Récepteur d'œstrogène/progestatif
Les récepteurs des œstrogènes et des progestogènes sont des récepteurs hormonaux nucléaires qui médiatisent les effets des œstrogènes et de la progestérone, respectivement. Ces récepteurs régulent divers processus physiologiques, notamment la fonction reproductrice, la densité osseuse et la santé cardiovasculaire. Les modulateurs des récepteurs des œstrogènes et des progestogènes sont largement étudiés pour leurs rôles dans le traitement hormonal substitutif, la contraception et le traitement des cancers sensibles aux hormones. Chez CymitQuimica, nous offrons une gamme complète de modulateurs de récepteurs des œstrogènes et des progestogènes de haute qualité pour soutenir vos recherches en endocrinologie, santé reproductive et biologie du cancer.
64 produits trouvés pour "Récepteur d'œstrogène/progestatif"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
(R)-Equol
CAS :(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.Formule :C15H14O3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :242.274,4'-Iminodiphenol
CAS :4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.Formule :C12H11NO2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :201.22Promestriene
CAS :Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation.Formule :C22H32O2Degré de pureté :99.35%Couleur et forme :White SolidMasse moléculaire :328.49Ethynodiol diacetate
CAS :Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with estrogens as an oral contraceptive.Formule :C24H32O4Degré de pureté :99.48% - 99.54%Couleur et forme :SolidMasse moléculaire :384.51Toremifene
CAS :Toremifene (GTx 006) is a selective estrogen-receptor modulator (SERM).Formule :C26H28ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White-To-Off-White SolidMasse moléculaire :405.96Gestrinone
CAS :Gestrinone (R 2323) 是一种合成类固醇激素，能够抑制平滑肌瘤(IC50:43.67 μM)，有用于子宫内膜异位症的研究潜力。Formule :C21H24O2Degré de pureté :99.21%Couleur et forme :Light Yellow SolidMasse moléculaire :308.41SLU-PP-332
CAS :SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,Formule :C18H14N2O2Degré de pureté :97.53% - 98.60%Couleur et forme :SoildMasse moléculaire :290.32Clomiphene citrate
CAS :Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.Formule :C32H36ClNO8Degré de pureté :98.67% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :598.1Dienestrol
CAS :Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist.Formule :C18H18O2Degré de pureté :96.73% - 98%Couleur et forme :Minute Needles From Dilute Alc SolidMasse moléculaire :266.33Giredestrant
CAS :Giredestrant (GDC-9545) is a potent oral anti-tumor ER antagonist competing with estradiol.Formule :C27H31F5N4ODegré de pureté :98.96% - 99.56%Couleur et forme :SolidMasse moléculaire :522.55Ref: TM-T11399
1mg105,00€5mg212,00€10mg334,00€25mg643,00€50mg1.018,00€100mg1.611,00€1mL*10mM (DMSO)245,00€Quinestrol
CAS :Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer andFormule :C25H32O2Degré de pureté :99.36% - 99.72%Couleur et forme :SolidMasse moléculaire :364.52Elacestrant
CAS :Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is an orally available selective estrogen receptor degrader .Formule :C30H38N2O2Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :458.63Ref: TM-T13674
1mg124,00€5mg235,00€10mg376,00€25mg645,00€50mg913,00€100mg1.216,00€1mL*10mM (DMSO)235,00€Gestodene
CAS :Gestodene (WL 70) is a progestogen hormonal contraceptive.Formule :C21H26O2Degré de pureté :98% - 99.68%Couleur et forme :White Crystalline SolidMasse moléculaire :310.43Mestranol
CAS :Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.Formule :C21H26O2Degré de pureté :99.16%Couleur et forme :Crystals From Methanol Or Acetone SolidMasse moléculaire :310.43Ethisterone
CAS :Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.Formule :C21H28O2Degré de pureté :97.96% - 99.50%Couleur et forme :Off-White PowderMasse moléculaire :312.45Panomifene TFA
Panomifene TFA（GYKl13504 TFA） is a antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases.Formule :C27H25F6NO4Degré de pureté :99.74%Couleur et forme :SoildMasse moléculaire :541.48Altrenogest
CAS :Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.Formule :C21H26O2Degré de pureté :98.98% - 99.66%Couleur et forme :Slightly Yellow PowderMasse moléculaire :310.43Methylpiperidino pyrazole
CAS :Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.Formule :C29H31N3O3Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :469.57AC-186
CAS :AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.
Formule :C18H17F3ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :306.32Endoxifen Z-isomer hydrochloride
CAS :Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.Formule :C25H28ClNO2Couleur et forme :SolidMasse moléculaire :409.95Bazedoxifene
CAS :Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.Formule :C30H34N2O3Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :470.61Nestoron
CAS :Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).Formule :C23H30O4Degré de pureté :99.83% - 99.92%Couleur et forme :SolidMasse moléculaire :370.48Ulipristal
CAS :Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.Formule :C28H35NO3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :433.584-Hydroxytamoxifen
CAS :4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.Formule :C26H29NO2Degré de pureté :99.37% - 99.93%Couleur et forme :SolidMasse moléculaire :387.51Elacestrant dihydrochloride
CAS :Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM forFormule :C30H40Cl2N2O2Degré de pureté :99.59% - 99.99%Couleur et forme :SolidMasse moléculaire :531.56Ref: TM-T13675
1mg113,00€5mg225,00€10mg356,00€25mg598,00€50mg852,00€100mg1.153,00€1mL*10mM (DMSO)264,00€Medroxyprogesterone
CAS :Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.Formule :C22H32O3Degré de pureté :99.18% - 99.51%Couleur et forme :Crystals From Chloroform SolidMasse moléculaire :344.49Desogestrel
CAS :Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
Formule :C22H30ODegré de pureté :99.8%Couleur et forme :Crystals SolidMasse moléculaire :310.47Ferrous Bisglycinate
CAS :Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.Formule :C4H8FeN2O4Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :203.96Norgestrel
CAS :Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.
Formule :C21H28O2Degré de pureté :99.71% - 99.72%Couleur et forme :Crystals From Methanol White Crystalline PowderMasse moléculaire :312.45GSK5182
CAS :GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)Formule :C27H31NO3Degré de pureté :97.63% - 99.42%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T8370
1mg52,00€2mg74,00€5mg96,00€10mg153,00€25mg274,00€50mg416,00€100mg615,00€1mL*10mM (DMSO)114,00€SNG-1153
CAS :SNG-1153 is a estrogen receptor ER-alpha36 modulator.Formule :C21H17F3O5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :406.35Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS :Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.
Formule :C18H18O3Degré de pureté :99.85% - 99.96%Couleur et forme :SolidMasse moléculaire :282.33Estradiol dipropionate
CAS :Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.Formule :C24H32O4Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :384.51WAY-200070
CAS :WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).Formule :C13H8BrNO3Degré de pureté :99.45% - 99.75%Couleur et forme :SolidMasse moléculaire :306.11Ref: TM-T3958
2mg42,00€5mg62,00€10mg96,00€25mg188,00€50mg311,00€100mg502,00€200mg715,00€1mL*10mM (DMSO)67,00€PROTAC ERRα ligand 2
CAS :PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)Formule :C20H13F6NO4Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :445.31Ref: TM-T5835
1mg43,00€5mg96,00€10mg116,00€25mg198,00€50mg299,00€100mg449,00€200mg627,00€1mL*10mM (DMSO)96,00€DY131
CAS :DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.Formule :C18H21N3O2Degré de pureté :98.65% - 99.66%Couleur et forme :SolidMasse moléculaire :311.38STF-62247
CAS :STF-62247 is TGN inhibitor with IC50 of 0.625 μM and 16 μM in RCC4 and RCC4/VHL cells, respectively.
Formule :C15H13N3SDegré de pureté :99.6% - 99.67%Couleur et forme :SolidMasse moléculaire :267.35Brilanestrant
CAS :Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).Formule :C26H20ClFN2O2Degré de pureté :99.07% - 99.17%Couleur et forme :Solid PowderMasse moléculaire :446.9Ref: TM-T5118
1mg50,00€2mg73,00€5mg101,00€10mg142,00€25mg245,00€50mg405,00€100mg582,00€1mL*10mM (DMSO)120,00€FLTX1
CAS :FLTX1, a Tamoxifen derivative, fluoresces to mark estrogen receptors and acts as a strong antiestrogen in breast cancer without affecting the uterus.Formule :C31H28N4O4Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :520.58Ref: TM-T8984
1mg55,00€5mg119,00€10mg182,00€25mg313,00€50mg442,00€100mg627,00€200mg845,00€1mL*10mM (DMSO)137,00€Hexestrol
CAS :Hexestrol (Hexanoestrol) binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.Formule :C18H22O2Degré de pureté :98.93% - 99.2%Couleur et forme :Needles From Benzene Thin Plates From Dil Alc Crystalline SolidMasse moléculaire :270.37Propyl pyrazole triol
CAS :PPT is a selective ERα agonist with 410x higher affinity than for ERβ.Formule :C24H22N2O3Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :386.44Ref: TM-T16566
1mg43,00€5mg93,00€10mg133,00€25mg250,00€50mg378,00€100mg570,00€200mg800,00€1mL*10mM (DMSO)90,00€Bazedoxifene acetate
CAS :Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).Formule :C32H38N2O5Degré de pureté :99.24% - 99.97%Couleur et forme :SolidMasse moléculaire :530.67Ref: TM-T2544
5mg44,00€10mg57,00€25mg86,00€50mg105,00€100mg152,00€200mg219,00€500mg358,00€1200mg618,00€1mL*10mM (DMSO)50,00€AZD9496
CAS :AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.Formule :C25H25F3N2O2Degré de pureté :97.28% - 98.47%Couleur et forme :SolidMasse moléculaire :442.47Ref: TM-T3975
1mg52,00€2mg73,00€5mg110,00€10mg178,00€25mg334,00€50mg494,00€100mg712,00€1mL*10mM (DMSO)105,00€SR 19881
CAS :SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).Formule :C19H24N2O2Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :312.41Ref: TM-T7904
1mg97,00€2mg149,00€5mg202,00€10mg324,00€25mg548,00€50mg785,00€100mg1.074,00€1mL*10mM (DMSO)220,00€Serba-2
CAS :Serba-2 is an agonist of benzopyran selective estrogen receptor beta.Formule :C18H18O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :282.33Fulvestrant-d3
Fulvestrant-d3 is a isotope labeled compound of Fulvestrant.an estrogen receptor (ER) antagonist and GPR30 agonist thatinduces apoptosis and autophagy.
Formule :C32H47F5O3SCouleur et forme :SolidMasse moléculaire :609.79Endoxifen E-isomer hydrochloride
CAS :Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).Formule :C25H28ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :409.95OP-1074
CAS :OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.Formule :C29H31NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.56DS20362725
CAS :DS20362725 is a selective estrogen-related receptor alpha (ERRα) agonist, commonly used in the study of metabolic disorders.Formule :C19H22N2O2Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :310.39Capesaris
CAS :Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.Formule :C19H13F2NO3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :341.31Bisphenol Z
CAS :Bisphenol Z is a bisphenol compound and high-performance monomer used in advanced engineering plastics, having antagonistic activity towards ERα.Formule :C18H20O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :268.35ERRγ Inverse Agonist 1
CAS :ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].Formule :C30H38Cl2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.54ERRα antagonist-1
CAS :ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα).Formule :C21H19N3S2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :377.53Norethisterone enanthate
CAS :Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.Formule :C27H38O3Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :410.59SIM-688
CAS :SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).Formule :C34H31F3N2O2Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :556.62NXT629
CAS :NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.Formule :C35H39N5O3SDegré de pureté :99.07% - 99.07%Couleur et forme :SolidMasse moléculaire :609.78Estrogen receptor antagonist 8
CAS :Estrogen Receptor Antagonist 8 is an ER antagonist with anti-uterine activity and may be used in the study of ovarian dysfunction.CASNETIN SODIUM (CasN)Formule :C25H21N3O4Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :427.45Zindoxifene
CAS :Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer.Formule :C21H21NO4Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :351.4Palazestrant
CAS :Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.Formule :C28H36FN3ODegré de pureté :97.55%Couleur et forme :SolidMasse moléculaire :449.6Ref: TM-T72945
1mg87,00€5mg159,00€10mg226,00€25mg378,00€50mg547,00€100mg747,00€1mL*10mM (DMSO)170,00€LY88074
CAS :LY88074, a raloxifene analog sans basic side chain, is an ERβ agonist (EC50 = 232 nM) that promotes uterine cell growth.
Formule :C21H14O4SDegré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :362.4H3B-6545
CAS :H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.Formule :C30H29F4N5O2Couleur et forme :SolidMasse moléculaire :567.58ERRα antagonist-2
CAS :ERRα antagonist-2 is an estrogen-related receptor α inverse agonist, inhibiting migration and invasion in ER-negative MDA-MB-231,breast cancer.Formule :C19H16N2O6SDegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :400.41(E/Z)-GSK5182
CAS :GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Formule :C27H31NO3Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T7709
1mg77,00€5mg167,00€10mg260,00€25mg477,00€50mg707,00€100mg1.063,00€1mL*10mM (DMSO)177,00€ERB-196
CAS :Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.Formule :C17H10FNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.27
![Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9800.webp&w=3840&q=75)
