413.45

    Ref: TM-T62113

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BLK-IN-1

    CAS :
    BLK-IN-1 selectively blocks BLK and BTK with IC50s of 18.8 and 20.5 nM, used in cancer research.
    Formule :C29H23F3N6O3
    Couleur et forme :Solid
    Masse moléculaire :560.53

    Ref: TM-T63959

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CPL304110

    CAS :
    CPL304110: oral, selective FGFR 1-3 inhibitor; IC50 - FGFR1: 0.75nM, FGFR2: 0.5nM, FGFR3: 3.05nM.
    Formule :C25H30N6O2
    Couleur et forme :Solid
    Masse moléculaire :446.54

    Ref: TM-T62652

    25mg
    690,00€
    50mg
    897,00€
    100mg
    1.476,00€
  • PHM16

    CAS :
    PHM16 is an ATP competitive FAK and FGFR2 inhibitor.
    Formule :C20H22N6O4
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :410.43

    Ref: TM-T24634

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-31

    CAS :
    EGFR-IN-31: Potent EGFR inhibitor, targets mutations & overexpression in NSCLC; potential cancer research compound. (WO2021185298A1, 2)
    Formule :C32H36FN7O2
    Couleur et forme :Solid
    Masse moléculaire :569.67

    Ref: TM-T64030

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FLT3/D835Y-IN-1

    CAS :
    FLT3/D835Y-IN-1, an oral FLT3 inhibitor (IC50: FLT3 - 0.26 nM, D835Y - 0.18 nM), shows anticancer potential in AML research.
    Formule :C22H21N5O3
    Couleur et forme :Solid
    Masse moléculaire :403.43

    Ref: TM-T61977

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • EGFR-IN-57

    CAS :
    EGFR-IN-57: potent EGFR-TK blocker, IC50 0.054 μM, oral. Halts VEGFR-2, CK2α, topo IIβ, tubulin. Causes G2/M, pre-G1 arrest, cancer cell death.
    Formule :C22H15N3O2S
    Couleur et forme :Solid
    Masse moléculaire :385.44

    Ref: TM-T61696

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JAK3-IN-1

    CAS :
    JAK3-IN-1 is an orally active, selective and potent JAK3 inhibitor for the study of immune system disorders.
    Formule :C26H30ClN7O2
    Couleur et forme :Solid
    Masse moléculaire :508.02

    Ref: TM-T15607

    5mg
    205,00€
    25mg
    690,00€
    50mg
    897,00€
    100mg
    1.251,00€
  • FGFR3-IN-1

    CAS :
    FGFR3-IN-1 (compound 1) is a fibroblast growth factor receptor (FGFR) inhibitor that inhibits FGFR1 (IC50: 40 nM), FGFR2 (IC50: 5.1 nM) and FGFR3 (IC50: 12 nM).
    Formule :C28H39N9O3S
    Couleur et forme :Solid
    Masse moléculaire :581.73

    Ref: TM-T64107

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • TRK/ALK-IN-1


    TRK/ALK-IN-1: Potent dual TRK & ALK inhibitor; IC50s: 2.2nM (TRKA), 9.3nM (ALK WT), 38nM (ALK L1196M); cancer research potential.
    Formule :C31H35ClF2N8O2S
    Couleur et forme :Solid
    Masse moléculaire :657.18

    Ref: TM-T72931

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • EGFR-IN-60

    CAS :
    EGFR-IN-60: oral anticancer drug, inhibits EGFR/JAK3, effective on H1975/A431 cells, promotes apoptosis.
    Formule :C28H28Cl2N6O
    Couleur et forme :Solid
    Masse moléculaire :535.47

    Ref: TM-T63769

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • ProMMP-9 inhibitor-3c

    CAS :
    ProMMP-9 inhibitor-3c hinders MMP-9 homodimers, blocks proMMP-9/α4β1 integrin/CD44 binding, and detaches EGFR.
    Formule :C18H20FN3O2S
    Couleur et forme :Solid
    Masse moléculaire :361.43

    Ref: TM-T69875

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BTK-IN-9

    CAS :
    BTK-IN-9 reversibly inhibits BTK, disrupts mitochondria, boosts ROS, and triggers apoptosis in Z138 cells, impeding condyloma cell growth.
    Formule :C25H19N7O4
    Couleur et forme :Solid
    Masse moléculaire :481.46

    Ref: TM-T63179

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • ZT55

    CAS :
    ZT55: Oral JAK2 inhibitor, IC50: 0.031 μM, hinders JAK2 V617F HEL cell growth, induces apoptosis, arrests cell cycle, effective in mice HEL tumor studies.
    Formule :C17H16N2O3
    Couleur et forme :Solid
    Masse moléculaire :296.32

    Ref: TM-T73567

    25mg
    642,00€
    50mg
    1.026,00€
    100mg
    1.648,00€
  • VEGFR-2-IN-24

    CAS :
    VEGFR-2-IN-24 is a potent inhibitor of VEGFR-2 (IC50: 0.22 μM) and can be used to study tumors.
    Formule :C28H23N3O6S
    Couleur et forme :Solid
    Masse moléculaire :529.56

    Ref: TM-T63722

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FGFR4-IN-11

    CAS :
    FGFR4-IN-11: selective, covalent FGFR4 inhibitor; IC50=2.1 nM; blocks FGF19 pathway; anticancer.
    Formule :C29H29N5O5
    Couleur et forme :Solid
    Masse moléculaire :527.57

    Ref: TM-T63704

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • c-Met-IN-14

    CAS :
    c-Met-IN-14: selective c-Met kinase inhibitor, IC50 2.89 nM, anticancer, stops G2/M phase, induces A549 cell apoptosis.
    Formule :C34H38ClFN4O7S
    Couleur et forme :Solid
    Masse moléculaire :701.2

    Ref: TM-T73022

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BI-1622

    CAS :
    BI-1622, an oral HER2 inhibitor, IC50: 7 nM, >25x selectivity over EGFR, shows effective in vivo antitumor activity.
    Formule :C26H24N10O2
    Couleur et forme :Solid
    Masse moléculaire :508.53

    Ref: TM-T63492

    25mg
    1.260,00€
    50mg
    1.639,00€
    100mg
    2.250,00€
  • EGFR-IN-26

    CAS :
    EGFR-IN-26 is an EGFR inhibitor that can be used in cancer research.
    Formule :C29H34N6O3
    Couleur et forme :Solid
    Masse moléculaire :514.62

    Ref: TM-T63571

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • ON 146040

    CAS :
    ON 146040 is an effective inhibitor of PI3K isoforms with IC50s of 14 and 20 nM for PI3Kα and PI3Kδ, respectively.
    Formule :C24H23N7O3S
    Degré de pureté :97.39%
    Couleur et forme :Solid
    Masse moléculaire :489.55

    Ref: TM-T12310

    1mg
    46,00€
    5mg
    96,00€
    1mL*10mM (DMSO)
    104,00€
    10mg
    156,00€
    25mg
    245,00€
    50mg
    344,00€
    100mg
    460,00€
    200mg
    622,00€
  • Antiproliferative agent-20

    CAS :
    Antiproliferative agent-20: potent oral anticancer drug with anti-angiogenic properties.
    Formule :C23H18N2O6
    Couleur et forme :Solid
    Masse moléculaire :418.4

    Ref: TM-T72191

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Ansornitinib

    CAS :
    Ansornitinib (ANG-3070) is a KDR and PDGF receptor inhibitor with antifibrotic activity for the study of diseases caused by abnormal or excessive fibrosis.
    Formule :C30H32N6O4
    Degré de pureté :99.24%
    Couleur et forme :Solid
    Masse moléculaire :540.61

    Ref: TM-T63809

    1mg
    124,00€
    5mg
    286,00€
    10mg
    447,00€
    25mg
    964,00€
    50mg
    1.521,00€
    100mg
    2.250,00€
  • Atrinositol

    CAS :
    Atrinositol improves energy homeostasis in a mouse model of pancreatic cancer.
    Formule :C6H15O15P3
    Couleur et forme :Solid
    Masse moléculaire :420.1

    Ref: TM-T30203

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AFG206

    CAS :
    AFG206 is the novel first-generation type II" FLT3 inhibitor."
    Formule :C20H19N3O2
    Couleur et forme :Solid
    Masse moléculaire :333.38

    Ref: TM-T68967

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • ALK-IN-22

    CAS :
    ALK-IN-22 suppresses ALK and mutants (IC50: 2.3-3.7 nM), hinders phosphorylation, and induces apoptosis in tumor studies.
    Formule :C24H24ClN7O2
    Couleur et forme :Solid
    Masse moléculaire :477.95

    Ref: TM-T63130

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • CHMFL-ABL/KIT-155

    CAS :
    CHMFL-ABL/KIT-155 is a highly potent and orally active type II ABL/c-KIT dual kinase inhibitor (IC50s: 46 nM/75 nM).
    Formule :C33H38F3N5O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :609.68

    Ref: TM-T10801

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • AC710

    CAS :
    AC710 is a potent PDGFR inhibitor (Kds: 0.6, 1, 1.57, 1.3, 1 nM for FLT3, KIT, CSF1R, PDGFRα and PDGFRβ).
    Formule :C31H42N6O4
    Degré de pureté :99.67%
    Couleur et forme :Solid
    Masse moléculaire :562.7

    Ref: TM-TQ0235

    5mg
    43,00€
    1mL*10mM (DMSO)
    49,00€
    10mg
    62,00€
    25mg
    111,00€
    50mg
    166,00€
  • CAY10583

    CAS :
    CAY10583 is a selective BLT2 agonist that increases TGF-β1 and bFGF, promotes keratinocyte migration, accelerates wound healing in diabetic mice.
    Formule :C25H25NO3
    Degré de pureté :>99.99% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :387.47

    Ref: TM-T26958

    1mg
    50,00€
    2mg
    79,00€
    5mg
    207,00€
  • EGFR-IN-51

    CAS :
    EGFR-IN-51 effectively inhibits EGFR and mutations with IC50s of 0.493-461.63 μM; it induces apoptosis in cancer cells.
    Formule :C21H15N3O2S
    Couleur et forme :Solid
    Masse moléculaire :373.43

    Ref: TM-T61513

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JAK-IN-30

    CAS :
    JAK-IN-30 (compound 31) is a water-soluble inhibitor of Janus kinases (JAKs), demonstrating inhibitory potency with half-maximal inhibitory concentration (IC50
    Formule :C19H26N8S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :398.53

    Ref: TM-T79235

    1mg
    166,00€
    5mg
    627,00€
    10mg
    1.134,00€